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Bioorganic and Medicinal Chemistry

Volumn 23, Issue 16, 2015, Pages 5098-5119

Quinoline-based antimalarial hybrid compounds

(2) Vandekerckhove, Stéphanie a D'Hooghe, Matthias a

a GHENT UNIVERSITY (Belgium)

Author keywords

Antimalarial agents; Hybrids; Quinolines

Indexed keywords

7 CHLOROQUINOLINE CHALCONE; 7 CHLOROQUINOLINE GAMMA LACTAM ANTIBIOTIC; ANTIMALARIAL AGENT; ARTEMISININ; ARTESUNATE; CARBAPENEM DERIVATIVE; CEPHALOSPORIN DERIVATIVE; CHALCONE DERIVATIVE; CHLOROQUINE; DIHYDROARTEMISININ; FERROCENE DERIVATIVE; GLUTATHIONE; MALARIA VACCINE; MONOBACTAM DERIVATIVE; PIPERAZINE DERIVATIVE; PROTEIN DISULFIDE REDUCTASE (GLUTATHIONE); PYRIMETHAMINE; QUINOLINE; RHODANINE; SULFADOXINE; UNCLASSIFIED DRUG; QUINOLINE DERIVATIVE;

AMINATION; ANTIMALARIAL ACTIVITY; ARTICLE; COVALENT BOND; CROSS RESISTANCE; DISEASE ERADICATION; DRUG BIOAVAILABILITY; DRUG CYTOTOXICITY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TRANSFORMATION; ELECTRON TRANSPORT; HUMAN; ISOMERISM; LIPOPHILICITY; LOW DRUG DOSE; MALARIA; MEDICINAL CHEMISTRY; NONHUMAN; PLASMODIUM BERGHEI; PLASMODIUM FALCIPARUM; POLYMERIZATION; PROTEIN DEGRADATION; PROTEIN EXPRESSION; PROTEIN MOTIF; ANIMAL; CHEMISTRY; DRUG DEVELOPMENT; DRUG EFFECTS; PLASMODIUM; PROCEDURES; SYNTHESIS;

PLASMODIUM PARASITES;

ANIMALS; ANTIMALARIALS; DRUG DISCOVERY; HUMANS; MALARIA; PLASMODIUM; QUINOLINES;

EID: 84938991910 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2014.12.018 Document Type: Article

Times cited : (190)

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