Recent advances in malaria drug discovery

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 10, 2013, Pages 2829-2843

  Biamonte, Marco A ^a   Wanner, Jutta ^b   Le Roch, Karine G ^c  

^a Signal Pharmaceuticals   (United States)

^b HOFFMANN LA ROCHE INC   (United States)

^c UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

Malaria Antimalarial Plasmodium Drugs Review

Indexed keywords

4,6 DIAMINO 1,2 DIHYDRO 2,2 DIMETHYL 1 [3 (2,4,5 TRICHLOROPHENOXY)PROPOXY] 1,3,5 TRIAZINE; ACT 213615; ALBITIAZOLIUM BROMIDE; AMODIAQUINE; ANTIMALARIAL AGENT; ARTEMETHER; ARTEMETHER PLUS BENFLUMETOL; ARTEMISININ; ARTEMISONE; ARTEROLANE; ARTESUNATE; ATOVAQUONE PLUS PROGUANIL; BENFLUMETOL; BENZIMIDAZOLE; CDRI 97 78; CHLOROQUINE; CYCLOGUANIL; DIHYDROARTEMISININ PLUS PIPERAQUINE; DSM 190; DSM 265; DU 1302; GENZ 668764; GNF 156; GNF 179; GNF PF 5069; GSK 369796; GW 844520; ICI 56 780; MEFLOQUINE; ML 238; N (1 BENZYL 4 PIPERIDINYL) 2 (HEXAHYDRO 4 METHYL 1H 1,4 DIAZEPIN 1 YL) 6,7 DIMETHOXY 4 QUINAZOLINAMINE; N TERT BUTYL ISOQUINE; NAPHTHOQUINE; NITD 609; NITD 731; OZ 439; P 218; PIPERAQUINE; PRIMAQUINE; PYRIMETHAMINE; PYRIMETHAMINE PLUS SULFADOXINE; QUINOLINE DERIVATIVE; RKA 182; SL 2 25; SSJ 183; TDR 84420; TIPRANAVIR; TM 2 115; UNCLASSIFIED DRUG; UNINDEXED DRUG; WR621308;

AGRANULOCYTOSIS; ANTIMALARIAL ACTIVITY; ANTIPROTOZOAL ACTIVITY; BONE MARROW TOXICITY; DEPRESSION; DOSE RESPONSE; DRUG ABSORPTION; DRUG BLOOD LEVEL; DRUG COST; DRUG ELIMINATION; DRUG HALF LIFE; DRUG MEGADOSE; DRUG METABOLISM; DRUG POTENCY; DRUG RESEARCH; DRUG STRUCTURE; DRUG TOLERABILITY; HEPATITIS; HUMAN; IC 50; LIFE CYCLE; MALARIA; MALARIA CONTROL; NIGHTMARE; NONHUMAN; PATIENT COMPLIANCE; PLASMODIUM FALCIPARUM; PLASMODIUM KNOWLESI; PLASMODIUM MALARIAE; PLASMODIUM OVALE; PLASMODIUM VIVAX; PREGNANT WOMAN; PSYCHOSIS; RELAPSE; REVIEW; SINGLE DRUG DOSE;

ANIMALS; ANTIMALARIALS; DRUG DISCOVERY; HUMANS; LIVER; LIVER TRANSPLANTATION; MALARIA; MOLECULAR STRUCTURE;

EID: 84876685433     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.03.067     Document Type: Review

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