메뉴 건너뛰기




Volumn 19, Issue 4, 2012, Pages 488-517

Developments in chemical approaches to treat tuberculosis in the last decade

Author keywords

Antitubercular agents; Arabinogalactan; Chemotherapy; Extensively drug resistance (XDR); Fatty acid synthase; MultiDrug Resistance (MDR); Mycobacterium tuberculosis; Mycolic acid; Peptidoglycan; Tuberculosis (TB)

Indexed keywords

6,7 DIHYDRO 2 NITRO 6 (4 TRIFLUOROMETHOXYBENZYLOXY) 5H IMIDAZO[2,1 B][1,3]OXAZINE; AMIKACIN; AMINOSALICYLIC ACID; BEDAQUILINE; BENZOTHIAZOLINE DERIVATIVE; CAPREOMYCIN; CIPROFLOXACIN; CYCLOSERINE; DELAMANID; DIAMINE DERIVATIVE; ETHAMBUTOL; ETHIONAMIDE; GATIFLOXACIN; ISONIAZID; KANAMYCIN; LEVOFLOXACIN; LINEZOLID; MOXIFLOXACIN; N (2 ADAMANTYL) N' GERANYLETHYLENEDIAMINE; PROTIONAMIDE; PYRAZINAMIDE; PYRROLE DERIVATIVE; QUINOLINE DERIVATIVE; RIFAMPICIN; STREPTOMYCIN; SULFONYLUREA DERIVATIVE; SUTEZOLID; THIOLACTOMYCIN; TUBERCULOSTATIC AGENT; UNINDEXED DRUG;

EID: 84863421391     PISSN: 09298673     EISSN: 1875533X     Source Type: Journal    
DOI: 10.2174/092986712798918815     Document Type: Article
Times cited : (15)

References (385)
  • 1
    • 31344478259 scopus 로고    scopus 로고
    • Robert Koch and the white death: From tuberculosis to tuberculin
    • DOI 10.1016/j.micinf.2005.06.004, PII S1286457905002297
    • Gradmann, C. Robert Koch and the white death: From tuberculosis to tuberculin. Microbes. Infect., 2006, 8, 294-301. (Pubitemid 43139318)
    • (2006) Microbes and Infection , vol.8 , Issue.1 , pp. 294-301
    • Gradmann, C.1
  • 2
    • 84863413173 scopus 로고    scopus 로고
    • 2010/2011 Tuberculosis Global Facts, November 2010
    • 2010/2011 Tuberculosis Global Facts, http://www.who.int/tb/publications/ global-report/en/index.html (November 2010
  • 3
    • 84863411019 scopus 로고    scopus 로고
    • World Health Organization (2008). "Countries with XDR-TB confirmed cases as of June 2008
    • World Health Organization (2008). "Countries with XDR-TB confirmed cases as of June 2008. www.who.int/tb/challenges/xdr/xdr-map-june08.
  • 4
    • 77952326903 scopus 로고    scopus 로고
    • The population dynamics and control of tuberculosis
    • Dye, C.; Williams, B.G. The Population Dynamics and Control of Tuberculosis. Science, 2010, 328, 856-861.
    • (2010) Science , vol.328 , pp. 856-861
    • Dye, C.1    Williams, B.G.2
  • 6
    • 77952356637 scopus 로고    scopus 로고
    • Tuberculosis: What we don't know can, and does, hurt us
    • Russell, D.G.; Barry 3rd, C.E.; Flynn, J.L. Tuberculosis: What We Don't Know Can, and Does, Hurt Us. Science, 2010, 328, 852-856.
    • (2010) Science , vol.328 , pp. 852-856
    • Russell, D.G.1    Barry III, C.E.2    Flynn, J.L.3
  • 8
    • 77951745983 scopus 로고    scopus 로고
    • Combined drug medium with isoniazid and rifampicin for identification of multi-drugresistant mycobacterium tuberculosis
    • Nalini, S.L.; Devika, R.K.; Ravikumar, D.; Ramachandran, R. Combined drug medium with isoniazid and rifampicin for identification of multi-drugresistant mycobacterium tuberculosis. Indian J. Med. Microbiol., 2010, 28(2), 162-163.
    • (2010) Indian J. Med. Microbiol. , vol.28 , Issue.2 , pp. 162-163
    • Nalini, S.L.1    Devika, R.K.2    Ravikumar, D.3    Ramachandran, R.4
  • 10
    • 77951242451 scopus 로고    scopus 로고
    • Diagnosis and follow-up of treatment of latent tuberculosis; the utility of the Quantiferon-TB Gold In-tube assay in outpatients from a tuberculosis low-endemic country
    • Dyrhol-Riise, A.M.; Gran, G.; Wenzel-Larsen, T.; Blomberg, B.; Haanshuus, C.G.; Moerkve, O. Diagnosis and follow-up of treatment of latent tuberculosis; the utility of the Quantiferon-TB Gold In-tube assay in outpatients from a tuberculosis low-endemic country. BMC Infectious Diseases, 2010, 10, 1471-2334.
    • (2010) BMC Infectious Diseases , vol.10 , pp. 1471-2334
    • Dyrhol-Riise, A.M.1    Gran, G.2    Wenzel-Larsen, T.3    Blomberg, B.4    Haanshuus, C.G.5    Moerkve, O.6
  • 11
    • 84863411017 scopus 로고    scopus 로고
    • Method of prognosis and/or diagnosing an irs in a patient infected with M. tuberculosis, and optionally hiv
    • WO2010089377, December
    • Autran, B. Method of Prognosis and/or Diagnosing an Irs in A Patient Infected with M. tuberculosis, and Optionally Hiv, PCT Int. Appl, WO2010089377, December, 2010.
    • (2010) PCT Int. Appl
    • Autran, B.1
  • 13
    • 10444227369 scopus 로고    scopus 로고
    • Fighting tuberculosis: An old disease new challenges
    • DOI 10.1002/med.20017
    • Tripathi, R.P.; Tewari, N.; Dwivedi, N.; Tiwari, V.K. Fighting tuberculosis: An old disease with new challenges. Med. Res. Rev., 2005, 25, 93-131. (Pubitemid 39642233)
    • (2005) Medicinal Research Reviews , vol.25 , Issue.1 , pp. 93-131
    • Tripathi, R.P.1    Tewari, N.2    Dwivedi, N.3    Tiwari, V.K.4
  • 15
    • 33847681052 scopus 로고    scopus 로고
    • Antituberculosis drugs: Ten years of research
    • DOI 10.1016/j.bmc.2007.01.030, PII S0968089607000442
    • Janin, Y.L. Antituberculosis drugs: Ten years of research. Bioorg. Med. Chem., 2007, 15, 2479-2513. (Pubitemid 46367698)
    • (2007) Bioorganic and Medicinal Chemistry , vol.15 , Issue.7 , pp. 2479-2513
    • Janin, Y.L.1
  • 16
    • 0033637727 scopus 로고    scopus 로고
    • Main directions in the search for new antituberculous drugs (review
    • Kayukova, L.A.; Praliev, K.D. Main directions in the search for new antituberculous drugs (review). Pharm. Chem. J., 2000, 34, 11-18.
    • (2000) Pharm. Chem. J. , vol.34 , pp. 11-18
    • Kayukova, L.A.1    Praliev, K.D.2
  • 17
    • 0033842495 scopus 로고    scopus 로고
    • A review of antimycobacterial natural products
    • DOI 10.1002/1099-1573(200008)14:5<303::AID-PTR712>3.0.CO;2-N
    • Newton, S.M.; Lau, C.; Wright, C.W. A review of antimycobacterial natural products. Phytother. Res., 2002, 14, 303-322. (Pubitemid 30655514)
    • (2000) Phytotherapy Research , vol.14 , Issue.5 , pp. 303-322
    • Newton, S.M.1    Lau, C.2    Wright, C.W.3
  • 18
    • 0347063673 scopus 로고    scopus 로고
    • Antimycobacterial natural products
    • DOI 10.1039/b212154a
    • Copp, B.R. Antimycobacterial natural products. Nat. Prod. Rep., 2003, 20, 535-557. (Pubitemid 38024760)
    • (2003) Natural Product Reports , vol.20 , Issue.6 , pp. 535-557
    • Copp, B.R.1
  • 19
    • 2142639382 scopus 로고    scopus 로고
    • Natural antimycobacterial metabolites: Current status
    • DOI 10.1016/j.phytochem.2004.02.013, PII S003194220400086X
    • Okunade, A.L.; Elwin-Lewis, M.P.F.; Lewis, W.H. Natural antimycobacterial metabolites: Current status. Phytochemistry, 2004, 65, 1017-1032. (Pubitemid 38542737)
    • (2004) Phytochemistry , vol.65 , Issue.8 , pp. 1017-1032
    • Okunade, A.L.1    Elvin-Lewis, M.P.F.2    Lewis, W.H.3
  • 21
    • 77955500148 scopus 로고    scopus 로고
    • Antitubercular potential of plants: A brief account of some important molecules
    • Negi, A.S.; Kumar, J.K.; Luqman, S.; Saikia, D.; Khanuja, S.P.S. Antitubercular Potential of Plants: A Brief Account of Some Important Molecules. Med. Res. Rev., 2010, 30(4), 603-645.
    • (2010) Med. Res. Rev. , vol.30 , Issue.4 , pp. 603-645
    • Negi, A.S.1    Kumar, J.K.2    Luqman, S.3    Saikia, D.4    Khanuja, S.P.S.5
  • 22
    • 77953331533 scopus 로고    scopus 로고
    • Anti-tuberculosis activity of selected medicinal plants against multi-drug resistant Mycobacterium tuberculosis isolates
    • Gupta, R.; Thakur, B.; Singh, P.; Singh, H.B.; Sharma, V.D.; Katoch, V.M.; Chauhan, S.V.S. Anti-tuberculosis activity of selected medicinal plants against multi-drug resistant Mycobacterium tuberculosis isolates. Indian J. Med. Res., 2010, 131, 809-813.
    • (2010) Indian J. Med. Res. , vol.131 , pp. 809-813
    • Gupta, R.1    Thakur, B.2    Singh, P.3    Singh, H.B.4    Sharma, V.D.5    Katoch, V.M.6    Chauhan, S.V.S.7
  • 23
    • 77449132175 scopus 로고    scopus 로고
    • An antimycobacterial cyclodepsipeptide from the entomopathogenic fungus ophiocordycepscommunis BCC 16475
    • Haritakun, R.; Sappan, M.; Suvannakad, R.; Tasanathai, K.; Isaka, M. An Antimycobacterial Cyclodepsipeptide from the Entomopathogenic Fungus Ophiocordycepscommunis BCC 16475. J. Nat. Prod., 2010, 73, 75-78.
    • (2010) J. Nat. Prod. , vol.73 , pp. 75-78
    • Haritakun, R.1    Sappan, M.2    Suvannakad, R.3    Tasanathai, K.4    Isaka, M.5
  • 24
    • 77949664317 scopus 로고    scopus 로고
    • A new long-chain alkene and antituberculosis constituents from the leaves of pourthiaea lucida
    • Chen, J.J.; Lin, W.J.; Shieh, P.C.; Chen, I.S.; Peng, C.F.; Sung, P.J. A New Long-Chain Alkene and Antituberculosis Constituents from the Leaves of Pourthiaea lucida. Eichemistry & biodiversity, 2010, 7, 717-721.
    • (2010) Eichemistry & Biodiversity , vol.7 , pp. 717-721
    • Chen, J.J.1    Lin, W.J.2    Shieh, P.C.3    Chen, I.S.4    Peng, C.F.5    Sung, P.J.6
  • 25
    • 77955551505 scopus 로고    scopus 로고
    • A bioactive labdane diterpenoid from Curcuma amada and its semisynthetic analogues as antitubercular agents
    • Singh, S.; Kumar, J.K.; Shanker, D.S.K.; Thakur, J.P.; Negi, A.S.; Banerjee, S. A bioactive labdane diterpenoid from Curcuma amada and its semisynthetic analogues as antitubercular agents. Eur. J. Med. Chem., 2010, 45, 4379-4382.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 4379-4382
    • Singh, S.1    Kumar, J.K.2    Shanker, D.S.K.3    Thakur, J.P.4    Negi, A.S.5    Banerjee, S.6
  • 28
    • 77953017562 scopus 로고    scopus 로고
    • Secondary metabolites from the roots of litsea hypophaea and their antitubercular activity
    • Pan, P.C.; Cheng, M.J.; Peng, C.F.; Huang, H.Y.; Chen, J.J.; Chen, I.S. Secondary Metabolites from the Roots of Litsea hypophaea and Their Antitubercular Activity. J. Nat. Prod., 2010, 73, 890-896.
    • (2010) J. Nat. Prod. , vol.73 , pp. 890-896
    • Pan, P.C.1    Cheng, M.J.2    Peng, C.F.3    Huang, H.Y.4    Chen, J.J.5    Chen, I.S.6
  • 29
    • 77955274098 scopus 로고    scopus 로고
    • Evaluation of flavonoids from Dorstenia barteri for their antimycobacterial, antigonorrheal and anti-reverse transcriptase activities
    • Kuete, V.; Ngameni, B.; Mbaveng, A.T.; Ngadjui, B.; Marion, M.J.J.; Lall, N. Evaluation of flavonoids from Dorstenia barteri for their antimycobacterial, antigonorrheal and anti-reverse transcriptase activities. Acta Tropica 2010, 116(1), 100-104.
    • (2010) Acta Tropica , vol.116 , Issue.1 , pp. 100-104
    • Kuete, V.1    Ngameni, B.2    Mbaveng, A.T.3    Ngadjui, B.4    Marion, M.J.J.5    Lall, N.6
  • 31
    • 1842843660 scopus 로고    scopus 로고
    • Recent advances towards identification of new drug targets for Mycobacterium tuberculosis
    • DOI 10.1517/14728222.8.2.79
    • Sharma, K.; Chopra, P.; Singh, Y. Recent advances towards identification of new drug targets for Mycobacterium tuberculosis. Expert Opin. Ther. Targets, 2004, 8(2), 79-93. (Pubitemid 38489535)
    • (2004) Expert Opinion on Therapeutic Targets , vol.8 , Issue.2 , pp. 79-93
    • Sharma, K.1    Chopra, P.2    Singh, Y.3
  • 32
    • 0036220660 scopus 로고    scopus 로고
    • Tuberculosis drug targets
    • Zhang, Y.; Amzel, L. M. Tuberculosis Drug Targets. Curr. Drug Targets, 2002, 3, 131-154. (Pubitemid 34296204)
    • (2002) Current Drug Targets , vol.3 , Issue.2 , pp. 131-154
    • Zhang, Y.1    Amzel, L.M.2
  • 33
    • 0001995201 scopus 로고    scopus 로고
    • Approaches to tuberculosis drug development
    • Hatfull GF, Jacobs WRJ (Ed.), ASM Press, Washington DC
    • Duncan, K.; Sacchettini, J.C. Approaches to tuberculosis drug development. Molecular genetics of mycobacteria. In: Hatfull GF, Jacobs WRJ (Ed.), ASM Press, Washington DC, 2000, pp. 297-307.
    • (2000) Molecular Genetics of Mycobacteria , pp. 297-307
    • Duncan, K.1    Sacchettini, J.C.2
  • 34
    • 0347481469 scopus 로고    scopus 로고
    • Mycobacterium tuberculosis: A model system for structural genomics
    • DOI 10.1016/j.sbi.2003.10.004
    • Smith, C.V.; Sacchettini, J.C. Mycobacterium tuberculosis a model system for structural genomics. Curr. Opin. Struct. Biol., 2003, 13, 658-664. (Pubitemid 37522140)
    • (2003) Current Opinion in Structural Biology , vol.13 , Issue.6 , pp. 658-664
    • Smith, C.V.1    Sacchettini, J.C.2
  • 35
    • 4644349770 scopus 로고    scopus 로고
    • Identification and validation of novel drug targets in tuberculosis
    • DOI 10.2174/1381612043383223
    • Duncan, K. Identification and validation of novel drug targets in tuberculosis. Curr. Pharm. Des.; 2004, 10, 3185-3194. (Pubitemid 39276608)
    • (2004) Current Pharmaceutical Design , vol.10 , Issue.26 , pp. 3185-3194
    • Duncan, K.1
  • 36
    • 22544449537 scopus 로고    scopus 로고
    • Recent advances in new structural classes of anti-tuberculosis agents
    • DOI 10.2174/0929867054546654
    • Nayyar, A.; Jain, R. Recent Advances in New Structural Classes of Anti-Tuberculosis Agents. Curr. Med. Chem., 2005, 12, 1873-1886. (Pubitemid 41015184)
    • (2005) Current Medicinal Chemistry , vol.12 , Issue.16 , pp. 1873-1886
    • Nayyar, A.1    Jain, R.2
  • 37
    • 33748419613 scopus 로고    scopus 로고
    • Novel targets for tuberculosis drug discovery
    • DOI 10.1016/j.coph.2006.06.004, PII S1471489206001354, Anti-infectives/New Technologies
    • Mdluli, K.; Spigelman, M. Novel targets for tuberculosis drug discovery. Curr. Opin. Pharmacol., 2006, 6 (5), 459-467. (Pubitemid 44340669)
    • (2006) Current Opinion in Pharmacology , vol.6 , Issue.5 , pp. 459-467
    • Mdluli, K.1    Spigelman, M.2
  • 38
    • 33747852367 scopus 로고    scopus 로고
    • Current status of some antituberculosis drugs and the development of new antituberculous agents with special reference to their in vitro and in vivo antimicrobial activities
    • DOI 10.2174/138161206778743646
    • Tomioka, H. Current status of some antituberculosis drugs and the development of new antituberculous agents with special reference to their in vitro and in vivo antimicrobial activities. Curr. Pharm. Des., 2006, 12, 4047-4070. (Pubitemid 44669760)
    • (2006) Current Pharmaceutical Design , vol.12 , Issue.31 , pp. 4047-4070
    • Tomioka, H.1
  • 39
    • 33750077287 scopus 로고    scopus 로고
    • Tuberculosis: Current treatment and new drug development
    • Liu, J.; Ren, H.P. Tuberculosis current treatment and New Drug development Anti-Infective Agents Med. Chem., 2006, 5, 331-344. (Pubitemid 44574832)
    • (2006) Anti-Infective Agents in Medicinal Chemistry , vol.5 , Issue.4 , pp. 331-344
    • Liu, J.1    Ren, H.P.2
  • 40
    • 77954957267 scopus 로고    scopus 로고
    • Eicosanoid pathways regulate adaptive immunity to Mycobacterium tuberculosis
    • Maziar, D.; Danielle, D.; Claudio, N.A.; Remold, H.G.; Behar, S.M. Eicosanoid pathways regulate adaptive immunity to Mycobacterium tuberculosis. Nat. Immunol., 2010, 11(8), 751-758.
    • (2010) Nat. Immunol. , vol.11 , Issue.8 , pp. 751-758
    • Maziar, D.1    Danielle, D.2    Claudio, N.A.3    Remold, H.G.4    Behar, S.M.5
  • 41
    • 77955661920 scopus 로고    scopus 로고
    • Evasion of innate immunity by Mycobacterium tuberculosis: Is death an exit strategy?
    • Behar, S.M.; Divangahi, M.; Remold, H.G. Evasion of innate immunity by Mycobacterium tuberculosis: Is death an exit strategy? Nat. Rev. Microbiol., 2010, 8(9), 668-674.
    • (2010) Nat. Rev. Microbiol. , vol.8 , Issue.9 , pp. 668-674
    • Behar, S.M.1    Divangahi, M.2    Remold, H.G.3
  • 42
    • 11144229891 scopus 로고
    • The actinomycins and their importance in the treatment of tumors in animals and man. Historical background
    • Woodruff, H.B.; Waksman, S.A. The actinomycins and their importance in the treatment of tumors in animals and man. Historical background. Ann. N.Y. Acad. Sci., 1960, 89, 287-298.
    • (1960) Ann. N.Y. Acad. Sci. , vol.89 , pp. 287-298
    • Woodruff, H.B.1    Waksman, S.A.2
  • 43
    • 42949096272 scopus 로고
    • The first clinical trial of streptomycin in human tuberculosis
    • Lehmann, J. The first clinical trial of streptomycin in human tuberculosis. Dis. Chest, 1949, 16, 684-703.
    • (1949) Dis. Chest , vol.16 , pp. 684-703
    • Lehmann, J.1
  • 44
    • 33644535147 scopus 로고    scopus 로고
    • Natural products-The future scaffolds for novel antibiotics?
    • Mark, S.B.; Antony, D.B. Natural products-The future scaffolds for novel antibiotics? Biochem. Pharmacol., 2006, 71, 919-929.
    • (2006) Biochem. Pharmacol. , vol.71 , pp. 919-929
    • Mark, S.B.1    Antony, D.B.2
  • 45
    • 0014653136 scopus 로고
    • Successes and failures in the search for antibiotics
    • Waksman, S.A. Successes and Failures in the search for Antibiotics. Ad. Appl. Microbiol., 1969, 11, 1-16.
    • (1969) Ad. Appl. Microbiol. , vol.11 , pp. 1-16
    • Waksman, S.A.1
  • 46
    • 42949135760 scopus 로고
    • Modern methods of chemotherapy of tuberculosis
    • Domagk, G. Modern methods of chemotherapy of tuberculosis. An. R. Acad. Nac. Med. (Madr.)., 1952, 69, 504-513.
    • (1952) An. R. Acad. Nac. Med. (Madr. , vol.69 , pp. 504-513
    • Domagk, G.1
  • 48
    • 2942721689 scopus 로고
    • Cycloserine a new antibiotic, in the treatment of human pulmonary tuberculosis: A preliminary report
    • Epstein, I.G.; Nair, K.G.; Boyd, L.J. Cycloserine, a new antibiotic, in the treatment of human pulmonary tuberculosis: A preliminary report. Antibiot. Med. Clin. Ther., 1955, 1, 80-93.
    • (1955) Antibiot. Med. Clin. Ther. , vol.1 , pp. 80-93
    • Epstein, I.G.1    Nair, K.G.2    Boyd, L.J.3
  • 49
    • 14844356959 scopus 로고    scopus 로고
    • Rifamycin - Mode of action, resistance, and biosynthesis
    • DOI 10.1021/cr030112j
    • Floss, H.G.; Yu, T.W. Rifamycin: Mode of Action, Resistance, and Biosynthesis. Chem. Rev., 2005, 105, 621-632. (Pubitemid 40351636)
    • (2005) Chemical Reviews , vol.105 , Issue.2 , pp. 621-632
    • Floss, H.G.1    Yu, T.-W.2
  • 50
    • 11144250804 scopus 로고    scopus 로고
    • Tuberculosis - Metabolism and respiration in the absence of growth
    • DOI 10.1038/nrmicro1065
    • Boshoff, I.M.; Barry, C.E. III. Tuberculosiss Metabolism and respiration in the absence of growth. Nat. Rev. Microbiol., 2005, 3, 70-80. (Pubitemid 40028470)
    • (2005) Nature Reviews Microbiology , vol.3 , Issue.1 , pp. 70-80
    • Boshoff, H.I.M.1    Barry III, C.E.2
  • 53
    • 0037871813 scopus 로고    scopus 로고
    • Treatment of tuberculosis
    • American Thoracic Society Centers for Disease Control and Prevention and Infectious Diseases Society of America
    • American Thoracic Society, Centers for Disease Control and Prevention and Infectious Diseases Society of America. Treatment of tuberculosis. MMWR 52, 1-77 (2003
    • (2003) MMWR , vol.52 , pp. 1-77
  • 55
  • 56
    • 84863411020 scopus 로고    scopus 로고
    • World Health Organization, Treatment of Tuberculosis Guidelines. & http://www.who.int/tb.xdr/faqs/en/ (2007
    • World Health Organization, Treatment of Tuberculosis Guidelines. http://www.who. int/tb/publications/cds-tb-2003-313/en/index.html & http://www.who.int/tb.xdr/faqs/en/ (2007
  • 57
    • 0347722525 scopus 로고    scopus 로고
    • TB drug discovery: Addressing issues of persistence and resistance
    • DOI 10.1016/j.tube.2003.08.019
    • Smith, C.V.; Sharma, V.; Sacchettini, J.C. TB drug discovery: Addressing issues of persistence and resistance. Tuberculosis (Edinb.), 2004, 84, 45-55. (Pubitemid 38082932)
    • (2004) Tuberculosis , vol.84 , Issue.1-2 , pp. 45-55
    • Smith, C.V.1    Sharma, V.2    Sacchettini, J.C.3
  • 59
    • 0028008721 scopus 로고
    • Infection caused by Mycobacterium tuberculosis
    • Peloquin, C.A.; Berning, S.E. Infection caused by Mycobacterium tuberculosis. Ann. Pharmacother., 1994, 28, 72-84. (Pubitemid 24042494)
    • (1994) Annals of Pharmacotherapy , vol.28 , Issue.1 , pp. 72-84
    • Peloquin, C.A.1    Berning, S.E.2
  • 60
    • 33845349993 scopus 로고    scopus 로고
    • An evaluation of data quality in a network for surveillance of Mycobacterium tuberculosis resistance to antituberculosis drugs in Ile-de-France region-2001-2002
    • DOI 10.1007/s10654-006-9069-y
    • Guerrin-Tran, E.; Thiolet, J.M.; Rousseau, C.; Henry, S.; Poirier, C.; Che, D.; Vinas, J.M.; Jarlier, V.; Robert, J. An evaluation of data quality in a network for surveillance of Mycobacterium tuberculosis resistance to antituberculosis drugs in Ile-de-France region-2001-2002. Eur. J. Epidemiol., 2006, 21, 783-785. (Pubitemid 44885199)
    • (2006) European Journal of Epidemiology , vol.21 , Issue.10 , pp. 783-785
    • Guerrin-Tran, E.1    Thiolet, J.-M.2    Rousseau, C.3    Henry, S.4    Poirier, C.5    Che, D.6    Vinas, J.-M.7    Jarlier, V.8    Robert, J.9
  • 61
    • 0031781994 scopus 로고    scopus 로고
    • Tuberculosis and HIV infection: A global perspective
    • DOI 10.1159/000029291
    • Murray, J.F. Tuberculosis and HIV Infection: A Global Perspective. Respiration, 1998, 65, 335-342. (Pubitemid 28491266)
    • (1998) Respiration , vol.65 , Issue.5 , pp. 335-342
    • Murray, J.F.1
  • 64
    • 17744419324 scopus 로고    scopus 로고
    • National Survey of Tuberculosis in England and Wales
    • National Survey of Tuberculosis in England and Wales. Communicable Dis. Rep. Wkly. 8, 209-212 (1998
    • (1998) Communicable Dis. Rep. Wkly. , vol.8 , pp. 209-212
  • 65
    • 33748893668 scopus 로고    scopus 로고
    • Infectious disease: Extensively drug-resistant TB gets foothold in South Africa
    • Cohen, J. Infectious disease: Extensively Drug-Resistant TB Gets Foothold in South Africa. Science, 2006, 313, 1554.
    • (2006) Science , vol.313 , pp. 1554
    • Cohen, J.1
  • 66
    • 33645119729 scopus 로고    scopus 로고
    • Emergence of mycobacterium tuberculosis with extensive resistance to second line drugs worldwide 2000-2004
    • Wright, A. Emergence of Mycobacterium tuberculosis with Extensive Resistance to Second Line Drugs Worldwide 2000-2004. MMWR. 2006, 55, 301-305.
    • (2006) MMWR , vol.55 , pp. 301-305
    • Wright, A.1
  • 67
    • 77949416435 scopus 로고    scopus 로고
    • New tuberculosis lab hailed as breakthrough in health diplomacy
    • Stone, R. New Tuberculosis Lab Hailed as Breakthrough in Health Diplomacy. Science, 2010, 327, 1312-1313.
    • (2010) Science , vol.327 , pp. 1312-1313
    • Stone, R.1
  • 68
    • 77952880349 scopus 로고    scopus 로고
    • The HIV-associated tuberculosis epidemic-when will we act?
    • Harries, A.D.; Zachariah, R.; Corbett, E.L. The HIV-associated tuberculosis epidemic-when will we act? The Lancet, 2010, 375, 1906-1919.
    • (2010) The Lancet , vol.375 , pp. 1906-1919
    • Harries, A.D.1    Zachariah, R.2    Corbett, E.L.3
  • 71
    • 0036774642 scopus 로고    scopus 로고
    • Re-annotation of the genome sequence of Mycobacterium tuberculosis H37Rv
    • Camus, J.C.; Pryor, M.J.; Medigue, C.; Cole, S.T. Re-annotation of the genome sequence of Mycobacterium tuberculosis H37Rv. Microbiology, 2002, 148, 2967-2973. (Pubitemid 35243696)
    • (2002) Microbiology , vol.148 , Issue.10 , pp. 2967-2973
    • Camus, J.-C.1    Pryor, M.J.2    Medigue, C.3    Cole, S.T.4
  • 73
    • 77950787126 scopus 로고    scopus 로고
    • Dynamic active-site protection by the M. tuberculosis protein tyrosine phosphatase ptpb lid domain
    • Flynn, E.M.; Hanson, J.A.; Alber, T.; Yang, H. Dynamic Active-Site Protection by the M. tuberculosis Protein Tyrosine Phosphatase PtpB Lid Domain. J. Am. Chem. Soc., 2010, 132, 4772-4780.
    • (2010) J. Am. Chem. Soc. , vol.132 , pp. 4772-4780
    • Flynn, E.M.1    Hanson, J.A.2    Alber, T.3    Yang, H.4
  • 75
    • 77955574023 scopus 로고    scopus 로고
    • Identification of thiazolidinones spiro-fused to indolin-2-ones as potent and selective inhibitors of the mycobacterium tuberculosis protein tyrosine phosphatase B
    • Vintonyak, V.V.; Warburg, K.; Kruse, H.; Grimme, S.; Hübel, K.; Rauh, D.; Waldmann, H. Identification of Thiazolidinones Spiro-Fused to Indolin-2-ones as Potent and Selective Inhibitors of the Mycobacterium tuberculosis Protein Tyrosine Phosphatase B. Angew. Chem. Int. Ed., 2010, 49, 5902-5905.
    • (2010) Angew. Chem. Int. Ed. , vol.49 , pp. 5902-5905
    • Vintonyak, V.V.1    Warburg, K.2    Kruse, H.3    Grimme, S.4    Hübel, K.5    Rauh, D.6    Waldmann, H.7
  • 76
    • 77953138509 scopus 로고    scopus 로고
    • Inhibition of Mycobacterium tuberculosis tyrosine phosphatase PtpA by synthetic chalcones: Kinetics, molecular modeling, toxicity and effect on growth
    • Mascarello, A.; Chiaradia, L.D.; Vernal, J.; Grimme, S.; Hübel, K.; Rauh, D.; Waldmann, H. Inhibition of Mycobacterium tuberculosis tyrosine phosphatase PtpA by synthetic chalcones: Kinetics, molecular modeling, toxicity and effect on growth. Bioorg. Med. Chem., 2010, 18, 3783-3789.
    • (2010) Bioorg. Med. Chem. , vol.18 , pp. 3783-3789
    • Mascarello, A.1    Chiaradia, L.D.2    Vernal, J.3    Grimme, S.4    Hübel, K.5    Rauh, D.6    Waldmann, H.7
  • 77
    • 77950862522 scopus 로고    scopus 로고
    • Expression and characterization of Mycobacterium tuberculosis methionine aminopeptidase type
    • Lu, J.P.; Ye, Q.Z. Expression and characterization of Mycobacterium tuberculosis methionine aminopeptidase type. Bioor. Med. Chem. Lett., 2010, 20, 2776-2779.
    • (2010) Bioor. Med. Chem. Lett. , vol.20 , pp. 2776-2779
    • Lu, J.P.1    Ye, Q.Z.2
  • 80
    • 77954600569 scopus 로고    scopus 로고
    • New molecular scaffolds for the design of Mycobacterium tuberculosis type II dehydroquinase inhibitors identified using ligand and receptor based virtual screening
    • Kumar, A.; Siddiqi, M.I.; Miertus, S. New molecular scaffolds for the design of Mycobacterium tuberculosis type II dehydroquinase inhibitors identified using ligand and receptor based virtual screening. J. Mol. Model., 2010, 16, 693-712.
    • (2010) J. Mol. Model. , vol.16 , pp. 693-712
    • Kumar, A.1    Siddiqi, M.I.2    Miertus, S.3
  • 81
    • 77950816491 scopus 로고    scopus 로고
    • Optimization of the interligand overhauser effect for fragment linking: Application to inhibitor discovery against mycobacterium tuberculosis pantothenate synthetase
    • Sledz, P.; Silvestre, H.L.; Hung, A.W.; Ciulli, A.; Blundell, T.L.; Abell, C. Optimization of the Interligand Overhauser Effect for Fragment Linking: Application to Inhibitor Discovery against Mycobacterium tuberculosis Pantothenate Synthetase. J. Am. Chem. Soc., 2010, i 4544-4545.
    • (2010) J. Am. Chem. Soc. , vol.I , pp. 4544-4545
    • Sledz, P.1    Silvestre, H.L.2    Hung, A.W.3    Ciulli, A.4    Blundell, T.L.5    Abell, C.6
  • 83
    • 77953138779 scopus 로고    scopus 로고
    • Virtual screening, selection and development of a benzindolone structural scaffold for inhibition of lumazine synthase
    • Talukdar, A.; Morgunova, E.; Duan, J.; Meining, W.; Foloppe, N.; Nilsson, L. Virtual screening, selection and development of a benzindolone structural scaffold for inhibition of lumazine synthase. Bioorg. Med. Chem., 2010, 18, 3518-3534.
    • (2010) Bioorg. Med. Chem. , vol.18 , pp. 3518-3534
    • Talukdar, A.1    Morgunova, E.2    Duan, J.3    Meining, W.4    Foloppe, N.5    Nilsson, L.6
  • 84
    • 0000875326 scopus 로고    scopus 로고
    • Aminoglycosides and aminocyclitols
    • 7th Ed. Edinburgh: Churchill Livingstone
    • Phillips, I.; Shannon, K.P. Aminoglycosides and aminocyclitols. Antibiotic and Chemotherapy, 7th Ed. Edinburgh: Churchill Livingstone. 1997, pp. 164-201.
    • (1997) Antibiotic and Chemotherapy , pp. 164-201
    • Phillips, I.1    Shannon, K.P.2
  • 85
    • 0035018011 scopus 로고    scopus 로고
    • Formation of the glycan chains in the synthesis of bacterial peptidoglycan
    • Heijenoort, Jv. Formation of the glycan chains in the synthesis of bacterial peptidoglycan. Glycobiology, 2001, 11, 25-36.
    • (2001) Glycobiology , vol.11 , pp. 25-36
    • Heijenoort, J.V.1
  • 86
    • 76149108438 scopus 로고    scopus 로고
    • Exfoliative dermatitis to all four first line oral anti-tubercular drugs
    • Dua, R.; Sindhwani, G.; Rawat, J. Exfoliative Dermatitis to All Four First Line Oral Anti-Tubercular Drugs. Indian J. Tuberc.2010, 57, 53-56.
    • (2010) Indian J. Tuberc. , vol.57 , pp. 53-56
    • Dua, R.1    Sindhwani, G.2    Rawat, J.3
  • 89
    • 30744441922 scopus 로고    scopus 로고
    • Identification of an ABC transporter required for iron acquisition and virulence in Mycobacterium tuberculosis
    • DOI 10.1128/JB.188.2.424-430.2006
    • Rodriguez, G.; Smith, I. Identification of an ABC transporter required for iron acquisition and virulence in Mycobacterium tuberculosis. J. Bacteriol., 2006, 188, 424-430. (Pubitemid 43100529)
    • (2006) Journal of Bacteriology , vol.188 , Issue.2 , pp. 424-430
    • Rodriguez, G.M.1    Smith, I.2
  • 90
    • 0032703901 scopus 로고    scopus 로고
    • Cloning and expression of Mycobacterium tuberculosis and Mycobacterium leprae dihydropteroate synthase in Escherichia coli
    • Nopponpunth, V.; Sirawaraporn, W.; Greene, P.J.; Santi, D.V. Cloning and expression of Mycobacterium tuberculosis and Mycobacterium leprae dihydropteroate synthase in Escherichia coli. J. Bacteriol., 1999, 181, 6814-6821. (Pubitemid 29517998)
    • (1999) Journal of Bacteriology , vol.181 , Issue.21 , pp. 6814-6821
    • Nopponpunth, V.1    Sirawaraporn, W.2    Greene, P.J.3    Santi, D.V.4
  • 92
    • 63549142301 scopus 로고    scopus 로고
    • Fourth-generation fluoroquinolones in tuberculosis
    • Riede, H.L. Fourth-generation fluoroquinolones in tuberculosis. Lancet, 2009, 373, 1148-1149.
    • (2009) Lancet , vol.373 , pp. 1148-1149
    • Riede, H.L.1
  • 93
    • 0026705772 scopus 로고
    • The catalaseperoxidase gene and isoniazid resistance of Mycobacterium tuberculosis
    • Zhang, Y.; Heym, B.; Allen, B.; Young, D.; Cole, S.T. The catalaseperoxidase gene and isoniazid resistance of Mycobacterium tuberculosis. Nature, 1992, 358, 591-593.
    • (1992) Nature , vol.358 , pp. 591-593
    • Zhang, Y.1    Heym, B.2    Allen, B.3    Young, D.4    Cole, S.T.5
  • 94
    • 0027211111 scopus 로고
    • Transformation with katG restores isoniazid-sensitivity in Mycobacterium tuberculosis isolates resistant to a range of drug concentrations
    • DOI 10.1111/j.1365-2958.1993.tb01596.x
    • Zhang, Y.; Garbe, T.; Young, D. Transformation with katG restores isoniazid-sensitivity in Mycobacterium tuberculosis isolates resistant to a range of drug concentrations. Mol Microbiol., 1993, 8(3), 521-524. (Pubitemid 23156446)
    • (1993) Molecular Microbiology , vol.8 , Issue.3 , pp. 521-524
    • Zhang, Y.1    Garbe, T.2    Young, D.3
  • 95
    • 0028960179 scopus 로고
    • Missense mutations in the catalase-peroxidase gene, katG, are associated with isoniazid resistance in Mycobacterium tuberculosis
    • Heym, B.; Alzari, P.M.; Honore, N.; Cole, S.T. Missense mutations in the catalase-peroxidase gene, katG, are associated with isoniazid resistance in Mycobacterium tuberculosis. Mol. Microbiol.; 1995, 15(2), 235-245.
    • (1995) Mol. Microbiol. , vol.15 , Issue.2 , pp. 235-245
    • Heym, B.1    Alzari, P.M.2    Honore, N.3    Cole, S.T.4
  • 96
    • 0032486197 scopus 로고    scopus 로고
    • Inhibition of a Mycobacterium tuberculosis β-Ketoacyl ACP synthase by isoniazid
    • DOI 10.1126/science.280.5369.1607
    • Mdluli, K.; Slayden, R.A.; Zhu, Y.; Ramaswamy, S.; Pan, X.; Mead, D.; Crane, D.D.; Musser, J.M.; Barry, C.E 3rd. Inhibition of a Mycobacterium tuberculosis beta-ketoacyl ACP synthase by isoniazid. Science, 1998, 280(5369), 1607-1610. (Pubitemid 28277706)
    • (1998) Science , vol.280 , Issue.5369 , pp. 1607-1610
    • Mdluli, K.1    Slayden, R.A.2    Zhu, Y.3    Ramaswamy, S.4    Pan, X.5    Mead, D.6    Crane, D.D.7    Musser, J.M.8    Barry III, C.E.9
  • 97
    • 74049108181 scopus 로고    scopus 로고
    • Mode of binding of the tuberculosis prodrug isoniazid to heme peroxidases binding studies and crystal structure of bovine lactoperoxidase with isoniazid At 2.7 A resolution
    • Singh, A.K.; Kumar, R.P.; Pandey, N.; Singh, N.; Sinha, M.; Bhushan, A.; Kaur, P.; Sharma, S.; Singh, T.P. Mode of Binding of the Tuberculosis Prodrug Isoniazid to Heme Peroxidases Binding Studies and Crystal Structure of Bovine Lactoperoxidase with Isoniazid At 2.7 A Resolution. The Journal Biological Chemistry, 2010, 285(2), 1569-1576.
    • (2010) The Journal Biological Chemistry , vol.285 , Issue.2 , pp. 1569-1576
    • Singh, A.K.1    Kumar, R.P.2    Pandey, N.3    Singh, N.4    Sinha, M.5    Bhushan, A.6    Kaur, P.7    Sharma, S.8    Singh, T.P.9
  • 99
    • 0027993499 scopus 로고
    • Mechanistic studies of the oxidation of isoniazid by the catalase peroxidase from Mycobacterium tuberculosis
    • Johnson, K.; Schultz, P.G. Mechanistic studies of the oxidation of isoniazid by the catalase peroxidase from Mycobacterium tuberculosis. J. Am. Chem. Soc., 1994, 116, 7425-7426. (Pubitemid 24274243)
    • (1994) Journal of the American Chemical Society , vol.116 , Issue.16 , pp. 7425-7426
    • Johnsson, K.1    Schultz, P.G.2
  • 100
    • 0031409343 scopus 로고    scopus 로고
    • Molecular action of anti-mycobacterial agent
    • Chopra, I.; Brennan, P.J. Molecular action of anti-mycobacterial agent. Tubercle and Lung, 1998, 78, 89-98.
    • (1998) Tubercle and Lung , vol.78 , pp. 89-98
    • Chopra, I.1    Brennan, P.J.2
  • 101
    • 77749301260 scopus 로고    scopus 로고
    • Severe isoniazid-associated liver injuries among persons being treated for latent tuberculosis infection -United States,2004-2008
    • Centers for Disease Control and Prevention
    • Centers for Disease Control and Prevention. Severe Isoniazid-Associated Liver Injuries Among Persons Being Treated for Latent Tuberculosis Infection -United States, 2004-2008. MMWR, 2010, 59 (8), 224-229.
    • (2010) MMWR , vol.59 , Issue.8 , pp. 224-229
  • 102
    • 84863402494 scopus 로고    scopus 로고
    • Recent progress in the identification and development of InhA direct inhibitors of Mycobacterium tuberculosis
    • Lu, X.Y.; You, Q.D.; Chen, Y.D. Recent progress in the identification and development of InhA direct inhibitors of Mycobacterium tuberculosis. Mini. Rev. Med. Chem., 2010, 10(3), 182-193.
    • (2010) Mini. Rev. Med. Chem. , vol.10 , Issue.3 , pp. 182-193
    • Lu, X.Y.1    You, Q.D.2    Chen, Y.D.3
  • 103
    • 0029954860 scopus 로고    scopus 로고
    • Mutations in pncA, a gene encoding pyrazinamidase/nicotinamidase, cause resistance to the antituberculous drug pyrazinamide in tubercle bacillus
    • DOI 10.1038/nm0696-662
    • Scorpio, A.; Zhang, Y. Mutations in pncA, a gene encoding pyrazinamidase/nicotinamidase, cause resistance to the antituberculous drug pyrazinamide in tubercle bacillus. Nat. Med., 1996, 2(6), 662-667. (Pubitemid 26191953)
    • (1996) Nature Medicine , vol.2 , Issue.6 , pp. 662-667
    • Scorpio, A.1    Zhang, Y.2
  • 104
    • 0013888783 scopus 로고
    • Microbial persistence. I. The capacity of tubercle bacilli to survive sterilization in mouse tissues
    • McCune, R.M.; Feldman, F.M.; McDermat, W. Microbial persistence. I. The capacity of tubercle bacilli to survive sterilization in mouse tissues. J. Exp. Med., 1966, 123, 445-468.
    • (1966) J. Exp. Med. , vol.123 , pp. 445-468
    • McCune, R.M.1    Feldman, F.M.2    McDermat, W.3
  • 105
    • 79960073574 scopus 로고    scopus 로고
    • Targeted tuberculin testing and treatment of latent tuberculosis infection
    • Centers for Disease Control and Prevention
    • Centers for Disease Control and Prevention. "Targeted tuberculin testing and treatment of latent tuberculosis infection". MMWR, 2000, 49, 31-32.
    • (2000) MMWR , vol.49 , pp. 31-32
  • 106
    • 0014062867 scopus 로고
    • Pyrazinamide susceptibility and amidase activity of tubercle bacilli
    • Konno, K.; Feldmann, F.M.; McDermott, W. Pyrazinamide susceptibility and amidase activity of tubercle bacilli. Am. Rev. Respir. Dis., 1967, 95(3), 461-469.
    • (1967) Am. Rev. Respir. Dis. , vol.95 , Issue.3 , pp. 461-469
    • Konno, K.1    Feldmann, F.M.2    McDermott, W.3
  • 107
    • 0036207006 scopus 로고    scopus 로고
    • Effects of pyrazinamide on fatty acid synthesis by whole mycobacterial cells and purified fatty acid synthase I
    • DOI 10.1128/JB.184.8.2167-2172.2002
    • Boshoff, H.I.; Mizrahi, V.; Barry, C.E. III. Effects of pyrazinamide on fatty acid synthesis by whole mycobacterial cells and purified fatty acid synthase I. J. Bacteriol., 2002, 184, 2167-2172. (Pubitemid 34259666)
    • (2002) Journal of Bacteriology , vol.184 , Issue.8 , pp. 2167-2172
    • Boshoff, H.I.1    Mizrahi, V.2    Barry III, C.E.3
  • 108
    • 0242437861 scopus 로고    scopus 로고
    • Mode of action of pyrazinamide: Disruption of Mycobacterium tuberculosis membrane transport and energetics by pyrazinoic acid
    • DOI 10.1093/jac/dkg446
    • Zhang, Y.; Wade, M.M.; Scorpio, A.; Zhang, H.; Sun, Z. Mode of action of pyrazinamide: Disruption of Mycobacterium tuberculosis membrane transport and energetics by pyrazinoic acid. J. Antimicrob. Chemother. 2003, 52, 790-795. (Pubitemid 37407806)
    • (2003) Journal of Antimicrobial Chemotherapy , vol.52 , Issue.5 , pp. 790-795
    • Zhang, Y.1    Wade, M.M.2    Scorpio, A.3    Zhang, H.4    Sun, Z.5
  • 109
    • 77049188261 scopus 로고
    • Activation of pyrazinamide and nicotinamide in acidic environments in vitro
    • McDermott, W.; Tompsett, R. Activation of pyrazinamide and nicotinamide in acidic environments in vitro. Am. Rev. Tuberculosis, 1954, 70(4), 748-754.
    • (1954) Am. Rev. Tuberculosis , vol.70 , Issue.4 , pp. 748-754
    • McDermott, W.1    Tompsett, R.2
  • 111
    • 0026696665 scopus 로고
    • Antimycobacterial activity of a series of pyrazinoic acid esters
    • Cyanamon, M.H.; Klemmens, S.P. Antimycobacterial activity of a series of pyrazinoic acid esters. J. Med. Chem. 1982, 35, 1212-1215.
    • (1982) J. Med. Chem. , vol.35 , pp. 1212-1215
    • Cyanamon, M.H.1    Klemmens, S.P.2
  • 112
    • 10444260248 scopus 로고
    • Experimental evaluation of efficacy VII. Cycloserine (CS) and terizidone (TZ
    • In Bartman K. (Ed). Berlin: Springer Verlog
    • Otten, H. Experimental evaluation of efficacy VII. Cycloserine (CS) and terizidone (TZ). In Bartman K. (Ed). Antituberculosis drugs. Handbook of experimental Pharmacology, Berlin: Springer Verlog, 1988, Vol. 44, pp. 158-166.
    • (1988) Antituberculosis Drugs. Handbook of Experimental Pharmacology , vol.44 , pp. 158-166
    • Otten, H.1
  • 114
    • 0014589983 scopus 로고
    • Susceptibility of mycobacterial Dalanyl-D-alanine synthetase to D-cycloserine
    • David, H.L. Takayama K, Goldman DS. Susceptibility of mycobacterial Dalanyl-D-alanine synthetase to D-cycloserine. Am. Rev. Resp. Dis., 1969, 100(4), 579-581.
    • (1969) Am. Rev. Resp. Dis. , vol.100 , Issue.4 , pp. 579-581
    • David, H.L.1    Takayama, K.2    Goldman, D.S.3
  • 115
    • 0030872573 scopus 로고    scopus 로고
    • Overexpression of the D-alanine racemase gene confers resistance to D- cycloserine in Mycobacterium smegmatis
    • Cacers, N.E.; Harris, N.B.; Wellehen, J.F.; Feng, Z.; Kapur, V.; Barletta, R.G. Overexpression of the D-alanine racemase gene confers resistance to Dcycloserine in Mycobacterium smegmatis J. Bacteriol., 1997, 179, 5046-5055. (Pubitemid 27340537)
    • (1997) Journal of Bacteriology , vol.179 , Issue.16 , pp. 5046-5055
    • Caceres, N.E.1    Harris, N.B.2    Wellehan, J.F.3    Feng, Z.4    Kapur, V.5    Barletta, R.G.6
  • 118
    • 0037066702 scopus 로고    scopus 로고
    • The antituberculosis drug ethionamide is activated by a flavoprotein monooxygenase
    • DOI 10.1074/jbc.M110751200
    • Vannelli, T.A.; Dykman, A.; Ortiz de Montellano, P.R. The antituberculosis drug ethionamide is activated by a flavoprotein monooxygenase, J. Biol. Chem. 2002, 277, 12824-12829. (Pubitemid 34952646)
    • (2002) Journal of Biological Chemistry , vol.277 , Issue.15 , pp. 12824-12829
    • Vannelli, T.A.1    Dykman, A.2    Ortiz De Montellano, P.R.3
  • 119
    • 33645471799 scopus 로고    scopus 로고
    • Oxidative activation of thiacetazone by the Mycobacterium tuberculosis flavin monooxygenase Eta A and human FMO1 and FMO3
    • Qian, L.; Ortiz de Montellano, P.R. Oxidative activation of thiacetazone by the Mycobacterium tuberculosis flavin monooxygenase Eta A and human FMO1 and FMO3, Chem. Res. Toxicol. 2006, 19, 443-449.
    • (2006) Chem. Res. Toxicol. , vol.19 , pp. 443-449
    • Qian, L.1    Ortiz De Montellano, P.R.2
  • 121
    • 17244378938 scopus 로고    scopus 로고
    • 2-Deoxystreptamine: Central scaffold of aminoglycoside antibiotics
    • DOI 10.1021/cr0404085
    • Busscher, G.F.; Rutjes, F.P.; van Delft, F.L. 2-Deoxystreptamine: Central scaffold of aminoglycoside antibiotics, Chem. Rev. 2005, 105, 775-791. (Pubitemid 40527375)
    • (2005) Chemical Reviews , vol.105 , Issue.3 , pp. 775-791
    • Busscher, G.F.1    Rutjes, F.P.J.T.2    Van Delft, F.L.3
  • 122
    • 0034699519 scopus 로고    scopus 로고
    • Functional insights from the structure of the 30S ribosomal subunit and its interactions with antibiotics
    • Carter, A. P.; Clemons, W. M.; Brodersen, D. E.; Morgan-Warren, R. J.; Wimberly, B. T.; Ramakrishnan, V. Functional insights from the structure of the 30S ribosomal subunit and its interactions with antibiotics, Nature, 2000, 407, 340-348.
    • (2000) Nature , vol.407 , pp. 340-348
    • Carter, A.P.1    Clemons, W.M.2    Brodersen, D.E.3    Morgan-Warren, R.J.4    Wimberly, B.T.5    Ramakrishnan, V.6
  • 123
    • 33746106088 scopus 로고    scopus 로고
    • Capreomycin Binds across the Ribosomal Subunit Interface Using tlyA-Encoded 2'-O-Methylations in 16S and 23S rRNAs
    • DOI 10.1016/j.molcel.2006.05.044, PII S1097276506004333
    • Johansen, S. K.; Maus, C. E.; Plikaytis, B. B.; Douthwaite, S. Capreomycin Binds across the Ribosomal Subunit Interface Using tlyA-Encoded 2'-OMethylations in 16S and 23S rRNAs, Mol. Cell, 2006, 23, 173-182. (Pubitemid 44081881)
    • (2006) Molecular Cell , vol.23 , Issue.2 , pp. 173-182
    • Johansen, S.K.1    Maus, C.E.2    Plikaytis, B.B.3    Douthwaite, S.4
  • 124
    • 0036096326 scopus 로고    scopus 로고
    • Cellular impermeability and uptake of biocides and antibiotics in Gram-positive bacteria and mycobacteria
    • Lambert, P.A.J. Cellular impermeability and uptake of biocides and antibiotics in Gram-positive bacteria and mycobacteria. Appl. Microbiol. 2002, 92, 46S-54S.
    • (2002) Appl. Microbiol. , vol.92
    • Lambert, P.A.J.1
  • 126
    • 0141677886 scopus 로고    scopus 로고
    • Mycobacterial porins - New channel proteins in unique outer membranes
    • DOI 10.1046/j.1365-2958.2003.03662.x
    • Niederweis, M. Mycobacterial porins -new channel proteins in unique outer membranes. Mol. Microbiol. 2003, 49, 1167-1177. (Pubitemid 37153488)
    • (2003) Molecular Microbiology , vol.49 , Issue.5 , pp. 1167-1177
    • Niederweis, M.1
  • 127
    • 1942505736 scopus 로고    scopus 로고
    • The MspA porin promotes growth and increases antibiotic susceptibility of both Mycobacterium bovis BCG and Mycobacterium tuberculosis
    • Mailaender, C.; Reiling, N.; Engelhardt, H.; Bossmann, S.; Ehlers, S.; Niederweis, M. The MspA porin promotes growth and increases antibiotic susceptibility of both Mycobacterium bovis BCG and Mycobacterium tuberculosis, Microbiology, 2004, 150, 853-864. (Pubitemid 38519306)
    • (2004) Microbiology , vol.150 , Issue.4 , pp. 853-864
    • Mailaender, C.1    Reiling, N.2    Engelhardt, H.3    Bossmann, S.4    Ehlers, S.5    Niederweis, M.6
  • 128
    • 7244258919 scopus 로고    scopus 로고
    • Multidrug resistance of a porin deletion mutant of Mycobacterium smegmatis
    • DOI 10.1128/AAC.48.11.4163-4170.2004
    • Stephan, J.; Mailaender, C.; Etienne, G.; Daffe, M.; Niederweis, M. Multidrug Resistance of a Porin Deletion Mutant of Mycobacterium smegmatis, Antimicrob. Agents Chemother. 2004, 48, 4163-4170. (Pubitemid 39434870)
    • (2004) Antimicrobial Agents and Chemotherapy , vol.48 , Issue.11 , pp. 4163-4170
    • Stephan, J.1    Mailaender, C.2    Etienne, G.3    Daffe, M.4    Niederweis, M.5
  • 129
    • 39849103711 scopus 로고    scopus 로고
    • Design, synthesis, and evaluation of novel ethambutol analogues
    • DOI 10.1016/j.bmcl.2008.01.065, PII S0960894X08000826
    • Yendapally, R.; Lee, R.E. Synthesis and Evaluation of Novel Ethambutol Analogues. Bioorg. Med. Chem. Lett., 2008, 18(5), 1607-1611. (Pubitemid 351318253)
    • (2008) Bioorganic and Medicinal Chemistry Letters , vol.18 , Issue.5 , pp. 1607-1611
    • Yendapally, R.1    Lee, R.E.2
  • 130
    • 0026029948 scopus 로고
    • Extracellular and intracellular activities of clarithromycin used alone and in association with ethambutol and rifampicin against Mycobacterium avium complex
    • Rastogi, N.; Labrousse, V. Extracellular and intracellular activities of clarithromycin used alone and in association with ethambutol and rifampicin against Mycobacterium avium complex. Antimicrob. Agents Chemother., 1991, 35(3), 462-470.
    • (1991) Antimicrob. Agents Chemother. , vol.35 , Issue.3 , pp. 462-470
    • Rastogi, N.1    Labrousse, V.2
  • 131
    • 0028114141 scopus 로고
    • Activities of the benzoxazinorifamycin KRM 1648 and ethambutol against Mycobacterium avium complex in vitro and in macrophages
    • Inderlied, C.B.; Barbara-Burnham, L.; Wu, M.; Young, L.S.; Bermudez, L.E.M. Activities of the benzoxazinorifamycin KRM 1648 and ethambutol against Mycobacterium avium complex in vitro and in macrophages. Antimicrob. Agents Chemother., 1994, 38, 1838-1843. (Pubitemid 24250734)
    • (1994) Antimicrobial Agents and Chemotherapy , vol.38 , Issue.8 , pp. 1838-1843
    • Inderlied, C.B.1    Barbara-Burnham, L.2    Wu, M.3    Young, L.S.4    Bermudez, L.E.M.5
  • 133
    • 0034209078 scopus 로고    scopus 로고
    • Ofloxacin induced arthropathy in patients with multi-drug resistance tuberculosis
    • Tumbanatham, A.; Vinodkumar, S. Ofloxacin induced arthropathy in patients with multi-drug resistance tuberculosis. J. Assoc. of Physicians India, 2000, 48(6), 647-648.
    • (2000) J. Assoc. of Physicians India , vol.48 , Issue.6 , pp. 647-648
    • Tumbanatham, A.1    Vinodkumar, S.2
  • 135
    • 0026628327 scopus 로고
    • Cytotoxicity of quinolones toward eukaryotic cells. Identification of topoisomerase II as the primary cellular target for the quinolone CP-115,953 in yeast
    • Elsea, S.H.; Osheroff, N.; Nitiss, J.L. Cytotoxicity of quinolones toward eukaryotic cells. Identification of topoisomerase II as the primary cellular target for the quinolone CP-115,953 in yeast. J. Biol. Chem., 1992, 267(19), 13150-13153.
    • (1992) J. Biol. Chem. , vol.267 , Issue.19 , pp. 13150-13153
    • Elsea, S.H.1    Osheroff, N.2    Nitiss, J.L.3
  • 136
    • 0022359647 scopus 로고
    • The fluoroquinolones: Structures, mechanisms of action and resistance, and spectra of activity in vitro
    • Wolfson, J.S.; Hooper, D.C. The fluoroquinolones: Structures, mechanisms of action and resistance, and spectra of activity in vitro. Antimicrob. Agents Chemother., 1985, 28, 581-586. (Pubitemid 16236555)
    • (1985) Antimicrobial Agents and Chemotherapy , vol.28 , Issue.4 , pp. 581-586
    • Wolfson, J.S.1    Hooper, D.C.2
  • 137
    • 0032189275 scopus 로고    scopus 로고
    • DNA gyrase and topoisomerase IV: Biochemical activities, physiological roles during chromosome replication, and drug sensitivities
    • DOI 10.1016/S0167-4781(98)00126-2, PII S0167478198001262
    • Levine, C.; Hiasa, H.; Marians, K.J. DNA gyrase and topoisomerase IV: Biochemical activities physiological roles during chromosome replication and drug sentivities. Biochem. Biophys. Acta., 1998, 1400, 29-43. (Pubitemid 28475094)
    • (1998) Biochimica et Biophysica Acta - Gene Structure and Expression , vol.1400 , Issue.1-3 , pp. 29-43
    • Levine, C.1    Hiasa, H.2    Marians, K.J.3
  • 138
    • 0017744584 scopus 로고
    • Development of antibacterial agents of the nalidixic acid type
    • Albrecht, R. Development of antibacterial agents of the nalidixic acid type. Prog. Drug Res., 1977, 21, 9-104.
    • (1977) Prog. Drug Res. , vol.21 , pp. 9-104
    • Albrecht, R.1
  • 139
  • 140
    • 0020679387 scopus 로고
    • In vitro activity of Bay 0867, a new quinoline derivative, compared with those of other antimicrobial agents
    • Wise, R.; Andrews, J.M.; Edwards, L.J. In vitro Activity of Bay 09867, a New Quinoline Derivative, Compared with Those of Other Antimicrobial Agents. Antimicrob. Agents Chemother., 1983, 23, 559-564. (Pubitemid 13163297)
    • (1983) Antimicrobial Agents and Chemotherapy , vol.23 , Issue.4 , pp. 559-564
    • Wise, R.1    Andrews, J.M.2    Edwards, L.J.3
  • 141
    • 0020411041 scopus 로고
    • In vitro and in vivo activity of DL-8280, a new oxazine derivative
    • Sato, K.; Matsuura, Y.; Inoue, M.; Une, T.; Osada, Y.; Ogawa, H.; Mitsuhashi, S. In vitro and in vivo activity of DL-8280, a new oxazine derivative. Antimicrob. Agents Chemother., 1982, 22, 548-553. (Pubitemid 13206530)
    • (1982) Antimicrobial Agents and Chemotherapy , vol.22 , Issue.4 , pp. 548-553
    • Sato, K.1    Matsuura, Y.2    Inoue, M.3
  • 144
    • 0034089387 scopus 로고    scopus 로고
    • Moxifloxacin a new antibiotic designed to treat community-acquired respiratory tract infections: A review of microbiologic and pharmacokinetic- dynamic characteristics
    • Nightingale, C.H. Moxifloxacin, a new antibiotic designed to treat community-acquired respiratory tract infections: A review of microbiologic and pharmacokinetic-dynamic characteristics. Pharmacotherapy, 2000, 20, 245.
    • (2000) Pharmacotherapy , vol.20 , pp. 245
    • Nightingale, C.H.1
  • 146
    • 0025027077 scopus 로고
    • New topoisomerase essential for chromosome segregation in E. coli
    • Kato, J.; Nishimura, Y.; Imamura, R.; Niki, H.; Hiraga, S.; Suzuki, H. New topoisomerase essential for chromosome segregation in E. coli. Cell, 1990, 63, 393-404.
    • (1990) Cell , vol.63 , pp. 393-404
    • Kato, J.1    Nishimura, Y.2    Imamura, R.3    Niki, H.4    Hiraga, S.5    Suzuki, H.6
  • 147
    • 0035180501 scopus 로고    scopus 로고
    • Target preference of 15 quinolones against Staphylococcus aureus, based on antibacterial activities and target inhibition
    • DOI 10.1128/AAC.45.12.3544-3547.2001
    • Takei, M.; Fukuda, H.; Kishii, R.; Hosaka, M. Target Preference of 15 Quinolones against Staphylococcus aureus, Based on Antibacterial Activities and Target Inhibition. Antimicrob. Agents Chemother. 2001, 45, 3544-3547. (Pubitemid 33107875)
    • (2001) Antimicrobial Agents and Chemotherapy , vol.45 , Issue.12 , pp. 3544-3547
    • Takei, M.1    Fukuda, H.2    Kishii, R.3    Hosaka, M.4
  • 149
    • 77951249362 scopus 로고    scopus 로고
    • In vitro activity of a new isothiazoloquinolone, ACH-702, against mycobacterium tuberculosis and other mycobacteria
    • Molina-Torres, C.A.; Ocampo-Candiani, J.; Rendon, A.; Pucci, M.J.; Vera-Cabrera, L. In Vitro Activity of a New Isothiazoloquinolone, ACH-702, against Mycobacterium tuberculosis and Other Mycobacteria. Antimicrob. Agents Chemother., 2010, 54(5), 2188-2190.
    • (2010) Antimicrob. Agents Chemother. , vol.54 , Issue.5 , pp. 2188-2190
    • Molina-Torres, C.A.1    Ocampo-Candiani, J.2    Rendon, A.3    Pucci, M.J.4    Vera-Cabrera, L.5
  • 152
    • 0002415298 scopus 로고    scopus 로고
    • Rifamycins
    • In: O'Grady F, Lambert HP, Finch RG, Greenwood, D. eds., 7theds. Edinburg: Churchill Livingston
    • Parneti, F.; Lancini, G. Rifamycins In: O'Grady F, Lambert HP, Finch RG, Greenwood, D. eds. Antibitic and Chemotherapy, 7theds. Edinburg: Churchill Livingston, 1997, pp. 453-459.
    • (1997) Antibitic and Chemotherapy , pp. 453-459
    • Parneti, F.1    Lancini, G.2
  • 154
    • 0037417077 scopus 로고    scopus 로고
    • In vitro activities of rifamycin derivatives ABI-1648 (rifalazil, KRM-1648), ABI-1657, and ABI-1131 against Chlamydia trachomatis and recent clinical isolates of Chlamydia pneumoniae
    • DOI 10.1128/AAC.47.3.1135-1136.2003
    • Robin, P.M.; Reznik, T.; Kutlin, A.; Hammerschlag, M.R. In vitro Activities of Rifamycin Derivatives ABI-1648 (Rifalazil, KRM-1648), ABI-1657, and ABI-1131 against Chlamydia trachomatis and Recent Clinical Isolates of Chlamydia pneumonia. Antimicrob. Agents Chemother., 2003, 47, 1135-1136. (Pubitemid 36254248)
    • (2003) Antimicrobial Agents and Chemotherapy , vol.47 , Issue.3 , pp. 1135-1136
    • Roblin, P.M.1    Reznik, T.2    Kutlin, A.3    Hammerschlag, M.R.4
  • 162
    • 53249084552 scopus 로고    scopus 로고
    • New anti-tuberculosis drugs with novel mechanisms of action
    • Rivers, E.C.; Mancera, R.L. New Anti-Tuberculosis Drugs with Novel Mechanisms of Action. Curr. Med. Chem. 2008, 15, 1956-1967.
    • (2008) Curr. Med. Chem. , vol.15 , pp. 1956-1967
    • Rivers, E.C.1    Mancera, R.L.2
  • 165
    • 72949083267 scopus 로고    scopus 로고
    • Anderson RF. Release of nitrite from the antitubercular nitroimidazole drug PA-824 and analogues upon one-electron reduction in protic, nonaqueous solvent
    • Maroz, A.; Shinde, S.S.; Franzblau, S.G.; Ma, Z.; Denny, W.A.; Palmer, B.D. Anderson RF. Release of nitrite from the antitubercular nitroimidazole drug PA-824 and analogues upon one-electron reduction in protic, nonaqueous solvent. Org. Biomol. Chem., 2010, 8, 413-418.
    • (2010) Org. Biomol. Chem. , vol.8 , pp. 413-418
    • Maroz, A.1    Shinde, S.S.2    Franzblau, S.G.3    Ma, Z.4    Denny, W.A.5    Palmer, B.D.6
  • 167
    • 33750589018 scopus 로고    scopus 로고
    • Combinations of R207910 with drugs used to treat multidrug-resistant tuberculosis have the potential to shorten treatment duration
    • DOI 10.1128/AAC.00766-06
    • Lounis, N.; Veziris, N.; Chauffour, A.; Truffot-Pernot, C.; Andries, K.; Jarlier, V. Combinations of R207910 with Drugs Used To Treat Multidrug-Resistant Tuberculosis Have the Potential To Shorten Treatment Duration. Antimicrob. Agents Chemother., 2006, 50, 3543-3547. (Pubitemid 44684863)
    • (2006) Antimicrobial Agents and Chemotherapy , vol.50 , Issue.11 , pp. 3543-3547
    • Lounis, N.1    Veziris, N.2    Chauffeur, A.3    Truffot-Pernot, C.4    Andries, K.5    Jarlier, V.6
  • 168
    • 77953797826 scopus 로고    scopus 로고
    • In vitro interactions between new antitubercular drug candidates SQ109 and TMC207
    • Reddy, V.M.; Einck, L.; Andries, K.; Nacy, C.A. In Vitro Interactions between New Antitubercular Drug Candidates SQ109 and TMC207. Antimicrob. Agents Chemother., 2010, 54, 2840-2846.
    • (2010) Antimicrob. Agents Chemother. , vol.54 , pp. 2840-2846
    • Reddy, V.M.1    Einck, L.2    Andries, K.3    Nacy, C.A.4
  • 170
    • 77149123917 scopus 로고    scopus 로고
    • Rates and mechanisms of resistance development in mycobacterium tuberculosis to a novel diarylquinoline ATP synthase inhibitor
    • Huitric, E.; Verhasselt, P.; Koul, A.; Andries, K.; Hoffner, S.; Andersson, D.I. Rates and Mechanisms of Resistance Development in Mycobacterium tuberculosis to a Novel Diarylquinoline ATP Synthase Inhibitor. Antimicrob. Agents Chemother., 2010, 54(3), 1022-1028.
    • (2010) Antimicrob. Agents Chemother. , vol.54 , Issue.3 , pp. 1022-1028
    • Huitric, E.1    Verhasselt, P.2    Koul, A.3    Andries, K.4    Hoffner, S.5    Andersson, D.I.6
  • 171
    • 0031753303 scopus 로고    scopus 로고
    • Bactericidal activities of the pyrrole derivative BM212 against multidrug-resistant and intramacrophagic Mycobacterium tuberculosis strains
    • Deidda, D.; Lampis, G.; Fioravanti, R.; Biava, M.; Porretta, G.C.; Zanetti, S.; Pompei, R. Bactericidal Activities of the Pyrrole Derivative BM212 against Multidrug-Resistant and Intramacrophagic Mycobacterium tuberculosis Strains. Antimicrob. Agents Chemother., 1998, 42, 3035-3037. (Pubitemid 28501251)
    • (1998) Antimicrobial Agents and Chemotherapy , vol.42 , Issue.11 , pp. 3035-3037
    • Deidda, D.1    Lampis, G.2    Fioravanti, R.3    Biava, M.4    Porretta, G.C.5    Zanetti, S.6    Pompei, R.7
  • 174
    • 33748040742 scopus 로고    scopus 로고
    • Synergistic interactions of SQ109, a new ethylene diamine, with front-line antitubercular drugs in vitro
    • DOI 10.1093/jac/dkl227
    • Chen, P.; Gearhart, J.; Protopopova, M.; Einck, L.; Nacy, C.A. Synergistic interactions of SQ109, a new ethylene diamine, with front-line antitubercular drugs in vitro. J. Antimicro. Chemotherapy. 2006, 58, 332-337. (Pubitemid 44294944)
    • (2006) Journal of Antimicrobial Chemotherapy , vol.58 , Issue.2 , pp. 332-337
    • Chen, P.1    Gearhart, J.2    Protopopova, M.3    Einck, L.4    Nacy, C.A.5
  • 181
    • 0020680673 scopus 로고
    • Thiotetromycin, a new antibiotic. Taxonomy, production, isolation, and physicochemical and biological properties
    • Omura, S.; Nakagawa, A.; Iwata, R.; Takahashi, Y.; Shimizu, H.; Tanaka, H. Thiotetromycin, a new antibiotic. Taxonomy, production, isolation, and physicochemical and biological properties. J. Antibiot.(Tokyo), 1983, 36, 109-114. (Pubitemid 13148116)
    • (1983) Journal of Antibiotics , vol.36 , Issue.2 , pp. 109-114
    • Omura, S.1    Iwai, Y.2    Nakagawa, A.3
  • 182
    • 0019977450 scopus 로고
    • Thiolactomycin, a new antibiotic. III. In vitro antibacterial activity
    • Noto, T.; Miyakawa, S.; Oishi, H.; Endo, H.; Okazaki, H. Thiolactomycin, a new antibiotic. III. In vitro antibacterial activity. J Antibiot (Tokyo), 1982, 35(4), 401-410. (Pubitemid 12046394)
    • (1982) Journal of Antibiotics , vol.35 , Issue.4 , pp. 401-410
    • Noto, T.1    Miyakawa, S.2    Oishi, H.3
  • 183
    • 0021074097 scopus 로고
    • Structure of a new antibacterial antibiotic, thiotetromycin
    • Omura, S.; Nakagawa, A.; Iwata, R.; Hatano, A. Structure of a new antibacterial antibiotic, thiotetromycin. J. Antibiot., 1983, 36, 1781-1782. (Pubitemid 14182445)
    • (1983) Journal of Antibiotics , vol.36 , Issue.12 , pp. 1781-1782
    • Omura, S.1    Nakagawa, A.2    Iwata, R.3    Hatano, A.4
  • 184
    • 0022454141 scopus 로고
    • Effect of thiolactomycin on the individual enzymes of the fatty acid synthase system in Escherichia coli
    • Nishida, I.; Kawaguchi, A.; Yamada, M. Effect of thiolactomycin on the individual enzymes of the fatty acid synthase system in Escherichia coli. J. Biochem., 1986, 99, 1447-1454. (Pubitemid 16033515)
    • (1986) Journal of Biochemistry , vol.99 , Issue.5 , pp. 1447-1454
    • Nishida, I.1    Kawaguchi, A.2    Yamada, M.3
  • 186
    • 77949471491 scopus 로고    scopus 로고
    • 3D-QSAR, molecular docking studies, and binding mode prediction of thiolactomycin analogs as mtFabH inhibitors
    • Lu, X.; Chen, Y.; You, Q. 3D-QSAR, molecular docking studies, and binding mode prediction of thiolactomycin analogs as mtFabH inhibitors. J. Enzyme Inhib. Med. Chem., 2010, 25(2), 240-249.
    • (2010) J. Enzyme Inhib. Med. Chem. , vol.25 , Issue.2 , pp. 240-249
    • Lu, X.1    Chen, Y.2    You, Q.3
  • 187
    • 0020623895 scopus 로고
    • Isolation and structure of citreothiolactone, a novel metabolite of Penicillium citrea-viride B
    • DOI 10.1016/S0040-4039(00)81601-9
    • Shizuri, Y.; Niwa, M.; Furukawa, H.; Yamamura, S. Isolation and structure of citroethiolactone, a novel metabolite of Penicillium citreo-viridebe. Tetrahedron Lett., 1983, 24, 1053-1054. (Pubitemid 13124097)
    • (1983) Tetrahedron Letters , vol.24 , Issue.10 , pp. 1053-1054
    • Shizuri, Y.1    Niwa, M.2    Furukawa, H.3    Yamamura, S.4
  • 188
    • 0022643922 scopus 로고
    • Isolation and structure of antibiotic U-68,204, a new thiolactone
    • Dolak, L.A.; Castle, T.M.; Truesdell, S.E.; Sebek, O.K. Isolation and structure of antibiotic U-68,204, a new thiolactone. J. Antibiot., 1986, 39, 26-31. (Pubitemid 16174633)
    • (1986) Journal of Antibiotics , vol.39 , Issue.1 , pp. 26-31
    • Dolak, L.A.1    Castle, T.M.2    Truesdell, S.E.3    Sebek, O.K.4
  • 192
    • 29744457268 scopus 로고    scopus 로고
    • Synthesis and evaluation of cyclic secondary amine substituted phenyl and benzyl nitrofuranyl amides as novel antituberculosis agents
    • DOI 10.1021/jm050765n
    • Tangallapally, R.P.; Yendapally, R.; Lee, R.E.; Lenaerts, A.J. Synthesis and Evaluation of cyclic secondary amine substituted phenyl and benzyl nitrofuranyl amides as novel antituberculosis agents. J. Med. Chem., 2005, 48, 8261-8269. (Pubitemid 43032535)
    • (2005) Journal of Medicinal Chemistry , vol.48 , Issue.26 , pp. 8261-8269
    • Tangallapally, R.P.1    Yendapally, R.2    Lee, R.E.3    Lenaerts, A.J.M.4    Lee, R.E.5
  • 193
    • 33645887824 scopus 로고    scopus 로고
    • Synthesis of new and potent analogues of antituberculosis agent 5-nitro-furan-2carboxylic acid 4-(4-benzyl-piperazin-1-yl)-benzylamide with improved bioavailability
    • Tangallapally, R.P.; Lee, R.E.; Lenaerts, A.J. Synthesis of new and potent analogues of antituberculosis agent 5-nitro-furan-2carboxylic acid 4-(4-benzyl-piperazin-1-yl)-benzylamide with improved bioavailability. Bioorg. Med. Chem. Lett., 2006, 16, 2584-2589.
    • (2006) Bioorg. Med. Chem. Lett. , vol.16 , pp. 2584-2589
    • Tangallapally, R.P.1    Lee, R.E.2    Lenaerts, A.J.3
  • 194
    • 76249119957 scopus 로고    scopus 로고
    • Pharmacophore mapping and electronic feature analysis for a series of nitroaromatic compounds with antitubercular activity
    • Tawari, N.R.; Degani, M.S. Pharmacophore Mapping and Electronic Feature Analysis for a Series of Nitroaromatic Compounds with Antitubercular Activity. J. Comput. Chem., 2010, 31, 739-751.
    • (2010) J. Comput. Chem. , vol.31 , pp. 739-751
    • Tawari, N.R.1    Degani, M.S.2
  • 195
    • 77955415635 scopus 로고    scopus 로고
    • 5-Nitro-2-furoic acid hydrazones: Design, synthesis and in vitro antimycobacterial evaluation against log and starved phase cultures
    • Sriram, D.; Yogeeswari, P.; Vyas, D.R.K.; Senthilkumar, P.; Bhat, P.; Srividya, M. 5-Nitro-2-furoic acid hydrazones: Design, synthesis and in vitro antimycobacterial evaluation against log and starved phase cultures. Bioorg. Med. Chem. Lett., 2010, 20, 4313-4316.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 4313-4316
    • Sriram, D.1    Yogeeswari, P.2    Vyas, D.R.K.3    Senthilkumar, P.4    Bhat, P.5    Srividya, M.6
  • 197
    • 45749084929 scopus 로고    scopus 로고
    • 1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings
    • DOI 10.1021/jm701560p
    • Biava, M.; Porretta, G.C.; Poce, G.; De Logu, A.; Saddi, M.; Meleddu, R.; Manetti, F.; De Rossi, E.; Botta, M. 1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings. J. Med. Chem., 2008, 51, 3644-3648. (Pubitemid 351875020)
    • (2008) Journal of Medicinal Chemistry , vol.51 , Issue.12 , pp. 3644-3648
    • Biava, M.1    Porretta, G.C.2    Poce, G.3    De Logu, A.4    Saddi, M.5    Meleddu, R.6    Manetti, F.7    De Rossi, E.8    Botta, M.9
  • 198
    • 70349765643 scopus 로고    scopus 로고
    • 1,5-Diaryl-2ethyl pyrrole derivatives as antimycobacterial agents: Design, synthesis and microbiological evaluation
    • Biava, M.; Porretta, G.C.; Poce, G.; De Logu, A.; Meleddu, R.; De Rossi, E.; Manetti, F.; Botta, M. 1,5-Diaryl-2ethyl pyrrole derivatives as antimycobacterial agents: Design, synthesis and microbiological evaluation. European J. Med. Chem., 2009, 44, 4734-4738.
    • (2009) European J. Med. Chem. , vol.44 , pp. 4734-4738
    • Biava, M.1    Porretta, G.C.2    Poce, G.3    De Logu, A.4    Meleddu, R.5    De Rossi, E.6    Manetti, F.7    Botta, M.8
  • 199
    • 51149107005 scopus 로고    scopus 로고
    • Synthesis of new 4-pyrrol-1yl benzoic acid hydrazide analogs and derived oxadiazole, triazole and pyrrole ring systems: A novel class of potential antibacterial and antitubercular agents
    • Joshi, S.D.; Vagdevi, H.M.; Vaidya, V.P.; Gadaginamath, G.S. Synthesis of new 4-pyrrol-1yl benzoic acid hydrazide analogs and derived oxadiazole, triazole and pyrrole ring systems: A novel class of potential antibacterial and antitubercular agents. Eur. J. Med. Chem., 2008, 43, 1989-1996.
    • (2008) Eur. J. Med. Chem. , vol.43 , pp. 1989-1996
    • Joshi, S.D.1    Vagdevi, H.M.2    Vaidya, V.P.3    Gadaginamath, G.S.4
  • 200
    • 77952985516 scopus 로고    scopus 로고
    • Preparation and properties in vitro and in vivo of antitubercular pyrroles
    • Hearn, M.J.; Chen, M.F.; Terrot, M.S.; Webster, E.R.; Cynamon, M.H. Preparation and properties in vitro and in vivo of antitubercular pyrroles. J. Het. Chem., 2010, 47(3), 707-712.
    • (2010) J. Het. Chem. , vol.47 , Issue.3 , pp. 707-712
    • Hearn, M.J.1    Chen, M.F.2    Terrot, M.S.3    Webster, E.R.4    Cynamon, M.H.5
  • 201
    • 77957367740 scopus 로고    scopus 로고
    • Synthesis, charecterization, and biological activities of some new pyrazoline derivatives, derived from ethyl-2-(2, 5-dichloroanilido) acetohydrazide
    • Sharma, R.N.; Sharma, K.P.; Dixit, S.N. Synthesis, Charecterization, and Biological Activities of some New Pyrazoline Derivatives, derived from Ethyl-2-(2, 5-dichloroanilido) Acetohydrazide, Int. J. ChemTech Research, 2010, 2 (3), 1413-1425.
    • (2010) Int. J. ChemTech Research , vol.2 , Issue.3 , pp. 1413-1425
    • Sharma, R.N.1    Sharma, K.P.2    Dixit, S.N.3
  • 203
    • 79958855195 scopus 로고    scopus 로고
    • Synthesis of some new quinolinylpyrazoles as potential antibacterial and antitubercular agents
    • Joshi, S.D.; Joshi, A.; Vagdevi, H.M.; Vaidya, V.P.; Gadaginamath, G.S. Synthesis of some new quinolinylpyrazoles as potential antibacterial and antitubercular agents. Ind. J. Het. Chem., 2010, 19(3), 221-224.
    • (2010) Ind. J. Het. Chem. , vol.19 , Issue.3 , pp. 221-224
    • Joshi, S.D.1    Joshi, A.2    Vagdevi, H.M.3    Vaidya, V.P.4    Gadaginamath, G.S.5
  • 204
    • 0038700567 scopus 로고    scopus 로고
    • Combinatorial lead optimization of [1,2]-diamines based on ethambutol as potential antituberculosis preclinical candidates
    • DOI 10.1021/cc020071p
    • Lee, R.E.; Protopopova, M.; Crooks, E.; Slayden, R.A.; Terrot, M.; Barry, C.E III. Combinatorial Lead Optimization of [1, 2]-Diamines Based on Ethambutol as Potential Antituberculosis Preclinical Candidates. J. Comb. Chem., 2003, 5(2), 172-187. (Pubitemid 37123511)
    • (2003) Journal of Combinatorial Chemistry , vol.5 , Issue.2 , pp. 172-187
    • Lee, R.E.1    Protopopova, M.2    Crooks, E.3    Slayden, R.A.4    Terrot, M.5    Barry III, C.E.6
  • 206
    • 71749112435 scopus 로고    scopus 로고
    • Synthesis and evaluation of (S,S)-N,N'-bis-[3-(2,2',6,6'- tetramethylbenzhydryloxy)-2-hydroxy-propyl]-ethylenediamine (S2824) analogs with anti-tuberculosis activity
    • Zhang, X.; Hu, Y.; Chen, S.; Luo, R.; Yue, J.; Zhang, Y.; Duan, W.; Wang, H. Synthesis and evaluation of (S,S)-N,N'-bis-[3-(2,2',6,6'- tetramethylbenzhydryloxy)-2-hydroxy-propyl]-ethylenediamine (S2824) analogs with anti-tuberculosis activity. Bioorg. Med. Chem. Lett., 2009, 19, 6074-6077.
    • (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 6074-6077
    • Zhang, X.1    Hu, Y.2    Chen, S.3    Luo, R.4    Yue, J.5    Zhang, Y.6    Duan, W.7    Wang, H.8
  • 207
    • 68349125246 scopus 로고    scopus 로고
    • Parallel synthesis of chiral pentamines and pyrrolidine containing bis-heterocyclic libraries. Multiple scaffolds with multiple building blocks: A double diversity for the identification for the identification of new antitubercular compounds
    • Nefzi, A.; Appel, J.; Arutyunyan, S.; Houghten, R.A. Parallel synthesis of chiral pentamines and pyrrolidine containing bis-heterocyclic libraries. Multiple scaffolds with multiple building blocks: A double diversity for the identification for the identification of new antitubercular compounds. Bioorg. Med. Chem. Lett., 2009, 19, 5169-5175.
    • (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 5169-5175
    • Nefzi, A.1    Appel, J.2    Arutyunyan, S.3    Houghten, R.A.4
  • 211
    • 0037075792 scopus 로고    scopus 로고
    • Synthesis and antimycobacterial activity of 6-arylpurines: The requirements for the N-9 substituent in active antimycobacterial purines
    • DOI 10.1021/jm0110284
    • Gundersen, L.L.; Nissen-Meyer, J.; Spilsberg, B. Synthesis and antimycobacterial activity of 6-arylpurines: The requirements for the N-9 substituent in active antimycobacterial purines. J. Med. Chem., 2002, 45, 1383-1386. (Pubitemid 34263575)
    • (2002) Journal of Medicinal Chemistry , vol.45 , Issue.6 , pp. 1383-1386
    • Gundersen, L.-L.1    Nissen-Meyer, J.2    Spilsberg, B.3
  • 212
    • 0035093384 scopus 로고    scopus 로고
    • Antimycobacterial activity of new quinoxaline-2-carbonitrile and quinoxaline-2-carbonitrile 1,4-di-N-oxide derivatives
    • Ortega, M.A.; Montoya, M.E.; Jaso, A.; Zarranz, B.; Tirapu, I.; Aldana, I.; Monge, A. Antimycobacterial activity of new quinoxaline-2-carbonitrile and quinoxaline-2-carbonitrile 1,4-di-N-oxide derivatives. Pharmazie, 2001, 56, 205-207. (Pubitemid 32209943)
    • (2001) Pharmazie , vol.56 , Issue.3 , pp. 205-207
    • Ortega, M.A.1    Montoya, M.E.2    Jaso, A.3    Zarranz, B.4    Tirapu, I.5    Aldana, I.6    Monge, A.7
  • 213
    • 0036242821 scopus 로고    scopus 로고
    • Novel substituted quinoxaline 1,4-dioxides with in vitro antimycobacterial and anticandida activity
    • DOI 10.1016/S0223-5234(02)01346-6, PII S0223523402013466
    • Carta, A.; Paglietti, G.; Rahbar Nikookar, M.E.; Sanna, P.; Sechi, L.; Zanetti, S. Original article Novel substituted quinoxaline 1,4-dioxides with in vitro antimycobacterial and anticandida activity. Eur. J. Med. Chem., 2002, 37, 355-366. (Pubitemid 34465545)
    • (2002) European Journal of Medicinal Chemistry , vol.37 , Issue.5 , pp. 355-366
    • Carta, A.1    Paglietti, G.2    Rahbar Nikookar, M.E.3    Sanna, P.4    Sechi, L.5    Zanetti, S.6
  • 215
    • 72049084988 scopus 로고    scopus 로고
    • In vitro antitubercular and antimicrobial activities of 1-substituted 2,3(1H,4H)-quinoxalinediones
    • Ramalingam, P.; Ganapaty, S.; Rao, Ch.; Babu, R. In vitro antitubercular and antimicrobial activities of 1-substituted 2,3(1H,4H)-quinoxalinediones. Bioorg. Med. Chem. Lett., 2010, 20(1), 406-408.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , Issue.1 , pp. 406-408
    • Ramalingam, P.1    Ganapaty, S.2    Rao, Ch.3    Babu, R.4
  • 216
    • 0036241998 scopus 로고    scopus 로고
    • Synthesis and antitubercular evaluation of 4-quinolylhydrazines
    • Savini, L.; Chiasserini, L.; Gaeta, A.; Pellerano, C. Synthesis and antitubercular evaluation of 4-quinolylhydrazines. Bioorg. Med. Chem., 2002, 10, 2193-2198.
    • (2002) Bioorg. Med. Chem. , vol.10 , pp. 2193-2198
    • Savini, L.1    Chiasserini, L.2    Gaeta, A.3    Pellerano, C.4
  • 218
    • 66449132135 scopus 로고    scopus 로고
    • Design synthesis and biological evaluation of novel triazole, urea and thiourea derivatives of quinoline against Mycobaterium tuberculosis
    • Upadhayaya, R.S.; Kulkarni, G.M.; Vasireddy, N.R.; Vandavasi, J.K.; Dixit, S.S.; Sharma, V.; Chattopadhyaya, J. Design synthesis and biological evaluation of novel triazole, urea and thiourea derivatives of quinoline against Mycobaterium tuberculosis. Bioorg. Med. Chem., 2009, 17, 4681-4692.
    • (2009) Bioorg. Med. Chem. , vol.17 , pp. 4681-4692
    • Upadhayaya, R.S.1    Kulkarni, G.M.2    Vasireddy, N.R.3    Vandavasi, J.K.4    Dixit, S.S.5    Sharma, V.6    Chattopadhyaya, J.7
  • 220
    • 74349084588 scopus 로고    scopus 로고
    • Design and synthesis of some new quinoline-3-carbohydrazone derivatives as potential antimycobacterial agents
    • Eswaran, S.; Adhikari, A.V.; Pal, N.K.; Chowdhury, I.H. Design and synthesis of some new quinoline-3-carbohydrazone derivatives as potential antimycobacterial agents. Bioorg. Med. Chem. Lett., 2010, 20, 1040-1044.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 1040-1044
    • Eswaran, S.1    Adhikari, A.V.2    Pal, N.K.3    Chowdhury, I.H.4
  • 221
    • 73549093364 scopus 로고    scopus 로고
    • A microwave-assisted, facile, regioselective Friedlander synthesis and antitubercular evaluation of 2,9-diaryl-2,3-dihydrothieno-[3,2-b]quinolines
    • Balamurugan, K.; Jeyachandran, V.S.; Perumal, T.H.; Manjashetty, P.; Yogeeswari, D.S. A microwave-assisted, facile, regioselective Friedlander synthesis and antitubercular evaluation of 2,9-diaryl-2,3-dihydrothieno-[3,2-b] quinolines. Eur. J. Med. Chem., 2010, 45, 682-688.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 682-688
    • Balamurugan, K.1    Jeyachandran, V.S.2    Perumal, T.H.3    Manjashetty, P.4    Yogeeswari, D.S.5
  • 224
    • 77954313777 scopus 로고    scopus 로고
    • New quinoline derivatives: Synthesis and investigation of antibacterial and antituberculosis properties
    • Eswaran, S.; Adhikari, A.V.; Chowdhury, I.H.; Pal, N.K.; Thomas, K.D. New quinoline derivatives: Synthesis and investigation of antibacterial and antituberculosis properties. Eur. J. Med. Chem., 2010, 45, 3374-3383.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 3374-3383
    • Eswaran, S.1    Adhikari, A.V.2    Chowdhury, I.H.3    Pal, N.K.4    Thomas, K.D.5
  • 225
    • 76049098678 scopus 로고    scopus 로고
    • New 1,3-oxazolo[4,5-c]quinoline derivatives: Synthesis and evaluation of antibacterial and antituberculosis properties
    • Eswaran, S.; Adhikari, A.V.; Kumar, A.R. New 1,3-oxazolo[4,5-c]quinoline derivatives: Synthesis and evaluation of antibacterial and antituberculosis properties. Eur. J. Med. Chem., 2010, 45(3), 957-966.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.3 , pp. 957-966
    • Eswaran, S.1    Adhikari, A.V.2    Kumar, A.R.3
  • 226
    • 74049097181 scopus 로고    scopus 로고
    • Synthesis and antituberculosis activity of novel mefloquine-isoxazole carboxylic esters as prodrugs
    • Jialin, M.; Hai, Y.; Yuehong, W. Synthesis and antituberculosis activity of novel mefloquine-isoxazole carboxylic esters as prodrugs. Bioorg. Med. Chem. Lett., 2010, 20(3), 1263-1268.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , Issue.3 , pp. 1263-1268
    • Jialin, M.1    Hai, Y.2    Yuehong, W.3
  • 227
    • 74349084588 scopus 로고    scopus 로고
    • Design and synthesis of some new quinoline-3-carbohydrazone derivatives as potential antimycobacterial agents
    • Eswaran, S.; Adhikari, A.V.; Pal, N.K.; Chowdhury, I.H. Design and synthesis of some new quinoline-3-carbohydrazone derivatives as potential antimycobacterial agents. Bioorg. Med. Chem. Lett., 2010, 20(3), 1040-1044.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , Issue.3 , pp. 1040-1044
    • Eswaran, S.1    Adhikari, A.V.2    Pal, N.K.3    Chowdhury, I.H.4
  • 228
    • 73549093364 scopus 로고    scopus 로고
    • A microwave-assisted, facile, regioselective Friedlaender synthesis and antitubercular evaluation of 2,9-diaryl-2,3-dihydrothieno-[3,2-b]quinolines
    • Balamurugan, K.; Jeyachandran, V.; Perumal, S.; Manjashetty, T.H.; Yogeeswari, P.; Sriram, D. A microwave-assisted, facile, regioselective Friedlaender synthesis and antitubercular evaluation of 2,9-diaryl-2,3- dihydrothieno-[3,2-b]quinolines. Eur. J. Med. Chem, 2010, 45(2), 682-688.
    • (2010) Eur. J. Med. Chem , vol.45 , Issue.2 , pp. 682-688
    • Balamurugan, K.1    Jeyachandran, V.2    Perumal, S.3    Manjashetty, T.H.4    Yogeeswari, P.5    Sriram, D.6
  • 229
    • 73549088732 scopus 로고    scopus 로고
    • Identification of benzofuro[2,3-b]quinoline derivatives as a new class of antituberculosis agents
    • Yang, C.L.; Tseng, C.H.; Chen, Y.L.; Lu, C.M.; Kao, C.L.; Wu, M.H.; Tzeng, C.C. Identification of benzofuro[2,3-b]quinoline derivatives as a new class of antituberculosis agents. Eur. J. Med. Chem., 2010, 45(2), 602-607.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.2 , pp. 602-607
    • Yang, C.L.1    Tseng, C.H.2    Chen, Y.L.3    Lu, C.M.4    Kao, C.L.5    Wu, M.H.6    Tzeng, C.C.7
  • 230
    • 1842630349 scopus 로고    scopus 로고
    • Synthesis and preliminary evaluation of some pyrazine containing thiazolines and thiazolidinones as antimicrobial agents
    • DOI 10.1016/j.bmc.2004.02.024, PII S0968089604001464
    • Bonde, C.G.; Gaikwad, N.J. Synthesis and preliminary evaluation of some pyrazine containing thiazoline and thiazolidinones as antimicrobial agents. Bioorg. Med. Chem., 2004, 12, 2151-2161. (Pubitemid 38476974)
    • (2004) Bioorganic and Medicinal Chemistry , vol.12 , Issue.9 , pp. 2151-2161
    • Bonde, C.G.1    Gaikwad, N.J.2
  • 231
    • 71049161722 scopus 로고    scopus 로고
    • Searching for new cures for tuberculosis: Design, synthesis, and biological evaluation of 2-methylbenzothiazoles
    • Huang, Q.; Mao, J.; Wan, B.; Brun, R.; Franzblau, S.G.; Kozikowski, A.P. Searching for New Cures for Tuberculosis: Design, Synthesis, and Biological Evaluation of 2-Methylbenzothiazoles. J. Med. Chem., 2009, 52, 6757-6767.
    • (2009) J. Med. Chem. , vol.52 , pp. 6757-6767
    • Huang, Q.1    Mao, J.2    Wan, B.3    Brun, R.4    Franzblau, S.G.5    Kozikowski, A.P.6
  • 232
    • 77949489030 scopus 로고    scopus 로고
    • Synthesis and antituberculosis activity of some N-pyridyl-N'- thiazolylhydrazine derivatives
    • Turan-Zitouni, G.; Kaplancikli, Z.A.; Oezdemir, A. Synthesis and antituberculosis activity of some N-pyridyl-N'-thiazolylhydrazine derivatives. Eur. J. Med. Chem., 2010, 45(5), 2085-2088.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.5 , pp. 2085-2088
    • Turan-Zitouni, G.1    Kaplancikli, Z.A.2    Oezdemir, A.3
  • 233
    • 77949659737 scopus 로고    scopus 로고
    • Synthesis of some novel 2-substituted-5-[isopropylthiazole] clubbed 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents
    • Suresh, K.G.V.; Rajendraprasad, Y.; Mallikarjuna, B.P.; Chandrashekar, S.M.; Kistayya, C. Synthesis of some novel 2-substituted-5-[isopropylthiazole] clubbed 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents. Eur. J. Med. Chem., 2010, 45(5), 2063-2074.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.5 , pp. 2063-2074
    • Suresh, K.G.V.1    Rajendraprasad, Y.2    Mallikarjuna, B.P.3    Chandrashekar, S.M.4    Kistayya, C.5
  • 234
    • 72049090933 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activity evaluation of new 1,2,4-triazoles and 1,3,4-thiadiazoles bearing imidazo[2,1-b]thiazole moiety
    • Guzeldemirci, N.U.; Kucukbasmaci, O. Synthesis and antimicrobial activity evaluation of new 1,2,4-triazoles and 1,3,4-thiadiazoles bearing imidazo[2,1-b]thiazole moiety. Eur. J. Med. Chem., 2010, 45(1), 63-68.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.1 , pp. 63-68
    • Guzeldemirci, N.U.1    Kucukbasmaci, O.2
  • 235
    • 77249142359 scopus 로고    scopus 로고
    • Identification, synthesis and pharmacological evaluation of tetrahydroindazole based ligands as novel antituberculosis agents
    • Guo, S.; Song, Y.; Huang, Q.; Wang, Y.; Brun, R.; Franzblau, S.G.; Kozikowski, A.P. Identification, synthesis and pharmacological evaluation of tetrahydroindazole based ligands as novel antituberculosis agents. J. Med. Chem., 2010, 53, 649-659.
    • (2010) J. Med. Chem. , vol.53 , pp. 649-659
    • Guo, S.1    Song, Y.2    Huang, Q.3    Wang, Y.4    Brun, R.5    Franzblau, S.G.6    Kozikowski, A.P.7
  • 236
    • 72049083985 scopus 로고    scopus 로고
    • Application of Huisgen (3+2) cycloaddition reaction: Synthesis of 1-(2,3-dihydrobenzofuran-2-yl-methyl [1,2,3]-triazoles and their antitubercular evaluations
    • Tripathi, R.P.; Yadav, A.K.; Ajay, A.; Bisht, S.S.; Chaturvedi, V.; Sinha, S.K. Application of Huisgen (3+2) cycloaddition reaction: Synthesis of 1-(2,3-dihydrobenzofuran-2-yl-methyl [1,2,3]-triazoles and their antitubercular evaluations. Eur. J. Med. Chem., 2010, 45(1), 142-148.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.1 , pp. 142-148
    • Tripathi, R.P.1    Yadav, A.K.2    Ajay, A.3    Bisht, S.S.4    Chaturvedi, V.5    Sinha, S.K.6
  • 237
    • 77955669542 scopus 로고    scopus 로고
    • Synthesis and tuberculostatic activity of novel 1,2,4-triazoles obtained from heterocyclic carbohydrazides
    • Gobis, K.; Foks, H.; Zwolska, Z.; Augustynowicz-Kopec, E. Synthesis and tuberculostatic activity of novel 1,2,4-triazoles obtained from heterocyclic carbohydrazides. Heterocycles, 2010, 81(4), 917-934.
    • (2010) Heterocycles , vol.81 , Issue.4 , pp. 917-934
    • Gobis, K.1    Foks, H.2    Zwolska, Z.3    Augustynowicz-Kopec, E.4
  • 238
    • 41949106754 scopus 로고    scopus 로고
    • Preparation and reactions of sugar azides with alkynes: Synthesis of sugar triazoles as antitubercular agents
    • Singh, B.K.; Yadav, A.K.; Kumar, B.; Gaikwad, A.; Sinha, S.K.; Chaturvedi, V.; Tripathi, R.P. Preparation and reactions of sugar azides with alkynes: Synthesis of sugar triazoles as antitubercular agents. Carbohydr. Res., 2008, 343, 1153-1162.
    • (2008) Carbohydr. Res. , vol.343 , pp. 1153-1162
    • Singh, B.K.1    Yadav, A.K.2    Kumar, B.3    Gaikwad, A.4    Sinha, S.K.5    Chaturvedi, V.6    Tripathi, R.P.7
  • 239
    • 0035833072 scopus 로고    scopus 로고
    • Some 3-thioxo/alkylthio-1,2,4-triazoles with a substituted thiourea moiety as possible antimycobacterials
    • DOI 10.1016/S0960-894X(01)00283-9, PII S0960894X01002839
    • Kucukguzel, I.; Kucukguzel, S.G.; Rollas, S.; Kiraz, M. Some 3-Thioxo/alkylthio-1,2,4-triazoles with a substituted thiourea moiety as possible antimycobacterials. Bioorg. Med. Chem. Lett., 2001, 11, 1703-1707. (Pubitemid 32568302)
    • (2001) Bioorganic and Medicinal Chemistry Letters , vol.11 , Issue.13 , pp. 1703-1707
    • Kucukguzel, I.1    Kucukguzel S.Guniz2    Rollas, S.3    Kiraz, M.4
  • 241
    • 77949659737 scopus 로고    scopus 로고
    • Synthesis of some novel 2-substituted-5-[isopropylthiazole] clubbed 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents
    • Kumar, G.V.S.; Rajendraprasad, Y.; Mallikarjuna, B.P.; Chandrashekar, S.M.; Kistayya, C. Synthesis of some novel 2-substituted-5-[isopropylthiazole] clubbed 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents. Eur. J. Med. Chem., 2010, 45, 2063-2074.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 2063-2074
    • Kumar, G.V.S.1    Rajendraprasad, Y.2    Mallikarjuna, B.P.3    Chandrashekar, S.M.4    Kistayya, C.5
  • 242
    • 0037016645 scopus 로고    scopus 로고
    • Nucleoside analogues as inhibitors of thymidylate kinases: Possible therapeutic applications
    • DOI 10.1002/1439-7633(20020104)3:1<108::AID-CBIC108>3.0.CO;2-B
    • Pochet, S.; Dugue, L.; Douguet, D.; Labesse, G.; Munier-Lehmann, H. Nucleoside Analogues as Inhibitors of Thymidylate Kinases: Possible Therapeutic Applications. ChemBioChem, 2002, 3, 108-110. (Pubitemid 34464803)
    • (2002) ChemBioChem , vol.3 , Issue.1 , pp. 108-110
    • Pochet, S.1    Dugue, L.2    Douguet, D.3    Labesse, G.4    Munier-Lehmann, H.5
  • 243
    • 0037037402 scopus 로고    scopus 로고
    • Synthesis and evaluation of thymidine-5'-O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase
    • DOI 10.1016/S0960-894X(02)00551-6, PII S0960894X02005516
    • Vanheusden, V.; Munier-Lehmann, H.; Pochet, S.; Herdewijn, P.; Van Calenbergh, S. Synthesis and evaluation of thymidine-5'-O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase. Bioorg. Med. Chem. Lett., 2002, 12, 2695-2698. (Pubitemid 35247620)
    • (2002) Bioorganic and Medicinal Chemistry Letters , vol.12 , Issue.19 , pp. 2695-2698
    • Vanheusden, V.1    Munier-Lehmann, H.2    Pochet, S.3    Herdewijn, P.4    Van Calenbergh, S.5
  • 245
    • 0038136960 scopus 로고    scopus 로고
    • Enzymatic and structural analysis of inhibitors designed against Mycobacterium tuberculosis thymidylate kinase: New insights into the phosphoryl transfer mechanism
    • DOI 10.1074/jbc.M209630200
    • Haouz, A.; Vanheusden, V.; Munier-Lehmann, H.; Froeyen, M.; Herdewijn, P.; Van Calenbergh, S.; Delarue, M. Enzymatic and structural analysis of inhibitors designed against Mycobacterium tuberculosis thymidylate kinase. New insights into the phosphoryl transfer mechanism. J. Biol. Chem., 2003, 278, 4963-4971. (Pubitemid 36801005)
    • (2003) Journal of Biological Chemistry , vol.278 , Issue.7 , pp. 4963-4971
    • Haouz, A.1    Vanheusden, V.2    Munier-Lehmann, H.3    Froeyen, M.4    Herdewijn, P.5    Van Calenbergh, S.6    Delarue, M.7
  • 247
    • 9744241646 scopus 로고    scopus 로고
    • Discovery of bicyclic thymidine analogues as selective and high-affinity inhibitors of Mycobacterium tuberculosis thymidine monophosphate kinase
    • DOI 10.1021/jm040847w
    • Vanheusden, V.; Munier-Lehmann, H.; Froeyen, M.; Busson, R.; Rozenski, J.; Herdewijn, P.; Van Calenbergh, S. Discovery of Bicyclic Thymidine analogues as selective and high-affinity inhibitors of Mycobacterium tuberculosis thymidine monophosphate kinase. J. Med. Chem., 2004, 47, 6187-6194. (Pubitemid 39587243)
    • (2004) Journal of Medicinal Chemistry , vol.47 , Issue.25 , pp. 6187-6194
    • Vanheusden, V.1    Munier-Lehmann, H.2    Froeyen, M.3    Busson, R.4    Rozenski, J.5    Herdewijn, P.6    Van Calenbergh, S.7
  • 250
    • 0028825294 scopus 로고
    • New benzylpyrimidines: Inhibition of DHFR from various species. QSAR, CoMFA and PC analysis
    • Czaplinski, K.H.; Hansel, W.; Wiese, M.; Seydel, J.K. New benzylpyrimidines: Inhibition of DHFR from various species. QSAR, CoMFA and PC analysis. Eur. J. Med. Chem., 1995, 30, 779-787.
    • (1995) Eur. J. Med. Chem. , vol.30 , pp. 779-787
    • Czaplinski, K.H.1    Hansel, W.2    Wiese, M.3    Seydel, J.K.4
  • 251
    • 77954217431 scopus 로고    scopus 로고
    • Crystallographic and docking studies of purine nucleoside phosphorylase from Mycobacterium tuberculosis
    • Ducati, R.G.; Basso, L.A.; Santos, D.S.; de Azevedo, Jr. W.F. Crystallographic and docking studies of purine nucleoside phosphorylase from Mycobacterium tuberculosis. Bioorg. Med. Chem., 2010, 18, 4769-4774.
    • (2010) Bioorg. Med. Chem. , vol.18 , pp. 4769-4774
    • Ducati, R.G.1    Basso, L.A.2    Santos, D.S.3    De Azevedo Jr., W.F.4
  • 252
    • 0028825294 scopus 로고
    • New benzylpyrimidines: Inhibition of DHFR from various species. QSAR, CoMFA and PC analysis
    • Czaplinski, K.H.; Hansel, W.; Wiese, M.; Seydel, J.K. New benzylpyrimidines: Inhibition of DHFR from various species. QSAR, CoMFA and PC analysis. Eur. J. Med. Chem.; 1995, 30, 779-787.
    • (1995) Eur. J. Med. Chem. , vol.30 , pp. 779-787
    • Czaplinski, K.H.1    Hansel, W.2    Wiese, M.3    Seydel, J.K.4
  • 253
    • 0035121462 scopus 로고    scopus 로고
    • Experimental in vitro efficacy study on the interaction of epiroprim plus isoniazid against Mycobacterium tuberculosis
    • DOI 10.1159/000048511
    • Dosso, M.; Ouattara, L.; Cherif, A.M.; Bouzid, S.A.; Haller, L.; Fernex, M. Experimental in vitro Efficacy Study on the Interaction of Epiroprim plus Isoniazid against Mycobacterium tuberculosis. Chemotherapy, 2001, 47, 123-127. (Pubitemid 32149703)
    • (2001) Chemotherapy , vol.47 , Issue.2 , pp. 123-127
    • Dosso, M.1    Ouattara, L.2    Cherif, A.M.3    Bouzid, S.A.4    Haller, L.5    Fernex, M.6
  • 255
    • 77955856678 scopus 로고    scopus 로고
    • Effect of halogen atom localization on the level of antimycobacterial activity of 2-Amino-4-arylamino-6-methylpyrimidines
    • Erkin, A.V.; Krutikov, V.I. Effect of Halogen Atom Localization on the Level of Antimycobacterial Activity of 2-Amino-4-arylamino-6-methylpyrimidines. Russian Journal of General Chemistry. 2010, 80(4), 818-824.
    • (2010) Russian Journal of General Chemistry. , vol.80 , Issue.4 , pp. 818-824
    • Erkin, A.V.1    Krutikov, V.I.2
  • 256
    • 77953130147 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of pyrimidine analogs of antimycobacterial purines
    • Read, M.L.; Braendvang, M.; Miranda, P.O.; Gundersen, L.L. Synthesis and biological evaluation of pyrimidine analogs of antimycobacterial purines. Bioorg. Med. Chem., 2010, 18, 3885-3897.
    • (2010) Bioorg. Med. Chem. , vol.18 , pp. 3885-3897
    • Read, M.L.1    Braendvang, M.2    Miranda, P.O.3    Gundersen, L.L.4
  • 257
    • 77954349411 scopus 로고    scopus 로고
    • Synthesis and in vitro evaluation of substituted pyrimido[5,4-d] pyrimidines as a novel class of Antimycobacterium tuberculosis agents
    • Bacelar, A.H.; Carvalho, M.A.; Proenca, M.F. Synthesis and in vitro evaluation of substituted pyrimido[5,4-d]pyrimidines as a novel class of Antimycobacterium tuberculosis agents Eur. J. Med. Chem., 2010, 45 , 3234-3239.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 3234-3239
    • Bacelar, A.H.1    Carvalho, M.A.2    Proenca, M.F.3
  • 259
    • 0035048959 scopus 로고    scopus 로고
    • Antimycobacterial activity of 1-deaza-7,8-dihydropteridine derivatives against Mycobacterium tuberculosis and Mycobacterium avium complex in vitro
    • Suling, W.J.; Maddry, J.A. Antimycobacterial activity of 1-deaza-7,8-dihydropteridine derivatives against Mycobacterium tuberculosis and Mycobacterium avium complex in vitro. J. Antimicrob. Chemother., 2001, 47, 451-454. (Pubitemid 32303412)
    • (2001) Journal of Antimicrobial Chemotherapy , vol.47 , Issue.4 , pp. 451-454
    • Suling, W.J.1    Maddry, J.A.2
  • 260
    • 77954316167 scopus 로고    scopus 로고
    • Discovery of new 1,3,5-triazine scaffolds withpotent activity against Mycobacterium tuberculosis H37Rv
    • Sunduru, N.; Gupta, L.; Chaturvedi, V.; Dwivedi, R.; Sinha, S.; Chauhan, P.M.S. Discovery of new 1,3,5-triazine scaffolds withpotent activity against Mycobacterium tuberculosis H37Rv. Eur. J. Med. Chem., 2010, 45, 3335-3345.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 3335-3345
    • Sunduru, N.1    Gupta, L.2    Chaturvedi, V.3    Dwivedi, R.4    Sinha, S.5    Chauhan, P.M.S.6
  • 261
    • 0029780824 scopus 로고    scopus 로고
    • Quantitative structure-activity relationships for the in vitro antimycobacterial activity of pyrazinoic acid esters
    • DOI 10.1021/jm950538t
    • Bergmann, K.E.; Cynamon, M.H.; Welch, J.T. Quantitative Structure-Activity Relationships for the in Vitro Antimycobacterial Activity of Pyrazinoic Acid Esters. J. Med. Chem., 1996, 39, 3394-3400. (Pubitemid 26322865)
    • (1996) Journal of Medicinal Chemistry , vol.39 , Issue.17 , pp. 3394-3400
    • Bergmann, K.E.1    Cynamon, M.H.2    Welch, J.T.3
  • 262
    • 0032543736 scopus 로고    scopus 로고
    • Antimycobacterial activity of substituted isosteres of pyridine- and pyrazinecarboxylic acids
    • DOI 10.1021/jm9708745
    • Wachter, G.A.; Davis, M.C. Martin AR, Franzblan SG. Antimycobacterial Activity of Substituted Isosteres of Pyridine-and Pyrazinecarboxylic Acids. J. Med. Chem. 1998, 41, 2436-2438. (Pubitemid 28285745)
    • (1998) Journal of Medicinal Chemistry , vol.41 , Issue.13 , pp. 2436-2438
    • Wachter, G.A.1    Davis, M.C.2    Martin, A.R.3    Franzblau, S.G.4
  • 263
    • 0035837067 scopus 로고    scopus 로고
    • Antimycobacterial activity of substituted isosteres of pyridine- and pyrazinecarboxylic acids. 2
    • DOI 10.1021/jm000350w
    • Gezginci, M.H.; Martin, A.R.; Franzblau, S.G. Antimycobacterial activity of substituted isosteres of pyridine and pyrazinecarboxylic acids. 2. J. Med. Chem., 2001, 44(10), 1560-1563. (Pubitemid 32852198)
    • (2001) Journal of Medicinal Chemistry , vol.44 , Issue.10 , pp. 1560-1563
    • Gezginci, M.H.1    Martin, A.R.2    Franzblau, S.G.3
  • 264
    • 0036046387 scopus 로고    scopus 로고
    • Synthesis of pyrazinoyl and related heterocycles as possible antitubercular agents
    • Govindarajan, R.; Bhat, A.R. Synthesis of pyrazinyl and related heterocycles as possible antitubercular agents. Indian J. Heterocyclic Chemistry. 2002, 11(4), 337-338. (Pubitemid 40768213)
    • (2002) Indian Journal of Heterocyclic Chemistry , vol.11 , Issue.4 , pp. 337-338
    • Govindarajan, R.1    Bhat, A.R.2
  • 265
    • 77949681145 scopus 로고    scopus 로고
    • 3D-QSAR study on ring substituted imidazoles for their antitubercular activity
    • Sharma, G.K.; Pathak, D. 3D-QSAR study on ring substituted imidazoles for their antitubercular activity. Lett. Drug Design Discovery, 2010, 7(2), 128-132.
    • (2010) Lett. Drug Design Discovery , vol.7 , Issue.2 , pp. 128-132
    • Sharma, G.K.1    Pathak, D.2
  • 266
    • 76649098896 scopus 로고    scopus 로고
    • Identification of triazinoindol-benzimidazolones as nanomolar inhibitors of the Mycobacterium tuberculosis enzyme TDP-6-deoxy-D-xylo-4-hexopyranosid-4- ulose 3,5-epimerase (RmlC
    • Sivendran, S.; Jones, V.; Sun, D.; Wang, Y.; Grzegorzewicz, A.E.; Scherman, M.S.; Napper, A.D.; McCammon, J.A.; Lee, R.E.; Diamond, S.L.; McNeil, M. Identification of triazinoindol-benzimidazolones as nanomolar inhibitors of the Mycobacterium tuberculosis enzyme TDP-6-deoxy-D-xylo-4-hexopyranosid-4-ulose 3,5-epimerase (RmlC). Bioorg. Med. Chem., 2010, 18(2), 896-908.
    • (2010) Bioorg. Med. Chem. , vol.18 , Issue.2 , pp. 896-908
    • Sivendran, S.1    Jones, V.2    Sun, D.3    Wang, Y.4    Grzegorzewicz, A.E.5    Scherman, M.S.6    Napper, A.D.7    McCammon, J.A.8    Lee, R.E.9    Diamond, S.L.10    McNeil, M.11
  • 268
    • 52449097257 scopus 로고    scopus 로고
    • Discovery of antimycobacterial spiro-piperidin-4ones: An atom economic, stereoselective synthesis, and biological intervention
    • 2008
    • Kumar, R.R.; Perumal, S.; Senthilkumar, P.; Yogeeswari, P.; Sriram, D. Discovery of antimycobacterial spiro-piperidin-4ones: An atom economic, stereoselective synthesis, and biological intervention. J. Med. Chem., 2008, 51, 5731-5735 (2008
    • (2008) J. Med. Chem. , vol.51 , pp. 5731-5735
    • Kumar, R.R.1    Perumal, S.2    Senthilkumar, P.3    Yogeeswari, P.4    Sriram, D.5
  • 269
    • 72049094262 scopus 로고    scopus 로고
    • A highly atom economic, chemo-region-and stereoselective synthesis and evaluation of spiro-pyrrolothiazoles as antitubercular agents
    • Karthikeyan, S.V.; Bala, B.D.; Raja, V.P.A.; Perumal, S.; Yogeeswari, P.; Sriram, D. A highly atom economic, chemo-region-and stereoselective synthesis and evaluation of spiro-pyrrolothiazoles as antitubercular agents. Bioorg. Med. Chem. Lett., 2010, 20, 350-353.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 350-353
    • Karthikeyan, S.V.1    Bala, B.D.2    Raja, V.P.A.3    Perumal, S.4    Yogeeswari, P.5    Sriram, D.6
  • 270
    • 41649096500 scopus 로고    scopus 로고
    • N-Aroyl-3,5-bis(benzylidene)-4-piperidones: A novel class of antimycobacterial agents
    • DOI 10.1016/j.bmc.2008.02.009, PII S0968089608001156
    • Das, U.; Das, S.; Bandy, B.; Stables, J.P.; Dimmocka, J.R. N-Aroyl-3,5-bis(bezylidene)-4-piperidones: A novel class of antimycobacterial agents. Bioorg. Med. Chem., 2008, 16, 3602-3607. (Pubitemid 351484043)
    • (2008) Bioorganic and Medicinal Chemistry , vol.16 , Issue.7 , pp. 3602-3607
    • Das, U.1    Das, S.2    Bandy, B.3    Stables, J.P.4    Dimmock, J.R.5
  • 271
    • 56249114531 scopus 로고    scopus 로고
    • A facile synthesis, antibacterial, and antitubercular studies of some piperin-4-one and tetrahydropyridine derivatives
    • Aridoss, G.; Amirthaganesan, S.; Kumar, N.A.; Kim, J.T.; Lim, K.T.; Kabilan, S.; Jeong, Y.T. A facile synthesis, antibacterial, and antitubercular studies of some piperin-4-one and tetrahydropyridine derivatives. Bioorg. Med. Chem. Lett., 2008, 18, 6542-6548.
    • (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 6542-6548
    • Aridoss, G.1    Amirthaganesan, S.2    Kumar, N.A.3    Kim, J.T.4    Lim, K.T.5    Kabilan, S.6    Jeong, Y.T.7
  • 272
    • 72249100101 scopus 로고    scopus 로고
    • 1,3-Dipolar cycloaddition of C-aryl-N-phenylnitrones to (R)-1-(1-phenylethyl)-3-[(E)-arylmethylidene]tetrahydro-4(1H)-pyridinones: Synthesis and antimycobacterial evaluation of enantiomerically pure spiroisoxazolidines
    • Kumar, R.S.; Perumal, S.; Shetty, K.A.; Yogeeswari, P.; Sriram, D. 1,3-Dipolar cycloaddition of C-aryl-N-phenylnitrones to (R)-1-(1-phenylethyl)-3- [(E)-arylmethylidene]tetrahydro-4(1H)-pyridinones: Synthesis and antimycobacterial evaluation of enantiomerically pure spiroisoxazolidines. Eur. J. Med. Chem., 2010, 45(1), 124-133.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.1 , pp. 124-133
    • Kumar, R.S.1    Perumal, S.2    Shetty, K.A.3    Yogeeswari, P.4    Sriram, D.5
  • 276
    • 77951138907 scopus 로고    scopus 로고
    • Utilization of the Suzuki coupling to enhance the antituberculosis activity of aryloxazoles
    • Moraski, G.C.; Franzblau, S.G.; Miller, M.J. Utilization of the Suzuki coupling to enhance the antituberculosis activity of aryloxazoles. Heterocycles, 2010, 80(2), 977-988.
    • (2010) Heterocycles , vol.80 , Issue.2 , pp. 977-988
    • Moraski, G.C.1    Franzblau, S.G.2    Miller, M.J.3
  • 279
    • 77949487512 scopus 로고    scopus 로고
    • Structure-activity relationship of new antituberculosis agents derived from oxazoline and oxazole benzyl esters
    • Moraski, G.C.; Chang, M.; Villegas-Estrada, A.; Franzblau, S.G.; Moellmann, U.; Miller, M.J. Structure-activity relationship of new antituberculosis agents derived from oxazoline and oxazole benzyl esters. Eur. J. Med. Chem., 2010, 45(5), 1703-1716.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.5 , pp. 1703-1716
    • Moraski, G.C.1    Chang, M.2    Villegas-Estrada, A.3    Franzblau, S.G.4    Moellmann, U.5    Miller, M.J.6
  • 282
    • 77950037279 scopus 로고    scopus 로고
    • Substituted hydrazinecarbothioamide as potent antitubercular agents: Synthesis and quantitative structure-activity relationship (QSAR
    • Singh, S.; Mandal, P.K.; Singh, N.; Misra, A.K.; Singh, S.; Chaturvedi, V.; Sinha, S.; Saxena, A.K. Substituted hydrazinecarbothioamide as potent antitubercular agents: Synthesis and quantitative structure-activity relationship (QSAR) Bioorg. Med. Chem. Lett., 2010, 20, 2597-2600.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 2597-2600
    • Singh, S.1    Mandal, P.K.2    Singh, N.3    Misra, A.K.4    Singh, S.5    Chaturvedi, V.6    Sinha, S.7    Saxena, A.K.8
  • 283
    • 0037019175 scopus 로고    scopus 로고
    • Synthesis, characterization and evaluation of antituberculosis activity of some hydrazones
    • Kocyigit, K.B.; Rollas, S. Synthesis, characterization and evaluation of antituberculosis activity of some hydrazones. Farmaco., 2010, 57(7), 595-599.
    • (2010) Farmaco. , vol.57 , Issue.7 , pp. 595-599
    • Kocyigit, K.B.1    Rollas, S.2
  • 284
    • 0036241998 scopus 로고    scopus 로고
    • Synthesis and antitubercular evaluation of 4-quinolylhydrazones
    • Savini, L.; Chiasserini, L.; Gaeta, A.; Pellerano, C. Synthesis and antitubercular evaluation of 4-quinolylhydrazones. Bioorg. Med. Chem., 2010, 10, 2193-2198.
    • (2010) Bioorg. Med. Chem. , vol.10 , pp. 2193-2198
    • Savini, L.1    Chiasserini, L.2    Gaeta, A.3    Pellerano, C.4
  • 285
    • 0037019131 scopus 로고    scopus 로고
    • Synthesis and antitubercular activity of 4-(3-coumarinyl)-3-cyclohexyl-4- thiazolin-2-one benzylidenehydrazones
    • DOI 10.1016/S0014-827X(02)01254-5, PII S0014827X02012545
    • Karali, N.; Kocabalkanli, A.; Gursoy, A.; Ates, O. Synthesis and antitubercular activity of 4-(3-coumarinyl)-3-cyclohexyl-4-thiazolin-2-one benzylidenehydrazones. Farmaco., 2002, 57, 589-593. (Pubitemid 34765753)
    • (2002) Farmaco , vol.57 , Issue.7 , pp. 589-593
    • Karal, N.1    Kocabalkanl, A.2    Gursoy, A.3    Ates, O.4
  • 287
    • 0024458038 scopus 로고
    • Synthesis and antitubercular activity of N-(2-naphthyl)glycine hydrazide analogues
    • Ramamurthy, B.; Bhatt, M.V. Synthesis and antitubercular activity of N-(2-naphthyl)glycine hydrazide analogs. J. Med. Chem., 1989, 32, 2421-2426. (Pubitemid 19269969)
    • (1989) Journal of Medicinal Chemistry , vol.32 , Issue.11 , pp. 2421-2426
    • Ramamurthy, B.1    Bhatt, M.V.2
  • 288
    • 0033675098 scopus 로고    scopus 로고
    • Synthesis of new fluorine substituted hydrazinecarboxamides and hydrazine carbothioamides having antitubercular and fungicidal activity
    • Nalavde, Y.M.; Josho, V. Synthesis of new fluorine substituted hydrazinecarboxamides and hydrazine carbothioamides having antitubercular and fungicidal activity. Ind. J. Chem., 2000, 39B, 634-637.
    • (2000) Ind. J. Chem. , vol.39 B , pp. 634-637
    • Nalavde, Y.M.1    Josho, V.2
  • 289
    • 0033258877 scopus 로고    scopus 로고
    • Pyrazinoic acid hydrazide derivatives: Synthesis and antimycobacterial activities
    • Miniyar, P.B.; Bhat, A.R. Pyrazinoic acid hydrazide derivatives: Synthesis and antimycobacterial activities. Ind J Het Chem., 1999, 9, 155-156.
    • (1999) Ind J Het Chem. , vol.9 , pp. 155-156
    • Miniyar, P.B.1    Bhat, A.R.2
  • 290
    • 74349108294 scopus 로고    scopus 로고
    • 5-Nitrothiazolylthiosemicarbazones: Synthesis and antimycobacterial evaluation against tubercular and non-tubercular mycobacterial species
    • Sriram, D.; Yogeeswari, P.; Senthilkumar, P.; Sangaraju, D. 5-Nitrothiazolylthiosemicarbazones: Synthesis and antimycobacterial evaluation against tubercular and non-tubercular mycobacterial species. J. Enzyme Inhib. Med. Chem., 2010, 25(1), 105-110.
    • (2010) J. Enzyme Inhib. Med. Chem. , vol.25 , Issue.1 , pp. 105-110
    • Sriram, D.1    Yogeeswari, P.2    Senthilkumar, P.3    Sangaraju, D.4
  • 291
    • 0025553897 scopus 로고
    • Studies on aryl thiosemicarbazones and 2-oxo-2-thiazolin-2-ylhydrazones
    • Jolly, V.S.; Sharma, K.P. Studies on aryl thiosemicarbazones and 2-oxo-2-thiazolin-2-ylhydrazones. J. Ind. Chem. Soc., 1990, 67(5), 412-413.
    • (1990) J. Ind. Chem. Soc. , vol.67 , Issue.5 , pp. 412-413
    • Jolly, V.S.1    Sharma, K.P.2
  • 292
    • 0035170176 scopus 로고    scopus 로고
    • Synthesis and in vitro tuberculostatic activity of Co (II), Cu (II) and Ni (II) complexes of dialdehyde starch dithiosemicarbazone
    • Para, A.; Klisiewicz-Panszczyk, T.; Jurek, I. Synthesis and in vitro tuberculostatic activity of Co (II), Cu (II) and Ni (II) complexes of dialdehyde starch dithiosemicarbazone. Acta Pol Pharm., 2001, 58, 405-408. (Pubitemid 33076823)
    • (2001) Acta Poloniae Pharmaceutica - Drug Research , vol.58 , Issue.5 , pp. 405-408
    • Para, A.1    Klisiewicz-Panszczyk, T.2    Jurek, I.3
  • 293
    • 0020319879 scopus 로고
    • Correlations between structure and antimycobacterial activity in a series of 2-acetylpyridine thiosemicarbazones
    • Collins, F.M.; Klayman, D.L.; Morrison, N.E. Correlations between Structure and Antimycobacterial Activity in a Series of 2-Acetylpyridine Thiosemicarbazones. J. Gen. Microbiol., 1982, 128, 1349-1356. (Pubitemid 12037168)
    • (1982) Journal of General Microbiology , vol.128 , Issue.6 , pp. 1349-1356
    • Collins, F.M.1    Klayman, D.L.2    Morrison, N.E.3
  • 294
    • 20744446480 scopus 로고    scopus 로고
    • In vitro antimycobacterial activity of newly synthesised S-alkylisothiosemicarbazone derivatives and synergistic interactions in combination with rifamycins against Mycobacterium avium
    • DOI 10.1016/j.ijantimicag.2005.03.005, PII S0924857905001068
    • Logua, A.D.; Saddi, M.; Onnis, V.; Sanna, C.; Congiu, C.; Borgna, R.; Cocco, M.T. In vitro antimycobacterial activity of newly synthesised Salkylisothiosemicarbazone derivatives and synergistic interactions in combination with rifamycins against Mycobacterium avium. Int. J. Antimicrob. Agents, 2005, 26, 28-32. (Pubitemid 40854112)
    • (2005) International Journal of Antimicrobial Agents , vol.26 , Issue.1 , pp. 28-32
    • De Logu, A.1    Saddi, M.2    Onnis, V.3    Sanna, C.4    Congiu, C.5    Borgna, R.6    Cocco, M.T.7
  • 295
    • 0036155349 scopus 로고    scopus 로고
    • Synthesis and antimycobacterial activity of new S- alkylisothiosemicarbazone derivatives
    • DOI 10.1016/S0968-0896(01)00310-8, PII S0968089601003108
    • Cocco, M.T.; Congiu, C.; Onnis, V.; Pellerano, M.L.; Logu, A.D. Synthesis and antimycobacterial activity of new S-alkylisothiosemicarbazone derivatives. Bioorg. Med. Chem., 2002, 10, 501-506. (Pubitemid 34112441)
    • (2002) Bioorganic and Medicinal Chemistry , vol.10 , Issue.3 , pp. 501-506
    • Cocco, M.T.1    Congiu, C.2    Onnis, V.3    Pellerano, M.L.4    Logu, A.D.5
  • 296
    • 10444236165 scopus 로고
    • Reactions of cyclic anhydrides with thiosemicarbazides: Synthesis and antituberculosis activity of glutaconylthiosemicarbazide and its cyclic analogs
    • Deshmukh, N.J.; Kulkarni, R.A.; Deodhar, K.D. Reactions of cyclic anhydrides with thiosemicarbazides: Synthesis and antituberculosis activity of glutaconylthiosemicarbazide and its cyclic analogs. Ind. J. Chem., 1985, 24B(3), 330-332.
    • (1985) Ind. J. Chem. , vol.24 B , Issue.3 , pp. 330-332
    • Deshmukh, N.J.1    Kulkarni, R.A.2    Deodhar, K.D.3
  • 298
    • 0142105859 scopus 로고    scopus 로고
    • Treatment of Mycobacterium avium-intracellulare complex lung disease with a macrolide, ethambutol, and clofazimine
    • Field, S.K.; Cowie, R.L. Treatment of Mycobacterium avium-intracellulare complex lung disease with a macrolide, ethambutol, and clofazimine. Chest, 2003, 124, 1482-1786.
    • (2003) Chest , vol.124 , pp. 1482-1786
    • Field, S.K.1    Cowie, R.L.2
  • 299
    • 0028283172 scopus 로고
    • In vitro and in vivo synergistic effect of isoniazid with streptomycin and clofazimine against Mycobacterium avium complex (MAC)
    • DOI 10.1016/0962-8479(94)90010-8
    • Reddy, V.M.; Srinivasan, S.; Gangadharam, P.R. In vitro and in vivo synergistic effect of isoniazid with streptomycin and clofazimine against Mycobacterium avium complex (MAC). Tuber. Lung Dis., 1994, 75, 208-212. (Pubitemid 24217279)
    • (1994) Tubercle and Lung Disease , vol.75 , Issue.3 , pp. 208-212
    • Venkata Reddy, M.1    Srinivasan, S.2    Gangadharam, P.R.J.3
  • 302
    • 0035098674 scopus 로고    scopus 로고
    • Enhancement of antibiotic activity against poly-drug resistant Mycobacterium tuberculosis by phenothiazines
    • DOI 10.1016/S0924-8579(00)00343-5, PII S0924857900003435
    • Viveiros, M.; Amaral, L. Enhancement of antibiotic activity against polydrug-resistant Mycobacterium tuberculosis by phenothiazines. Int J. Antimicro. Agents, 2001, 17, 225-228. (Pubitemid 32229901)
    • (2001) International Journal of Antimicrobial Agents , vol.17 , Issue.3 , pp. 225-228
    • Viveiros, M.1    Amaral, L.2
  • 303
    • 0030462751 scopus 로고    scopus 로고
    • Inhibition of the respiration of multi-drug resistant clinical isolates of Mycobacterium tuberculosis by thioridazine: Potential use for initial therapy of freshly diagnosed tuberculosis
    • DOI 10.1093/jac/38.6.1049
    • Amaral, L.; Kristiansen, J.E.; Abebe, L.S.; Millett, W. Inhibition of the respiration of multi-drug resistant clinical isolates of Mycobacterium tuberculosis by thioridazine: Potential use for initial therapy of freshly diagnosed tuberculosis. J. Antimicrob. Chemother., 1996, 38, 1049-1053. (Pubitemid 27073284)
    • (1996) Journal of Antimicrobial Chemotherapy , vol.38 , Issue.6 , pp. 1049-1053
    • Amaral, L.1    Kristiansen, J.E.2    Abebe, L.S.3    Millett, W.4
  • 304
    • 0035010729 scopus 로고    scopus 로고
    • Activity of phenothiazines against antibiotic-resistant Mycobacterium tuberculosis: A review supporting further studies that may elucidate the potential use of thioridazine as anti-tuberculosis therapy
    • Amaral, L.; Kristiansen, J.E.; Viveiros, M.; Atougui, J. Activity of phenothiazines against antibiotic-resistant Mycobacterium tuberculosis: A review supporting further studies that may elucidate the potential use of thioridazine as an anti-tuberculosis therapy. J. Antimicrob. Chemother., 2001, 47, 505-511. (Pubitemid 32447635)
    • (2001) Journal of Antimicrobial Chemotherapy , vol.47 , Issue.5 , pp. 505-511
    • Amaral, L.1    Kristiansen, J.E.2    Viveiros, M.3    Atouguia, J.4
  • 305
    • 77950849122 scopus 로고    scopus 로고
    • Thioridazine cures extensively drug-resistant tuberculosis (XDR-TB) and the need for global trials is now!
    • Amarala, L.; Boereeb, M.J.; Gillespie, S.H.; Udwadiad, Z.F.; Soolingene, D.V. Thioridazine cures extensively drug-resistant tuberculosis (XDR-TB) and the need for global trials is now! Int J. Antimicro. Agents, 2010, 35, 524-526.
    • (2010) Int J. Antimicro. Agents , vol.35 , pp. 524-526
    • Amarala, L.1    Boereeb, M.J.2    Gillespie, S.H.3    Udwadiad, Z.F.4    Soolingene, D.V.5
  • 307
    • 0034501311 scopus 로고    scopus 로고
    • Pleuromutilin antibiotics
    • Hunt, E. Pleuromutilin antibiotics. Drugs Future, 2000, 25, 1163-1168. (Pubitemid 32094765)
    • (2000) Drugs of the Future , vol.25 , Issue.11 , pp. 1163-1168
    • Hunt, E.1
  • 308
    • 33645767206 scopus 로고    scopus 로고
    • Interaction of pleuromutilin derivatives with the ribosomal peptidyl transferase center
    • Long, K.S.; Hansen, L.H.; Jakobsen, L.; Vester, B. Interaction of Pleuromutilin Derivatives with the Ribosomal Peptidyl Transferase Center. Antimicrob. Agents Chemother., 2006, 50, 1458-1462.
    • (2006) Antimicrob. Agents Chemother. , vol.50 , pp. 1458-1462
    • Long, K.S.1    Hansen, L.H.2    Jakobsen, L.3    Vester, B.4
  • 309
    • 9644281855 scopus 로고    scopus 로고
    • Inhibition of peptide bond formation by pleuromutilins: The structure of the 50S ribosomal subunit from Deinococcus radiodurans in complex with tiamulin
    • DOI 10.1111/j.1365-2958.2004.04346.x
    • Schluenzen, F.; Pyetan, E.; Fucini, P.; Yonath, A.; Harms, J.M. Inhibition of peptide bond formation by pleuromutilins: The structure of the 50S ribosomal subunit from Deinococcus radiodurans in complex with tiamulin. Mol. Microbiol., 2004, 54, 1287-1294. (Pubitemid 39578271)
    • (2004) Molecular Microbiology , vol.54 , Issue.5 , pp. 1287-1294
    • Schlunzen, F.1    Pyetan, E.2    Fucini, P.3    Yonath, A.4    Harms, J.M.5
  • 312
    • 17144376741 scopus 로고    scopus 로고
    • Synthesis, biological activity, and SAR of antimycobacterial 9-aryl-, 9-arylsulfonyl-, and 9-benzyl-6-(2-furyl)purines
    • Bakkestuen, A.K.; Gundersen, L.L.; Utenova, B.T. Synthesis, biological activity, and SAR of antimycobacterial 9-aryl-, 9-arylsulfonyl-, and 9-benzyl-6-(2-furyl)purines. J. Med. Chem., 2005, 48, 2710-2723.
    • (2005) J. Med. Chem. , vol.48 , pp. 2710-2723
    • Bakkestuen, A.K.1    Gundersen, L.L.2    Utenova, B.T.3
  • 313
    • 27544509944 scopus 로고    scopus 로고
    • Selective anti-tubercular purines: Synthesis and chemotherapeutic properties of 6-aryl- and 6-heteroaryl-9-benzylpurines
    • DOI 10.1016/j.bmc.2005.06.054, PII S0968089605005961
    • Braendvang, M.; Gundersen, L.L. Selective anti-tubercular purines: Synthesis and chemotherapeutic properties of 6-aryl-and 6-heteroaryl-9- benzylpurines. Bioorg. Med. Chem., 2005, 13, 6360-6373. (Pubitemid 41539300)
    • (2005) Bioorganic and Medicinal Chemistry , vol.13 , Issue.23 , pp. 6360-6373
    • Braendvang, M.1    Gundersen, L.-L.2
  • 315
    • 1342324049 scopus 로고    scopus 로고
    • Synthesis, anti-mycobacterial, anti-trichomonas and anti-candida in vitro activities of 2-substituted-6,7-difluoro-3-methylquinoxaline 1,4-dioxides
    • DOI 10.1016/j.ejmech.2003.11.008
    • Carta, A.; Loriga, M.; Paglietti, G.; Mattana, A.; Fiori, P.L.; Mollicotti, P.; Sechi, L.; Zanetti, S. Synthesis, anti-mycobacterial, anti-trichomonas and anti-candida in vitro activities of 2-substituted-6,7- difluoro-3-methylquinoxaline 1,4-dioxides. Eur. J. Med. Chem.; 2004, 39, 195-203. (Pubitemid 38249532)
    • (2004) European Journal of Medicinal Chemistry , vol.39 , Issue.2 , pp. 195-203
    • Carta, A.1    Loriga, M.2    Paglietti, G.3    Mattana, A.4    Fiori, P.L.5    Mollicotti, P.6    Sechi, L.7    Zanetti, S.8
  • 316
    • 0037361604 scopus 로고    scopus 로고
    • Studies on novel bacterial translocase I inhibitors, A-500359s. II. Biological activities of A-500359 A, C, D and G
    • Muramatsu, Y.; Ishii, M.M.; Inukai, M. Studies on novel bacterial translocase I inhibitors, A-500359s. II. Biological activities of A-500359 A, C, D and G. J. Antibiot., 2003, 56, 253-258. (Pubitemid 36443393)
    • (2003) Journal of Antibiotics , vol.56 , Issue.3 , pp. 253-258
    • Muramatsu, Y.1    Ishii, M.M.2    Inukai, M.3
  • 317
    • 0037363273 scopus 로고    scopus 로고
    • Studies on novel bacterial translocase I inhibitors, A-500359s. III. Deaminocaprolactam derivatives of capuramycin: A-500359 E, F, H, M-1 and M-2
    • Muramatsu, Y.; Miyakoshi, S.; Ogawa, Y.; Ohnuki, T.; Ishii, M.M.; Arai, M.; Takatsu, T.; Inukai, M. Studies on novel bacterial translocase I inhibitors, A-500359s. III. Deaminocaprolactam derivatives of capuramycin: A-500359 E, F, H; M-1 and M-2. J. Antibiot., 2003, 56, 259-267. (Pubitemid 36443394)
    • (2003) Journal of Antibiotics , vol.56 , Issue.3 , pp. 259-267
    • Muramatsu, Y.1    Miyakoshi, S.2    Ogawa, Y.3    Ohnuki, T.4    Ishii, M.M.5    Arai, M.6    Takatsu, T.7    Inukai, M.8
  • 331
    • 61349152974 scopus 로고    scopus 로고
    • A facile synthesis of α,α'-(EE)-bis(benzylidene)- cycloalkanones and their antitubercular evaluations
    • Singh, N.; Pandey, J.; Yadav, A. A facile synthesis of α,α'-(EE)-bis(benzylidene)-cycloalkanones and their antitubercular evaluations. Eur. J. Med. Chem., 2009, 44, 1705-1709.
    • (2009) Eur. J. Med. Chem. , vol.44 , pp. 1705-1709
    • Singh, N.1    Pandey, J.2    Yadav, A.3
  • 333
    • 1342345087 scopus 로고    scopus 로고
    • Bauhinoxepins A and B: New Antimycobacterial Dibenzo[b,f]oxepins from Bauhinia saccocalyx
    • DOI 10.1002/hlca.200490006
    • Kittakoop, P.; Nopichai, S.; Thongon, N.; Charoenchai, P.; Thebtaranonth, Y.; Bauhinoxepins, A. B. New antimycobacterial dibenzo[b,f]oxepins from Bauhinia saccocalyx. Helvetica chimica acta, 2004, 87, 175-179. (Pubitemid 38250123)
    • (2004) Helvetica Chimica Acta , vol.87 , Issue.1 , pp. 175-179
    • Kittakoop, P.1    Nopichai, S.2    Thongon, N.3    Charoenchai, P.4    Thebtaranonth, Y.5
  • 334
    • 73449131179 scopus 로고    scopus 로고
    • 2-aryl-3-(1H-azol-1-yl)-1H-indole derivatives: A new class of antimycobacterial compounds conventional heating in comparison with MWassisted synthesis
    • Zampieri, D.; Mamolo, M.G.; Laurini, E.; Scialino, G.; Banfi, E. Vio L. 2-aryl-3-(1H-azol-1-yl)-1H-indole derivatives: A new class of antimycobacterial compounds conventional heating in comparison with MWassisted synthesis. Arch. Pharm. Chem. Life Sci., 2009, 342, 716-722.
    • (2009) Arch. Pharm. Chem. Life Sci. , vol.342 , pp. 716-722
    • Zampieri, D.1    Mamolo, M.G.2    Laurini, E.3    Scialino, G.4    Banfi, E.5    Vio, L.6
  • 335
    • 0019868222 scopus 로고
    • Synthesis and antibacterial activity of 1-(arylamino)-1H-pyrroles and 4-(1H-pyrrol-1-ylimino)-2,5-cyclohexadienes
    • Johnson, R.E.; Soria, A.E.; O'Connor, J.R.; Dobson, R.A. Synthesis and antibacterial activity of 1-(arylamino)-1H-pyrroles and 4-(1H-pyrrol-1-ylimino)- 2,5-cyclohexadienes. J. Med. Chem., 1981, 24, 1314-1319. (Pubitemid 12209062)
    • (1981) Journal of Medicinal Chemistry , vol.24 , Issue.11 , pp. 1314-1319
    • Johnson, R.E.1    Soria, A.E.2    O'Connor, J.R.3    Dobson, R.A.4
  • 336
    • 0000245437 scopus 로고
    • Synthesis of methyl/ethyl 4-substituted-benzoylthiazole-2-carbamates as potential chemotherapeutic agents
    • Manian, A.K.; Khadse, B.G.; Sengupta, S.R. Synthesis of methyl/ethyl 4-substituted-benzoylthiazole-2-carbamates as potential chemotherapeutic agents. Ind. J. Chem.; 1993, 32B, 407-409.
    • (1993) Ind. J. Chem. , vol.32 B , pp. 407-409
    • Manian, A.K.1    Khadse, B.G.2    Sengupta, S.R.3
  • 337
    • 0002561888 scopus 로고
    • Synthesis and antimicrobial activity of some dithiocarbamates, 2-arylimino-4-oxothiazolidines and their 5-arylidene derivatives
    • Desai, N.C. Synthesis and antimicrobial activity of some dithiocarbamates, 2-arylimino-4-oxothiazolidines and their 5-arylidene derivatives. Ind. J. Chem., 1993, 32, 343-346.
    • (1993) Ind. J. Chem. , vol.32 , pp. 343-346
    • Desai, N.C.1
  • 338
    • 0345228677 scopus 로고
    • Synthesis of N-aryl/substituted-methyl/heteroaryl pyrrolidino/ piperidinosuccinimides as antituberculosis agents
    • Rangnekar, V.M.; Lokhande, S.R.; Bhamaria, R.P.; Khadse, B.G. Synthesis of N-aryl/substituted-methyl/heteroaryl pyrrolidino/piperidinosuccinimides as antituberculosis agents. Ind. J. Chem., 1983, 22B, 1070-1071.
    • (1983) Ind. J. Chem. , vol.22 B , pp. 1070-1071
    • Rangnekar, V.M.1    Lokhande, S.R.2    Bhamaria, R.P.3    Khadse, B.G.4
  • 339
    • 0022380271 scopus 로고
    • Studies on synthesis and antitubercular activity of some (+) -α-aceto-N,N-diarylsuccinamide
    • Dave, M.P.; Patel, J.M.; Langalia, N.A.; Shah, S.R.; Thaker, K.A. Studies on the synthesis and antitubercular activity of some aceto-N,N'- diarylsuccinamide. J. Ind. Chem. Soc., 1985, 62(5), 386-387. (Pubitemid 16170736)
    • (1985) Journal of the Indian Chemical Society , vol.62 , Issue.5 , pp. 386-387
    • Dave, M.P.1    Patel, J.M.2    Langalia, N.A.3
  • 340
    • 0022357254 scopus 로고
    • Synthesis and antibacterial activity of 2,2'-dithiobis(benzamide) derivatives against Mycobacterium species
    • DOI 10.1021/jm00150a006
    • Okachi, R.; Nijno, H.; Kitaura, K.; Mineura, K.; Nakamizo, Y.; Murayama, Y.; Ono, T.; Nakamizo, A. Synthesis and antibacterial activity of 2,2'-dithiobis(benzamide) derivatives against Mycobacterium species. J. Med. Chem., 1985, 28, 1772-1779. (Pubitemid 16176830)
    • (1985) Journal of Medicinal Chemistry , vol.28 , Issue.12 , pp. 1772-1779
    • Okachi, R.1    Niino, H.2    Kitaura, K.3
  • 341
    • 0037294865 scopus 로고    scopus 로고
    • Synthesis and investigation of tuberculosis inhibition activities of some 1,2,3-triazole derivatives
    • DOI 10.1016/S0223-5234(02)01445-9
    • Dabak K, Sezer O, Akar A, Anac O. Synthesis and investigation of tuberculosis inhibition activities of some 1,2,3-triazole derivatives. Eur. J. Med. Chem., 2003, 38, 215-218. (Pubitemid 36288475)
    • (2003) European Journal of Medicinal Chemistry , vol.38 , Issue.2 , pp. 215-218
    • Dabak, K.1    Sezer, O.2    Akar, A.3    Anac, O.4
  • 342
    • 0032885734 scopus 로고    scopus 로고
    • Synthesis and biological activity of 2-azetidinones, sulphonamides, arylamides and thiourea derivatives
    • Patel, P.; Korgaokar, S.; Parikh, K.; Parekh, H. Synthesis and biological activity of 2-azetidinones, sulphonamides, arylamides and thiourea derivatives. Ind. J. Chem., 1999, 38B, 696-700.
    • (1999) Ind. J. Chem. , vol.38 B , pp. 696-700
    • Patel, P.1    Korgaokar, S.2    Parikh, K.3    Parekh, H.4
  • 345
    • 0343478173 scopus 로고    scopus 로고
    • Synthesis of 2-benzylthiopyridine-4-carbothioamide derivatives and their antimycobacterial, antifungal and photosynthesis-inhibiting activity
    • Klimesova, V.; Svoboda, M.; Waisser, K.; Kaustova, J.; Buchta, V.; Kralova, K. Synthesis of 2-benzylthiopyridine-4-carbothioamide derivatives and their antimycobacterial, antifungal and photosynthesis-inhibiting activity. Eur. J. Med. Chem., 1999, 34, 433-440.
    • (1999) Eur. J. Med. Chem. , vol.34 , pp. 433-440
    • Klimesova, V.1    Svoboda, M.2    Waisser, K.3    Kaustova, J.4    Buchta, V.5    Kralova, K.6
  • 347
    • 0034862337 scopus 로고    scopus 로고
    • Novel triheterocyclic systems by Mannich reaction on 3- arylsydnones: Synthesis of 3-aryl-4-[2'(8'-hydroxy-7'-quinolinyl-methylamino)- thiazol-4'-yl]sydnones and 3-aryl-4-[2'-(3'-acetyl-2'-hydroxybenzylamino)- thiazol-4'-yl] sydnones as possible antimicrobial agents
    • Mallur, S.G.; Badami, B.V. Novel triheterocyclic systems by Mannich reaction on 3-arylsydnones: Synthesis of 3-aryl-4-[2'-(8"-hydroxy-7"- quinolinylmethylamino)-thiazol-4'-yl]sydnones and 3-aryl-4-[2'-(3"-acetyl- 2"-hydroxybenzylamino)-thiazol-4'-yl]sydnones as possible antimicrobial agents. Ind. J. Chem.; 2001, 40B, 742-747. (Pubitemid 32808165)
    • (2001) Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry , vol.40 , Issue.8 , pp. 742-747
    • Mallur, S.G.1    Badami, B.V.2
  • 348
    • 0032265027 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of certain pyrazoline derivatives of 2-[6-methoxy naphthyl]-propionic acid (naproxen)
    • Udupi, R.H.; Kushnoor, A.S.; Bhat, A.R. Synthesis and biological evaluation of certain pyrazoline derivatives of naproxen. Ind. J. Het. Chem., 1998, 8, 63-66. (Pubitemid 128540664)
    • (1998) Indian Journal of Heterocyclic Chemistry , vol.8 , Issue.1 , pp. 63-66
    • Udupi, R.H.1    Kushnoor, A.S.2    Bhat, A.R.3
  • 349
    • 0042244475 scopus 로고    scopus 로고
    • Synthesis, anticancer, antitubercular and amtimicrobial activity of some new pyrimidine derivatives
    • Nimavat, K.S.; Popat, K.H.; Joshi, H.S. Synthesis, anticancer, antitubercular and amtimicrobial activity of some new pyrimidine derivatives. Ind. J. Het. Chem., 2003, 12, 225-228.
    • (2003) Ind. J. Het. Chem. , vol.12 , pp. 225-228
    • Nimavat, K.S.1    Popat, K.H.2    Joshi, H.S.3
  • 351
    • 0037052030 scopus 로고    scopus 로고
    • Antimycobacterial activity of 5-arylidene aromatic derivatives of hydantoin
    • DOI 10.1016/S0014-827X(01)01194-6, PII S0014827X01011946
    • Szymanska, E.; Kiec-Kononowicz, K. Antimycobacterial activity of 5-arylidene derivatives of hydantoin. Farmaco, 2002, 57, 355-362. (Pubitemid 34460500)
    • (2002) Farmaco , vol.57 , Issue.5 , pp. 355-362
    • Szymanska, E.1    Kiec-Kononowicz, K.2
  • 353
    • 72049094262 scopus 로고    scopus 로고
    • A highly atom economic, chemo-, regio-and stereoselective synthesis and evaluation of spiro-pyrrolothiazoles as antitubercular agents
    • Karthikeyan, S.V.; Bala, B.D.; Raja, V.P.A.; Perumal, S.; Yogeeswari, P.; Sriram, D. A highly atom economic, chemo-, regio-and stereoselective synthesis and evaluation of spiro-pyrrolothiazoles as antitubercular agents. Bioorg. Med. Chem. Lett., 2010, 20(1), 350-353.
    • (2010) Bioorg. Med. Chem. Lett. , vol.20 , Issue.1 , pp. 350-353
    • Karthikeyan, S.V.1    Bala, B.D.2    Raja, V.P.A.3    Perumal, S.4    Yogeeswari, P.5    Sriram, D.6
  • 354
    • 77955556522 scopus 로고    scopus 로고
    • Design synthesis, and antitubercular evaluation of novel series of 3-benzofuran-5-aryl-1-pyrazolyl-pyridylmethanone and 3-benzofuran-5-aryl-1- pyrazolylcarbonyl-4-oxo-naphthyridin analogs
    • Manna, K.; Agrawal, Y.K. Design, synthesis, and antitubercular evaluation of novel series of 3-benzofuran-5-aryl-1-pyrazolyl-pyridylmethanone and 3-benzofuran-5-aryl-1-pyrazolylcarbonyl-4-oxo-naphthyridin analogs. Eur. J. Med. Chem., 2010, 45, 3831-3839.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 3831-3839
    • Manna, K.1    Agrawal, Y.K.2
  • 356
    • 79958817048 scopus 로고    scopus 로고
    • Synthesis of some N-(4-oxo-2-substituted-phenylquinazolin-3-(4H)-yl)-2- [(5-aryl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamides as antitub -ercular agents
    • Rao, G.K.; Rajasekaran, S.; Pai, P.N.S. Synthesis of some N-(4-oxo-2-substituted-phenylquinazolin-3-(4H)-yl)-2-[(5-aryl-1,3, 4-oxadiazol-2-yl)sulfanyl]acetamides as antitub -ercular agents. Ind. J. Het. Chem., 2010, 19(3), 293-294.
    • (2010) Ind. J. Het. Chem. , vol.19 , Issue.3 , pp. 293-294
    • Rao, G.K.1    Rajasekaran, S.2    Pai, P.N.S.3
  • 358
    • 77349123954 scopus 로고    scopus 로고
    • Synthesis and anti-tuberculosis activity of new hetero(Mn, Co, Ni)trinuclear iron(III) furoates
    • Melnic, S.; Prodius, D.; Stoeckli-Evans, H.; Shova, S.; Turta, C. Synthesis and anti-tuberculosis activity of new hetero(Mn, Co, Ni)trinuclear iron(III) furoates. Eur. J. Med. Chem., 2010, 45(4), 1465-1469.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.4 , pp. 1465-1469
    • Melnic, S.1    Prodius, D.2    Stoeckli-Evans, H.3    Shova, S.4    Turta, C.5
  • 359
    • 75849153770 scopus 로고    scopus 로고
    • Pharmacophoric model building for antitubercular activity of the individual Schiff bases of small combinatorial library
    • Abdel-Aal, W.S.; Hassan, H.Y.; Aboul-Fadl, T.; Youssef, A.F. Pharmacophoric model building for antitubercular activity of the individual Schiff bases of small combinatorial library. Eur. J. Med. Chem., 2010, 45(3), 1098-1106.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.3 , pp. 1098-1106
    • Abdel-Aal, W.S.1    Hassan, H.Y.2    Aboul-Fadl, T.3    Youssef, A.F.4
  • 363
    • 72049097924 scopus 로고    scopus 로고
    • Novel three-component domino reactions of ketones, isatin and amino acids: Synthesis and discovery of antimycobacterial activity of highly functionalised novel dispiropyrrolidines
    • Kumar, R.S.; Rajesh, S.M.; Perumal, S.; Banerjee, D.; Yogeeswari, P.; Sriram, D. Novel three-component domino reactions of ketones, isatin and amino acids: Synthesis and discovery of antimycobacterial activity of highly functionalised novel dispiropyrrolidines. Eur. J. Med. Chem., 2010, 45(1), 411-422.
    • (2010) Eur. J. Med. Chem. , vol.45 , Issue.1 , pp. 411-422
    • Kumar, R.S.1    Rajesh, S.M.2    Perumal, S.3    Banerjee, D.4    Yogeeswari, P.5    Sriram, D.6
  • 367
    • 33646112903 scopus 로고    scopus 로고
    • Antibacterial drug discovery and structure-based design
    • and references cited therein
    • Barker, J.J. Antibacterial drug discovery and structure-based design. Drug Discov. Today, 2006, 11, 391-404 and references cited therein.
    • (2006) Drug Discov. Today , vol.11 , pp. 391-404
    • Barker, J.J.1
  • 368
    • 4644371689 scopus 로고    scopus 로고
    • Structural bioinformatic approaches to the discovery of new antimycobacterial drugs
    • Kantardjieff, K.; Rupp, B. Structural Bioinformatic Approaches to the Discovery of New Antimycobacterial Drugs. Current Pharma. Des., 2004, 10, 1-17.
    • (2004) Current Pharma. Des. , vol.10 , pp. 1-17
    • Kantardjieff, K.1    Rupp, B.2
  • 369
    • 0242330263 scopus 로고    scopus 로고
    • Structure-based design of hepatitis C virus inhibitors
    • DOI 10.1046/j.1365-2893.2003.00443.x
    • Smith, R.M.; Wu, G.Y. Structure-based design of hepatitis C virus inhibitors. J. Viral Hepat., 2003, 10, 405-412. (Pubitemid 37352580)
    • (2003) Journal of Viral Hepatitis , vol.10 , Issue.6 , pp. 405-412
    • Smith, R.M.1    Wu, G.Y.2
  • 370
    • 0038606190 scopus 로고    scopus 로고
    • Structure-based design of AIDS drugs and the development of resistance
    • Wlodawer, A. Structure-based design of AIDS drugs and the development of resistance. Vox Sang., 2002, 83, 23-26.
    • (2002) Vox Sang. , vol.83 , pp. 23-26
    • Wlodawer, A.1
  • 371
    • 0034567210 scopus 로고    scopus 로고
    • Comparative protein structure modeling. Introduction and practical examples with modeller Methods
    • Sanchez, R.; Sali, A. Comparative protein structure modeling. Introduction and practical examples with modeller Methods. Mol Biol., 2000, 143, 97-129.
    • (2000) Mol Biol. , vol.143 , pp. 97-129
    • Sanchez, R.1    Sali, A.2
  • 373
    • 0035342428 scopus 로고    scopus 로고
    • Ligand-protein inverse docking and its use in the computer search of protein targets of a small molecule
    • Chen, Y.Z.; Zhi, D.G. Ligand-protein inverse docking and its use in the computer search of protein targets of a small molecule. Proteins, 2001, 43, 217-226.
    • (2001) Proteins , vol.43 , pp. 217-226
    • Chen, Y.Z.1    Zhi, D.G.2
  • 374
    • 17344380633 scopus 로고    scopus 로고
    • ICM-DISCO docking by global energy optimization with fully flexible side-chains
    • DOI 10.1002/prot.10383
    • Fernandez-Recio, J.; Totrov, M.; Abagyan, R. ICM-DISCO docking by global energy optimizaton with fully flexible side-chains. Proteins, 2003, 52, 113-117. (Pubitemid 36648859)
    • (2003) Proteins: Structure, Function and Genetics , vol.52 , Issue.1 , pp. 113-117
    • Fernandez-Recio, J.1    Totrov, M.2    Abagyan, R.3
  • 376
    • 12344293492 scopus 로고    scopus 로고
    • Identification of 4-substituted 1,2,3-triazoles as novel oxazolidinone antibacterial agents with reduced activity against monoamine oxidase A
    • DOI 10.1021/jm0400810
    • Reck, F.; Zhou, F.; Girardot, M.; Kern, G.; Eyermann, C.J.; Hales, N.J.; Ramsay, R.R.; Gravestock, M.B. Identification of 4-substituted 1,2,3-triazoles as novel oxazolidinone antibacterial agents with reduced activity against monoamine oxidase A. J. Med. Chem., 2005, 48, 499-506. (Pubitemid 40139792)
    • (2005) Journal of Medicinal Chemistry , vol.48 , Issue.2 , pp. 499-506
    • Reck, F.1    Zhou, F.2    Girardot, M.3    Kern, G.4    Eyermann, C.J.5    Hales, N.J.6    Ramsay, R.R.7    Gravestock, M.B.8
  • 377
  • 379
    • 85047175465 scopus 로고    scopus 로고
    • FAD-independent and herbicide-resistant mutants of tobacco acetohydroxy acid synthase
    • Le, D.T.; Choi, J.D. FAD-independent and Herbicide-resistant Mutants of Tobacco Acetohydroxy Acid Synthase. Bull. Korean Chem. Soc., 2005, 26, 1-6.
    • (2005) Bull. Korean Chem. Soc. , vol.26 , pp. 1-6
    • Le, D.T.1    Choi, J.D.2
  • 381
    • 0043123259 scopus 로고    scopus 로고
    • Acetohydroxyacid synthase from Mycobacterium avium and its inhibition by sulfonylureas and imidazolinones
    • Zohar, Y.; Einav, M.; Chipman, D.M.; Barak, Z. Acetohydroxyacid synthase from Mycobacterium avium and its inhibition by sulfonylureas and imidazolinones. Biochim. Biophys. Acta., 2003, 1649, 97.
    • (2003) Biochim. Biophys. Acta. , vol.1649 , pp. 97
    • Zohar, Y.1    Einav, M.2    Chipman, D.M.3    Barak, Z.4
  • 382
    • 34250816250 scopus 로고    scopus 로고
    • Virtual screening of tubercular acetohydroxy acid synthase inhibitors through analysis of structural models
    • Le, D.T.; Lee, H.S.; Chung, Y.J.; Yoon, M.Y.; Choi, J.D. Virtual Screening of Tubercular Acetohydroxy Acid Synthase Inhibitors through Analysis of Structural Models. Bull. Korean Chem. Soc., 2007, 28, 947-952.
    • (2007) Bull. Korean Chem. Soc. , vol.28 , pp. 947-952
    • Le, D.T.1    Lee, H.S.2    Chung, Y.J.3    Yoon, M.Y.4    Choi, J.D.5
  • 383
    • 24044541011 scopus 로고    scopus 로고
    • Quinolone alkaloids from Evodia rutaecarpa: A potent new group of antimycobacterial compounds [2]
    • DOI 10.1016/j.ijantimicag.2005.06.003, PII S0924857905001664
    • Adams, M.; Wube, A.A.; Bucar, F.; Bauer, R.; Kunert, O.; Haslinger, E. Quinoline alkaloids from Evodia rutaecarpa: Apotent new group of antimycobacterial compounds. Int. J. Antimicrob. Agents, 2005, 26, 262-264. (Pubitemid 41219616)
    • (2005) International Journal of Antimicrobial Agents , vol.26 , Issue.3 , pp. 262-264
    • Adams, M.1    Wube, A.A.2    Bucar, F.3    Bauer, R.4    Kunert, O.5    Haslinger, E.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.