Synthesis and investigation of tuberculosis inhibition activities of some 1,2,3-triazole derivatives

European Journal of Medicinal Chemistry

Volumn 38, Issue 2, 2003, Pages 215-218

  Dabak, Kadir ^a   Sezer, Özkan ^a   Akar, Ahmet ^a   Anaç, Olcay ^a  

^a ISTANBUL TECHNICAL UNIVERSITY   (Turkey)

Author keywords

1,2,3 Triazoles; Tuberculosis inhibition

Indexed keywords

1,2,3 TRIAZOLE DERIVATIVE; 4 (2 FURANCARBONYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (2 FURANCARBONYL) 1 PHENYL 1H 1,2,3 TRIAZOLE; 4 (2 METHYLPROPANOYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (2 METHYLPROPANOYL) 1 (NAPHTH 1 YL) 1H 1,2,3 TRIAZOLE; 4 (2 NAPHTHOYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (2 NAPHTHOYL) 1 (NAPHTH 1 YL) 1H 1,2,3 TRIAZOLE; 4 (2 THIOPHENECARBONYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (2 THIOPHENECARBONYL) 1 (BROMOETHYL) 1H 1,2,3 TRIAZOLE; 4 (2 THIOPHENECARBONYL) 1 (NAPHTH 1 YL) 1H 1,2,3 TRIAZOLE; 4 (2',4' DICHLOROBENZOYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (2',4' DICHLOROBENZOYL) 1 (NAPHTH 1 YL) 1H 1,2,3 TRIAZOLE; 4 (2,5 DIMETHYL 3 FURANCARBONYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (2,5 DIMETHYL 3 FURANCARBONYL) 1 PHENYL 1H 1,2,3 TRIAZOLE; 4 (4' BROMOBENZOYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (4' BROMOBENZOYL) 1 PHENYL 1H 1,2,3 TRIAZOLE; 4 (4' METHOXYBENZOYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (BENZOYL) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (BENZOYL) 1 (NAPHTH 1 YL) 1H 1,2,3 TRIAZOLE; 4 (ETHYLCARBOXYLATE) 1 (4 CHLOROPHENYL) 1H 1,2,3 TRIAZOLE; 4 (ETHYLCARBOXYLATE) 1 PHENYL 1H 1,2,3 TRIAZOLE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG RESEARCH; DRUG SCREENING; DRUG SYNTHESIS; INFECTION PREVENTION; TUBERCULOSIS; TUBERCULOSIS CONTROL;

EID: 0037294865     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(02)01445-9     Document Type: Article

References (11)

1. Clarke D., Mares R.W., McNab H. J. Chem. Soc. Chem. Commun. 1993;1026.
2. Sezer Ö., Dabak K., Anaç O., Akar A. Helv. Chim. Acta. 79:1996;449.
3. Gilchrist T.L., Geymer G.E. Katritzky A.R., Boulton A.J. Advances in Heterocyclic Chemistry. 16:1974;33 Academic Press, New York.
4. Stojanovic F.M., Arnold Z. Collect. Czech. Chem. Commun. 32:1967;2155.
5. Sezer Ö., Dabak K., Anaç O., Akar A. Helv. Chim. Acta. 80:1997;960.
6. Collins L., Franzblau S.G. Antimicrob. Agents Chemother. 40:1997;2809.
7. Dabak K., Akar A. Heterocycl. Commun. 8:(1):2002;61-64.
8. Biagi G., Giorgi I., Livi O., Lucacchini A., Martini C., Scartoni V. J. Pharm. Sci. 82:(9):1993;893.
9. L'abbe G., Verbeke M., Dehaen W., Toppet S. J. Chem. Soc. Perkin Trans. 1. 15:1993;1719.
10. Abu-Orabi T., Sultan M.A., Athaf I., Jibril F.M., Mari'i A., Ali A.L.-S. J. Heterocycl. Chem. 26:(5):1989;1461.
11. L'abbe G., Bruynseels M., Delbeke P., Toppet S. J. Heterocycl. Chem. 27:(7):1990;2021.