Synthesis and preliminary evaluation of some pyrazine containing thiazolines and thiazolidinones as antimicrobial agents

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 9, 2004, Pages 2151-2161

  Bonde, Chandrakant G ^a   Gaikwad, Naresh J ^a  

^a RTM NAGPUR UNIVERSITY   (India)

Author keywords

Antimicrobial; Hemolytic assay; Thiazolidinones; Thiazoline

Indexed keywords

ANTIINFECTIVE AGENT; ANTIMYCOBACTERIAL AGENT; N' [3 (4 BROMOPHENYL) 4 OXO 1,3 THIAZOLIDINYLIDENE] 2 (PYRAZIN 2 YLOXY)ACETOHYDRAZIDE; PYRAZINE DERIVATIVE; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; BACILLUS SUBTILIS; BACTERIAL STRAIN; CONCENTRATION RESPONSE; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; HEMOLYSIS; IN VITRO STUDY; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; SALMONELLA TYPHI; STANDARDIZATION; STAPHYLOCOCCUS AUREUS; TOXICITY;

ANTI-BACTERIAL AGENTS; DRUG EVALUATION, PRECLINICAL; HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; MICROBIAL SENSITIVITY TESTS; PYRAZINES; SPECIES SPECIFICITY; THIAZOLES;

MYCOBACTERIUM; MYCOBACTERIUM TUBERCULOSIS; NEGIBACTERIA; POSIBACTERIA;

EID: 1842630349     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.02.024     Document Type: Article

References (25)

1. Rouhi A.M. Chem. Eng. News. 17:1999;52.
2. Clarck C., Jacobs M., Appelbaum P. J. Clin. Microbiol. 36:1998;3579.
3. Davidson P.T., Le H.Q. Drugs. 43:1992;651.
4. Vincent T.A. Int. J. Antimicrob. Agents. 16:2000;317.
5. Tan Y.T., Tillett D.J., Mckay I.A. Mol. Med. Today. 6:2000;309.
6. MacManus M.C. Am. J. Health-Syst. Pharm. 54:1997;1420.
7. Heinemann J.A. Drug Discov. Today. 4:1999;72.
8. Chopra I., Hodgson J., Metcalf B., Poste G. Antimicrob. Agents Chemother. 41:1997;497.
9. Sander P., Bottger E.C. Chemotherapy. 45:1999;95.
10. Chan W.C., Li R.C., Ling J.M. J. Antimicrob. Chemother. 43:1999;55.
11. Bush K. Curr. Opin. Chem. Biol. 1:1997;169.
12. Stapleton P., Shannon K., Phillips I. J. Antimicrob. Chemother. 36:1995;483.
13. Chopra I.J. Antimicrob. Chemother. 30:1992;737.
14. Coleman K., Athalye M., Clancey A., Davison M., Payne D.J., Perry C.R., Chopra I.J. Antimicrob. Chemother. 33:1994;1091.
15. Sykes R.B., Bonner D.P. Br. Med. Bull. 40:1984;96.
16. Bonde C.G., Nadkarni B.A., Khadse B.G. Indian J. Heter. Chem. 10:2001;271.
17. Sihgh S.P., Parmar S.S., Raman K., Stenherb V.I. Chem. Pharm. Bull. 81:1981;197.
18. Patel P.B., Trivedi J.T. Ind. Chem. Soc. 54:1987;765.
19. Vittoria D.M., Mazzoni O., Piscopo E., Caligmano A., Bolognese A. J. Med. Chem. 35:1992;2910.
20. Omar A.M., Eshba N.H. J. Pharm. Sci. 73:1984;1166.
21. Chaudhary M., Parmar S.S., Chaudhari S.K., Ramasastry B.V. J. Pharm. Sci. 65:1976;443.
22. Ragab F.A., Hussain m.M., Hanna M.m., Hassan G.S. J. Pharm. Sci. 34:1993;387.
23. Hassan I.Y., Koussi A.A., Farghaly Z.S. Chem. Pharm. Bull. 46(5):1998;863.
24. Sahm D.F., Washington J.A., Ballows A., Housler W.J., Herrmann K.L., Isenberg H.D., Shadomy H.J. A Manual of Clinical Microbiology. fifth ed. 1991;1105 ASM, Washington, DC.
25. Kikuchi K.E., Bernard M., Sadownik A., Regen S.L., Armstrong D. Antimicrob. Agents Chemother. 41:1997;1433.