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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 9, 2011, Pages 2606-2610

Potent antiprotozoal activity of a novel semi-synthetic berberine derivative

(12) Bahar, Mark a Deng, Ye a Zhu, Xiaohua a He, Shanshan a Pandharkar, Trupti a Drew, Mark E a,b Navarro Vázquez, Armando c Anklin, Clemens e Gil, Roberto R d Doskotch, Raymond W a Werbovetz, Karl A a Kinghorn, A Douglas a

a OHIO STATE UNIVERSITY (United States)

b THE OHIO STATE UNIVERSITY COLLEGE OF MEDICINE (United States)

c UNIVERSITY OF VIGO (Spain)

d CARNEGIE MELLON UNIVERSITY (United States)

e BRUKER BIOSPIN CORPORATION (United States)

Author keywords

5,6 Didehydro 8,8 diethyl 13 oxodihydroberberine chloride; African trypanosomiasis; Berberine; Inhibitory activity; Leishmaniasis; Malaria

Indexed keywords

5,6 DIDEHYDRO 8,8 DIETHYL 13 OXODIHYDROBERBERINE CHLORIDE; AMPHOTERICIN B; BERBERINE DERIVATIVE; MILTEFOSINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIPROTOZOAL ACTIVITY; CONFERENCE PAPER; CONTROLLED STUDY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; MALARIA; MOUSE; NONHUMAN; TRYPANOSOMIASIS; VERO CELL; VISCERAL LEISHMANIASIS;

ANIMALS; ANTIPROTOZOAL AGENTS; BERBERINE; CERCOPITHECUS AETHIOPS; DISEASE MODELS, ANIMAL; INHIBITORY CONCENTRATION 50; LEISHMANIA; LEISHMANIASIS; MALARIA; MICE; MODELS, MOLECULAR; PARASITES; PLASMODIUM FALCIPARUM; PROTOZOAN INFECTIONS; TRYPANOSOMA BRUCEI BRUCEI; TRYPANOSOMIASIS; VERO CELLS;

EID: 79955460123 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2011.01.101 Document Type: Conference Paper

Times cited : (48)

References (40)

1
- 65349181925
- P.J. Hotez , A. Fenwick , L. Savioli , and D.H. Molyneux Lancet 373 2009 1570
- (2009) Lancet , vol.373 , pp. 1570
- Hotez, P.J.¹ Fenwick, A.² Savioli, L.³ Molyneux, D.H.⁴

2
- 72949115014
- B. Liese , M. Rosenberg , and A. Schratz Lancet 375 2010 67
- (2010) Lancet , vol.375 , pp. 67
- Liese, B.¹ Rosenberg, M.² Schratz, A.³

3
- 74049146746
- L. Conteh , T. Engels , and D.H. Molyneux Lancet 375 2010 239
- (2010) Lancet , vol.375 , pp. 239
- Conteh, L.¹ Engels, T.² Molyneux, D.H.³

4
- 0037157590
- P. Trouiller , P. Olliaro , E. Torreele , J. Orbinski , R. Laing , and N. Ford Lancet 359 2002 2188
- (2002) Lancet , vol.359 , pp. 2188
- Trouiller, P.¹ Olliaro, P.² Torreele, E.³ Orbinski, J.⁴ Laing, R.⁵ Ford, N.⁶

5
- 0037183163
- G. Yamey , and E. Torreele Br. Med. J. 325 2002 176
- (2002) Br. Med. J. , vol.325 , pp. 176
- Yamey, G.¹ Torreele, E.²

6
- 79955372969
- World Health Organization Geneva
- E. Toreele , M. Usdin , and P.A. Chirac Needs-based Pharmaceutical R&D Agenda for Neglected Diseases 2004 World Health Organization Geneva
- (2004) Needs-based Pharmaceutical R&D Agenda for Neglected Diseases
- Toreele, E.¹ Usdin, M.² Chirac, P.A.³

7
- 84934441783
- P. Hotez , E. Ottesen , A. Fenwick , and D. Molyneux Adv. Exp. Med. Biol. 582 2006 23
- (2006) Adv. Exp. Med. Biol. , vol.582 , pp. 23
- Hotez, P.¹ Ottesen, E.² Fenwick, A.³ Molyneux, D.⁴

8
- 34548422845
- P.J. Hotez , D.H. Molyneux , A. Fenwick , J. Kumaresan , S.E. Sachs , J.D. Sachs , and L. Savioli N. Eng. J. Med. 357 2007 1018
- (2007) N. Eng. J. Med. , vol.357 , pp. 1018
- Hotez, P.J.¹ Molyneux, D.H.² Fenwick, A.³ Kumaresan, J.⁴ Sachs, S.E.⁵ Sachs, J.D.⁶ Savioli, L.⁷

9
- 79955424508
- Neglected Tropical Diseases (accessed Aug 2010)
- Neglected Tropical Diseases. http://whqlibdoc.who.int/publications/ (accessed Aug 2010).

10
- 0003438149
- 2nd ed. John Wiley and Sons Ltd Chichester, UK
- P.M. Dewick Medicinal Natural Products: A Biosynthetic Approach 2nd ed. 2002 John Wiley and Sons Ltd Chichester, UK
- (2002) Medicinal Natural Products: A Biosynthetic Approach
- Dewick, P.M.¹

11
- 70349665346
- R. Sinha , and G.S. Kumar J. Phys. Chem. B 113 2009 13410
- (2009) J. Phys. Chem. B , vol.113 , pp. 13410
- Sinha, R.¹ Kumar, G.S.²

12
- 71749102883
- Y.X. Wang , Y.P. Wang , H. Zhang , W.J. Kong , Y.H. Li , F. Liu , R.M. Gao , T. Liu , J.D. Jiang , and D.Q. Song Bioorg. Med. Chem. Lett. 19 2009 6004
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 6004
- Wang, Y.X.¹ Wang, Y.P.² Zhang, H.³ Kong, W.J.⁴ Li, Y.H.⁵ Liu, F.⁶ Gao, R.M.⁷ Liu, T.⁸ Jiang, J.D.⁹ Song, D.Q.¹⁰

13
- 74049139484
- H. Zhang , J. Wei , R. Xue , J.D. Wu , W. Zhao , Z.Z. Wang , S.K. Wang , Z.X. Zhou , D.Q. Song , Y.M. Wang , H.N. Pan , W.J. Kong , and J.D. Jiang Metabolism 59 2010 285
- (2010) Metabolism , vol.59 , pp. 285
- Zhang, H.¹ Wei, J.² Xue, R.³ Wu, J.D.⁴ Zhao, W.⁵ Wang, Z.Z.⁶ Wang, S.K.⁷ Zhou, Z.X.⁸ Song, D.Q.⁹ Wang, Y.M.¹⁰ Pan, H.N.¹¹ Kong, W.J.¹² Jiang, J.D.¹³

14
- 76949094803
- M.Y. Qi , Y. Feng , D.Z. Dai , N. Li , Y.S. Cheng , and Y. Dai Acta Pharmacol. Sin. 31 2010 165
- (2010) Acta Pharmacol. Sin. , vol.31 , pp. 165
- Qi, M.Y.¹ Feng, Y.² Dai, D.Z.³ Li, N.⁴ Cheng, Y.S.⁵ Dai, Y.⁶

15
- 77649186191
- R.S. Iwazaki , E.H. Endo , T. Ueda-Nakamura , C.V. Nakamura , L.B. Garcia , and B.P. Filho Antonie van Leeuwenhoek 97 2010 201
- (2010) Antonie Van Leeuwenhoek , vol.97 , pp. 201
- Iwazaki, R.S.¹ Endo, E.H.² Ueda-Nakamura, T.³ Nakamura, C.V.⁴ Garcia, L.B.⁵ Filho, B.P.⁶

16
- 0022369270
- A.K. Ghosh , F.K. Bhattacharyya , and D.K. Ghosh Exp. Parasitol. 60 1985 404
- (1985) Exp. Parasitol. , vol.60 , pp. 404
- Ghosh, A.K.¹ Bhattacharyya, F.K.² Ghosh, D.K.³

17
- 0023888151
- J.L. Vennerstrom , and D.L. Klayman J. Med. Chem. 31 1988 1084
- (1988) J. Med. Chem. , vol.31 , pp. 1084
- Vennerstrom, J.L.¹ Klayman, D.L.²

18
- 0025320783
- J.L. Vennerstrom , J.K. Lovelace , V.B. Waits , W.L. Hanson , and D.L. Klayman Antimicrob. Agents Chemother. 34 1990 918
- (1990) Antimicrob. Agents Chemother. , vol.34 , pp. 918
- Vennerstrom, J.L.¹ Lovelace, J.K.² Waits, V.B.³ Hanson, W.L.⁴ Klayman, D.L.⁵

19
- 0036082293
- B. Nyasse , E. Nkwengoua , B. Sondengam , C. Denier , and M. Willson Pharmazie 57 2002 358
- (2002) Pharmazie , vol.57 , pp. 358
- Nyasse, B.¹ Nkwengoua, E.² Sondengam, B.³ Denier, C.⁴ Willson, M.⁵

20
- 55249117688
- V. Rosenkranz , and M. Wink Molecules 13 2008 2462
- (2008) Molecules , vol.13 , pp. 2462
- Rosenkranz, V.¹ Wink, M.²

21
- 70350525419
- P. Saha , R. Sen , C. Hariharan , D. Kumar , P. Das , and M. Chatterjee Free Radical Res. 43 2009 1101
- (2009) Free Radical Res. , vol.43 , pp. 1101
- Saha, P.¹ Sen, R.² Hariharan, C.³ Kumar, D.⁴ Das, P.⁵ Chatterjee, M.⁶

22
- 70349511962
- E.T. Nkwengoua , I. Ngantchou , B. Nyasse , C. Denier , C. Blonski , and B. Schneider Nat. Prod. Res. 23 2009 1144
- (2009) Nat. Prod. Res. , vol.23 , pp. 1144
- Nkwengoua, E.T.¹ Ngantchou, I.² Nyasse, B.³ Denier, C.⁴ Blonski, C.⁵ Schneider, B.⁶

23
- 0018356232
- J.L. Moniot , T.M. Kravetz , A.H. Abd el Rahman , and M. Shamma J. Pharm. Sci. 68 1979 705
- (1979) J. Pharm. Sci. , vol.68 , pp. 705
- Moniot, J.L.¹ Kravetz, T.M.² Abd El Rahman, A.H.³ Shamma, M.⁴

24
- 79955429783
- +, 374.1004)
- +, 374.1004)

25
- 79955431323
- +, 370.0846)
- +, 370.0846)

26
- 79955442646
- note
- 5, 406.1654)

27
- 18144404174
- W.-D.Z. Li , and H. Yang Tetrahedron 61 2005 5037
- (2005) Tetrahedron , vol.61 , pp. 5037
- Li, W.-D.Z.¹ Yang, H.²

28
- 0031661329
- K. Iwasa , D.-U. Lee , S.-I. Kang , and W. Wiegrebe J. Nat. Prod. 61 1998 1150
- (1998) J. Nat. Prod. , vol.61 , pp. 1150
- Iwasa, K.¹ Lee, D.-U.² Kang, S.-I.³ Wiegrebe, W.⁴

29
- 77955465923
- Z. Cheng , A.-F. Chen , F. Wu , L. Sheng , H.-K. Zhang , M. Gu , Y.-Y. Li , L.-N. Zhang , L.-H. Hu , J.-Y. Li , and J. Li Bioorg. Med. Chem. 18 2010 5915
- (2010) Bioorg. Med. Chem. , vol.18 , pp. 5915
- Cheng, Z.¹ Chen, A.-F.² Wu, F.³ Sheng, L.⁴ Zhang, H.-K.⁵ Gu, M.⁶ Li, Y.-Y.⁷ Zhang, L.-N.⁸ Hu, L.-H.⁹ Li, J.-Y.¹⁰ Li, J.¹¹

30
- 33847086721
- A. Bax , R. Freeman , and S.P. Kempsell J. Am. Chem. Soc. 102 1980 4849
- (1980) J. Am. Chem. Soc. , vol.102 , pp. 4849
- Bax, A.¹ Freeman, R.² Kempsell, S.P.³

31
- 43049141516
- Y. Zhao , and D.G. Truhlar Theor. Chem. Acc. 120 2008 215
- (2008) Theor. Chem. Acc. , vol.120 , pp. 215
- Zhao, Y.¹ Truhlar, D.G.²

32
- 84961980477
- J. Tomasi , B. Mennucci , and R. Cammi Chem. Rev. 105 2005 2999
- (2005) Chem. Rev. , vol.105 , pp. 2999
- Tomasi, J.¹ Mennucci, B.² Cammi, R.³

33
- 77952819729
- Rev. A.02 Gaussian, Wallingford, CT
- gaussian09, Rev. A.02: Frisch, M. J. et al. Gaussian, Wallingford, CT, 2004.
- (2004) Gaussian09
- Frisch, M.J.¹

34
- 49349113509
- F. Jensen J. Chem. Theor. Comput. 4 2008 719
- (2008) J. Chem. Theor. Comput. , vol.4 , pp. 719
- Jensen, F.¹

35
- 49349095278
- Y. Zhao , and D.G. Truhlar J. Phys. Chem. A 112 2008 6794
- (2008) J. Phys. Chem. A , vol.112 , pp. 6794
- Zhao, Y.¹ Truhlar, D.G.²

36
- 35148813913
- G. Bifulco , P. Dambruoso , L. Gómez-Paloma , and R. Riccio Chem. Rev. 107 2007 3744
- (2007) Chem. Rev. , vol.107 , pp. 3744
- Bifulco, G.¹ Dambruoso, P.² Gómez-Paloma, L.³ Riccio, R.⁴

37
- 58549093170
- D. Delfín , R. Morgan , X. Zhu , and K. Werbovetz Bioorg. Med. Chem. 17 2009 820
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 820
- Delfín, D.¹ Morgan, R.² Zhu, X.³ Werbovetz, K.⁴

38
- 0346996811
- K. Werbovetz , D. Sackett , D. Delfin , G. Bhattacharya , M. Salem , T. Obrzut , D. Rattendi , and C. Bacchi Mol. Pharmacol. 64 2003 1325
- (2003) Mol. Pharmacol. , vol.64 , pp. 1325
- Werbovetz, K.¹ Sackett, D.² Delfin, D.³ Bhattacharya, G.⁴ Salem, M.⁵ Obrzut, T.⁶ Rattendi, D.⁷ Bacchi, C.⁸

39
- 12544251879
- J. Liu , I.Y. Gluzman , M.E. Drew , and D.E. Goldberg J. Biol. Chem. 280 2005 1432
- (2005) J. Biol. Chem. , vol.280 , pp. 1432
- Liu, J.¹ Gluzman, I.Y.² Drew, M.E.³ Goldberg, D.E.⁴

40
- 12944293007
- M. Salem , and K. Werbovetz J. Nat. Prod. 68 2005 108
- (2005) J. Nat. Prod. , vol.68 , pp. 108
- Salem, M.¹ Werbovetz, K.²

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