Evolution, structure, and activation mechanism of family 3/C G-protein-coupled receptors

Pharmacology and Therapeutics

Volumn 98, Issue 3, 2003, Pages 325-354

  Pin, Jean Philippe ^a   Galvez, Thierry ^a,b   Prézeau, Laurent ^a  

^a CCIPE   (France)

^b STANFORD UNIVERSITY MEDICAL CENTER   (United States)

Author keywords

Dimerization; G protein coupled receptors; GABAB receptors; Metabotropic glutamate receptors; Pheromones; Taste

Indexed keywords

1 AMINOCYCLOPENTANE 1,3,4 TRICARBOXYLATE; 2 AMINO 2 (2 CARBOXYCYCLOPROPYL) 3 (XANTHEN 9 YL)PROPIONIC ACID; 2 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID B RECEPTOR BLOCKING AGENT; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; 6A NAPHTHALEN 2 YLMETHYL 5 METHYLIDENEHEXAHYDROCYCLOPENTA[C]FURAN 1 ONE; 7 HYDROXYIMINOCYCLOPROPAN[B]CHROMEN 1A CARBOXYLIC ACID ETHYL ESTER; ALPHA METHYLAMINOPHOSPHONOBUTYRATE; AMINO ACID RECEPTOR; BACLOFEN; CALCIUM ION; CALCIUM SENSING RECEPTOR; CALMODULIN; CYSTEINE; DIMER; G PROTEIN COUPLED RECEPTOR; G PROTEIN COUPLED RECEPTOR AGONIST; GLUTAMIC ACID; HOMER PROTEIN; HORMONE RECEPTOR; METABOTROPIC RECEPTOR AGONIST; METABOTROPIC RECEPTOR ANTAGONIST; N ACETYLASPARTYLGLUTAMIC ACID; PHEROMONE; PHOSPHOSERINE; PROTEIN; RECEPTOR SUBTYPE; RHODOPSIN; TRANSCRIPTION FACTOR; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ALLOSTERISM; AMINO ACID SUBSTITUTION; ANXIETY DISORDER; BINDING AFFINITY; BINDING SITE; CARBOXY TERMINAL SEQUENCE; CYTOPLASM; DRUG DEPENDENCE; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; HUMAN; LIGAND BINDING; NONHUMAN; NUCLEOTIDE SEQUENCE; ODOR; PHARMACOPHORE; PHYLOGENY; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN FAMILY; PROTEIN FUNCTION; PROTEIN INTERACTION; PROTEIN STRUCTURE; PROTEIN TARGETING; RECEPTOR BINDING; REGULATORY MECHANISM; REVIEW; SCHIZOPHRENIA; SEQUENCE HOMOLOGY; SWEETNESS; TASTE; TASTE BUD;

EID: 0038662595     PISSN: 01637258     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0163-7258(03)00038-X     Document Type: Review

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