Ca2+ requirement for high-affinity γ-aminobutyric acid (GABA) binding at GABA(B) receptors: Involvement of serine 269 of the GABA(B)R1 subunit

Molecular Pharmacology

Volumn 57, Issue 3, 2000, Pages 419-426

  Galvez, Thierry ^a,c   Urwyler, Stephan ^b   Prézeau, Laurent ^a   Mosbacher, Johannes ^b   Joly, Cécile ^a   Malitschek, Barbara ^b   Heid, Jakob ^b   Brabet, Isabelle ^a   Froestl, Wolfgang ^b   Bettler, Bernhard ^b   Kaupmann, Klemens ^b   Pin, Jean Philippe ^a  

^a INSERM   (France)

^b NOVARTIS PHARMA AG   (Switzerland)

^c CNRS   (France)

Author keywords

[No Author keywords available]

Indexed keywords

3 AMINOPROPANEPHOSPHONIC ACID; 4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; BACLOFEN; CALCIUM ION; CALCIUM SENSING RECEPTOR; CGP 56999A; CGP 64213; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); IODINE 125; METABOTROPIC RECEPTOR; RECEPTOR SUBUNIT; SERINE; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ANIMAL TISSUE; ARTICLE; BRAIN MEMBRANE; CAENORHABDITIS ELEGANS; CONCENTRATION RESPONSE; CONTROLLED STUDY; DISSOCIATION; DRUG RECEPTOR BINDING; NONHUMAN; POINT MUTATION; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; SEQUENCE HOMOLOGY;

EID: 18144452059     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.57.3.419     Document Type: Article

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