Positive allosteric modulators for γ-aminobutyric acidB receptors open new routes for the development of drugs targeting family 3 G-protein-coupled receptors

Molecular Pharmacology

Volumn 60, Issue 5, 2001, Pages 881-884

  Pin, Jean Philippe ^a,b   Parmentier, Marie Laure ^a   Prézeau, Laurent ^a  

^a CNRS   (France)

^b INSERM   (France)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID B RECEPTOR STIMULATING AGENT; ADENYLATE CYCLASE; BACLOFEN; BENZODIAZEPINE DERIVATIVE; CALCIUM CHANNEL; CALCIUM SENSING RECEPTOR; CGP 13501; CGP 7930; CHLORIDE CHANNEL; G PROTEIN COUPLED RECEPTOR; METABOTROPIC RECEPTOR; POTASSIUM CHANNEL; RHODOPSIN; UNCLASSIFIED DRUG;

ALLOSTERISM; DRUG BINDING SITE; EPILEPSY; HUMAN; KNOCKOUT MOUSE; MULTIPLE SCLEROSIS; NERVE CELL EXCITABILITY; NEUROTRANSMITTER RELEASE; PRIORITY JOURNAL; PROTEIN TARGETING; RECEPTOR DOWN REGULATION; REVIEW;

EID: 0034757740     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.60.5.881     Document Type: Review

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