Structural insights into G-protein-coupled receptor allostery

Nature

Volumn 559, Issue 7712, 2018, Pages 45-53

  Thal, David M ^a   Glukhova, Alisa ^a   Sexton, Patrick M ^a   Christopoulos, Arthur ^a  

^a MONASH UNIVERSITY   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

G PROTEIN COUPLED RECEPTOR;

BIOCHEMICAL COMPOSITION; BIOCHEMISTRY; DRUG; ENVIRONMENTAL CUE; MEMBRANE; MOLECULAR ANALYSIS; PROTEIN;

ALLOSTERISM; AMINO TERMINAL SEQUENCE; CYTOSOL; DIMERIZATION; LIGAND BINDING; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN DOMAIN; PROTEIN INTERACTION; PROTEIN QUATERNARY STRUCTURE; PROTEIN STABILITY; PROTEIN STRUCTURE; REVIEW; SIGNAL TRANSDUCTION; STRUCTURE ACTIVITY RELATION; AGONISTS; ANIMAL; BINDING SITE; CHEMISTRY; CLASSIFICATION; DRUG EFFECT; HUMAN; METABOLISM; MOLECULAR MODEL; PROTEIN MULTIMERIZATION;

ALLOSTERIC REGULATION; ANIMALS; BINDING SITES; CYTOSOL; HUMANS; MODELS, MOLECULAR; PROTEIN CONFORMATION; PROTEIN MULTIMERIZATION; RECEPTORS, G-PROTEIN-COUPLED;

EID: 85049650721     PISSN: 00280836     EISSN: 14764687     Source Type: Journal    
DOI: 10.1038/s41586-018-0259-z     Document Type: Review

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