Crystal structures of a stabilized β1-adrenoceptor bound to the biased agonists bucindolol and carvedilol

Structure

Volumn 20, Issue 5, 2012, Pages 841-849

  Warne, Tony ^a   Edwards, Patricia C ^a   Leslie, Andrew G W ^a   Tate, Christopher G ^a  

^a MRC LABORATORY OF MOLECULAR BIOLOGY   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ADRENALIN; BETA 1 ADRENERGIC RECEPTOR; BISOPROLOL; BUCINDOLOL; CARAZOLOL; CARMOTEROL; CARVEDILOL; CYANOPINDOLOL; DOBUTAMINE; FORMOTEROL; GUANINE NUCLEOTIDE BINDING PROTEIN; METOPROLOL;

ARTICLE; CRYSTAL STRUCTURE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; EXTRACELLULAR SPACE; PRIORITY JOURNAL; PROTEIN POLYMORPHISM; SIGNAL TRANSDUCTION; THERMOSTABILITY;

ADRENERGIC BETA-ANTAGONISTS; ANIMALS; CARBAZOLES; CRYSTALLOGRAPHY, X-RAY; HUMANS; MODELS, MOLECULAR; PROPANOLAMINES; RECEPTORS, ADRENERGIC, BETA-1; TURKEYS;

AVES;

EID: 84861064804     PISSN: 09692126     EISSN: 18784186     Source Type: Journal    
DOI: 10.1016/j.str.2012.03.014     Document Type: Article

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