Antimalarial drug discovery: Recent progress and future directions

Progress in Medicinal Chemistry

Volumn 52, Issue , 2013, Pages 97-151

  Calderón, Félix ^a   Wilson, David M ^a   Gamo, Francisco Javier ^a  

^a GLAXOSMITHKLINE   (Spain)

Author keywords

Antimalarial; Drug discovery; Malaria; Mode of action; Plasmodium; Resistance; Whole cell screening

Indexed keywords

3 (N ACETYL N HYDROXYAMINO)PROPYLPHOSPHONIC ACID; 4,6 DIAMINO 1,2 DIHYDRO 2,2 DIMETHYL 1 [3 (2,4,5 TRICHLOROPHENOXY)PROPOXY] 1,3,5 TRIAZINE; ANTIMALARIAL AGENT; ARTEMETHER; ARTEMETHER PLUS BENFLUMETOL; ARTEMISININ; ARTEROLANE; ATOVAQUONE; BENFLUMETOL; CHLOROQUINE; DECOQUINATE; FOSMIDOMYCIN; HALOFANTRINE; JPC 2056; MEFLOQUINE; N [3 (2,4,5 TRICHLOROPHENOXY)PROPOXY] N' ISOPROPYLIMIDOCARBONIMIDIC DIAMIDE; OZ 439; P 218; PHOSPHOTRANSFERASE INHIBITOR; PIPERAQUINE; PRIMAQUINE; PROGUANIL; PYRIMETHAMINE; PYRONARIDINE; SULFADOXINE; TEBUQUINE; UNCLASSIFIED DRUG;

ARTICLE; BIOSYNTHESIS; CELL SCREENING; CROSS RESISTANCE; ENZYME ACTIVITY; HUMAN; MALARIA; MALARIA FALCIPARUM; METABOLISM; NONHUMAN; PLASMODIUM; PRIORITY JOURNAL; SINGLE DRUG DOSE; X RAY CRYSTALLOGRAPHY;

EID: 84873398285     PISSN: 00796468     EISSN: 18757863     Source Type: Book Series    
DOI: 10.1016/B978-0-444-62652-3.00003-X     Document Type: Chapter

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