4-Aminoquinoline analogs of chloroquine with shortened side chains retain activity against chloroquine-resistant Plasmodium falciparum

Antimicrobial Agents and Chemotherapy

Volumn 40, Issue 8, 1996, Pages 1846-1854

  Ridley, Robert G ^a   Hofheinz, Werner ^a   Matile, Hugues ^a   Jaquet, Catherine ^a   Dorn, Arnulf ^a   Masciadri, Raffaello ^a   Jolidon, Synèse ^a   Richter, Wolfgang F ^b   Guenzi, Alberto ^b   Girometta, Maria Angela ^b   Urwyler, Heinrich ^b   Huber, Werner ^c   Thaithong, Sodsri ^d   Peters, Wallace ^e  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

^b F HOFFMANN LA ROCHE LTD   (Switzerland)

^c SWISS TROPICAL AND PUBLIC HEALTH INSTITUTE   (Switzerland)

^d CHULALONGKORN UNIVERSITY   (Thailand)

^e UNIVERSITY OF OXFORD   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOQUINOLINE DERIVATIVE; CHLOROQUINE; RO 413118; RO 470543; RO 479396; RO 480346; UNCLASSIFIED DRUG;

ANIMAL MODEL; ANTIMALARIAL ACTIVITY; AREA UNDER THE CURVE; ARTICLE; CONTROLLED STUDY; CROSS RESISTANCE; DOSE RESPONSE; DRUG RESISTANCE; INTRAVENOUS DRUG ADMINISTRATION; MALARIA FALCIPARUM; MALE; MOUSE; NONHUMAN; ORAL DRUG ADMINISTRATION; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; SUBCUTANEOUS DRUG ADMINISTRATION;

EID: 9444258557     PISSN: 00664804     EISSN: None     Source Type: Journal    
DOI: 10.1128/aac.40.8.1846     Document Type: Article

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