Palladium-catalysed reactions in solid phase organic synthesis

Tetrahedron

Volumn 59, Issue 7, 2003, Pages 885-939

  Bräse, Stefan ^a   Kirchhoff, Jan H ^b   Köbberling, Johannes ^c  

^a UNIVERSITY OF BONN   (Germany)

^b CLARIANT PRODUKTE DEUTSCHLAND GMBH   (Germany)

^c BAYER AG   (Germany)

Author keywords

Combinatorial chemistry; Cross coupling reactions; Heck reaction; Palladium; Solid support; Suzuki coupling

Indexed keywords

ALCOHOL DERIVATIVE; ALKYNE DERIVATIVE; ALLYL COMPOUND; AMINE; CARBONYL DERIVATIVE; ESTER DERIVATIVE; ETHER DERIVATIVE; HALIDE; PALLADIUM; PALLADIUM COMPLEX; POLYCYCLIC AROMATIC HYDROCARBON DERIVATIVE; SILICON DERIVATIVE; SULFONIC ACID DERIVATIVE; THIOL DERIVATIVE; ZINC DERIVATIVE;

ALKENYLATION; ARTICLE; ARYLATION; CARBOMETALLATION; CATALYSIS; CHEMICAL BOND; CHEMICAL REACTION; CROSS COUPLING REACTION; CYANATION; DEGRADATION; DEPROTECTION REACTION; DERIVATIZATION; HECK REACTION; HYDROGENATION; NEGISHI REACTION; ORGANIC CHEMISTRY; PRIORITY JOURNAL; SOLID; SONOGASHIRA REACTION; STILLE REACTION; SUZUKI REACTION; SYNTHESIS; WACKER REACTION;

LATEOLABRAX JAPONICUS;

EID: 0037429030     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4020(02)01425-4     Document Type: Review

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278. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
279. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
280. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
281. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
282. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation
283. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
284. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
285. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
286. Suzuki reactions: Gravel, M.; Thompson, K. A.; Zak, M.; Bérubé, C.; Hall, D. G. Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids, J. Org. Chem. 2002, 67, 3-15. Baudoin, O.; Cesario, M.; Guenard, D.; Gueritte, F. Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams, J. Org. Chem. 2002, 67, 1199-1207. Haag, R.; Sunder, A.; Hebel, A.; Roller, S. Dendritic Aliphatic Polyethers as High-Loading Soluble Supports for Carbonyl Compounds and Parallel Membrane Separation Techniques, J. Comb. Chem. 2002, 4, 112-119. Lutz, C.; Bleicher, K. H. Multipin solid-phase synthesis of biaryls via Suzuki cross coupling reaction of aryltriflates, Tetrahedron Lett. 2002, 43, 2211-2214. Spivey, A. C.; Turner, D. J.; Turner, M. L.; Yeates, S. A Novel "Double-Coupling" Strategy for Iterative Oligothiophene Synthesis Using Orthogonal Si/Ge Protection, Org. Lett. 2002, 4, 1899-1902. Phoon, C. W.; Sim, M. M. Solid-Phase Syntheses of 1,2,4-Trisubstituted Urazole and Thiourazole Derivatives, J. Comb. Chem. 2002, 4, 491-495. Kell, R. J.; Hodge, P.; Nisar, M.; Watson, D. Towards more Chemically Robust Polymer-supported Chiral Catalysts for the Reactions of Aldehydes with Dialkylzincs, Bioorg. Med. Chem. Lett. 2002, 12, 1803-1807. Briehn, C. A.; Bäuerle, P. Design and Synthesis of a 256-Membered π-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s, J. Comb. Chem 2002, 4, 457-469. Revell, J. D.; Ganesan, A. Ionic Liquid Acceleration of Solid-Phase Suzuki-Miyaura Cross-Coupling Reactions, Org. Lett. 2002, 4, 3071-3073. Lew, A.; Chamberlin, A. R. The Preparation of Phenyl-stilbene Derivatives using the Safety Catch Linker, Meth. Mol. Biol. 2002, 201, 93-109. Wu, T. Y. H.; Schultz, P. G. A Versatile Linkage Strategy for Solid-Phase Synthesis of N,N-Dimethyltryptamines and β-Carbolines, Org. Lett. 2002, 4, 4033-4036.
287. Hudson R.H.E., Li G., Tse J. The Use of Sonogashira Coupling for the Synthesis of Modified Uracil Peptide Nucleic Acid. Tetrahedron Lett. 43:2002;1381-1386. Sonogashira reaction.
288. Carbonylation reactions: Liao, Y.; Reitman, M.; Zhang, Y.; Fathi, R.; Yang, Z. Palladium(II)-Mediated Cascade Carbonylative Annulation of o-Alkynylphenols on Silyl Linker-Based Macrobeads: A Combinatorial Synthesis of a 2,3-Disubstituted Benzo[b]furan Library, Org. Lett. 2002, 4, 2607-2609. Allylic substitution and removal of allylic protecting groups: Royo, M.; Farrera-Sinfreu, J.; Sole, L.; Albericio, F. Four-dimensional Orthogonal Solid-phase Synthesis of new Scaffolds based on Cyclic Tetra-β-peptides, Tetrahedron Lett. 2002, 43, 2029-2032. Kan, T.; Kobayashi, H.; Fukuyama, T. Highly Versatile Synthesis of Polyamines by Ns-Strategy on a Novel Trityl Chloride Resin, Synlett 2002, 1338-1340. Farrera-Sinfreu, J.; Royo, M.; Albericio, F. Undesired Removal of the Fmoc Group by the free ε-Amino Function of a Lysine Residue, Tetrahedron Lett. 2002, 43, 7813-7815. Spinelli, N.; Meyer, A.; Hayakawa, Y.; Imbach, J.-L.; Vasseur, J.-J. Use of Allylic Protecting Groups for the Synthesis of Base-sensitive Prooligonucleotides, Eur. J. Org. Chem. 2002, 1, 49-56.
289. Carbonylation reactions: Liao, Y.; Reitman, M.; Zhang, Y.; Fathi, R.; Yang, Z. Palladium(II)-Mediated Cascade Carbonylative Annulation of o-Alkynylphenols on Silyl Linker-Based Macrobeads: A Combinatorial Synthesis of a 2,3-Disubstituted Benzo[b]furan Library, Org. Lett. 2002, 4, 2607-2609. Allylic substitution and removal of allylic protecting groups: Royo, M.; Farrera-Sinfreu, J.; Sole, L.; Albericio, F. Four-dimensional Orthogonal Solid-phase Synthesis of new Scaffolds based on Cyclic Tetra-β-peptides, Tetrahedron Lett. 2002, 43, 2029-2032. Kan, T.; Kobayashi, H.; Fukuyama, T. Highly Versatile Synthesis of Polyamines by Ns-Strategy on a Novel Trityl Chloride Resin, Synlett 2002, 1338-1340. Farrera-Sinfreu, J.; Royo, M.; Albericio, F. Undesired Removal of the Fmoc Group by the free ε-Amino Function of a Lysine Residue, Tetrahedron Lett. 2002, 43, 7813-7815. Spinelli, N.; Meyer, A.; Hayakawa, Y.; Imbach, J.-L.; Vasseur, J.-J. Use of Allylic Protecting Groups for the Synthesis of Base-sensitive Prooligonucleotides, Eur. J. Org. Chem. 2002, 1, 49-56.
290. Carbonylation reactions: Liao, Y.; Reitman, M.; Zhang, Y.; Fathi, R.; Yang, Z. Palladium(II)-Mediated Cascade Carbonylative Annulation of o-Alkynylphenols on Silyl Linker-Based Macrobeads: A Combinatorial Synthesis of a 2,3-Disubstituted Benzo[b]furan Library, Org. Lett. 2002, 4, 2607-2609. Allylic substitution and removal of allylic protecting groups: Royo, M.; Farrera-Sinfreu, J.; Sole, L.; Albericio, F. Four-dimensional Orthogonal Solid-phase Synthesis of new Scaffolds based on Cyclic Tetra-β-peptides, Tetrahedron Lett. 2002, 43, 2029-2032. Kan, T.; Kobayashi, H.; Fukuyama, T. Highly Versatile Synthesis of Polyamines by Ns-Strategy on a Novel Trityl Chloride Resin, Synlett 2002, 1338-1340. Farrera-Sinfreu, J.; Royo, M.; Albericio, F. Undesired Removal of the Fmoc Group by the free ε-Amino Function of a Lysine Residue, Tetrahedron Lett. 2002, 43, 7813-7815. Spinelli, N.; Meyer, A.; Hayakawa, Y.; Imbach, J.-L.; Vasseur, J.-J. Use of Allylic Protecting Groups for the Synthesis of Base-sensitive Prooligonucleotides, Eur. J. Org. Chem. 2002, 1, 49-56.
291. Carbonylation reactions: Liao, Y.; Reitman, M.; Zhang, Y.; Fathi, R.; Yang, Z. Palladium(II)-Mediated Cascade Carbonylative Annulation of o-Alkynylphenols on Silyl Linker-Based Macrobeads: A Combinatorial Synthesis of a 2,3-Disubstituted Benzo[b]furan Library, Org. Lett. 2002, 4, 2607-2609. Allylic substitution and removal of allylic protecting groups: Royo, M.; Farrera-Sinfreu, J.; Sole, L.; Albericio, F. Four-dimensional Orthogonal Solid-phase Synthesis of new Scaffolds based on Cyclic Tetra-β-peptides, Tetrahedron Lett. 2002, 43, 2029-2032. Kan, T.; Kobayashi, H.; Fukuyama, T. Highly Versatile Synthesis of Polyamines by Ns-Strategy on a Novel Trityl Chloride Resin, Synlett 2002, 1338-1340. Farrera-Sinfreu, J.; Royo, M.; Albericio, F. Undesired Removal of the Fmoc Group by the free ε-Amino Function of a Lysine Residue, Tetrahedron Lett. 2002, 43, 7813-7815. Spinelli, N.; Meyer, A.; Hayakawa, Y.; Imbach, J.-L.; Vasseur, J.-J. Use of Allylic Protecting Groups for the Synthesis of Base-sensitive Prooligonucleotides, Eur. J. Org. Chem. 2002, 1, 49-56.
292. Carbonylation reactions: Liao, Y.; Reitman, M.; Zhang, Y.; Fathi, R.; Yang, Z. Palladium(II)-Mediated Cascade Carbonylative Annulation of o-Alkynylphenols on Silyl Linker-Based Macrobeads: A Combinatorial Synthesis of a 2,3-Disubstituted Benzo[b]furan Library, Org. Lett. 2002, 4, 2607-2609. Allylic substitution and removal of allylic protecting groups: Royo, M.; Farrera-Sinfreu, J.; Sole, L.; Albericio, F. Four-dimensional Orthogonal Solid-phase Synthesis of new Scaffolds based on Cyclic Tetra-β-peptides, Tetrahedron Lett. 2002, 43, 2029-2032. Kan, T.; Kobayashi, H.; Fukuyama, T. Highly Versatile Synthesis of Polyamines by Ns-Strategy on a Novel Trityl Chloride Resin, Synlett 2002, 1338-1340. Farrera-Sinfreu, J.; Royo, M.; Albericio, F. Undesired Removal of the Fmoc Group by the free ε-Amino Function of a Lysine Residue, Tetrahedron Lett. 2002, 43, 7813-7815. Spinelli, N.; Meyer, A.; Hayakawa, Y.; Imbach, J.-L.; Vasseur, J.-J. Use of Allylic Protecting Groups for the Synthesis of Base-sensitive Prooligonucleotides, Eur. J. Org. Chem. 2002, 1, 49-56.