-
1
-
-
0003178552
-
-
For a review on linkers: (a) Morphy, J. R. Curr. Opin. Drug Discovery Dev. 1998, 1, 59. (b) Eggenweiler, H.-M. Drug Discovery Today 1998, 3, 552.
-
(1998)
Curr. Opin. Drug Discovery Dev.
, vol.1
, pp. 59
-
-
Morphy, J.R.1
-
2
-
-
0031792553
-
-
For a review on linkers: (a) Morphy, J. R. Curr. Opin. Drug Discovery Dev. 1998, 1, 59. (b) Eggenweiler, H.-M. Drug Discovery Today 1998, 3, 552.
-
(1998)
Drug Discovery Today
, vol.3
, pp. 552
-
-
Eggenweiler, H.-M.1
-
3
-
-
0020724415
-
-
(a) Prasad, V. V. K.; Warne, P. A.; Lieberman, S. J. Steroid Biochem. 1983, 18, 257.
-
(1983)
J. Steroid Biochem.
, vol.18
, pp. 257
-
-
Prasad, V.V.K.1
Warne, P.A.2
Lieberman, S.3
-
5
-
-
8744310757
-
-
(c) Hodge, P.; Kemp, J.; Khoshdel, E.; Perry, G. M. React. Polym. 1985, 299.
-
(1985)
React. Polym.
, pp. 299
-
-
Hodge, P.1
Kemp, J.2
Khoshdel, E.3
Perry, G.M.4
-
7
-
-
0024989259
-
-
(e) Blossey, E. C.; Cannon, R. G.; Ford, W. T.; Periyasamy, M.; Mohanraj, S. J. Org. Chem. 1990, 55, 4664.
-
(1990)
J. Org. Chem.
, vol.55
, pp. 4664
-
-
Blossey, E.C.1
Cannon, R.G.2
Ford, W.T.3
Periyasamy, M.4
Mohanraj, S.5
-
9
-
-
0028100318
-
-
(g) Boyce, R.; Li, G.; Nestler, H. P.; Suenaga, T.; Still, W. C. J. Am. Chem. Soc. 1994, 776, 7955.
-
(1994)
J. Am. Chem. Soc.
, vol.776
, pp. 7955
-
-
Boyce, R.1
Li, G.2
Nestler, H.P.3
Suenaga, T.4
Still, W.C.5
-
10
-
-
8744261958
-
-
(h) Lebl, M.; Krchnak, V.; Sepetov, N. F.; Seligman, B.; Strop, P.; Felder, S.; Lam, K. S. Peptide Sci. 1995.
-
(1995)
Peptide Sci.
-
-
Lebl, M.1
Krchnak, V.2
Sepetov, N.F.3
Seligman, B.4
Strop, P.5
Felder, S.6
Lam, K.S.7
-
11
-
-
0029925955
-
-
(i) Cheng, Y.; Suenaga, T.; Still, W. C. J. Am. Chem. Soc. 1996, 118, 1813.
-
(1996)
J. Am. Chem. Soc.
, vol.118
, pp. 1813
-
-
Cheng, Y.1
Suenaga, T.2
Still, W.C.3
-
12
-
-
0030445091
-
-
(j) Wess, G.; Bock, K.; Kleine, H.; Kurz, M.; Guba, W.; Hemmerle, H.; Lopez-Calle, E.; Baringhaus, K.-H.; Glombik, H.; Enhsen, A.; Kramer, W. Angew. Chem., Int. Ed. Engl. 1996, 35, 2222.
-
(1996)
Angew. Chem., Int. Ed. Engl.
, vol.35
, pp. 2222
-
-
Wess, G.1
Bock, K.2
Kleine, H.3
Kurz, M.4
Guba, W.5
Hemmerle, H.6
Lopez-Calle, E.7
Baringhaus, K.-H.8
Glombik, H.9
Enhsen, A.10
Kramer, W.11
-
15
-
-
0000905921
-
-
(a) Ramage, R.; Barron, C. A.; Bielecki, S.; Thomas, D. W. Tetrahedron Lett. 1987, 28, 4105.
-
(1987)
Tetrahedron Lett.
, vol.28
, pp. 4105
-
-
Ramage, R.1
Barron, C.A.2
Bielecki, S.3
Thomas, D.W.4
-
17
-
-
0032474703
-
-
(c) Reggelin, M.; Brenig, V.; Welcker, R. Tetrahedron Lett. 1998, 39, 4801. (molecular weight of 8) = 46.5 mg. After the reaction, 275.5 mg of resin was recovered. Therefore, 275.5 - 238.4 (theoretical starting weight) = 37.1 mg of 8 was coupled. The yield of the reaction is (37.1/46.5) × 100% = 80%. The loading of the resulting resin is (37.1/310)/0.2755 = 0.43 mmol/g.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 4801
-
-
Reggelin, M.1
Brenig, V.2
Welcker, R.3
-
21
-
-
0000725865
-
-
(d) Scott, W. J.; Crisp, G. T.; Stille, J. K. J. Am. Chem. Soc. 1984, 106, 4630.
-
(1984)
J. Am. Chem. Soc.
, vol.106
, pp. 4630
-
-
Scott, W.J.1
Crisp, G.T.2
Stille, J.K.3
-
22
-
-
0009394369
-
-
(e) Crisp, G. T.; Scott, W. J.; Stille, J. K. J. Am. Chem. Soc. 1984, 106, 7500.
-
(1984)
J. Am. Chem. Soc.
, vol.106
, pp. 7500
-
-
Crisp, G.T.1
Scott, W.J.2
Stille, J.K.3
-
23
-
-
0000202518
-
-
(f) Scott, W. J.; Peña, M. R.; Swärd, K.; Stoessel, S. J.; Stille, J. K. J. Org. Chem. 1985, 50, 2302.
-
(1985)
J. Org. Chem.
, vol.50
, pp. 2302
-
-
Scott, W.J.1
Peña, M.R.2
Swärd, K.3
Stoessel, S.J.4
Stille, J.K.5
-
25
-
-
0000807122
-
-
(a) Harnisch, W.; Morera, E.; Ortar, G. J. Org. Chem. 1985, 50, 1990.
-
(1985)
J. Org. Chem.
, vol.50
, pp. 1990
-
-
Harnisch, W.1
Morera, E.2
Ortar, G.3
-
27
-
-
0000978284
-
-
(c) Ciattini, P. R.; Morera, E.; Ortar, G. Synth. Commun. 1990, 20, 1293.
-
(1990)
Synth. Commun.
, vol.20
, pp. 1293
-
-
Ciattini, P.R.1
Morera, E.2
Ortar, G.3
-
28
-
-
0028594037
-
-
(d) Skoda-Földes, R.; Kollár, L.; Marinelli, F.; Arcadi, A. Steroids 1994, 59, 691.
-
(1994)
Steroids
, vol.59
, pp. 691
-
-
Skoda-Földes, R.1
Kollár, L.2
Marinelli, F.3
Arcadi, A.4
-
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note
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This chemistry has been used for the synthesis of several libraries, which for patenting reasons will be reported in due course.
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