Combinatorial synthesis and biological evaluation of library of small-molecule Ser/Thr-protein phosphatase inhibitors

Bioorganic and Medicinal Chemistry

Volumn 5, Issue 1, 1997, Pages 165-177

  Wipf, Peter ^a   Cunningham, April ^a   Rice, Robert L ^b   Lazo, John S ^b  

^a UNIVERSITY OF PITTSBURGH   (United States)

^b UNIVERSITY OF PITTSBURGH SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; PHOSPHOPROTEIN PHOSPHATASE; PHOSPHOPROTEIN PHOSPHATASE INHIBITOR;

ANTINEOPLASTIC ACTIVITY; BREAST CANCER; CELL CYCLE; CELL CYCLE G1 PHASE; CONFERENCE PAPER; CONTROLLED STUDY; DRUG DESIGN; ENZYME INHIBITION; FLOW CYTOMETRY; HUMAN; HUMAN CELL; IN VITRO STUDY; PEPTIDE SYNTHESIS; PROTEIN PROCESSING; QUANTITATIVE STRUCTURE ACTIVITY RELATION; SIGNAL TRANSDUCTION;

BREAST NEOPLASMS; CELL CYCLE; CELL DIVISION; DRUG DESIGN; ENZYME INHIBITORS; HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; OXAZOLES; PHOSPHOPROTEIN PHOSPHATASE; SERINE; THREONINE; TUMOR CELLS, CULTURED;

EID: 0031030829     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(96)00199-X     Document Type: Conference Paper

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