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For 2-Cl-trityl resin attachment to the imidazole of histidine, see: Cody, D. M. R.; DeWitt, S. H.; Hodges, J. C.; Kiely, J. S.; Moos, W. M.; Pavia, M. R.; Roth, B. D.; Schroeder, M. C.; Stankovic, C. J.; U.S. Patent, 5,324,483(1994).
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For biological results on a broader sampling of analogues, including urethanes, see Hoekstra, W. J.; Maryanoff, B. E.; Andrade-Gordon, P.; Cohen, J. H.; Costanzo, M. J.; Damiano, B. P.; Haertlein, B. J.; Harris, B. D.; Kauffman, J. A.; Keane, P. M.; McComsey, D. F.; Villani, F. J.; Yabut, S. C. Bioorg. Med. Chem. Lett. 1996, 6, 2371.
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0342600237
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note
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1H NMR. Representative examples also gave satisfactory combustion analysis.
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16
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0030062528
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For a synthesis of Leu-Trp thiazoles cyclized from Leu-β-keto-Trp ester precursors, see von Geldern, T. W.; Hutchins, C.; Kester, J. A.; Wu-Wong, J. R.; Chiou, W.; Dixon, D. B.; Opgenorth, T. J. J. Med. Chem. 1996, 39, 957.
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