Allosteric ligands and their binding sites define γ-aminobutyric acid (gaba) type a receptor subtypes

Advances in Pharmacology

Volumn 73, Issue , 2015, Pages 167-202

  Olsen, Richard W ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

Anxiolytics; Chloride channels; Convulsants; Ethanol; GABA receptors; General anesthetics; Ligand gated ion channels; Positive allosteric modulators

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; ALCOHOL; ANESTHETIC AGENT; BENZODIAZEPINE; PICROTOXIN; PICROTOXININ; 4 AMINOBUTYRIC ACID A RECEPTOR STIMULATING AGENT; LIGAND;

AFFINITY LABELING; ALLOSTERISM; ANXIETY; ARTICLE; BINDING AFFINITY; BINDING SITE; CENTRAL NERVOUS SYSTEM; CRYSTAL STRUCTURE; EPILEPSY; HUMAN; LIGAND BINDING; MEMORY DISORDER; MUTAGENESIS; NEUROCHEMISTRY; NONHUMAN; PHOTOAFFINITY LABELING; PRIORITY JOURNAL; RECEPTOR BINDING; SLEEP DISORDER; SUBSTANCE ABUSE; ANIMAL; BRAIN; DRUG EFFECTS; METABOLISM;

ALLOSTERIC REGULATION; ALLOSTERIC SITE; ANIMALS; BINDING SITES; BRAIN; GABA-A RECEPTOR AGONISTS; HUMANS; LIGANDS; RECEPTORS, GABA-A;

EID: 84921653616     PISSN: 10543589     EISSN: 15578925     Source Type: Book Series    
DOI: 10.1016/bs.apha.2014.11.005     Document Type: Chapter

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