-
1
-
-
84986959314
-
A bioautographic agar overlay method for the detection of antifungal compounds from higher plants
-
Rahalison, L.; Hamburger, M.; Monod, M.; Frenk, E.; Hostettman, K. A bioautographic agar overlay method for the detection of antifungal compounds from higher plants. Phytochem. Anal., 1991, 2, 199-203.
-
(1991)
Phytochem. Anal
, vol.2
, pp. 199-203
-
-
Rahalison, L.1
Hamburger, M.2
Monod, M.3
Frenk, E.4
Hostettman, K.5
-
2
-
-
0026090223
-
Plants used in Guatemala for the treatment of dermatomucosal infections. 1: Screening of 38 plant extracts for anticandidal activity
-
Caceres, A.; Lopez, B.R.; Giron, M.A.; Logemann, H. Plants used in Guatemala for the treatment of dermatomucosal infections. 1: Screening of 38 plant extracts for anticandidal activity. J. Ethnopharmacol., 1991, 31, 263-276.
-
(1991)
J. Ethnopharmacol
, vol.31
, pp. 263-276
-
-
Caceres, A.1
Lopez, B.R.2
Giron, M.A.3
Logemann, H.4
-
3
-
-
0022133070
-
Cryptococcosis in the acquired immunodeficiency syndrome
-
Kovacs, J.A.; Kovacs, A.A.; Polis, M.; Wright, W.C.; Gill, V.J.; Tuazon, C.U.; Gelmann, E.P.; Lane, H.C.; Longfield, R.; Overturf, G.; Macher, A.M.; Fauci, A.S.; Parillo, J.E.; Bennett, J.E.; Masur, H. Cryptococcosis in the acquired immunodeficiency syndrome. Ann. Int. Med., 1985, 103, 533-538.
-
(1985)
Ann. Int. Med
, vol.103
, pp. 533-538
-
-
Kovacs, J.A.1
Kovacs, A.A.2
Polis, M.3
Wright, W.C.4
Gill, V.J.5
Tuazon, C.U.6
Gelmann, E.P.7
Lane, H.C.8
Longfield, R.9
Overturf, G.10
Macher, A.M.11
Fauci, A.S.12
Parillo, J.E.13
Bennett, J.E.14
Masur, H.15
-
4
-
-
73549103962
-
Evaluation of SAR for Amphotericin B Derivatives by Artificial Neural Network
-
Sardari, S.; Dezfulian, M. Evaluation of SAR for Amphotericin B Derivatives by Artificial Neural Network. Trop. J. Pharm. Res., 2005, 4, 517-521.
-
(2005)
Trop. J. Pharm. Res
, vol.4
, pp. 517-521
-
-
Sardari, S.1
Dezfulian, M.2
-
5
-
-
0027483015
-
Fungicidal properties of defensin NP-1 and activity against Cryptococcus neoformans in vitro
-
Alcouloumre, M.S.; Ghannoum, M.A.; Ibrahim, A.S.; Selsted, M.E.; Edwards, J.E. Fungicidal properties of defensin NP-1 and activity against Cryptococcus neoformans in vitro. Antimicrob. Agents Chemother., 1993, 37, 2628-2632.
-
(1993)
Antimicrob. Agents Chemother
, vol.37
, pp. 2628-2632
-
-
Alcouloumre, M.S.1
Ghannoum, M.A.2
Ibrahim, A.S.3
Selsted, M.E.4
Edwards, J.E.5
-
6
-
-
1642545489
-
Anti-microbial peptides: From invertebrates to vertebrates
-
Bulet, P.; Stocklin, R.; Menin, L. Anti-microbial peptides: from invertebrates to vertebrates. Immunol. Rev., 2004, 198, 169-184.
-
(2004)
Immunol. Rev
, vol.198
, pp. 169-184
-
-
Bulet, P.1
Stocklin, R.2
Menin, L.3
-
7
-
-
0019386682
-
Sequence and specificity of two antibacterial proteins involved in insect immunity
-
Steiner, H.; Hultmark, D.; Engstrom, A.; Bennich, H.; Boman, H.G. Sequence and specificity of two antibacterial proteins involved in insect immunity. Nature, 1981, 292, 246-248.
-
(1981)
Nature
, vol.292
, pp. 246-248
-
-
Steiner, H.1
Hultmark, D.2
Engstrom, A.3
Bennich, H.4
Boman, H.G.5
-
8
-
-
0022402545
-
-
Ganz, T.; Selsted, M.E.; Szklarek, D.; Harwig, S.S.; Daher, K.; Bainton, D.F.; Lehrer, R.I. Defensins. Natural peptide antibiotics of human neuitrophils. J. Clin. Invest., 1985, 76, 1427-1435.
-
Ganz, T.; Selsted, M.E.; Szklarek, D.; Harwig, S.S.; Daher, K.; Bainton, D.F.; Lehrer, R.I. Defensins. Natural peptide antibiotics of human neuitrophils. J. Clin. Invest., 1985, 76, 1427-1435.
-
-
-
-
9
-
-
0036252092
-
Cationic peptides: Distribution and mechanisms of resistance
-
Devine, D.A.; Hancock, R.E.W. Cationic peptides: distribution and mechanisms of resistance. Curr. Pharm. Des., 2002, 8, 703-714.
-
(2002)
Curr. Pharm. Des
, vol.8
, pp. 703-714
-
-
Devine, D.A.1
Hancock, R.E.W.2
-
10
-
-
0042381670
-
Novel properties of antimicrobial peptides
-
Kamysz, W.; Okruj, M.; Lukasiak, J. Novel properties of antimicrobial peptides. Acta. Biochim., 2003, 50, 461-469.
-
(2003)
Acta. Biochim
, vol.50
, pp. 461-469
-
-
Kamysz, W.1
Okruj, M.2
Lukasiak, J.3
-
11
-
-
0030967077
-
Signaling in plant-microbe interactions
-
Baker, B., Zambryski, P.; Staskawicz, B.; Dinesh-Kumar, S.P. Signaling in plant-microbe interactions. Science, 1997, 276, 726-33.
-
(1997)
Science
, vol.276
, pp. 726-733
-
-
Baker, B.1
Zambryski, P.2
Staskawicz, B.3
Dinesh-Kumar, S.P.4
-
12
-
-
0033763238
-
Transgenic plants expressing cationic peptide chimeras exhibit broad-spectrum resistance to phytopathogens
-
Osusky, M.; Zhou, G; Osuska, L.; Hancock, R.E.; Kay, W.W.; Misra, S. Transgenic plants expressing cationic peptide chimeras exhibit broad-spectrum resistance to phytopathogens. Nat. Biotechnol., 2000, 18, 1162-1166.
-
(2000)
Nat. Biotechnol
, vol.18
, pp. 1162-1166
-
-
Osusky, M.1
Zhou, G.2
Osuska, L.3
Hancock, R.E.4
Kay, W.W.5
Misra, S.6
-
13
-
-
0036158878
-
Peptides as drugs: Is there a market?
-
Loffet, A. Peptides as drugs: is there a market?. J. Pept. Sci., 2002, 8, 1-7.
-
(2002)
J. Pept. Sci
, vol.8
, pp. 1-7
-
-
Loffet, A.1
-
14
-
-
0034098916
-
Bactericidal activity of mammalian cathelicidin-derived peptides
-
Travis, S.M.; Anderson, N.N.; Forsyth, W.R. Bactericidal activity of mammalian cathelicidin-derived peptides. Infect. Immun., 2000, 68, 2748-55.
-
(2000)
Infect. Immun
, vol.68
, pp. 2748-2755
-
-
Travis, S.M.1
Anderson, N.N.2
Forsyth, W.R.3
-
15
-
-
0028289032
-
Characterization of a rabbit cationic protein (CAP18) with lipopolysaccharide-inhibitory activity
-
Hirata, M.; Shimomura, Y.; Yoshida, M. Characterization of a rabbit cationic protein (CAP18) with lipopolysaccharide-inhibitory activity. Infect. Immun., 1994, 62, 1421-6.
-
(1994)
Infect. Immun
, vol.62
, pp. 1421-1426
-
-
Hirata, M.1
Shimomura, Y.2
Yoshida, M.3
-
16
-
-
0028844134
-
-
Zanetti, M.; Gennaro, R.; Romeo, D. Cathelicidins: A novel protein family with a common proregion and a variable C-terminal antimicrobial domain. FEBS Lett., 1995, 374, 1-5.
-
Zanetti, M.; Gennaro, R.; Romeo, D. Cathelicidins: A novel protein family with a common proregion and a variable C-terminal antimicrobial domain. FEBS Lett., 1995, 374, 1-5.
-
-
-
-
17
-
-
0031729624
-
Evaluation of antimicrobial and lipopolysaccharide-neutralizing effects of a synthetic CAP18 fragment against Pseudomonas aeruginosa in a mouse model
-
Sawa, T.; Kurahashi. K.; Ohara, M. Evaluation of antimicrobial and lipopolysaccharide-neutralizing effects of a synthetic CAP18 fragment against Pseudomonas aeruginosa in a mouse model. Antimicrob. Agents Chemother., 1998, 42, 3269-75.
-
(1998)
Antimicrob. Agents Chemother
, vol.42
, pp. 3269-3275
-
-
Sawa, T.1
Kurahashi, K.2
Ohara, M.3
-
19
-
-
0037371597
-
Mechanisms of antimicrobial peptide action and resistance
-
Yeaman, R.M.; Yount Y.N. Mechanisms of antimicrobial peptide action and resistance. Pharmacol. Rev., 2003, 55, 27-55.
-
(2003)
Pharmacol. Rev
, vol.55
, pp. 27-55
-
-
Yeaman, R.M.1
Yount, Y.N.2
-
20
-
-
0034824597
-
From "carpet" mechanism to de novo designed diastereomeric cell-selective antimicrobial peptides
-
Shai, Y.; Oren, Z. From "carpet" mechanism to de novo designed diastereomeric cell-selective antimicrobial peptides. Peptides, 2001, 22, 1629 -1641.
-
(2001)
Peptides
, vol.22
, pp. 1629-1641
-
-
Shai, Y.1
Oren, Z.2
-
21
-
-
0037371597
-
Mechanisms of antimicrobial peptide action and resistance
-
Yeaman, M.R.; Yount, N.Y. Mechanisms of antimicrobial peptide action and resistance. Pharmacol. Rev., 2003, 55, 27-55.
-
(2003)
Pharmacol. Rev
, vol.55
, pp. 27-55
-
-
Yeaman, M.R.1
Yount, N.Y.2
-
22
-
-
1242306544
-
Antimicrobial peptides from ranid frogs: Taxonomic and phylogenetic markers and a potential source of new therapeutic agents
-
Conlon, J.M.; Kolodziejek, J.; Nowotny, N. Antimicrobial peptides from ranid frogs: taxonomic and phylogenetic markers and a potential source of new therapeutic agents. Biochim. Biophys. Acta., 2004, 1696, 1-14.
-
(2004)
Biochim. Biophys. Acta
, vol.1696
, pp. 1-14
-
-
Conlon, J.M.1
Kolodziejek, J.2
Nowotny, N.3
-
23
-
-
0033569408
-
Beta-defensins: Linking innate and adaptive immunity through dendritic and T cell CCR6
-
Yang, D.; Chertov, O.; Bykovskaia, S. N.; Chen, Q.; Buffo, M. J.; Shogan, J.; Anderson, M.; Schroder, J. M.; Wang, J. M.; Howard, O. M. Z.; Oppenheim, J. J. Beta-defensins: linking innate and adaptive immunity through dendritic and T cell CCR6. Science., 1999, 286, 525-528.
-
(1999)
Science
, vol.286
, pp. 525-528
-
-
Yang, D.1
Chertov, O.2
Bykovskaia, S.N.3
Chen, Q.4
Buffo, M.J.5
Shogan, J.6
Anderson, M.7
Schroder, J.M.8
Wang, J.M.9
Howard, O.M.Z.10
Oppenheim, J.J.11
-
24
-
-
0025372569
-
All-D amino acid-containing channel-forming antibiotic peptides
-
Wade, D.; Boman, A.; Wåhlin, B.; Drain, C. M.; Andreu, D.; Boman, H. G.; Merrifield, R. B. All-D amino acid-containing channel-forming antibiotic peptides. Proc. Natl. Acad. Sci. U.S.A., 1990, 87, 4761-4765.
-
(1990)
Proc. Natl. Acad. Sci. U.S.A
, vol.87
, pp. 4761-4765
-
-
Wade, D.1
Boman, A.2
Wåhlin, B.3
Drain, C.M.4
Andreu, D.5
Boman, H.G.6
Merrifield, R.B.7
-
25
-
-
0030738014
-
Interactions of an antimicrobial peptide, magainin 2, with outer and inner membranes of Gram-negative bacteria
-
Matsuzaki, K.; Sugishita, K.; Harada, M.; Fujii, N.; Miyajima, K. Interactions of an antimicrobial peptide, magainin 2, with outer and inner membranes of Gram-negative bacteria. Biochim. Biophys. Acta, 1997, 1327, 119-130.
-
(1997)
Biochim. Biophys. Acta
, vol.1327
, pp. 119-130
-
-
Matsuzaki, K.1
Sugishita, K.2
Harada, M.3
Fujii, N.4
Miyajima, K.5
-
26
-
-
0003225524
-
Molecular Structure and Function
-
Gennis, R. B. Molecular Structure and Function. Biomembrane, 1989, 1, 51-158.
-
(1989)
Biomembrane
, vol.1
, pp. 51-158
-
-
Gennis, R.B.1
-
27
-
-
0023864293
-
Binding and action of cecropin and cecropin analogues: Antibacterial peptides from insects
-
Steiner, H.; Andreu, D.; Merrifield, R. B. Binding and action of cecropin and cecropin analogues: antibacterial peptides from insects. Biochim. Biophys. Acta, 1988, 939, 260-266.
-
(1988)
Biochim. Biophys. Acta
, vol.939
, pp. 260-266
-
-
Steiner, H.1
Andreu, D.2
Merrifield, R.B.3
-
28
-
-
0035719931
-
Amphipathic α-helical antimicrobial peptides, a systematic study of the effects of structural and physical properties on biological activity
-
Giangasparo, A.; Sandri, L.; Tossi, A. Amphipathic α-helical antimicrobial peptides, a systematic study of the effects of structural and physical properties on biological activity. Eur. J. Biochem., 2001, 268, 5589-5600.
-
(2001)
Eur. J. Biochem
, vol.268
, pp. 5589-5600
-
-
Giangasparo, A.1
Sandri, L.2
Tossi, A.3
-
29
-
-
0343503006
-
The comparison of characteristic between membrane-active antifungal peptide and its pseudo peptides
-
Eunoh, J.; Hong S.U.; Lee, K.H. The comparison of characteristic between membrane-active antifungal peptide and its pseudo peptides. Bioorg. Med. Chem., 1999, 7, 2509-2515.
-
(1999)
Bioorg. Med. Chem
, vol.7
, pp. 2509-2515
-
-
Eunoh, J.1
Hong, S.U.2
Lee, K.H.3
-
30
-
-
0036948138
-
Mode of action of membrane active antimicrobial peptides
-
Shai, Y. Mode of action of membrane active antimicrobial peptides. Biopolymers, 2002, 66, 236-248.
-
(2002)
Biopolymers
, vol.66
, pp. 236-248
-
-
Shai, Y.1
-
31
-
-
0034859096
-
Barrel-stave model or toroidal model? A case study on melittin pores
-
Yang, L.; Harroun, T.A.; Weiss, T.M. L.; Ding, H.W. Barrel-stave model or toroidal model? A case study on melittin pores. Biophys. J., 2001, 81, 1475-1485.
-
(2001)
Biophys. J
, vol.81
, pp. 1475-1485
-
-
Yang, L.1
Harroun, T.A.2
Weiss, T.M.L.3
Ding, H.W.4
-
32
-
-
0017363554
-
Electrically gated ionic channels in lipid bilayers
-
Ehrenstein, G.; Lecar, H. Q. Electrically gated ionic channels in lipid bilayers. Rev. Biophys., 1977, 10, 1-34.
-
(1977)
Rev. Biophys
, vol.10
, pp. 1-34
-
-
Ehrenstein, G.1
Lecar, H.Q.2
-
33
-
-
0036296712
-
Expression of insect cystein-rich antifungal peptides in transgenic tobacco enhances resistance to a fungal disease
-
Banzet, N.; Lotris, M.P.; Bulet, P.; Francosis, E.; Deropierre, C.; Dubald, M. Expression of insect cystein-rich antifungal peptides in transgenic tobacco enhances resistance to a fungal disease. Plant Sci., 2002, 162, 995-1006.
-
(2002)
Plant Sci
, vol.162
, pp. 995-1006
-
-
Banzet, N.1
Lotris, M.P.2
Bulet, P.3
Francosis, E.4
Deropierre, C.5
Dubald, M.6
-
34
-
-
32344443212
-
Antifungal activity of synthetic peptide derived from halocidin, antimicrobial peptide from the tunicate, Halocynthia aurantium
-
Jang, W.S.; Kim H.K.; Lee K.Y.; Kim S.A.; Han Y.S.; Lee, I.H. Antifungal activity of synthetic peptide derived from halocidin, antimicrobial peptide from the tunicate, Halocynthia aurantium. FEBS Lett., 2006, 580, 1490-1496.
-
(2006)
FEBS Lett
, vol.580
, pp. 1490-1496
-
-
Jang, W.S.1
Kim, H.K.2
Lee, K.Y.3
Kim, S.A.4
Han, Y.S.5
Lee, I.H.6
-
35
-
-
0027169823
-
-
Kokryakov, V.N.; Harwig, S.S.; Panyutich, E.A.; Shevchenko, A.A.; Aleshina, G.M.; Shamova, O.; Korneva, H.A.; Lehrer, R.I. Protegrins: leukocyte antimicrobial peptides that combine features of corticostatic defensins and tachyplesins. FEBS Lett., 1993, 327(2), 23,1-6.
-
Kokryakov, V.N.; Harwig, S.S.; Panyutich, E.A.; Shevchenko, A.A.; Aleshina, G.M.; Shamova, O.; Korneva, H.A.; Lehrer, R.I. Protegrins: leukocyte antimicrobial peptides that combine features of corticostatic defensins and tachyplesins. FEBS Lett., 1993, 327(2), 23,1-6.
-
-
-
-
36
-
-
32644478817
-
Concurrent isolation of a Kunitz-type trypsin inhibitor with antifungal activity and a novel lectin from Pseudostellaria heterophylla roots
-
Wang, H.X.; Ng, T.B. Concurrent isolation of a Kunitz-type trypsin inhibitor with antifungal activity and a novel lectin from Pseudostellaria heterophylla roots. Biochem. Biophys. Res. Commun., 2006, 342, 349-353.
-
(2006)
Biochem. Biophys. Res. Commun
, vol.342
, pp. 349-353
-
-
Wang, H.X.1
Ng, T.B.2
-
37
-
-
15244344778
-
Identification of a novel antifungal nonapeptide generated by combinatorial approach
-
Kumar, M.; Chaturvedi, A.K.; Kavishavar, A.; Shukla, P.K.; Kesarwani, A.P.; Kundu, B. Identification of a novel antifungal nonapeptide generated by combinatorial approach. Int. J. Antimicrob. Agent., 2005, 25, 313-320.
-
(2005)
Int. J. Antimicrob. Agent
, vol.25
, pp. 313-320
-
-
Kumar, M.1
Chaturvedi, A.K.2
Kavishavar, A.3
Shukla, P.K.4
Kesarwani, A.P.5
Kundu, B.6
-
38
-
-
0021846352
-
Primary structures of six antimicrobial peptides of rabbit peritoneal neutrophils
-
Selsted, M.E.; Brown, D.M.; DeLange, R.J.; Harwig, S.S.; Lehrer, R.I. Primary structures of six antimicrobial peptides of rabbit peritoneal neutrophils. J. Biol. Chem., 1985, 260(8), 4579-84.
-
(1985)
J. Biol. Chem
, vol.260
, Issue.8
, pp. 4579-4584
-
-
Selsted, M.E.1
Brown, D.M.2
DeLange, R.J.3
Harwig, S.S.4
Lehrer, R.I.5
-
39
-
-
0033433992
-
SMAP-29: A potent antibacterial and antifungal peptide from sheep leukocytes
-
Skerlavaj, B.; Benincasa, M.; Risso, A.; Zanetti, M.; Renato, G. SMAP-29: a potent antibacterial and antifungal peptide from sheep leukocytes. FEBS Lett., 1999, 463, 58-62.
-
(1999)
FEBS Lett
, vol.463
, pp. 58-62
-
-
Skerlavaj, B.1
Benincasa, M.2
Risso, A.3
Zanetti, M.4
Renato, G.5
-
40
-
-
7244221533
-
Inhibition of Adherence and Killing of Candida albicans with a 23-Mer Peptide (Fn/23) with Dual Antifungal Properties
-
Klotz, S.A.; Gaur, N.K.; Rauceo, J.; Lake, D.F.; Park, Y.; Hahm, S. Inhibition of Adherence and Killing of Candida albicans with a 23-Mer Peptide (Fn/23) with Dual Antifungal Properties. Antimicrob. Agent Chemother., 2004, 48 (11), 4337-4341.
-
(2004)
Antimicrob. Agent Chemother
, vol.48
, Issue.11
, pp. 4337-4341
-
-
Klotz, S.A.1
Gaur, N.K.2
Rauceo, J.3
Lake, D.F.4
Park, Y.5
Hahm, S.6
-
41
-
-
0034450462
-
Cecropins, antibacterial peptides from insects and mammals, are potently fungicidal against Candida albicans
-
Andra, J.; Berninghausen, O.; LEIPPE, M. Cecropins, antibacterial peptides from insects and mammals, are potently fungicidal against Candida albicans. Med. Microbiol. Immunol., 2001, 189, 169-173.
-
(2001)
Med. Microbiol. Immunol
, vol.189
, pp. 169-173
-
-
Andra, J.1
Berninghausen, O.2
LEIPPE, M.3
-
42
-
-
0035842069
-
Molecular scaffold of a new pokeweed antifungal peptide deduced by 1H nuclear magnetic resonance
-
Gao, G.H.; Liu, W.; Dai, J.X.; Wang, J.F.; Hu, Z.; Zhang, Y.; Wang, D.C. Molecular scaffold of a new pokeweed antifungal peptide deduced by 1H nuclear magnetic resonance. Int. J. Bio. Macromol., 2001, 29, 251-258..
-
(2001)
Int. J. Bio. Macromol
, vol.29
, pp. 251-258
-
-
Gao, G.H.1
Liu, W.2
Dai, J.X.3
Wang, J.F.4
Hu, Z.5
Zhang, Y.6
Wang, D.C.7
-
43
-
-
0026736540
-
Magainin 2, a natural antibiotic from frog skin, forms ion channels in lipid bilayer membranes
-
Cruciani, R.A.; Barker, J.L.; Durell, S.R.; Raghunathan, G.; Guy, H.R.; Zasloff, M.; Stanley, E.F. Magainin 2, a natural antibiotic from frog skin, forms ion channels in lipid bilayer membranes. Eur. J. Pharmacol., 1992, 226(4), 287-96
-
(1992)
Eur. J. Pharmacol
, vol.226
, Issue.4
, pp. 287-296
-
-
Cruciani, R.A.1
Barker, J.L.2
Durell, S.R.3
Raghunathan, G.4
Guy, H.R.5
Zasloff, M.6
Stanley, E.F.7
-
44
-
-
0030583613
-
Determination of the disulfide array of the first inducible antifungal peptide from insects: Drosomycin from Drosophila melanogaster
-
Michut, L.; Fehlbaum, P.; Moniatte, M.; Dorsselaer, A.V.; Reichhart, J.M.; Bulet, P. Determination of the disulfide array of the first inducible antifungal peptide from insects: drosomycin from Drosophila melanogaster. FEBS Lett., 1996, 395, 6 -10.
-
(1996)
FEBS Lett
, vol.395
, pp. 6-10
-
-
Michut, L.1
Fehlbaum, P.2
Moniatte, M.3
Dorsselaer, A.V.4
Reichhart, J.M.5
Bulet, P.6
-
45
-
-
0032585345
-
Bacterial expression of tenecin 3, an insect antifungal protein isolated from Tenebrio molitor, and its efficient purification
-
Kim, D. H.; Lee, Y.T.; Lee, Y. J.; Chung, J. H.; Lee, B. L.; Choi, B.S.; Lee, Y. Bacterial expression of tenecin 3, an insect antifungal protein isolated from Tenebrio molitor, and its efficient purification. Mol. Cell., 1998, 8(6), 786-9
-
(1998)
Mol. Cell
, vol.8
, Issue.6
, pp. 786-789
-
-
Kim, D.H.1
Lee, Y.T.2
Lee, Y.J.3
Chung, J.H.4
Lee, B.L.5
Choi, B.S.6
Lee, Y.7
-
46
-
-
0037134784
-
Two novel antifungal peptides distinct with a five-disulfide motif from the bark of Eucommiaulmoides Oliv
-
Huang, R.H.; Xiang, Y.; Liu, X.Z.; Zhang, Y.; Hu, Z.; Wang, D. C. Two novel antifungal peptides distinct with a five-disulfide motif from the bark of Eucommiaulmoides Oliv. FEBS Lett., 2002, 521, 87-90.
-
(2002)
FEBS Lett
, vol.521
, pp. 87-90
-
-
Huang, R.H.1
Xiang, Y.2
Liu, X.Z.3
Zhang, Y.4
Hu, Z.5
Wang, D.C.6
-
47
-
-
0036152594
-
Isolation of cicadin, a novel and potent antifungal peptide from Juvenile cicadas
-
Wang, H.; Ng, T.B. Isolation of cicadin, a novel and potent antifungal peptide from Juvenile cicadas. Peptides, 2002, 23, 7 -11.
-
(2002)
Peptides
, vol.23
, pp. 7-11
-
-
Wang, H.1
Ng, T.B.2
-
48
-
-
1242306544
-
Antimicrobial peptides from rained frogs: Taxonomic and phylogenic markers and a potential source of new therapeutic agents
-
Conlon, L.M.; Kolodziejek, J.; Nowontny, N. Antimicrobial peptides from rained frogs: Taxonomic and phylogenic markers and a potential source of new therapeutic agents. Biochim. Biophys. Acta, 2004, 1696, 1-14.
-
(2004)
Biochim. Biophys. Acta
, vol.1696
, pp. 1-14
-
-
Conlon, L.M.1
Kolodziejek, J.2
Nowontny, N.3
-
49
-
-
3042814737
-
Antifungal proteins and peptides of leguminous and nonleguminous origin
-
Ng, T.B. Antifungal proteins and peptides of leguminous and nonleguminous origin. Peptides, 2000, 25, 1215-1222.
-
(2000)
Peptides
, vol.25
, pp. 1215-1222
-
-
Ng, T.B.1
-
50
-
-
0345363252
-
Isolation and characterization of a novel antifungal peptide from Aspergillus niger
-
Lee, D.G.; Shin, S.Y.; Maeng, C.Y.; Jin, Z.Z.; Kim, K.L.; Hahm, K.S. Isolation and characterization of a novel antifungal peptide from Aspergillus niger. Biochem. Biophys. Res. Commun., 1999, 263, 646 -651.
-
(1999)
Biochem. Biophys. Res. Commun
, vol.263
, pp. 646-651
-
-
Lee, D.G.1
Shin, S.Y.2
Maeng, C.Y.3
Jin, Z.Z.4
Kim, K.L.5
Hahm, K.S.6
-
51
-
-
0028352996
-
Fungicin M4: A narrow spectrum peptide antibiotic from Bacillus licheniformis M-4
-
Lebbadi, M.; Gálvez, A.; Maqueda, M.; Martínez-Bueno, M.; Valdivia, E. Fungicin M4: a narrow spectrum peptide antibiotic from Bacillus licheniformis M-4. J. Appl. Bacteriol., 1994, 77(1), 49-53.
-
(1994)
J. Appl. Bacteriol
, vol.77
, Issue.1
, pp. 49-53
-
-
Lebbadi, M.1
Gálvez, A.2
Maqueda, M.3
Martínez-Bueno, M.4
Valdivia, E.5
-
52
-
-
33646402378
-
Biological activity of Tat (47-58) peptide on human pathogenic fungi
-
Jung, H. J.; Park, Y.; Hahm, K. S.; Lee, D.G. Biological activity of Tat (47-58) peptide on human pathogenic fungi. Biochem. Biophys. Res. Commun., 2006, 345, 222 -228.
-
(2006)
Biochem. Biophys. Res. Commun
, vol.345
, pp. 222-228
-
-
Jung, H.J.1
Park, Y.2
Hahm, K.S.3
Lee, D.G.4
-
53
-
-
0028925597
-
-
Gräfe, U.; Ihn, W.; Ritzau, M.; Schade, W.; Stengel, C.; Schlegel, B.; Fleck, W. F.; Künkel, W.; Härtl, A.; Gutsche, W. Helioferins, novel antifungal lipopeptides from Mycogone rosea: screening, isolation, structure, and biological properties. J. Antibiot., 1995, 48(2), 128-133.
-
Gräfe, U.; Ihn, W.; Ritzau, M.; Schade, W.; Stengel, C.; Schlegel, B.; Fleck, W. F.; Künkel, W.; Härtl, A.; Gutsche, W. Helioferins, novel antifungal lipopeptides from Mycogone rosea: screening, isolation, structure, and biological properties. J. Antibiot., 1995, 48(2), 128-133.
-
-
-
-
54
-
-
0028486247
-
-
Klich, A.; Arthur, K. S.; Lax, A.R.; Bland, J. M. Iturin A: a potential new fungicide for stored grains. Mycopathology, 1994, 127 (2), 453-460.
-
Klich, A.; Arthur, K. S.; Lax, A.R.; Bland, J. M. Iturin A: a potential new fungicide for stored grains. Mycopathology, 1994, 127 (2), 453-460.
-
-
-
-
55
-
-
0034660429
-
Antimicrobial Nonapeptide Leucinostatin A-Dependent Effects on the Physical Properties of Phospholipid Model Membranes
-
Fresta, M.; Ricci, M.; Rossi, C.; Furneri, P.M.; Puglisi, G. Antimicrobial Nonapeptide Leucinostatin A-Dependent Effects on the Physical Properties of Phospholipid Model Membranes. J. Coll. Inter. Sci., 2000, 226 (2), 222-230.
-
(2000)
J. Coll. Inter. Sci
, vol.226
, Issue.2
, pp. 222-230
-
-
Fresta, M.1
Ricci, M.2
Rossi, C.3
Furneri, P.M.4
Puglisi, G.5
-
56
-
-
0025281052
-
Conformational studies of nikkomycin X in aqueous solution
-
Krainer, E.; Naider, F.; Becker, J. M. Conformational studies of nikkomycin X in aqueous solution. Biopolymers, 1990, 29 (8), 1297 -1306.
-
(1990)
Biopolymers
, vol.29
, Issue.8
, pp. 1297-1306
-
-
Krainer, E.1
Naider, F.2
Becker, J.M.3
-
57
-
-
0014868818
-
Mechanism of Action of the Antifugal Agent Polyoxin D
-
Endo, A.; Kakiki, K.; Misato, T. Mechanism of Action of the Antifugal Agent Polyoxin D. J Bacteriol., 1970, 104(1), 189-196.
-
(1970)
J Bacteriol
, vol.104
, Issue.1
, pp. 189-196
-
-
Endo, A.1
Kakiki, K.2
Misato, T.3
-
58
-
-
0032958766
-
Antifungal peptides: Novel therapeutic compounds against emerging pathogens
-
De Lucca, A. J.; Walsh, T. J. Antifungal peptides: novel therapeutic compounds against emerging pathogens. Antimicrob. Agents Chemother., 1999, 43(1), 1-11.
-
(1999)
Antimicrob. Agents Chemother
, vol.43
, Issue.1
, pp. 1-11
-
-
De Lucca, A.J.1
Walsh, T.J.2
-
59
-
-
73549107340
-
New antibiotics, trichopolyns A and B: Isolation and biological activity
-
Fuji, E.; Fujita, Y.; Takaishi, T.; Fujita, I.; Arita, M.; Hiratsuka, N. New antibiotics, trichopolyns A and B: isolation and biological activity. Cel. Mol. Life Sci., 1978, 34(2), 253-361.
-
(1978)
Cel. Mol. Life Sci
, vol.34
, Issue.2
, pp. 253-361
-
-
Fuji, E.1
Fujita, Y.2
Takaishi, T.3
Fujita, I.4
Arita, M.5
Hiratsuka, N.6
-
60
-
-
0027057467
-
Pneumocandins from Zalerion arboricola. V. Glutamic acid- and leucine-derived amino acids in pneumocandin A0 (L-671,329) and distinct origins of the substituted proline residues in pneumocandins A0 and B0
-
Adefarati, A.A.; Hensens, O.D.; Jones, E.T.; Tkacz, J.S. Pneumocandins from Zalerion arboricola. V. Glutamic acid- and leucine-derived amino acids in pneumocandin A0 (L-671,329) and distinct origins of the substituted proline residues in pneumocandins A0 and B0. J. Antibiot., 1992, 45(12), 1953-7.
-
(1992)
J. Antibiot
, vol.45
, Issue.12
, pp. 1953-1957
-
-
Adefarati, A.A.1
Hensens, O.D.2
Jones, E.T.3
Tkacz, J.S.4
-
61
-
-
0025123312
-
-
Iwamoto, T.; Fujie, A.; Tsurumi, Y.; Nitta, K.; Hashimoto, S.; Okuhara, M. WF11899A, B and C, novel antifungal lipopeptides. I. Taxonomy, fermentation, isolation and physico-chemical properties. J. Antibiot., 1990, 43(9), 1183-5.
-
Iwamoto, T.; Fujie, A.; Tsurumi, Y.; Nitta, K.; Hashimoto, S.; Okuhara, M. WF11899A, B and C, novel antifungal lipopeptides. I. Taxonomy, fermentation, isolation and physico-chemical properties. J. Antibiot., 1990, 43(9), 1183-5.
-
-
-
-
62
-
-
0001134345
-
Purification and properties of a new chitin-binding antifungal CB-1 from Bacillus licheniformis
-
Shigeru, O.; Mitsuo, H.; Sonoe, Y. Purification and properties of a new chitin-binding antifungal CB-1 from Bacillus licheniformis. Biosci. Biotechnol. Biochem., 1996, 60 (3), 481-483.
-
(1996)
Biosci. Biotechnol. Biochem
, vol.60
, Issue.3
, pp. 481-483
-
-
Shigeru, O.1
Mitsuo, H.2
Sonoe, Y.3
-
63
-
-
0033964034
-
Pilot-scale purification of zeamatin, an antifungal protein from maize
-
Wilson, S.; Mahiou, B.; Reiger, R.; Tentler, S.; Schimmoler, R.; Orndorff, S.; Selitrennikoff, C. P. Pilot-scale purification of zeamatin, an antifungal protein from maize. Biotechnol. Prog., 2000, 16(1), 38-43.
-
(2000)
Biotechnol. Prog
, vol.16
, Issue.1
, pp. 38-43
-
-
Wilson, S.1
Mahiou, B.2
Reiger, R.3
Tentler, S.4
Schimmoler, R.5
Orndorff, S.6
Selitrennikoff, C.P.7
-
64
-
-
0032539972
-
Solution structure of Ace-AMP1, a potent antimicrobial protein extracted from onion seeds. Structural analogies with plant nonspecific lipid transfer proteins
-
Tassin, S.; Broekaert, W. F.; Marion, D.; Acland, D. P.; Ptak, M.; Vovelle, F.; Sodano, P. Solution structure of Ace-AMP1, a potent antimicrobial protein extracted from onion seeds. Structural analogies with plant nonspecific lipid transfer proteins. Biochemistry, 1998, 37(11), 3623-37.
-
(1998)
Biochemistry
, vol.37
, Issue.11
, pp. 3623-3637
-
-
Tassin, S.1
Broekaert, W.F.2
Marion, D.3
Acland, D.P.4
Ptak, M.5
Vovelle, F.6
Sodano, P.7
-
65
-
-
33846781508
-
An antifungal peptide from red lentil seeds
-
Wang, H.X.; Ng, T.B. An antifungal peptide from red lentil seeds. Peptides, 2007, 28 (3), 547-552.
-
(2007)
Peptides
, vol.28
, Issue.3
, pp. 547-552
-
-
Wang, H.X.1
Ng, T.B.2
-
66
-
-
9644264232
-
Coccinin, an antifungal peptide with antiproliferative and HIV-1 reverse transcriptase inhibitory activities from large scarlet runner beans
-
Ngai, P.H.K..; Ng, TB. Coccinin, an antifungal peptide with antiproliferative and HIV-1 reverse transcriptase inhibitory activities from large scarlet runner beans. Peptides, 2004, 25, 2063-2068.
-
(2004)
Peptides
, vol.25
, pp. 2063-2068
-
-
Ngai, P.H.K.1
Ng, T.B.2
-
67
-
-
0043207427
-
-
Chu, K.T.; Liu, K.H.; Ng, T.B. Cicerann, a novel antifungal peptide from the green chickpea. Pep., 2003, 24, 659-663.
-
Chu, K.T.; Liu, K.H.; Ng, T.B. Cicerann, a novel antifungal peptide from the green chickpea. Pep., 2003, 24, 659-663.
-
-
-
-
68
-
-
0141518452
-
-
Wong, J.H.; Ng, T.B. Gymnin, a potent defensin-like antifungal peptide from the Yunnan bean (Gymnocladus chinensis Baill). Peptides, 2003, 24, 963-968.
-
Wong, J.H.; Ng, T.B. Gymnin, a potent defensin-like antifungal peptide from the Yunnan bean (Gymnocladus chinensis Baill). Peptides, 2003, 24, 963-968.
-
-
-
-
69
-
-
0347990380
-
Insect diapuse-specific peptide from the leaf beetle has consensus with a putative iridovirus peptide
-
Tanaka, H.; Satio, K.; Satio, Y.; Yamashita, T.; Agoh, M.; Okkunishi, J. Insect diapuse-specific peptide from the leaf beetle has consensus with a putative iridovirus peptide. Peptides, 2003, 24, 1327-1333.
-
(2003)
Peptides
, vol.24
, pp. 1327-1333
-
-
Tanaka, H.1
Satio, K.2
Satio, Y.3
Yamashita, T.4
Agoh, M.5
Okkunishi, J.6
-
70
-
-
0032940371
-
LY303366 exhibits rapid and potent fungicidal activity in flow cytometric assays of yeast viability
-
Green, L.J.; Marder, P.; Mann, L. L.; Chio, L.; Current, W. L. LY303366 exhibits rapid and potent fungicidal activity in flow cytometric assays of yeast viability. Antimicrob. Agents Chemother., 1999, 43 (4), 830-835.
-
(1999)
Antimicrob. Agents Chemother
, vol.43
, Issue.4
, pp. 830-835
-
-
Green, L.J.1
Marder, P.2
Mann, L.L.3
Chio, L.4
Current, W.L.5
-
71
-
-
0031865111
-
-
De Lucca, A.J.; Bland, J.M.; Grimm, C.; Jacks, T.J.; Cary, J.W.; Jaynes, J.M.; Cleveland,T.E.; Walsh.; T.J. Fungicidal and binding properties of the natural peptides cecropin B and dermaseptin. J. Microbiol., 1998, 44, 514.520.
-
De Lucca, A.J.; Bland, J.M.; Grimm, C.; Jacks, T.J.; Cary, J.W.; Jaynes, J.M.; Cleveland,T.E.; Walsh.; T.J. Fungicidal and binding properties of the natural peptides cecropin B and dermaseptin. J. Microbiol., 1998, 44, 514.520.
-
-
-
-
72
-
-
0343503006
-
The comparison of characteristics between membrane-active antifungal peptide and its pseudopeptides
-
Oh, J.E.; Hong, S.U.; Lee, K.H. The comparison of characteristics between membrane-active antifungal peptide and its pseudopeptides. Bioorg. Med. Chem., 1999, 7, 2509-2515.
-
(1999)
Bioorg. Med. Chem
, vol.7
, pp. 2509-2515
-
-
Oh, J.E.1
Hong, S.U.2
Lee, K.H.3
-
73
-
-
0037971557
-
Release of antimicrobial peptide Dhvar-5 from polymethylmethacrylate beads
-
Faber, C.; Stallmann, H. P.; Lyaruu, D. M.; Blieck, J. M. A.; Bervoets, J. M.; Wuisman, P. I. J. M. Release of antimicrobial peptide Dhvar-5 from polymethylmethacrylate beads. J. Antimicrob. Chemother., 2003, 51, 1359-1364
-
(2003)
J. Antimicrob. Chemother
, vol.51
, pp. 1359-1364
-
-
Faber, C.1
Stallmann, H.P.2
Lyaruu, D.M.3
Blieck, J.M.A.4
Bervoets, J.M.5
Wuisman, P.I.J.M.6
-
74
-
-
0025678163
-
Activity of cilofungin (LY 121019), a new lipopeptide antibiotic, on the cell wall and cytoplasmic membrane of Candida albicans. Structural modifications in scanning and transmission electron microscopy
-
Drouhet, E.; Dupont, B.; Improvisi, L.; Lesourd, M.; Prevost, M. C. Activity of cilofungin (LY 121019), a new lipopeptide antibiotic, on the cell wall and cytoplasmic membrane of Candida albicans. Structural modifications in scanning and transmission electron microscopy. J. Med. Vet. Mycol., 1990, 28(6), 425-36.
-
(1990)
J. Med. Vet. Mycol
, vol.28
, Issue.6
, pp. 425-436
-
-
Drouhet, E.1
Dupont, B.2
Improvisi, L.3
Lesourd, M.4
Prevost, M.C.5
-
75
-
-
1642359643
-
Energetics of pore formation induced by membrane active peptides
-
Lee, M.T.; Chen, F.Y.; Huang, H.W. Energetics of pore formation induced by membrane active peptides. Biochemistry, 2004, 433, 590-3599.
-
(2004)
Biochemistry
, vol.433
, pp. 590-3599
-
-
Lee, M.T.1
Chen, F.Y.2
Huang, H.W.3
-
76
-
-
68149136602
-
Evidence of pores and thinned lipid bilayers induced in oriented lipid membranes interacting with the antimicrobial peptides, magainin-2 and aurein-3
-
Kim, C.; Spano, J.; Park, E.K.; Wi, S. Evidence of pores and thinned lipid bilayers induced in oriented lipid membranes interacting with the antimicrobial peptides, magainin-2 and aurein-3. BBABiomembr., 2009, 1788 (7), 1482-1496.
-
(2009)
BBABiomembr
, vol.1788
, Issue.7
, pp. 1482-1496
-
-
Kim, C.1
Spano, J.2
Park, E.K.3
Wi, S.4
-
77
-
-
0036897824
-
Mimicry of bioactive peptides via nonnatural, sequence-specific peptidomimetic oligomers
-
Patch, J.A.; Barron, A.E. Mimicry of bioactive peptides via nonnatural, sequence-specific peptidomimetic oligomers. Cur. Opin. Chem. Biol., 2002, 6, 872-877
-
(2002)
Cur. Opin. Chem. Biol
, vol.6
, pp. 872-877
-
-
Patch, J.A.1
Barron, A.E.2
-
78
-
-
0542421525
-
A Manifesto
-
Gellman, S.H. Foldamers: A Manifesto. Acc. Chem. Res., 1998, 31, 173-180
-
(1998)
Acc. Chem. Res
, vol.31
, pp. 173-180
-
-
Gellman, S.H.F.1
-
79
-
-
13944277208
-
-
P.E. Nielsen, Ed. Weinheim, Germany: Wiley-VCH Verlag
-
Guichard, G. In Pseudopeptides in Drug Development; P.E. Nielsen, Ed. Weinheim, Germany: Wiley-VCH Verlag, 2004; pp. 33-120.
-
(2004)
In Pseudopeptides in Drug Development
, pp. 33-120
-
-
Guichard, G.1
-
80
-
-
0037202210
-
Structureactivity studies of 14-helical antimicrobial beta-peptides: Probing the relationship between conformational stability and antimicrobial potency
-
Raguse, T.L.; Porter, E.A.; Weisblum, B.; Gellman, S.H. Structureactivity studies of 14-helical antimicrobial beta-peptides: probing the relationship between conformational stability and antimicrobial potency. J. Am. Chem. Soc., 2002, 124, 12774-12785.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 12774-12785
-
-
Raguse, T.L.1
Porter, E.A.2
Weisblum, B.3
Gellman, S.H.4
-
81
-
-
57549101729
-
Peptoid architectures: Elaboration, actuation, and application
-
Yoo, B.; Kirshenbaum, K. Peptoid architectures: elaboration, actuation, and application. Curr. Opin. Chem. Biol., 2008, 12 (6), 714-721.
-
(2008)
Curr. Opin. Chem. Biol
, vol.12
, Issue.6
, pp. 714-721
-
-
Yoo, B.1
Kirshenbaum, K.2
-
82
-
-
4444243683
-
A small molecule Smac mimic potentiates TRAIL- and TNFalpha-mediated cell death
-
Li, L., Thomas, R.M.; Suzuki, H.; De Brabander, J.K.; Wang, X.; Harran, P.G. A small molecule Smac mimic potentiates TRAIL- and TNFalpha-mediated cell death. Science, 2004, 3, 305, 1471-74.
-
(2004)
Science
, vol.3
, Issue.305
, pp. 1471-1474
-
-
Li, L.1
Thomas, R.M.2
Suzuki, H.3
De Brabander, J.K.4
Wang, X.5
Harran, P.G.6
-
83
-
-
0033851469
-
Conformational and topographical considerations in designing agonist peptidomimetics from peptide leads
-
Hruby, V. J.; Balse, P. M. Conformational and topographical considerations in designing agonist peptidomimetics from peptide leads. Curr. Med. Chem., 2000, 7, 945-970.
-
(2000)
Curr. Med. Chem
, vol.7
, pp. 945-970
-
-
Hruby, V.J.1
Balse, P.M.2
-
84
-
-
0030884435
-
Design of peptides, proteins, and peptidomimetics in chi space
-
Hruby, V. J.; Li, G.; Haskell-Luevano, C.; Shenderovich, M. Design of peptides, proteins, and peptidomimetics in chi space. Biopolymers, 1997, 43, 219-266.
-
(1997)
Biopolymers
, vol.43
, pp. 219-266
-
-
Hruby, V.J.1
Li, G.2
Haskell-Luevano, C.3
Shenderovich, M.4
-
86
-
-
0037187386
-
Design, synthesis, and evaluation of opioid analogues with nonpeptidic beta-turn scaffold: Enkephalin and endomorphin mimetics
-
Eguchi, M.; Shen, R. Y. W.; Shea, J. P.; Lee, M.S.; Kahn, M. Design, synthesis, and evaluation of opioid analogues with nonpeptidic beta-turn scaffold: enkephalin and endomorphin mimetics. J. Med. Chem., 2002, 45, 1395-1398.
-
(2002)
J. Med. Chem
, vol.45
, pp. 1395-1398
-
-
Eguchi, M.1
Shen, R.Y.W.2
Shea, J.P.3
Lee, M.S.4
Kahn, M.5
-
87
-
-
0037031636
-
-
Wang, W.; Yang, J.; Ying, J.; Xiong, C.; Zhang, J.; Cai, C.; Hruby, V. J. Stereoselective synthesis of dipeptide beta-turn mimetics: 7-benzyl and 8-phenyl substituted azabicyclo[4.3.0]nonane amino acid esters. J. Org. Chem., 2002, 67, 6353-6360.
-
Wang, W.; Yang, J.; Ying, J.; Xiong, C.; Zhang, J.; Cai, C.; Hruby, V. J. Stereoselective synthesis of dipeptide beta-turn mimetics: 7-benzyl and 8-phenyl substituted azabicyclo[4.3.0]nonane amino acid esters. J. Org. Chem., 2002, 67, 6353-6360.
-
-
-
-
88
-
-
0031802413
-
Synthesis and structural and functional evaluation of a protein modified with a beta-turn mimic
-
Jean, F.; Buisine, E.; Melnyk, O.; Drobecq, H.; Odaert, B.; Hugues, M.; Lippens, G.; Tartar, A. Synthesis and structural and functional evaluation of a protein modified with a beta-turn mimic. J. Am. Chem. Soc., 1998, 120, 6076-6083.
-
(1998)
J. Am. Chem. Soc
, vol.120
, pp. 6076-6083
-
-
Jean, F.1
Buisine, E.2
Melnyk, O.3
Drobecq, H.4
Odaert, B.5
Hugues, M.6
Lippens, G.7
Tartar, A.8
-
89
-
-
0037048625
-
Synthesis of a negatively charged dibenzofuran-based beta-turn mimetic and its incorporation into the WW miniprotein-enhanced solubility without a loss of thermodynamic stability
-
Kaul, R.; Deechongkit, S.; Kelly, J. W. Synthesis of a negatively charged dibenzofuran-based beta-turn mimetic and its incorporation into the WW miniprotein-enhanced solubility without a loss of thermodynamic stability. J. Am. Chem. Soc., 2002, 124, 11900-11907.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 11900-11907
-
-
Kaul, R.1
Deechongkit, S.2
Kelly, J.W.3
-
90
-
-
0037178340
-
Ni-to-Ni+3-ethylene- bridged partially modified retro-inverso tetrapeptide betaturn mimetic: Design, synthesis, and structural characterization
-
Han, Y.; Giragossian, C.; Mierke, D. F.; Chorev, M. Ni-to-Ni+3-ethylene- bridged partially modified retro-inverso tetrapeptide betaturn mimetic: design, synthesis, and structural characterization. J. Org. Chem., 2002, 67, 5085-5097.
-
(2002)
J. Org. Chem
, vol.67
, pp. 5085-5097
-
-
Han, Y.1
Giragossian, C.2
Mierke, D.F.3
Chorev, M.4
-
91
-
-
0019958486
-
Potent new inhibitors of human renin
-
Szelke, M.; Leckie, B.; Hallett, A; Jones, D.M.; Sueiras, J.; Atrash, B. Potent new inhibitors of human renin. Nature, 1982, 299, 555-557.
-
(1982)
Nature
, vol.299
, pp. 555-557
-
-
Szelke, M.1
Leckie, B.2
Hallett, A.3
Jones, D.M.4
Sueiras, J.5
Atrash, B.6
-
92
-
-
0027478912
-
Peptidomimetics derived from natural products
-
Wiley, R.A.; Rich, D.H. Peptidomimetics derived from natural products. Med. Res. Rev. 1993, 13, 327-384.
-
(1993)
Med. Res. Rev
, vol.13
, pp. 327-384
-
-
Wiley, R.A.1
Rich, D.H.2
-
93
-
-
0030576323
-
-
Maibaum, V.; Cohen, N.C.; Rijeger, H.; Gschke, .R; Maibaum, J.; Cumin, F.; Fuhrer, W.; Wood, J.M. Bioactive hydroxyethylene dipeptide isosteres with hydrophobic (P3-P1)-moieties. A novel strategy towards small non-peptide renin inhibitors. Bioorg. Med. Chem. Lett., 1996, 6, 1589-l 594.
-
Maibaum, V.; Cohen, N.C.; Rijeger, H.; Gschke, .R; Maibaum, J.; Cumin, F.; Fuhrer, W.; Wood, J.M. Bioactive hydroxyethylene dipeptide isosteres with hydrophobic (P3-P1)-moieties. A novel strategy towards small non-peptide renin inhibitors. Bioorg. Med. Chem. Lett., 1996, 6, 1589-l 594.
-
-
-
-
94
-
-
0141608479
-
Design and synthesis of novel 2,7-dialkyl substituted 5(S)-amino-4(S)-hydroxy-8-phenyl- octanecarboxamides as in vitro potent peptidomimetic inhibitors of human rennin
-
Goschke, R.; Cohen, N.C.; Wood, J.M.; Maibaum, J. Design and synthesis of novel 2,7-dialkyl substituted 5(S)-amino-4(S)-hydroxy-8-phenyl- octanecarboxamides as in vitro potent peptidomimetic inhibitors of human rennin. Bioorg. Med. Chem. Lett., 1997, 7, 2735-2740.
-
(1997)
Bioorg. Med. Chem. Lett
, vol.7
, pp. 2735-2740
-
-
Goschke, R.1
Cohen, N.C.2
Wood, J.M.3
Maibaum, J.4
-
95
-
-
17144451277
-
-
Dolle, R.E.; Prasad, C.V.C.; Prouty, C.P.; Salvino, J.M.; Awad, M.M.A.; Schmidt, S.J.; Hoyer, D.; Ross, T.M.; Graybill, T.L.; Speier, G.J. Pyridazinodiazepines as a high-affinity, P2-P3 peptidomimetic class of interleukin-1 beta-converting enzyme inhibitor. J. Med. Chem., 1997, 40, 1941-l 946.
-
Dolle, R.E.; Prasad, C.V.C.; Prouty, C.P.; Salvino, J.M.; Awad, M.M.A.; Schmidt, S.J.; Hoyer, D.; Ross, T.M.; Graybill, T.L.; Speier, G.J. Pyridazinodiazepines as a high-affinity, P2-P3 peptidomimetic class of interleukin-1 beta-converting enzyme inhibitor. J. Med. Chem., 1997, 40, 1941-l 946.
-
-
-
-
96
-
-
0030598676
-
-
McKittrick, B.A.; Stamford, A.W.; Weng, X.; Ma, K.; Chackalamannil, S.; Czarniecki, M.; Cleven, R.M.; Fawzi, A.B. Design and synthesis of phosphinic acids that triply inhibit endothelin converting enzyme, angiotensin converting enzyme and neutral endopeptidase 24.11. Bioorg. Med. Chem. Lett., 1996, 6, 1629-l 634.
-
McKittrick, B.A.; Stamford, A.W.; Weng, X.; Ma, K.; Chackalamannil, S.; Czarniecki, M.; Cleven, R.M.; Fawzi, A.B. Design and synthesis of phosphinic acids that triply inhibit endothelin converting enzyme, angiotensin converting enzyme and neutral endopeptidase 24.11. Bioorg. Med. Chem. Lett., 1996, 6, 1629-l 634.
-
-
-
-
97
-
-
0031552096
-
Replacements for lysine in L-seryl-L-lysyl dipeptide amide inhibitors of candida albicans myristoyl-CoA:protein N-myristoyltransferase
-
Brown, D.L.; Devadas, B.; Lu, H.F.; Nagarajan, S.; Zupec, M.E.; Freeman, S.K.; McWherter, C.A.; Getman, D.P.; Sikorski, J.A. Replacements for lysine in L-seryl-L-lysyl dipeptide amide inhibitors of candida albicans myristoyl-CoA:protein N-myristoyltransferase. Bioorg. Med. Chem. Lett., 1997, 7, 379-382.
-
(1997)
Bioorg. Med. Chem. Lett
, vol.7
, pp. 379-382
-
-
Brown, D.L.1
Devadas, B.2
Lu, H.F.3
Nagarajan, S.4
Zupec, M.E.5
Freeman, S.K.6
McWherter, C.A.7
Getman, D.P.8
Sikorski, J.A.9
-
98
-
-
9444264701
-
Neuropeptide Y and the nonpeptide antagonist BIBP 3226 share an overlapping binding site at the human Y1 receptor
-
Saute, M.; Rudolf, K.; Wittneben, H.; Herzog, H.; Martinez, R.; Munoz, M.; Eberlein, W.; Engel, W.; Walker, P.; Beck-Sickinger, A.G. Neuropeptide Y and the nonpeptide antagonist BIBP 3226 share an overlapping binding site at the human Y1 receptor. Pharmacology, 1996, 50, 285-292.
-
(1996)
Pharmacology
, vol.50
, pp. 285-292
-
-
Saute, M.1
Rudolf, K.2
Wittneben, H.3
Herzog, H.4
Martinez, R.5
Munoz, M.6
Eberlein, W.7
Engel, W.8
Walker, P.9
Beck-Sickinger, A.G.10
-
99
-
-
0032864224
-
Synthesis of conformationally restricted mimetics of gamma-turns and incorporation into desmopressin, an analogue of the peptide hormone vasopressin
-
Brickmann, K.; Yuan, Z.; Sethson, I.; Somfai, P.; Kihlberg, J. Synthesis of conformationally restricted mimetics of gamma-turns and incorporation into desmopressin, an analogue of the peptide hormone vasopressin. Chem. Eur. J., 1999, 5, 2241-2253.
-
(1999)
Chem. Eur. J
, vol.5
, pp. 2241-2253
-
-
Brickmann, K.1
Yuan, Z.2
Sethson, I.3
Somfai, P.4
Kihlberg, J.5
-
100
-
-
0037030644
-
Synthesis and pharmacological evaluation of an analogue of the peptide hormone oxytocin that contains a mimetic of an inverse gamma-turn
-
Yuan, Z.; Blomberg, D.; Sethson, I.; Brickmann, K.; Ekholm, K.; Johansson, B.; Nilsson, A.; Kihlberg, J. Synthesis and pharmacological evaluation of an analogue of the peptide hormone oxytocin that contains a mimetic of an inverse gamma-turn. J. Med. Chem., 2002, 45, 2512-2519.
-
(2002)
J. Med. Chem
, vol.45
, pp. 2512-2519
-
-
Yuan, Z.1
Blomberg, D.2
Sethson, I.3
Brickmann, K.4
Ekholm, K.5
Johansson, B.6
Nilsson, A.7
Kihlberg, J.8
-
101
-
-
18144419714
-
Synthesis of a β-turn mimetic suitable for incorporation in the peptide hormone LHRH
-
Yuan, Z.; Kihlberg, J. Synthesis of a β-turn mimetic suitable for incorporation in the peptide hormone LHRH. Tetrahedron, 2005, 61, 4901-4909.
-
(2005)
Tetrahedron
, vol.61
, pp. 4901-4909
-
-
Yuan, Z.1
Kihlberg, J.2
-
102
-
-
0033869114
-
Comparison of three γ-turn mimetic scaffolds incorporated into angiotensin II
-
Lindman, S.; Lindeberg, G.; Nyberg, F.; Karlén, A.; Hallberg, A. Comparison of three γ-turn mimetic scaffolds incorporated into angiotensin II. Bioorg. Med. Chem., 2000, 8, 2375-2383.
-
(2000)
Bioorg. Med. Chem
, vol.8
, pp. 2375-2383
-
-
Lindman, S.1
Lindeberg, G.2
Nyberg, F.3
Karlén, A.4
Hallberg, A.5
-
103
-
-
0029084673
-
Macrocyclic peptidomimetics-forcing peptides into bioactive conformations
-
Fairlie, D.P.; Abbenante, G.; March, D.R. Macrocyclic peptidomimetics-forcing peptides into bioactive conformations. Curr. Med. Chem., 1995, 2, 654-686.
-
(1995)
Curr. Med. Chem
, vol.2
, pp. 654-686
-
-
Fairlie, D.P.1
Abbenante, G.2
March, D.R.3
-
104
-
-
0030768259
-
-
Hanessian, S.; McNaughton-Smith, G.; Lombart, H.G.; Lubell, W.D. Design and Synthesis of Conformationally Constrained Amino Acids as Versatile Scaffolds and Peptide Mimetics. Tetrahedron, 1997, 53, 12789-l 2854.
-
Hanessian, S.; McNaughton-Smith, G.; Lombart, H.G.; Lubell, W.D. Design and Synthesis of Conformationally Constrained Amino Acids as Versatile Scaffolds and Peptide Mimetics. Tetrahedron, 1997, 53, 12789-l 2854.
-
-
-
-
105
-
-
0032478055
-
Nonpeptide glycoprotein IIb/IIIa inhibitors: Substituted quinazolinediones and quinazolinones as potent fibrinogen receptor antagonists
-
Liverton, N.J.; Armstrong, D.J; Claremon, D.A; Remy, D.C.; Baldwin, J.J.; Lynch, R.J.; Zhang, G.; Gould, R.J. Nonpeptide glycoprotein IIb/IIIa inhibitors: substituted quinazolinediones and quinazolinones as potent fibrinogen receptor antagonists. Bioorg. Med. Chem. Lett., 1998, 8, 483-486.
-
(1998)
Bioorg. Med. Chem. Lett
, vol.8
, pp. 483-486
-
-
Liverton, N.J.1
Armstrong, D.J.2
Claremon, D.A.3
Remy, D.C.4
Baldwin, J.J.5
Lynch, R.J.6
Zhang, G.7
Gould, R.J.8
-
106
-
-
0141869940
-
Clinically validated peptides as templates for de novo peptidomimetic drug design at G-protein-coupled receptors
-
Jones, M.R; Boatman, P.D; Semple, G.; Shin, Y.; Tamura, Y.S. Clinically validated peptides as templates for de novo peptidomimetic drug design at G-protein-coupled receptors. J. Curr. Opin. Pharmacol., 2003, 3, 530-543.
-
(2003)
J. Curr. Opin. Pharmacol
, vol.3
, pp. 530-543
-
-
Jones, M.R.1
Boatman, P.D.2
Semple, G.3
Shin, Y.4
Tamura, Y.S.5
-
107
-
-
0030764541
-
Approaches to the Synthesis of Ureapeptoid. Peptidomimetics
-
Kruijtzer, J.A.W.; Lefeber, D.J.; Liskamp, R.M.J. Approaches to the Synthesis of Ureapeptoid. Peptidomimetics. Tetrahedron Lett., 1997, 38 (30), 5335-5338,
-
(1997)
Tetrahedron Lett
, vol.38
, Issue.30
, pp. 5335-5338
-
-
Kruijtzer, J.A.W.1
Lefeber, D.J.2
Liskamp, R.M.J.3
-
108
-
-
73549105142
-
Combinatorial Chemistry Online
-
Terrett, N.K. Combinatorial Chemistry Online. J. Comb. Chem., 2008, 10 (8), 31-34.
-
(2008)
J. Comb. Chem
, vol.10
, Issue.8
, pp. 31-34
-
-
Terrett, N.K.1
-
109
-
-
0030943416
-
Solid Phase Syntheses of Oligoureas
-
Burgess, K.; Ibarzo, J.; Linthicum, D. S.; Russell, D. H.; Shin, H.; Shitangkoon, A.; Totani, R.; Zhang, A. J. Solid Phase Syntheses of Oligoureas. J. Am. Chem. Soc, 1997, 119, 1556- 1564
-
(1997)
J. Am. Chem. Soc
, vol.119
, pp. 1556-1564
-
-
Burgess, K.1
Ibarzo, J.2
Linthicum, D.S.3
Russell, D.H.4
Shin, H.5
Shitangkoon, A.6
Totani, R.7
Zhang, A.J.8
-
110
-
-
0029988589
-
-
Han, H.; Janda, K. D. Azatides: Solution and Liquid Phase Syntheses of a New Peptidomimetic. J. Am. Chem. Soc, 1996, 118, 2539-2544.
-
Han, H.; Janda, K. D. Azatides: Solution and Liquid Phase Syntheses of a New Peptidomimetic. J. Am. Chem. Soc, 1996, 118, 2539-2544.
-
-
-
-
111
-
-
0035496146
-
On the Antimicrobial and Hemolytic Activities of Amphiphilic beta-peptides
-
Arvidsson, P.I.; Frackenpohl, J.; Ryder, N.S.; Liechty, B.; Petersen, F.; Zimmermann, H.; Camenisch, G.P.; Woessner, R.; Seebach, D. On the Antimicrobial and Hemolytic Activities of Amphiphilic beta-peptides. ChemBiochem., 2001, 2, 771-773.
-
(2001)
ChemBiochem
, vol.2
, pp. 771-773
-
-
Arvidsson, P.I.1
Frackenpohl, J.2
Ryder, N.S.3
Liechty, B.4
Petersen, F.5
Zimmermann, H.6
Camenisch, G.P.7
Woessner, R.8
Seebach, D.9
-
112
-
-
0030967686
-
A second-generation synthesis of scalemic 3,5,5-trisubstituted pyrrolin-4-ones: Incorporation of functionalized amino acid side-chains
-
Smith, A. B.; Benowitz, A. B.; Favor, D. A.; Sprengeler, P. A.; Hirschmann, R. A second-generation synthesis of scalemic 3,5,5-trisubstituted pyrrolin-4-ones: Incorporation of functionalized amino acid side-chains. Tetrahedron Lett., 1997,38, 3809-3812.
-
(1997)
Tetrahedron Lett
, vol.38
, pp. 3809-3812
-
-
Smith, A.B.1
Benowitz, A.B.2
Favor, D.A.3
Sprengeler, P.A.4
Hirschmann, R.5
-
113
-
-
0029953649
-
Molecular diversity of peptidomimetics: Approaches to the solid-phase synthesis of peptidosulfonamides
-
Bont, D. B. A.; Moree, W. J.; Liskamp, R. M. Molecular diversity of peptidomimetics: Approaches to the solid-phase synthesis of peptidosulfonamides . J. Bioorg. Med. Chem., 1996, 4, 667-672.
-
(1996)
J. Bioorg. Med. Chem
, vol.4
, pp. 667-672
-
-
Bont, D.B.A.1
Moree, W.J.2
Liskamp, R.M.3
-
114
-
-
0031561062
-
HIV-1 TAR RNA Recognition by an Unnatural Biopolymer
-
Wang, X.; Huq, I.; Rana, T. M. HIV-1 TAR RNA Recognition by an Unnatural Biopolymer. J. Am. Chem. Soc., 1997, 119, 6444-6445.
-
(1997)
J. Am. Chem. Soc
, vol.119
, pp. 6444-6445
-
-
Wang, X.1
Huq, I.2
Rana, T.M.3
-
115
-
-
0030810207
-
Synthesis of Diverse Ethoxyformacetal Oligomers. Toward Libraries of Metal-Coordinating Unnatural Biopolymers
-
Hall, D. G.; Schultz, P. G. Synthesis of Diverse Ethoxyformacetal Oligomers. Toward Libraries of Metal-Coordinating Unnatural Biopolymers. Tetrahedron Lett., 1997, 38, 7825-7529.
-
(1997)
Tetrahedron Lett
, vol.38
, pp. 7825-7529
-
-
Hall, D.G.1
Schultz, P.G.2
-
116
-
-
33746888689
-
Mimicking helical antibacterial peptides with nonpeptidic folding oligomers
-
Violette, A.; Fournel, S.; Lamour, L.; Chaloin, O.; Frisch, B.; Briand, J.; Monteil, H.; Guichard, G. Mimicking helical antibacterial peptides with nonpeptidic folding oligomers. J. Chem. Biol., 2006, 13, 531-538.
-
(2006)
J. Chem. Biol
, vol.13
, pp. 531-538
-
-
Violette, A.1
Fournel, S.2
Lamour, L.3
Chaloin, O.4
Frisch, B.5
Briand, J.6
Monteil, H.7
Guichard, G.8
-
117
-
-
25444476499
-
Inhibiting HIV fusion with a β-peptide foldamer
-
Stephens, O.M.; Kim, S.; Welch, B.D.; Hodsdon, M.E.; Kay, M.S.; Schepartz, A. Inhibiting HIV fusion with a β-peptide foldamer. J. Am. Chem. Soc., 2005, 127, 13126-13127.
-
(2005)
J. Am. Chem. Soc
, vol.127
, pp. 13126-13127
-
-
Stephens, O.M.1
Kim, S.2
Welch, B.D.3
Hodsdon, M.E.4
Kay, M.S.5
Schepartz, A.6
-
118
-
-
9644273958
-
-
Kritzer, J.A.; Stephens, O.M.; Guarracino, D.A.; Reznik, S.K.; Schepartz, A. beta-peptides as inhibitors of protein-protein interactions. Bioorg. Med. Chem., 2005, 13, 11-16.
-
Kritzer, J.A.; Stephens, O.M.; Guarracino, D.A.; Reznik, S.K.; Schepartz, A. beta-peptides as inhibitors of protein-protein interactions. Bioorg. Med. Chem., 2005, 13, 11-16.
-
-
-
-
119
-
-
3543098742
-
Helical ßpeptide inhibitors of the p53-hDM2 interaction
-
Kritzer, J.A.; Lear, J.D.; Hodsdon, M.E.; Schepartz, A. Helical ßpeptide inhibitors of the p53-hDM2 interaction. Chem. Soc., 2004, 126, 9468-9469.
-
(2004)
Chem. Soc
, vol.126
, pp. 9468-9469
-
-
Kritzer, J.A.1
Lear, J.D.2
Hodsdon, M.E.3
Schepartz, A.4
-
120
-
-
15444348427
-
Identification and initial structure-activity relationships of a novel class of nonpeptide inhibitors of blood coagulation factor Xa
-
Klein, S.I.; Czekaj, M.; Gardner, C.J.; Guertin, K.R.; Cheney, D.L.; Spada, A.P.; Bolton, S.A.; Brown, K.; Colussi, D.; Heran, C.L. Identification and initial structure-activity relationships of a novel class of nonpeptide inhibitors of blood coagulation factor Xa. J. Med. Chem., 1998, 41, 437-450.
-
(1998)
J. Med. Chem
, vol.41
, pp. 437-450
-
-
Klein, S.I.1
Czekaj, M.2
Gardner, C.J.3
Guertin, K.R.4
Cheney, D.L.5
Spada, A.P.6
Bolton, S.A.7
Brown, K.8
Colussi, D.9
Heran, C.L.10
-
121
-
-
73549103512
-
-
Las Vegas. Washington, DC: American Chemical Society;
-
Sall, D.J.; Bastian, J.A.; Briggs, S.L.; Buben, J.A.; Chirgadze, N.Y.; Clawson, D.K.; Denney, M.L.; Gierra, D.D.; Gifford-Moore, D.S.; Harper, R.W. Book of Abstracts. 214th American Chemical Society National Meeting: 1997 Sept 7-11: Las Vegas. Washington, DC: American Chemical Society; 1997:A58.
-
(1997)
Book of Abstracts. 214th American Chemical Society National Meeting: 1997 Sept 7-11
-
-
Sall, D.J.1
Bastian, J.A.2
Briggs, S.L.3
Buben, J.A.4
Chirgadze, N.Y.5
Clawson, D.K.6
Denney, M.L.7
Gierra, D.D.8
Gifford-Moore, D.S.9
Harper, R.W.10
-
122
-
-
0030835791
-
-
Chirgadze, N.Y.; Sal, D.J.; Klimkowski, V.J.; Clawson, D,K.; Briggs, S.L.; Hermann, R.; Smith, G.F.; Gifford-Moore, D.S.; Werv, J.P. The crystal structure of human alpha-thrombin complexed with LY178550, a nonpeptidyl, active site-directed inhibitor. Protein Sci., 1997, 6, 1412-l 417.
-
Chirgadze, N.Y.; Sal, D.J.; Klimkowski, V.J.; Clawson, D,K.; Briggs, S.L.; Hermann, R.; Smith, G.F.; Gifford-Moore, D.S.; Werv, J.P. The crystal structure of human alpha-thrombin complexed with LY178550, a nonpeptidyl, active site-directed inhibitor. Protein Sci., 1997, 6, 1412-l 417.
-
-
-
-
123
-
-
0030034763
-
Potent cell active not-thiol tetrapeptide inhibitors of Farnesyl transferase
-
Hunt ,J.T.; Lee, V.G.; Leftheris, K.; Seizinaer, B.; Carboni, J.; Mabus, J.; Ricca, A.; Yan, N.; Manne V. Potent cell active not-thiol tetrapeptide inhibitors of Farnesyl transferase. J. Med. Chem., 1996, 39, 353-358.
-
(1996)
J. Med. Chem
, vol.39
, pp. 353-358
-
-
Hunt, J.T.1
Lee, V.G.2
Leftheris, K.3
Seizinaer, B.4
Carboni, J.5
Mabus, J.6
Ricca, A.7
Yan, N.8
Manne, V.9
-
124
-
-
18544398961
-
-
Nioroae, F.G.; Doll, R.J.; Vibulbhan, B.; Alvarez, C.S.; Bishoo, W.R.; Pktrin, J.; Kirschmeier, P.; Carruthers, N.I.; Wong, J. Discovery of Novel Nonpeptide Tricyclic Inhibitors of Ras Farnesyl Protein Transferase. Bioorg. Med. Chem., 1997, 5, 101-l 13.
-
Nioroae, F.G.; Doll, R.J.; Vibulbhan, B.; Alvarez, C.S.; Bishoo, W.R.; Pktrin, J.; Kirschmeier, P.; Carruthers, N.I.; Wong, J. Discovery of Novel Nonpeptide Tricyclic Inhibitors of Ras Farnesyl Protein Transferase. Bioorg. Med. Chem., 1997, 5, 101-l 13.
-
-
-
-
125
-
-
0029586503
-
Novel tricyclic inhibitors of farnesyl protein transferase. Biochemical characterization and inhibition of Ras modification in transfected Cos cells
-
l-30618
-
Bishop, W.R.; Bond, R.; Petrin, J.; Wang, L.; Patton, R.; Doll, R.; Njoroge, G.; Catino, J.; Schwartz, J.; Windsor, W. Novel tricyclic inhibitors of farnesyl protein transferase. Biochemical characterization and inhibition of Ras modification in transfected Cos cells. J. Biol. Chem., 1995, 270, 3061 l-30618.
-
(1995)
J. Biol. Chem
, vol.270
, pp. 3061
-
-
Bishop, W.R.1
Bond, R.2
Petrin, J.3
Wang, L.4
Patton, R.5
Doll, R.6
Njoroge, G.7
Catino, J.8
Schwartz, J.9
Windsor, W.10
-
126
-
-
0032478160
-
Solid-phase synthesis of peptidomimetic oligomers with a phosphodiester backbone
-
Lin, P.; Ganesan, A. Solid-phase synthesis of peptidomimetic oligomers with a phosphodiester backbone. Bioorg. Med. Chem. Lett., 1998, 8, 511-514.
-
(1998)
Bioorg. Med. Chem. Lett
, vol.8
, pp. 511-514
-
-
Lin, P.1
Ganesan, A.2
-
127
-
-
17344384874
-
Non-haemolytic beta-amino-acid oligomers
-
Porter, E.A.; Wang, X.; Lee, H.S.; Weisblum, B.; Gellman, S.H. Non-haemolytic beta-amino-acid oligomers. Nature, 2000, 404 (6778), 565.
-
(2000)
Nature
, vol.404
, Issue.6778
, pp. 565
-
-
Porter, E.A.1
Wang, X.2
Lee, H.S.3
Weisblum, B.4
Gellman, S.H.5
-
128
-
-
0037178109
-
Mimicry of hostdefense peptides by unnatural oligomers: Antimicrobial betapeptides
-
Porter, E.A.; Weisblum, B.; Gellman, S.H. Mimicry of hostdefense peptides by unnatural oligomers: antimicrobial betapeptides. J. Am. Chem. Soc., 2002, 124, 7324-7330.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 7324-7330
-
-
Porter, E.A.1
Weisblum, B.2
Gellman, S.H.3
-
129
-
-
0037202210
-
Structureactivity studies of 14-helical antimicrobial beta-peptides: Probing the relationship between conformational stability and antimicrobial potency
-
Raguse, T.L.; Porter, E.A.; Weisblum, B.; Gellman, S.H. Structureactivity studies of 14-helical antimicrobial beta-peptides: probing the relationship between conformational stability and antimicrobial potency. J. Am. Chem. Soc., 2002, 124, 12774-12785.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 12774-12785
-
-
Raguse, T.L.1
Porter, E.A.2
Weisblum, B.3
Gellman, S.H.4
-
130
-
-
58149190056
-
Lipid domains in bacterial membranes and the action of antimicrobial agents
-
Epand, R.M.; Epand, R.F. Lipid domains in bacterial membranes and the action of antimicrobial agents. BBA-Biomembranes, 2009, 1788 (1), 289-294.
-
(2009)
BBA-Biomembranes
, vol.1788
, Issue.1
, pp. 289-294
-
-
Epand, R.M.1
Epand, R.F.2
-
131
-
-
0347417960
-
Antibiotic and hemolytic activity of a beta2/beta3 peptide capable of folding into a 12/10-helical secondary structure
-
Arvidsson, P.I.; Ryder, N.S.; Weiss, H.M.; Gross, G.; Kretz, O., Woessner, R.; Seebach, D. Antibiotic and hemolytic activity of a beta2/beta3 peptide capable of folding into a 12/10-helical secondary structure. ChemBioChem., 2003, 4, 1345-1347.
-
(2003)
ChemBioChem
, vol.4
, pp. 1345-1347
-
-
Arvidsson, P.I.1
Ryder, N.S.2
Weiss, H.M.3
Gross, G.4
Kretz, O.5
Woessner, R.6
Seebach, D.7
-
132
-
-
0141888597
-
Helical peptoid mimics of magainin-2 amide
-
Patch, J.A.; Barron, A.E. Helical peptoid mimics of magainin-2 amide. J. Am. Chem. Soc., 2003, 125, 12092-12093.
-
(2003)
J. Am. Chem. Soc
, vol.125
, pp. 12092-12093
-
-
Patch, J.A.1
Barron, A.E.2
-
133
-
-
34447278135
-
Infectious disease: Connecting innate immunity to biocidal polymers
-
Gabriel, J.G.; Som, A.; Madkour, E.A.; Eren, T.; Tew, N.T. Infectious disease: Connecting innate immunity to biocidal polymers. Mater. Sci. Eng., 2007, 57, 28-64.
-
(2007)
Mater. Sci. Eng
, vol.57
, pp. 28-64
-
-
Gabriel, J.G.1
Som, A.2
Madkour, E.A.3
Eren, T.4
Tew, N.T.5
-
134
-
-
0035471135
-
-
Cheng, R.P.; Gellman, S.H.; DeGrado, W.F. beta-Peptides: from structure to function. Chem. Rev., 2001, 101, 3219-3232.
-
Cheng, R.P.; Gellman, S.H.; DeGrado, W.F. beta-Peptides: from structure to function. Chem. Rev., 2001, 101, 3219-3232.
-
-
-
-
135
-
-
0347417960
-
-
Arvidsson, P.I,; Ryder, Neil.S,; Weiss, H.M,; Gross, G,; Kretz, O,; Woessner, R,; Seebach, D. Antibiotic and hemolytic activity of a beta2/beta3 peptide capable of folding into a 12/10-helical secondary structure. ChemBioChem, 2003, 4 (12), 1345-1347.
-
Arvidsson, P.I,; Ryder, Neil.S,; Weiss, H.M,; Gross, G,; Kretz, O,; Woessner, R,; Seebach, D. Antibiotic and hemolytic activity of a beta2/beta3 peptide capable of folding into a 12/10-helical secondary structure. ChemBioChem, 2003, 4 (12), 1345-1347.
-
-
-
-
136
-
-
0030995823
-
Residue-based control of helix shape in β-peptide oligomers
-
Appella, D.H.; Christianson, L.A.; Klein, D.A.; Powell, D.R.; Huang, X.; Joseph, J.; Barchi, J.; Gellman, S.H. Residue-based control of helix shape in β-peptide oligomers. Nature, 1997, 387, 381-384.
-
(1997)
Nature
, vol.387
, pp. 381-384
-
-
Appella, D.H.1
Christianson, L.A.2
Klein, D.A.3
Powell, D.R.4
Huang, X.5
Joseph, J.6
Barchi, J.7
Gellman, S.H.8
-
137
-
-
0000088927
-
The twists and turns of beta-peptides
-
DeGrado, W.F,; Schneider, J.P,; Hamuro, Y . The twists and turns of beta-peptides. J. Pept. Res., 1999, 54 (3), 206-217.
-
(1999)
J. Pept. Res
, vol.54
, Issue.3
, pp. 206-217
-
-
DeGrado, W.F.1
Schneider, J.P.2
Hamuro, Y.3
-
138
-
-
0034802565
-
De novo design, synthesis, and characterization of antimicrobial beta-peptides
-
Liu, D.; DeGrado, W.F. De novo design, synthesis, and characterization of antimicrobial beta-peptides. J. Am. Chem. Soc., 2001, 123, 7553-7559.
-
(2001)
J. Am. Chem. Soc
, vol.123
, pp. 7553-7559
-
-
Liu, D.1
DeGrado, W.F.2
-
139
-
-
33748929145
-
Antimicrobial activity of an abiotic host defense peptide mimic
-
Tew, G.N.; Clements, D.; Tang, H.; Arnt, L.; Scott, R.W. Antimicrobial activity of an abiotic host defense peptide mimic. Biochim. Biophys. Acta Biomembr., 2006, 1758, 1387-1392.
-
(2006)
Biochim. Biophys. Acta Biomembr
, vol.1758
, pp. 1387-1392
-
-
Tew, G.N.1
Clements, D.2
Tang, H.3
Arnt, L.4
Scott, R.W.5
-
140
-
-
0030785114
-
β-Peptides: A surprise at every turn
-
Seebach, D.; Matthews, J. L. β-Peptides: a surprise at every turn. Chem. Commun., 1997, 1, 2015-2022.
-
(1997)
Chem. Commun
, vol.1
, pp. 2015-2022
-
-
Seebach, D.1
Matthews, J.L.2
-
141
-
-
0037134881
-
Tolerance of acyclic residues in the beta-peptide 12-helix: Access to diverse side-chain arrays for biological applications
-
LePlae, P.R.; Fisk, J.D.; Porter, E.A.; Weisblum, B.; Gellman, S.H. Tolerance of acyclic residues in the beta-peptide 12-helix: access to diverse side-chain arrays for biological applications. J. Am. Chem. Soc., 2002, 124, 6820-6821.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 6820-6821
-
-
LePlae, P.R.1
Fisk, J.D.2
Porter, E.A.3
Weisblum, B.4
Gellman, S.H.5
-
142
-
-
0344928208
-
Helical Peptoid Mimics of Lung Surfactant Protein C
-
Wu, C.W.; Seurynck, S.L.; Lee, K.Y.C.; Barron, A.E. Helical Peptoid Mimics of Lung Surfactant Protein C. J. Chembiol., 2003, 10, 1057-1063.
-
(2003)
J. Chembiol
, vol.10
, pp. 1057-1063
-
-
Wu, C.W.1
Seurynck, S.L.2
Lee, K.Y.C.3
Barron, A.E.4
-
143
-
-
0029059507
-
Comparison of the proteolytic susceptibilities of homologous L-amino acid, D-amino acid, and N-substituted glycine peptide andpeptoid oligomers
-
Miller, S.M.; Simon, R.J.; Ng, S.; Zuckermann, R.N.; Kerr, J.M.; Moos, W.H. Comparison of the proteolytic susceptibilities of homologous L-amino acid, D-amino acid, and N-substituted glycine peptide andpeptoid oligomers. Drug Dev. Res., 1995, 35, 20-32.
-
(1995)
Drug Dev. Res
, vol.35
, pp. 20-32
-
-
Miller, S.M.1
Simon, R.J.2
Ng, S.3
Zuckermann, R.N.4
Kerr, J.M.5
Moos, W.H.6
-
144
-
-
0030424369
-
Pharmacologic characterization of CHIR 2279, an N-substituted glycine peptoid with high-affinity binding for alpha 1-adrenoceptors
-
Gibbons, J.A.; Hancock, A.A.; Vitt, C.R.; Knepper; S.; Buckner, S.A.; Brune, M.E.; Milicic, I.; Kerwin, J.F.; Richter, L.S.; Taylor, E.W., Spear, K.L.; Zuckermann, R.N.; Spellmeyer, D.C.; Braeckman, R.A.; Moos, W.H. Pharmacologic characterization of CHIR 2279, an N-substituted glycine peptoid with high-affinity binding for alpha 1-adrenoceptors. J. Pharmacol. Exp. Ther., 1996, 277, 885-899.
-
(1996)
J. Pharmacol. Exp. Ther
, vol.277
, pp. 885-899
-
-
Gibbons, J.A.1
Hancock, A.A.2
Vitt, C.R.3
Knepper, S.4
Buckner, S.A.5
Brune, M.E.6
Milicic, I.7
Kerwin, J.F.8
Richter, L.S.9
Taylor, E.W.10
Spear, K.L.11
Zuckermann, R.N.12
Spellmeyer, D.C.13
Braeckman, R.A.14
Moos, W.H.15
-
145
-
-
0034822676
-
Peptoid oligomers with alpha-chiral, aromatic side chains: Effects of chain length on secondary structure
-
Wu, C.W.; Sanborn, T.J.; Zuckermann, R.N.; Barron, A.E. Peptoid oligomers with alpha-chiral, aromatic side chains: effects of chain length on secondary structure. J. Am. Chem. Soc., 2001, 123, 2958-2963.
-
(2001)
J. Am. Chem. Soc
, vol.123
, pp. 2958-2963
-
-
Wu, C.W.1
Sanborn, T.J.2
Zuckermann, R.N.3
Barron, A.E.4
-
146
-
-
0032515982
-
-
Kirshenbaum, K.; Barron, A.E.; Armand, P.; Goldsmith, R.; Bradley, E.; Cohen, F.E.; Dill, K.A.; Zuckermann, R.N. Sequencespecific polypeptoids: a diverse family of heteropolymers with stable secondary structure. Proc. Natl. Acad. Sci., 1998, 95, 4303-4308.
-
Kirshenbaum, K.; Barron, A.E.; Armand, P.; Goldsmith, R.; Bradley, E.; Cohen, F.E.; Dill, K.A.; Zuckermann, R.N. Sequencespecific polypeptoids: a diverse family of heteropolymers with stable secondary structure. Proc. Natl. Acad. Sci., 1998, 95, 4303-4308.
-
-
-
-
147
-
-
31344472510
-
Antimicrobial β-peptoids by a block synthesis approach
-
Shuey, S.W.; Delaney, W.J.; Shah, M.C.; Scialdone, M.A. Antimicrobial β-peptoids by a block synthesis approach. Bioorg. Med. Chem. Lett., 2006, 16 (5), 1245-1248.
-
(2006)
Bioorg. Med. Chem. Lett
, vol.16
, Issue.5
, pp. 1245-1248
-
-
Shuey, S.W.1
Delaney, W.J.2
Shah, M.C.3
Scialdone, M.A.4
-
148
-
-
0032705431
-
Bioinspired polymeric materials: In-between proteins and plastics
-
Barron, A.E.; Zuckermann, R.N. Bioinspired polymeric materials: in-between proteins and plastics. Curr. Opin. Chem. Biol., 1999, 3, 681-687.
-
(1999)
Curr. Opin. Chem. Biol
, vol.3
, pp. 681-687
-
-
Barron, A.E.1
Zuckermann, R.N.2
-
149
-
-
0034700141
-
The design, synthesis, and evaluation of molecules that enable or enhance cellular uptake: Peptoid molecular transporters
-
Wender, P.A.; Mitchell, D.J.; Pattabiraman, K.; Pelkey, E.T.; Steinman, L.; Rothbard, J.B. The design, synthesis, and evaluation of molecules that enable or enhance cellular uptake: peptoid molecular transporters. Proc. Natl. Acad. Sci., 2000, 97, 13003-13008.
-
(2000)
Proc. Natl. Acad. Sci
, vol.97
, pp. 13003-13008
-
-
Wender, P.A.1
Mitchell, D.J.2
Pattabiraman, K.3
Pelkey, E.T.4
Steinman, L.5
Rothbard, J.B.6
-
150
-
-
0000908874
-
Efficient Method for the Preparation of Peptoids [Oligo(N-substituted glycines)] by Submonomer Solid-Phase Synthesis
-
Zuckermann, R.N.; Kerr, J.M.; Kent, S.B.H.; Moos, W.H. Efficient Method for the Preparation of Peptoids [Oligo(N-substituted glycines)] by Submonomer Solid-Phase Synthesis.J. Am. Chem. Soc., 1992, 114, 10646-10647.
-
(1992)
J. Am. Chem. Soc
, vol.114
, pp. 10646-10647
-
-
Zuckermann, R.N.1
Kerr, J.M.2
Kent, S.B.H.3
Moos, W.H.4
-
151
-
-
20444366611
-
New peptidomimetic polymers for antifouling surfaces
-
Statz, A.R.; Meagher, R.J.; Barron, A.E.; Messersmith, P.B. New peptidomimetic polymers for antifouling surfaces. J. Am. Chem. Soc., 2005, 127, 7972-7973.
-
(2005)
J. Am. Chem. Soc
, vol.127
, pp. 7972-7973
-
-
Statz, A.R.1
Meagher, R.J.2
Barron, A.E.3
Messersmith, P.B.4
-
152
-
-
0033863173
-
Combinatorial libraries: A tool to design antimicrobial and antifungal peptide analogues having lytic specificities for structure-activity relationship studies
-
Blondelle, S.E.; Lohner, K. Combinatorial libraries: a tool to design antimicrobial and antifungal peptide analogues having lytic specificities for structure-activity relationship studies. Bio. Polymers, 2000, 55, 74-87.
-
(2000)
Bio. Polymers
, vol.55
, pp. 74-87
-
-
Blondelle, S.E.1
Lohner, K.2
-
153
-
-
0037014049
-
Stable helical secondary structure in short chain N,N'-linked oligoreas bearing proteinogenic side chain
-
Semetey, V.; Rognan, D.; Hemmerlin, C.; Graff, R., Briand; J.P.; Marraud, M.; Guichard, G. Stable helical secondary structure in short chain N,N'-linked oligoreas bearing proteinogenic side chain. Angew. Chem. Int. Ed. Engl., 2002, 41, 1893-1895.
-
(2002)
Angew. Chem. Int. Ed. Engl
, vol.41
, pp. 1893-1895
-
-
Semetey, V.1
Rognan, D.2
Hemmerlin, C.3
Graff, R.4
Briand, J.P.5
Marraud, M.6
Guichard, G.7
-
154
-
-
0036944713
-
Helix forming oligoureas: Temperaturedependent NMR, structure determination and circular dichroism of a nonomer with functionalised side chain
-
Hemmerlin, C.; Marraud, M.; Rognan, D.; Graff, R.; Semetey, V.; Briand; J.P.; Guichard, G. Helix forming oligoureas: temperaturedependent NMR, structure determination and circular dichroism of a nonomer with functionalised side chain. Helv. Chim. Acta, 2002, 85, 3692-3711.
-
(2002)
Helv. Chim. Acta
, vol.85
, pp. 3692-3711
-
-
Hemmerlin, C.1
Marraud, M.2
Rognan, D.3
Graff, R.4
Semetey, V.5
Briand, J.P.6
Guichard, G.7
-
155
-
-
13944267446
-
N'-linked oligoureas as foldamers: Chain length requirements for helix formation in protic solvent investigated by circular dichroism, NMR spectroscopy, and molecular dynamics
-
Violette, A.; Averlant-Petit, M.C.; Semetey, V.; Hemmerlin, C.; Casimir, R.; Graff, R.; Marraud, M.; Briand, J.P.; Rognan, D.; Guichard, G. N,N'-linked oligoureas as foldamers: chain length requirements for helix formation in protic solvent investigated by circular dichroism, NMR spectroscopy, and molecular dynamics. J. Am. Chem. Soc., 2005, 127, 2156-2164.
-
(2005)
J. Am. Chem. Soc
, vol.127
, pp. 2156-2164
-
-
Violette, A.1
Averlant-Petit, M.C.2
Semetey, V.3
Hemmerlin, C.4
Casimir, R.5
Graff, R.6
Marraud, M.7
Briand, J.P.8
Rognan, D.9
Guichard, G.N.10
-
156
-
-
0346665667
-
3-residues with side-chain branching adjacent to the β-carbon atom
-
3-residues with side-chain branching adjacent to the β-carbon atom. Helv. Chim. Acta, 2002, 85, 4154-4164.
-
(2002)
Helv. Chim. Acta
, vol.85
, pp. 4154-4164
-
-
Raguse, T.L.1
Lai, J.R.2
Gellman, S.H.3
-
157
-
-
0036950531
-
Genomics-based approaches to gene discovery in innate immunity
-
Scheetz, T.; Bartlett, J.A.; Walters, J.D.; Schutte, B.C.; Casavant, T. L.; McCray, P. B. Genomics-based approaches to gene discovery in innate immunity. Immunol. Rev., 2002, 190, 137-145.
-
(2002)
Immunol. Rev
, vol.190
, pp. 137-145
-
-
Scheetz, T.1
Bartlett, J.A.2
Walters, J.D.3
Schutte, B.C.4
Casavant, T.L.5
McCray, P.B.6
-
158
-
-
0037012402
-
NMR conformational analysis of antide, a potent antagonist of the gonadotropin releasing hormone
-
Digilio, G; Bracco, C; Barbero, L; Chicco, D; Del Curto, MD; Esposito, P; Traversa, S; Aime, S. NMR conformational analysis of antide, a potent antagonist of the gonadotropin releasing hormone. J. Am. Chem. Soc., 2002, 124, 3431-3442.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 3431-3442
-
-
Digilio, G.1
Bracco, C.2
Barbero, L.3
Chicco, D.4
Del Curto, M.D.5
Esposito, P.6
Traversa, S.7
Aime, S.8
-
159
-
-
0032196592
-
Patenting computerdesigned peptides
-
Patel, S.; Stott, I.P.; Bhakoo, M.; Elliott, P. Patenting computerdesigned peptides. J. Comp. Aided. Mol. Des., 1998, 12: 543-556.
-
(1998)
J. Comp. Aided. Mol. Des
, vol.12
, pp. 543-556
-
-
Patel, S.1
Stott, I.P.2
Bhakoo, M.3
Elliott, P.4
-
160
-
-
0035954729
-
Antibacterial agents based on the cyclic D,L-alpha-peptide architecture
-
Lopez, S.F.; Kim, H.S.; Choi, E.C.; Delgado, M.; Granja, J.R.; Khasanov, A.; Kraehenbuehl, K.; Long, G.; Weinberger, D.A.; Wilcoxen, K.M.; Ghadiri, M.R. Antibacterial agents based on the cyclic D,L-alpha-peptide architecture. Nature, 2001, 412, 452-455.
-
(2001)
Nature
, vol.412
, pp. 452-455
-
-
Lopez, S.F.1
Kim, H.S.2
Choi, E.C.3
Delgado, M.4
Granja, J.R.5
Khasanov, A.6
Kraehenbuehl, K.7
Long, G.8
Weinberger, D.A.9
Wilcoxen, K.M.10
Ghadiri, M.R.11
-
161
-
-
60249090449
-
Evaluation of structural features of membrane acting antifungal peptides by artificial neural networks
-
Soltani, S.; Keymanesh K.; Sardari, S. Evaluation of structural features of membrane acting antifungal peptides by artificial neural networks. J. Biol. Sci., 2008, 8, 834-845.
-
(2008)
J. Biol. Sci
, vol.8
, pp. 834-845
-
-
Soltani, S.1
Keymanesh, K.2
Sardari, S.3
-
162
-
-
33847769895
-
-
Sardari, S.; Dezfulian, M. Cheminformatics in Anti-infective Agents Discovery. Mini Rev. Med. Chem., 2007, 7, 181-189.
-
Sardari, S.; Dezfulian, M. Cheminformatics in Anti-infective Agents Discovery. Mini Rev. Med. Chem., 2007, 7, 181-189.
-
-
-
-
163
-
-
33749680215
-
Sequence requirements and an optimization strategy for short antimicrobial peptides
-
Hilpert, K.; Elliott, R. M.; Volkmer, R.; Henklein, P.; Donini, O.; Zhou, Q.; Winkler, F.H.D.; Hancock, W.R.E. Sequence requirements and an optimization strategy for short antimicrobial peptides. Chem. Biol., 2006, 13, 1101-1107.
-
(2006)
Chem. Biol
, vol.13
, pp. 1101-1107
-
-
Hilpert, K.1
Elliott, R.M.2
Volkmer, R.3
Henklein, P.4
Donini, O.5
Zhou, Q.6
Winkler, F.H.D.7
Hancock, W.R.E.8
-
164
-
-
60249093776
-
QSAR modeling and computer-aided design of antimicrobial peptides
-
Jenssen, H.; Fjell, C.D.; Cherkasov, A.; Hancock, R.E. QSAR modeling and computer-aided design of antimicrobial peptides. J. Pept. Sci., 2007, 10, 1784-7019.
-
(2007)
J. Pept. Sci
, vol.10
, pp. 1784-7019
-
-
Jenssen, H.1
Fjell, C.D.2
Cherkasov, A.3
Hancock, R.E.4
-
165
-
-
34548132041
-
Analysis of protegrin structurefunction- activity relationships: The structural characteristics important for antimicrobial activity using smoothed amino acid sequence descriptors
-
Fernandez, M.; Caballero, J. Analysis of protegrin structurefunction- activity relationships: the structural characteristics important for antimicrobial activity using smoothed amino acid sequence descriptors. Mol. Simul., 2007, 33, 689-702.
-
(2007)
Mol. Simul
, vol.33
, pp. 689-702
-
-
Fernandez, M.1
Caballero, J.2
-
166
-
-
32044458173
-
SuperMimic - Fitting peptide mimetics into protein structures
-
Goede, A.; Michalsky, E.; Schmidt, U.; Preissner, R. SuperMimic - Fitting peptide mimetics into protein structures. BMC Bioinformatics, 2006, 7, 11.
-
(2006)
BMC Bioinformatics
, vol.7
, pp. 11
-
-
Goede, A.1
Michalsky, E.2
Schmidt, U.3
Preissner, R.4
-
167
-
-
34447506602
-
Design and biological evaluation of photo-switchable inhibitors
-
Fullbeck, M.; Michalsky, E.; Jaeger, I. S.; Henklein; P.; Kuhn, H.; Ruck-Braun, K.; Preissner, R. Design and biological evaluation of photo-switchable inhibitors. Genome Informatics, 2006, 17, 141-151.
-
(2006)
Genome Informatics
, vol.17
, pp. 141-151
-
-
Fullbeck, M.1
Michalsky, E.2
Jaeger, I.S.3
Henklein, P.4
Kuhn, H.5
Ruck-Braun, K.6
Preissner, R.7
-
168
-
-
0141869940
-
Clinically validated peptides as templates for de novo peptidomimetic drug design at G-protein-coupled receptors
-
Jones, R. M.; Boatman, D.; Semple, G.; Shin, Y. J.; Tamura, S. Y. Clinically validated peptides as templates for de novo peptidomimetic drug design at G-protein-coupled receptors. Cur. Opin. Pharmacol., 2003, 3, 530-543.
-
(2003)
Cur. Opin. Pharmacol
, vol.3
, pp. 530-543
-
-
Jones, R.M.1
Boatman, D.2
Semple, G.3
Shin, Y.J.4
Tamura, S.Y.5
-
169
-
-
11844249386
-
Relationship between side chain structure and 14-helix stability of beta-peptides in water
-
Kritzer, J.A.; Tirado-Rives, J.; Hart, S.A.; Lear, J.D.; Jorgensen, W.L.; Schepartz, A. Relationship between side chain structure and 14-helix stability of beta-peptides in water. J. Am. Chem. Soc., 2005, 127, 167-178.
-
(2005)
J. Am. Chem. Soc
, vol.127
, pp. 167-178
-
-
Kritzer, J.A.1
Tirado-Rives, J.2
Hart, S.A.3
Lear, J.D.4
Jorgensen, W.L.5
Schepartz, A.6
-
170
-
-
0034624823
-
Consensus bioactive conformation of cyclic GnRH antagonists defined by NMR and molecular modeling
-
Koerber, S.C.; Rizo, J.; Struthers, R.S.; Rivier, J.E. C. Consensus bioactive conformation of cyclic GnRH antagonists defined by NMR and molecular modeling. J. Med. Chem., 2000, 43, 819-828.
-
(2000)
J. Med. Chem
, vol.43
, pp. 819-828
-
-
Koerber, S.C.1
Rizo, J.2
Struthers, R.S.3
Rivier, J.E.C.4
-
171
-
-
0037012402
-
NMR conformational analysis of antide, a potent antagonist of the gonadotropin releasing hormone
-
Digilio, G.; Bracco, C.; Barbero, L.; Chicco, D.; Del Curto, M. D. ; Esposito, P.; Traversa. S.; Aime, S. NMR conformational analysis of antide, a potent antagonist of the gonadotropin releasing hormone. J. Am. Chem. Soc., 2002, 124, 3431-3442.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 3431-3442
-
-
Digilio, G.1
Bracco, C.2
Barbero, L.3
Chicco, D.4
Del Curto, M.D.5
Esposito, P.6
Traversa, S.7
Aime, S.8
-
172
-
-
15444355594
-
Discovery of a novel, potent, and orally active nonpeptide antagonist of the human luteinizing hormone-releasing hormone (LHRH) receptor
-
Cho, N.; Harada, M.; Imaeda, T.; Imada, T.; Matsumoto, H.; Hayase, Y.; Sasaki, S.; Furuya, S.; Suzuki, N.; Okubo, S. Discovery of a novel, potent, and orally active nonpeptide antagonist of the human luteinizing hormone-releasing hormone (LHRH) receptor. J. Med. Chem., 1998, 41, 4190-4195.
-
(1998)
J. Med. Chem
, vol.41
, pp. 4190-4195
-
-
Cho, N.1
Harada, M.2
Imaeda, T.3
Imada, T.4
Matsumoto, H.5
Hayase, Y.6
Sasaki, S.7
Furuya, S.8
Suzuki, N.9
Okubo, S.10
-
173
-
-
0242684600
-
Structure-activity relationships for a series of peptidomimetic antimicrobial prodrugs containing glutamine analogues
-
Neil, J.M.; Andruszkiewicz, R.; Gupta, S.; Milewski, S.; Payne, J.W. Structure-activity relationships for a series of peptidomimetic antimicrobial prodrugs containing glutamine analogues. J. Antimicrob. Chemother., 2003, 51, 821-831.
-
(2003)
J. Antimicrob. Chemother
, vol.51
, pp. 821-831
-
-
Neil, J.M.1
Andruszkiewicz, R.2
Gupta, S.3
Milewski, S.4
Payne, J.W.5
-
174
-
-
0000801464
-
Annu. Nonpeptide agonists for peptide receptors: Lessons from ligands
-
Sugg, E.E. Annu. Nonpeptide agonists for peptide receptors: lessons from ligands. Rep. Med. Chem., 1997, 32, 277-283.
-
(1997)
Rep. Med. Chem
, vol.32
, pp. 277-283
-
-
Sugg, E.E.1
-
175
-
-
20544475205
-
Design, modelling, synthesis and biological evaluation of peptidomimetic phosphinates as inhibitors of matrix metalloproteinases MMP-2 and MMP-8
-
Bianchini, G.; Aschi, M.; Cavicchio, G.; Crucianelli, M.; Preziuso, S.; Gallina, G.; Nastari, A.; Gavuzzod, E.; Mazzaa, F. Design, modelling, synthesis and biological evaluation of peptidomimetic phosphinates as inhibitors of matrix metalloproteinases MMP-2 and MMP-8. Bioorg. Med. Chem., 2005, 13, 4740-4749.
-
(2005)
Bioorg. Med. Chem
, vol.13
, pp. 4740-4749
-
-
Bianchini, G.1
Aschi, M.2
Cavicchio, G.3
Crucianelli, M.4
Preziuso, S.5
Gallina, G.6
Nastari, A.7
Gavuzzod, E.8
Mazzaa, F.9
-
176
-
-
13944252004
-
Synthesis and evaluation of diverse analogs of amygdalin as potential peptidomimetics of peptide T
-
Araya, E.; Rodriguez, A.; Rubio, J.; Spada, A.; Joglar, J.; Llebaria, A.; Lagunas, C.; Fernandez, A.G.; Spisanie, S.; Perez, J.J. Synthesis and evaluation of diverse analogs of amygdalin as potential peptidomimetics of peptide T. Bioorg. Med. Chem. Lett., 2005, 15, 1493-1496.
-
(2005)
Bioorg. Med. Chem. Lett
, vol.15
, pp. 1493-1496
-
-
Araya, E.1
Rodriguez, A.2
Rubio, J.3
Spada, A.4
Joglar, J.5
Llebaria, A.6
Lagunas, C.7
Fernandez, A.G.8
Spisanie, S.9
Perez, J.J.10
-
177
-
-
27744456972
-
Modeling of farnesyltransferase inhibition by some thiol and non-thiol peptidomimetic inhibitors using genetic neural networks and RDF approaches
-
Gonzalez, M.P.; Caballero, J.; Tundidor-Camba, A.; Helguerab, A.M.; Fernandezc, M. Modeling of farnesyltransferase inhibition by some thiol and non-thiol peptidomimetic inhibitors using genetic neural networks and RDF approaches. Bioorg. Med. Chem., 2006, 14, 200-213.
-
(2006)
Bioorg. Med. Chem
, vol.14
, pp. 200-213
-
-
Gonzalez, M.P.1
Caballero, J.2
Tundidor-Camba, A.3
Helguerab, A.M.4
Fernandezc, M.5
-
178
-
-
33646358479
-
Design and Synthesis of a Novel Peptidomimetic Inhibitor of Caspase-3
-
Zhang, J.; Liu, L.; Guo, Y.; Yang, J.; Wei, L.; Zhong, D.; Wang, J. Design and Synthesis of a Novel Peptidomimetic Inhibitor of Caspase-3. Chem. Res. Chin. Univ., 2006, 22, 225-228.
-
(2006)
Chem. Res. Chin. Univ
, vol.22
, pp. 225-228
-
-
Zhang, J.1
Liu, L.2
Guo, Y.3
Yang, J.4
Wei, L.5
Zhong, D.6
Wang, J.7
-
179
-
-
21144453843
-
P2 pyridine N-oxide thrombin inhibitors: A novel peptidomimetic scaffold
-
Nantermet, P.G.; Burgey, C.S.; Robinson, K.A.; Pellicore, J.M.; Newton, C.N.; Deng, J.Z.; Selnick, H.G.; Lewis, S.D.; Lucas, B.J.; Krueger, J.A. P2 pyridine N-oxide thrombin inhibitors: a novel peptidomimetic scaffold. Bioorg. Med. Chem. Lett., 2005, 15, 2771-2775.
-
(2005)
Bioorg. Med. Chem. Lett
, vol.15
, pp. 2771-2775
-
-
Nantermet, P.G.1
Burgey, C.S.2
Robinson, K.A.3
Pellicore, J.M.4
Newton, C.N.5
Deng, J.Z.6
Selnick, H.G.7
Lewis, S.D.8
Lucas, B.J.9
Krueger, J.A.10
-
180
-
-
0042158268
-
Design, synthesis, and evaluation of azepine-based cryptophycin mimetics
-
Smith, A.B.; Cho, Y.S.; Pettitb, G.R.; Hirschmanna, R. Design, synthesis, and evaluation of azepine-based cryptophycin mimetics. Tetrahedron, 2003, 59, 6991-7009.
-
(2003)
Tetrahedron
, vol.59
, pp. 6991-7009
-
-
Smith, A.B.1
Cho, Y.S.2
Pettitb, G.R.3
Hirschmanna, R.4
-
181
-
-
0037430643
-
Modification of the N-terminus of peptidomimetic protein tyrosine phosphatase 1B (PTP1B) inhibitors: Identification of analogues with cellular activity
-
Larsen, S.D.; Stevens, F.G.; Lindberg, T.J.; Bodnar, P.M., O'Sullivan, T.J.; Schostarez, H.J.; Palazuk, B.J.; Bleasdaleb, J.E. Modification of the N-terminus of peptidomimetic protein tyrosine phosphatase 1B (PTP1B) inhibitors: identification of analogues with cellular activity. Bioorg. Med. Chem. Lett., 2003, 13, 971-975.
-
(2003)
Bioorg. Med. Chem. Lett
, vol.13
, pp. 971-975
-
-
Larsen, S.D.1
Stevens, F.G.2
Lindberg, T.J.3
Bodnar, P.M.4
O'Sullivan, T.J.5
Schostarez, H.J.6
Palazuk, B.J.7
Bleasdaleb, J.E.8
-
182
-
-
3543055012
-
Novel peptidomimetic inhibitors of signal transducer and activator of transcription 3 dimerization and biological activity
-
Turkson, J.; Kim, J.S.; Zhang, S.; Yuan, J.; Huang, M.; Glenn, M.; Haura, E.; Sebti, S,; Hamilton, A.D.; Jove, R. Novel peptidomimetic inhibitors of signal transducer and activator of transcription 3 dimerization and biological activity. Mol. Cancer Ther., 2004, 3 (3), p.261-269.
-
(2004)
Mol. Cancer Ther
, vol.3
, Issue.3
, pp. 261-269
-
-
Turkson, J.1
Kim, J.S.2
Zhang, S.3
Yuan, J.4
Huang, M.5
Glenn, M.6
Haura, E.7
Sebti, S.8
Hamilton, A.D.9
Jove, R.10
-
183
-
-
0034689595
-
Novel peptidomimetic hematoregulatory compounds
-
Heerding, D.A.; Abruzzese, M.; Alberts, D.; Burgess, J.; Callahan, J.F.; Huffman, W.F. Novel peptidomimetic hematoregulatory compounds. Bioorg. Med. Chem. Lett., 2000,10, 531-534.
-
(2000)
Bioorg. Med. Chem. Lett
, vol.10
, pp. 531-534
-
-
Heerding, D.A.1
Abruzzese, M.2
Alberts, D.3
Burgess, J.4
Callahan, J.F.5
Huffman, W.F.6
-
184
-
-
0035997944
-
Adenovirus inhibition by peptidomimetic integrin antagonists
-
Hippenmeyer, P.J.; Ruminski, P.G.; Rico, J.G.; Lu, H.S.; Griggs, D.W. Adenovirus inhibition by peptidomimetic integrin antagonists. Antivir. Res., 2002, 55, 169-178.
-
(2002)
Antivir. Res
, vol.55
, pp. 169-178
-
-
Hippenmeyer, P.J.1
Ruminski, P.G.2
Rico, J.G.3
Lu, H.S.4
Griggs, D.W.5
-
185
-
-
10844238962
-
Computational studies and peptidomimetic design for the human p53-MDM2 complex
-
Zhong, H.; Carlson, H.A. Computational studies and peptidomimetic design for the human p53-MDM2 complex. Proteins, 2005, 58, 222-234.
-
(2005)
Proteins
, vol.58
, pp. 222-234
-
-
Zhong, H.1
Carlson, H.A.2
-
186
-
-
19944367270
-
Structure-based design of P3 moieties in the peptide mimetic factor VIIa inhibitor
-
Kadono, S.; Sakamoto, A.; Kikuchi, Y.; Oheda, M.; Yabuta, N.; Yoshihashi, K.; Kitazawa, T. Structure-based design of P3 moieties in the peptide mimetic factor VIIa inhibitor. Biochem. Biophy. Res. Comm., 2005, 327, 589-596.
-
(2005)
Biochem. Biophy. Res. Comm
, vol.327
, pp. 589-596
-
-
Kadono, S.1
Sakamoto, A.2
Kikuchi, Y.3
Oheda, M.4
Yabuta, N.5
Yoshihashi, K.6
Kitazawa, T.7
-
187
-
-
34548079602
-
In Silico analysis of antifungal peptides (AFPs): Determining the lead template sequence of potent antifungal peptides
-
Soltani, S.; Keymanesh, K.; Sardari, S. In Silico analysis of antifungal peptides (AFPs): Determining the lead template sequence of potent antifungal peptides. Expert Opin. Drug. Discov., 2007, 2, 837-847.
-
(2007)
Expert Opin. Drug. Discov
, vol.2
, pp. 837-847
-
-
Soltani, S.1
Keymanesh, K.2
Sardari, S.3
-
188
-
-
0242684600
-
Structure-activity relationships for a series of peptidomimetic antimicrobial prodrugs containing glutamine analogues
-
Marshall, N.J.; Andruszkiewicz, R.; Gupta, S.; Milewski, S.; Payne, J.W. Structure-activity relationships for a series of peptidomimetic antimicrobial prodrugs containing glutamine analogues. J. Antimicrob. Chemother., 2003, 51, 821-831.
-
(2003)
J. Antimicrob. Chemother
, vol.51
, pp. 821-831
-
-
Marshall, N.J.1
Andruszkiewicz, R.2
Gupta, S.3
Milewski, S.4
Payne, J.W.5
-
189
-
-
0001239683
-
Peptidomimetic building blocks for drug discovery: An overview
-
Goodman, M; Shao, H. Peptidomimetic building blocks for drug discovery: an overview. Pure. Appl. Chem., 1996, 68, 1303-1308.
-
(1996)
Pure. Appl. Chem
, vol.68
, pp. 1303-1308
-
-
Goodman, M.1
Shao, H.2
|