TRPV1: A target for next generation analgesics

Current Neuropharmacology

Volumn 6, Issue 2, 2008, Pages 151-163

  Premkumar, Louis S ^a   Sikand, Parul ^a  

^a SOUTHERN ILLINOIS UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Inflammatory mediators; Nociceptive ion channels; Nociceptors; Pain; Protein kinases; TRPV1

Indexed keywords

(4 TERT BUTYLPHENYL) 4 (3 CHLOROPYRIDIN 2 YL)TETRAHYDROPYRAZINE 1(2H) CARBOXAMIDE; 1 [3 (TRIFLUOROMETHYL)PYRIDINE 2 YL] N [4 (TRIFLUOROMETHYLSULFONYL)PHENYL] 1,2,3,6 TETRAHYDROPYRIDINE 4 CARBOXAMIDE; 1 ISOQUINOLIN 5 YL 3 (4 TRIFLUOROMETHYLBENZYL)UREA; 4 CHLORO N (3 METHOXYPHENYL)CINNAMAMIDE; A 425619; A 784168; A 795614; AMG 0347; AMG 0347,; AMG 517; AMG 8163; AMG 9810; BOTULINUM TOXIN; CALCIUM; CAPSAICIN; CAPSAZEPINE; CATION CHANNEL; GRC 6211; IODORESINIFERATOXIN; JNJ 17203212; JYL 1421; KANAMYCIN; MK 2295; N (4 HYDROXYPHENYL)ARACHIDONAMIDE; N 1H INDAZOL 4 YL N' (5 PIPERIDIN 1 YL 2,3 DIHYDRO 1H INDEN 1 YL)UREA; N(G) NITROARGININE METHYL ESTER; NDG 8243; RECEPTOR BLOCKING AGENT; RESINIFERATOXIN; RUTHENIUM RED; SUBSTANCE P ANTAGONIST; UNINDEXED DRUG; VANILLOID RECEPTOR 1; VANILLOID RECEPTOR 1 ANTAGONIST;

ACTION POTENTIAL; AIDS RELATED COMPLEX; ANALGESIA; BLADDER DISEASE; BLOOD VESSEL INNERVATION; CANCER PAIN; CARDIOVASCULAR SYSTEM; CELL SUBPOPULATION; CENTRAL NERVOUS SYSTEM; CLINICAL TRIAL; DIABETIC NEUROPATHY; DIZZINESS; DRUG EFFICACY; DRUG MECHANISM; DRUG SELECTIVITY; DRUG TARGETING; FOOD INTAKE; GASTROINTESTINAL TRACT; GENE DELETION; HAIR; HEARING; HUMAN; HYPERALGESIA; HYPOTHERMIA; INTERSTITIAL CYSTITIS; LOW DRUG DOSE; MOTOR DYSFUNCTION; MUSCLE SPINDLE AFFERENT NERVE; MUSCULOSKELETAL PAIN; NERVE ENDING; NEUROMODULATION; NEUROPATHIC PAIN; NEUROPATHY; NEUROTRANSMISSION; NEUROTRANSMITTER RELEASE; NOCICEPTIVE STIMULATION; NONHUMAN; OINTMENT; PAIN THRESHOLD; PERIPHERAL NERVOUS SYSTEM; POSTHERPETIC NEURALGIA; PROTEIN ANALYSIS; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN LOCALIZATION; PROTEIN PHOSPHORYLATION; PRURITUS; RESPIRATORY SYSTEM; REVIEW; SENSORY NERVE CELL; TASTE; THERMOREGULATION; TINNITUS; URINE INCONTINENCE;

EID: 47749116508     PISSN: 1570159X     EISSN: None     Source Type: Journal    
DOI: 10.2174/157015908784533888     Document Type: Review

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