Neurogenic responses mediated by vanilloid receptor-1 (TRPV1) are blocked by the high affinity antagonist, iodo-resiniferatoxin

British Journal of Pharmacology

Volumn 138, Issue 5, 2003, Pages 977-985

  Rigoni, Michela ^a   Trevisani, Marcello ^a   Gazzieri, David ^a   Nadaletto, Riccardo ^a   Tognetto, Michele ^a   Creminon, Christophe ^b   Davis, John B ^c   Campi, Barbara ^a   Amadesi, Silvia ^a   Geppetti, Pierangelo ^a   Harrison, Selena ^a  

^a UNIVERSITY OF FERRARA   (Italy)

^b Institut National de la Recherche Agronomique   (France)

^c GLAXOSMITHKLINE   (United Kingdom)

Author keywords

Capsaicin; Capsazepine; Iodo resiniferatoxin; Resiniferatoxin; Vanilloid receptor 1

Indexed keywords

CAPSAICIN; CAPSAZEPINE; IODORESINIFERATOXIN; IONOMYCIN; POTASSIUM CHLORIDE; RESINIFERATOXIN; UNCLASSIFIED DRUG; VANILLOID RECEPTOR; VANILLOID RECEPTOR 1;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BLADDER; CALCIUM CELL LEVEL; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; GUINEA PIG; IC 50; MALE; MOUSE; NEUROGENIC INFLAMMATION; NOCICEPTION; NONHUMAN; PAIN; PRIORITY JOURNAL; RAT; RECEPTOR INTRINSIC ACTIVITY; RECEPTOR SENSITIVITY; TRIGEMINAL NERVE;

ANIMALS; CELL LINE; DITERPENES; DOSE-RESPONSE RELATIONSHIP, DRUG; GUINEA PIGS; HUMANS; MALE; MICE; MUSCLE CONTRACTION; NEURONS; PAIN MEASUREMENT; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, DRUG;

EID: 0037349190     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0705110     Document Type: Article

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