Thapsigargin binds to and inhibits the cloned vanilloid receptor-1

Biochemical and Biophysical Research Communications

Volumn 293, Issue 2, 2002, Pages 777-782

  Tóth, Attila ^a   Kedei, Noémi ^a   Szabó, Tamás ^a   Wang, Yun ^a   Blumberg, Peter M ^a  

^a NATIONAL CANCER INSTITUTE   (United States)

Author keywords

Capsaicin; Resiniferatoxin binding; Sarcoplasmatic reticulum ATPase; Thapsigargin; Vanilloid receptor subtype 1; VR1 transfected CHO cells

Indexed keywords

ADENOSINE TRIPHOSPHATASE INHIBITOR; CALCIUM ION; CAPSAICIN; THAPSIGARGIN; VANILLOID RECEPTOR;

ANIMAL CELL; ARTICLE; BINDING SITE; CALCIUM TRANSPORT; CHO CELL; CONTROLLED STUDY; DRUG EFFECT; DRUG STRUCTURE; ENZYME INHIBITION; NONHUMAN; PRIORITY JOURNAL; SARCOPLASMIC RETICULUM;

ANIMALS; CALCIUM; CALCIUM-TRANSPORTING ATPASES; CAPSAICIN; CHO CELLS; CLONING, MOLECULAR; CRICETINAE; DITERPENES; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; KINETICS; RECEPTORS, DRUG; SARCOPLASMIC RETICULUM CALCIUM-TRANSPORTING ATPASES; THAPSIGARGIN; TRPV CATION CHANNELS;

EID: 0036294731     PISSN: 0006291X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-291X(02)00293-0     Document Type: Article

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