SCOPUS 정보 검색 플랫폼

ChemMedChem

Volumn 9, Issue 2, 2014, Pages 256-275

Structure-based and fragment-based GPCR drug discovery

(3) Andrews, Stephen P a Brown, Giles A a Christopher, John A a

a Heptares Therapeutics Ltd (United Kingdom)

Author keywords

Fragment Based Drug Discovery; G Proteincoupled Receptors; Structural Biology; Structure Based Drug Discovery

Indexed keywords

ADENOSINE A2A RECEPTOR ANTAGONIST; ADENOSINE RECEPTOR; BETA 1 ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR; CHEMOKINE; DOPAMINE; G PROTEIN COUPLED RECEPTOR; HISTAMINE RECEPTOR;

CELL MEMBRANE; CRYSTAL STRUCTURE; DRUG DEVELOPMENT; FRAGMENT BASED DRUG DISCOVERY; NONHUMAN; PRIORITY JOURNAL; REVIEW; SCREENING;

FRAGMENT-BASED DRUG DISCOVERY; G PROTEIN-COUPLED RECEPTORS; STRUCTURAL BIOLOGY; STRUCTURE-BASED DRUG DISCOVERY;

ANIMALS; DRUG DESIGN; HUMANS; LIGANDS; MOLECULAR DOCKING SIMULATION; PROTEIN CONFORMATION; RECEPTORS, G-PROTEIN-COUPLED;

EID: 84897026211 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201300382 Document Type: Review

Times cited : (68)

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