[3H]ZM241385 - An antagonist radioligand for adenosine A2A receptors in rat brain

European Journal of Pharmacology

Volumn 411, Issue 3, 2001, Pages 205-210

  Alexander, Stephen P H ^a   Millns, Paul J ^a  

^a UNIVERSITY OF NOTTINGHAM   (United Kingdom)

Author keywords

Adenosine A2A receptor; Autoradiography; Radioligand binding; Striatum, rat

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); 4 [2 [7 AMINO 2 (2 FURYL) 1,2,4 TRIAZOLO[2,3 A][1,3,5]TRIAZIN 5 YLAMINO]ETHYL]PHENOL; 5 AMINO 2 (2 FURYL) 7 (2 PHENYLETHYL)PYRAZOLO[4,3 E][1,2,4]TRIAZOLO[1,5 C]PYRIMIDINE; 8 [4 (2 AMINOETHYLCARBAMOYL)METHOXYPHENYL] 1,3 DIPROPYLXANTHINE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2A RECEPTOR; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); THEOPHYLLINE;

ANIMAL TISSUE; ARTICLE; BINDING KINETICS; CONTROLLED STUDY; CORPUS STRIATUM; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; FEMALE; FRONTAL CORTEX; HIPPOCAMPUS; ISOTOPE LABELING; LIGAND BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BLOCKING; TEMPERATURE DEPENDENCE;

ANIMALS; AUTORADIOGRAPHY; BINDING, COMPETITIVE; BRAIN CHEMISTRY; FEMALE; HALF-LIFE; MALE; MEMBRANES; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTOR, ADENOSINE A2A; RECEPTORS, PURINERGIC P1; THERMODYNAMICS; TRIAZINES; TRIAZOLES;

EID: 0035847134     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(00)00899-2     Document Type: Article

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