Design of monoamine reuptake inhibitors: SSRIs, SNRIs and NRIs

Topics in Medicinal Chemistry

Volumn 4, Issue , 2009, Pages 53-94

  Whitlock, Gavin A ^a   Andrews, Mark D ^a   Brown, Alan D ^a   Fish, Paul V ^a   Stobie, Alan ^a   Wakenhut, Florian ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United Kingdom)

Author keywords

Design; Dual reuptake inhibitor; Monoamine; NRI; SAR; SNRI; SSRI

Indexed keywords

1 3,4 DIHYDRO 1H QUINOLIN 2 ONE; 4 (4 CHLOROPHENYL)PIPERIDINE; AMITRIPTYLINE; ATOMOXETINE; CITALOPRAM; COCAINE; DAPOXETINE; DOPAMINE; DULOXETINE; FLUOXETINE; MILNACIPRAN; MORPHOLINE DERIVATIVE; NORADRENALIN; NORADRENALIN UPTAKE INHIBITOR; PAROXETINE; PIPERAZINE DERIVATIVE; PIPERIDINE DERIVATIVE; PROPANAMINE DERIVATIVE; PYRROLIDINE DERIVATIVE; REBOXETINE; SEROTONIN; SEROTONIN NORADRENALIN REUPTAKE INHIBITOR; SEROTONIN UPTAKE INHIBITOR; SERTRALINE; TROPANE DERIVATIVE; UK 373911; UK 390957; UNCLASSIFIED DRUG; UNINDEXED DRUG; VENLAFAXINE; VILOXAZINE;

ATTENTION DEFICIT DISORDER; CHEMISTRY; CLINICAL TRIAL; DEPRESSION; DRUG BINDING; DRUG DESIGN; DRUG RESEARCH; DRUG SYNTHESIS; HUMAN; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PRIORITY JOURNAL; REVIEW; STRUCTURE ACTIVITY RELATION;

EID: 77950548585     PISSN: 18622461     EISSN: 1862247X     Source Type: Book Series    
DOI: 10.1007/7355_2008_028     Document Type: Review

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