N-Alkyl-N-arylmethylpiperidin-4-amines: Novel dual inhibitors of serotonin and norepinephrine reuptake

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 10, 2006, Pages 2714-2718

  Boot, J R ^a   Boulet, S L ^a   Clark, B P ^a   Cases Thomas, M J ^a   Delhaye, L ^b   Diker, K ^b   Fairhurst, J ^a   Findlay, J ^a   Gallagher, P T ^a   Gilmore, J ^a   Harris, J R ^a   Masters, J J ^a   Mitchell, S N ^a   Naik, M ^a   Simmonds, R G ^a   Smith, S M ^a   Richards, S J ^a   Timms, G H ^a   Whatton, M A ^a   Wolfe, C N ^a   Wood, V A ^a   more..

^a ELI LILLY AND COMPANY   (United States)

^b Eli Lilly Benelux   (Belgium)

Author keywords

Aminopiperidines; Inhibitors; Norepinephrine; Reuptake; Serotonin; Transporter

Indexed keywords

AMINE; NORADRENALIN UPTAKE INHIBITOR; PIPERIDINE DERIVATIVE; SEROTONIN UPTAKE INHIBITOR;

ARTICLE; DRUG SCREENING; DRUG SYNTHESIS; NORADRENALIN UPTAKE; RECEPTOR BINDING; SEROTONIN UPTAKE; STRUCTURE ACTIVITY RELATION;

NOREPINEPHRINE; PIPERIDINES; SEROTONIN UPTAKE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33645845143     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.02.008     Document Type: Article

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