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D'Cruz OJ, Samuel P, Uckun FM: Conceival, a novel noncontraceptive vaginal vehicle for lipophilic microbicides. AAPS PharmSciTech (2005) 6(1):E56-E64.
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In vivo evaluation of a gel formulation of stampidine, a novel nonspermicidal broad-spectrum anti-HIV microbicide
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D'Cruz OJ, Samuel P, Waurzyniak B, Uckun FM: In vivo evaluation of a gel formulation of stampidine, a novel nonspermicidal broad-spectrum anti-HIV microbicide. Am J Drug Deliv (2003) 1(4):275-285.
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Am J Drug Deliv
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191
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Development and evaluation of a thermoreversible ovule formulation of stampidine, a novel nonspermicidal broad-spectrum antihuman immunodeficiency virus microbicide
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D'Cruz OJ, Samuel P, Waurzyniak B, Uckun FM: Development and evaluation of a thermoreversible ovule formulation of stampidine, a novel nonspermicidal broad-spectrum antihuman immunodeficiency virus microbicide. Biol Reprod (2003) 69(6):1843-1851.
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Stampidine is a nonspermicidal broad-spectrum anti-human immunodeficiency virus microbicide
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This paper describes the unique features of a novel aryl phosphate derivative of stavudine with potent anti-HIV activity as a topical microbicide, •
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D'Cruz OJ, Uckun FM: Stampidine is a nonspermicidal broad-spectrum anti-human immunodeficiency virus microbicide. Fertil Steril (2003) 81(Suppl 1):831-841. • This paper describes the unique features of a novel aryl phosphate derivative of stavudine with potent anti-HIV activity as a topical microbicide.
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Fertil Steril
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Developmental safety profile of the anti-HIV agent stampidine in rabbits
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D'Cruz OJ, Erbeck D, Uckun FM: Developmental safety profile of the anti-HIV agent stampidine in rabbits. Arzneimittelforschung (2006) 56(2a):159-166.
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194
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A study of the potential of the pig as a model for the vaginal irritancy of benzalkonium chloride in comparison to the nonirritant microbicide PHI-443 and the spermicide vanadocene dithiocarbamate
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This paper reports the development of a physiologically relevant and sensitive animal model for the local tolerance of microbicide and spermicide formulations, •
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D'Cruz OJ, Erbeck D, Uckun FM: A study of the potential of the pig as a model for the vaginal irritancy of benzalkonium chloride in comparison to the nonirritant microbicide PHI-443 and the spermicide vanadocene dithiocarbamate. Toxicol Pathol (2005) 33(4):465-476. • This paper reports the development of a physiologically relevant and sensitive animal model for the local tolerance of microbicide and spermicide formulations.
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Toxicol Pathol
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Large-scale synthesis and formulation of GMP-grade stampidine, a new anti-HIV agent
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DuMez D, Venkatachalam TK, Uckun FM: Large-scale synthesis and formulation of GMP-grade stampidine, a new anti-HIV agent. Arzneimittelforschung (2006) 56(2a):136-151.
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196
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Large-scale synthesis of GMP grade N′-[2-(2-thiophene)ethyl]-N′- [2-(5-bromopyridyl)] thiourea [PHI-443], a new anti-HIV drug candidate
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Dumez D, Venkatachalam TK, Uckun FM: Large-scale synthesis of GMP grade N′-[2-(2-thiophene)ethyl]-N′- [2-(5-bromopyridyl)] thiourea [PHI-443], a new anti-HIV drug candidate. Arzneimittelforschung (2007) 57(6):330-339.
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