Large-scale synthesis and formulation of GMP-grade stampidine, a new anti-HIV agent

Arzneimittel-Forschung/Drug Research

Volumn 56, Issue 2 A, 2006, Pages 136-151

  DuMez, Darin ^a,b   Venkatachalam, Taracad K ^a,b   Uckun, Fatih M ^a,b,c  

^a PARKER HUGHES INSTITUTE   (United States)

^b Paradigm Pharmaceuticals   (United States)

^c Ikaros Enterprises   (United States)

Author keywords

Anti HIV agents; Antiretroviral therapy; CAS 217178 62 6; CAS 3056 17 5; DDE 113; HI 113; N p (4 bromophenyl) 2',3' didehydro 3' deoxy 5' thymidylyl L alanine methyl ester; Stampidine, formulation, GMP, synthesis; Stavudine

Indexed keywords

CAS 217178 62 6; CAS 3056 17 5; DDE 113; HI 113; RNA DIRECTED DNA POLYMERASE INHIBITOR; STAMPIDINE; STAVUDINE; UNCLASSIFIED DRUG; ZIDOVUDINE;

ARTICLE; DRUG CAPSULE; DRUG DOSAGE FORM; DRUG FORMULATION; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; GOOD MANUFACTURING PRACTICE; HIGHLY ACTIVE ANTIRETROVIRAL THERAPY; LARGE SCALE PRODUCTION; PARTICLE SIZE;

EID: 33645101334     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-0031-1296801     Document Type: Article

References (17)

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