The thiocarboxanilide nonnucleoside UC781 is a tight-binding inhibitor of HIV-1 reverse transcriptase

Biochemistry

Volumn 36, Issue 25, 1997, Pages 7786-7792

  Barnard, John ^b   Borkow, Gadi ^b   Parniak, Michael A ^a  

^a MCGILL UNIVERSITY   (Canada)

^b NONE

Author keywords

[No Author keywords available]

Indexed keywords

2',3' DIDEOXYNUCLEOSIDE DERIVATIVE; ANILIDE; N [4 CHLORO 3 (3 METHYL 2 BUTENYLOXY)PHENYL] 2 METHYL 3 FURANCARBOTHIOAMIDE; N [4 CHLORO 3 (3 METHYL 2 BUTENYLOXY)PHENYL] 2 METHYL 3 FURANOCARBOTHIAMIDE; NEVIRAPINE; RNA DIRECTED DNA POLYMERASE INHIBITOR; THIOCARBAMIC ACID DERIVATIVE; UNCLASSIFIED DRUG; VIRUS ENZYME; ZIDOVUDINE;

ANTIVIRAL ACTIVITY; ARTICLE; CONTROLLED STUDY; ENZYME ACTIVITY; FLUORESCENCE; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; PRIORITY JOURNAL; SEXUALLY TRANSMITTED DISEASE; VIRUS GENE; VIRUS REPLICATION;

ANILIDES; BENZODIAZEPINONES; FURANS; HIV-1 REVERSE TRANSCRIPTASE; KINETICS; NEVIRAPINE; PROTEIN BINDING; PYRIDINES; REVERSE TRANSCRIPTASE INHIBITORS; SPECTROMETRY, FLUORESCENCE;

HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0030751673     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi970140u     Document Type: Article

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