-
2
-
-
4444355871
-
-
H.-J. Bohm, D. Banner, S. Bendels, M. Kansy, B. Kuhn, K. Mueller, U. O-bst-Sander, and M. Stahl Chem. Biol. Chem. 5 2004 637 643
-
(2004)
Chem. Biol. Chem.
, vol.5
, pp. 637-643
-
-
Bohm, H.-J.1
Banner, D.2
Bendels, S.3
Kansy, M.4
Kuhn, B.5
Mueller, K.6
O-Bst-Sander, U.7
Stahl, M.8
-
6
-
-
4544318450
-
-
J.A. Olsen, D.W. Banner, P. Seiler, B. Wagner, T. Tschopp, U. Obst-Sander, M. Kansy, K. Mueller, and F. Diederich Chem. Biol. Chem. 5 2004 666 675
-
(2004)
Chem. Biol. Chem.
, vol.5
, pp. 666-675
-
-
Olsen, J.A.1
Banner, D.W.2
Seiler, P.3
Wagner, B.4
Tschopp, T.5
Obst-Sander, U.6
Kansy, M.7
Mueller, K.8
Diederich, F.9
-
10
-
-
0029156922
-
-
G.J. Peters, C.L. van der Wilt, B. van der Triest, G. Cadacci-Pisanelli, P.G. Johnston, C.J. van Groeningen, and H.M. Pinedo Eur. J. Cancer 31A 1995 1299 1305
-
(1995)
Eur. J. Cancer
, vol.31
, pp. 1299-1305
-
-
Peters, G.J.1
Van Der Wilt, C.L.2
Van Der Triest, B.3
Cadacci-Pisanelli, G.4
Johnston, P.G.5
Van Groeningen, C.J.6
Pinedo, H.M.7
-
11
-
-
0037130282
-
-
G.J. Peters, H.H.J. Backus, S. Freemanthle, B. van der Triest, G. Cadacci-Pisanelli, C.L. van der Wilt, K. Smid, J. Lumec, A.H. Calvert, S. March, H.L. McLeod, E. Bloemena, S. Meijer, G. Jansen, C.J. van Groeningen, and H.M. Pinedo Biochem. Biophys. Acta 1587 2002 194 205
-
(2002)
Biochem. Biophys. Acta
, vol.1587
, pp. 194-205
-
-
Peters, G.J.1
Backus, H.H.J.2
Freemanthle, S.3
Van Der Triest, B.4
Cadacci-Pisanelli, G.5
Van Der Wilt, C.L.6
Smid, K.7
Lumec, J.8
Calvert, A.H.9
March, S.10
McLeod, H.L.11
Bloemena, E.12
Meijer, S.13
Jansen, G.14
Van Groeningen, C.J.15
Pinedo, H.M.16
-
14
-
-
0034060753
-
-
C.L. Piedbois, I.D. Zaleski, H. Juhel, C. Schmitt, A. Bellanger, and P. Piedbois Ann. Oncol. 11 2000 157 161
-
(2000)
Ann. Oncol.
, vol.11
, pp. 157-161
-
-
Piedbois, C.L.1
Zaleski, I.D.2
Juhel, H.3
Schmitt, C.4
Bellanger, A.5
Piedbois, P.6
-
18
-
-
0031842077
-
-
C.J.A. Punt Cancer 83 1998 679 689
-
(1998)
Cancer
, vol.83
, pp. 679-689
-
-
Punt, C.J.A.1
-
21
-
-
10844241474
-
-
J. Feliu, J.M. Vincent, C.G. Giron, M. Costella, E. Fonseca, J. Aparicho, M. Lomas, L.A. Aparicio, F.J. Dorta, and M.G. Baron Br. J. Cancer 91 2004 1758 1762
-
(2004)
Br. J. Cancer
, vol.91
, pp. 1758-1762
-
-
Feliu, J.1
Vincent, J.M.2
Giron, C.G.3
Costella, M.4
Fonseca, E.5
Aparicho, J.6
Lomas, M.7
Aparicio, L.A.8
Dorta, F.J.9
Baron, M.G.10
-
22
-
-
9344248389
-
-
T. Shirasaka, K. Nakano, T. Takechi, H. Statake, J. Uchda, and A. Fujioka Cancer Res. 56 1996 2602 2606
-
(1996)
Cancer Res.
, vol.56
, pp. 2602-2606
-
-
Shirasaka, T.1
Nakano, K.2
Takechi, T.3
Statake, H.4
Uchda, J.5
Fujioka, A.6
-
28
-
-
17144361816
-
-
K. Tanabe, Y. Makijura, Y. Tachi, A.I. Sato, and S.I. Nishimoto Biorg. Med. Chem. Lett. 15 2005 2321 2324
-
(2005)
Biorg. Med. Chem. Lett.
, vol.15
, pp. 2321-2324
-
-
Tanabe, K.1
Makijura, Y.2
Tachi, Y.3
Sato, A.I.4
Nishimoto, S.I.5
-
29
-
-
33645461180
-
-
R.K. Herrlinger, F.R.J. Cummings, M.N.C. Martin, M. Schwab, T. Ahmad, and P.D. Jewell Pharm. Genomics 15 2005 2005
-
(2005)
Pharm. Genomics
, vol.15
, pp. 2005
-
-
Herrlinger, R.K.1
Cummings, F.R.J.2
Martin, M.N.C.3
Schwab, M.4
Ahmad, T.5
Jewell, P.D.6
-
31
-
-
0037130283
-
-
A.L. Jackman, C.J. Melin, R. Kimbell, L. Brunton, G.W. Aherne, D.S. Theti, and M. Walton Biochim. Biophys. Acta 1587 2002 215 223
-
(2002)
Biochim. Biophys. Acta
, vol.1587
, pp. 215-223
-
-
Jackman, A.L.1
Melin, C.J.2
Kimbell, R.3
Brunton, L.4
Aherne, G.W.5
Theti, D.S.6
Walton, M.7
-
34
-
-
0032973498
-
-
H. Brackwitz, J. Bergmann, Y. Thoms, T. Wollny, and P. Langen Biorg. Chem. Med. Lett. 7 1999 1195 1200
-
(1999)
Biorg. Chem. Med. Lett.
, vol.7
, pp. 1195-1200
-
-
Brackwitz, H.1
Bergmann, J.2
Thoms, Y.3
Wollny, T.4
Langen, P.5
-
35
-
-
10044259855
-
-
W.E. Bauta, B.E. Schlmeier, B. Burke, J.F. Puente, W.R. Cantrell Jr., D. Lovett, J. Goebel, B. Anderson, D. Ionescu, and R. Guo Org. Process. Res. Dev. 8 2004 889 896
-
(2004)
Org. Process. Res. Dev.
, vol.8
, pp. 889-896
-
-
Bauta, W.E.1
Schlmeier, B.E.2
Burke, B.3
Puente, J.F.4
Cantrell Jr., W.R.5
Lovett, D.6
Goebel, J.7
Anderson, B.8
Ionescu, D.9
Guo, R.10
-
36
-
-
0036023405
-
-
P. Pourquier, C. Gioffre, G. Kohlhagen, Y. Urasaki, F. Goldwasser, L.W. Hertel, S. Yu, R.T. Pon, W.H. Gmeiner, and Y. Pomimier Clin. Cancer Res. 8 2002 2499 2504
-
(2002)
Clin. Cancer Res.
, vol.8
, pp. 2499-2504
-
-
Pourquier, P.1
Gioffre, C.2
Kohlhagen, G.3
Urasaki, Y.4
Goldwasser, F.5
Hertel, L.W.6
Yu, S.7
Pon, R.T.8
Gmeiner, W.H.9
Pomimier, Y.10
-
39
-
-
18244395551
-
-
S.M. Ali, A.R. Khan, M.U. Ahmad, P. Chen, S. Sheik, and I. Ahmad Biorg. Med. Chem. Lett. 15 2005 2571 2574
-
(2005)
Biorg. Med. Chem. Lett.
, vol.15
, pp. 2571-2574
-
-
Ali, S.M.1
Khan, A.R.2
Ahmad, M.U.3
Chen, P.4
Sheik, S.5
Ahmad, I.6
-
42
-
-
33645450874
-
Phase One Clinical Trials, Recent Phase I Trial Show Promise for Sarcoma
-
Summer
-
Phase One Clinical Trials, Recent Phase I Trial Show Promise for Sarcoma, CTRC Report, Summer 2005.
-
(2005)
CTRC Report
-
-
-
47
-
-
0032486436
-
-
K.C. Nicolaou, S. Kim, J. Pfefferkorn, J. Xu, T. Ohshima, S. Hosokawa, D. Vourloumis, and T. Li Angew. Chem. Int. Ed. 37 1998 1418 1420
-
(1998)
Angew. Chem. Int. Ed.
, vol.37
, pp. 1418-1420
-
-
Nicolaou, K.C.1
Kim, S.2
Pfefferkorn, J.3
Xu, J.4
Ohshima, T.5
Hosokawa, S.6
Vourloumis, D.7
Li, T.8
-
48
-
-
1942490811
-
-
S. Honore, K. Kamath, D. Braguer, L. Wilson, C. Briand, and M.A. Jordan Mol. Cancer Ther. 2 2003 1303 1311
-
(2003)
Mol. Cancer Ther.
, vol.2
, pp. 1303-1311
-
-
Honore, S.1
Kamath, K.2
Braguer, D.3
Wilson, L.4
Briand, C.5
Jordan, M.A.6
-
49
-
-
0033083045
-
-
S.L. Mooberry, G. Tien, A.H. Hernandez, A. Plubrukarn, and B.S. Davidson Cancer Res. 59 1999 653 660
-
(1999)
Cancer Res.
, vol.59
, pp. 653-660
-
-
Mooberry, S.L.1
Tien, G.2
Hernandez, A.H.3
Plubrukarn, A.4
Davidson, B.S.5
-
50
-
-
0037096807
-
-
K.A. Hood, L.M. West, B. Rouwe, P.T. Northcote, M.V. Berridge, S.W. Wakefield, J.H. Miller, and A. Peloruside Cancer Res. 62 2002 3356 3360
-
(2002)
Cancer Res.
, vol.62
, pp. 3356-3360
-
-
Hood, K.A.1
West, L.M.2
Rouwe, B.3
Northcote, P.T.4
Berridge, M.V.5
Wakefield, S.W.6
Miller, J.H.7
Peloruside, A.8
-
51
-
-
0035832113
-
-
S.L. Gwaltney, H.M. Imade, K.J. Barr, Q.L. Laura Gehrke, R.B. Credo, R.B. Warner, J.Y. Lee, P. Kovar, J. Wang, M.A. Nukkala, N.A. Zielinski, D. Forst, S.C. Ng, and H.L. Sham Biorg. Med. Chem. Lett. 11 2001 871 874
-
(2001)
Biorg. Med. Chem. Lett.
, vol.11
, pp. 871-874
-
-
Gwaltney, S.L.1
Imade, H.M.2
Barr, K.J.3
Laura Gehrke, Q.L.4
Credo, R.B.5
Warner, R.B.6
Lee, J.Y.7
Kovar, P.8
Wang, J.9
Nukkala, M.A.10
Zielinski, N.A.11
Forst, D.12
Ng, S.C.13
Sham, H.L.14
-
52
-
-
20444410402
-
-
H. Gao, X. Zhang, Y. Chen, H. Shen, T. Pang, J. Sun, C. XU, J. Ding, C. Li, and W. Lu Biorg. Med. Chem. Lett. 15 2005 3233 3236
-
(2005)
Biorg. Med. Chem. Lett.
, vol.15
, pp. 3233-3236
-
-
Gao, H.1
Zhang, X.2
Chen, Y.3
Shen, H.4
Pang, T.5
Sun, J.6
Xu, C.7
Ding, J.8
Li, C.9
Lu, W.10
-
55
-
-
0028036429
-
-
L. Li, K.H. Wang, S.C. Kuo, T.S. Wu, D. Lednicer, C.M. Lin, E. Hamel, and K.H. Lee J. Med. Chem. 37 1994 3400 3407
-
(1994)
J. Med. Chem.
, vol.37
, pp. 3400-3407
-
-
Li, L.1
Wang, K.H.2
Kuo, S.C.3
Wu, T.S.4
Lednicer, D.5
Lin, C.M.6
Hamel, E.7
Lee, K.H.8
-
56
-
-
0035829462
-
-
Y. Xia, Z. Yu, P. Xia, T. Hacki, E. Hamel, A. Mauger, J.H. Wu, and K.H. Lee J. Med. Chem. 44 2001 3932 3936
-
(2001)
J. Med. Chem.
, vol.44
, pp. 3932-3936
-
-
Xia, Y.1
Yu, Z.2
Xia, P.3
Hacki, T.4
Hamel, E.5
Mauger, A.6
Wu, J.H.7
Lee, K.H.8
-
59
-
-
0036895024
-
-
E.H. Rubin, D.P. de Alwis, I. Pouliquen, L. Green, P. Marder, Y. Lin, R. Musanti, S.L. Grospe, S.L. Smith, D.L. Toppmeyer, J. Much, M. Kane, A. Chaudhary, C. Jordan, M. Burgess, and C.A. Slapak Clin. Cancer Res. 8 2002 3710 3717
-
(2002)
Clin. Cancer Res.
, vol.8
, pp. 3710-3717
-
-
Rubin, E.H.1
De Alwis, D.P.2
Pouliquen, I.3
Green, L.4
Marder, P.5
Lin, Y.6
Musanti, R.7
Grospe, S.L.8
Smith, S.L.9
Toppmeyer, D.L.10
Much, J.11
Kane, M.12
Chaudhary, A.13
Jordan, C.14
Burgess, M.15
Slapak, C.A.16
-
60
-
-
12144287074
-
-
S. Wang, A. Folkes, I. Chuckowree, X. Cockroft, S. Sohal, W. Miler, J. Milton, S.P. Wren, N. Vicker, P. Depledge, J. Scott, L. Smith, H. Jones, P. Mistry, R. Faint, D. Thompson, and S. Cocks J. Med. Chem. 47 2004 1329 1338
-
(2004)
J. Med. Chem.
, vol.47
, pp. 1329-1338
-
-
Wang, S.1
Folkes, A.2
Chuckowree, I.3
Cockroft, X.4
Sohal, S.5
Miler, W.6
Milton, J.7
Wren, S.P.8
Vicker, N.9
Depledge, P.10
Scott, J.11
Smith, L.12
Jones, H.13
Mistry, P.14
Faint, R.15
Thompson, D.16
Cocks, S.17
-
61
-
-
21744447836
-
-
A. Boumendjel, H.B. Cortay, D. Trmpier, T. Perrotton, and A. Di Pietro Med. Res. Rev. 25 2005 453 472
-
(2005)
Med. Res. Rev.
, vol.25
, pp. 453-472
-
-
Boumendjel, A.1
Cortay, H.B.2
Trmpier, D.3
Perrotton, T.4
Di Pietro, A.5
-
62
-
-
12144290723
-
-
S. Wang, N.C. Wan, J. Harrison, W. Miller, I. Chuckowree, S. Sohal, T.C. Hancox, S. Baker, A. Folkes, F. Wilson, D. Thompson, S. Cocks, H. Farmer, A. Boyce, C. Freathy, J. Broadbridge, J. Scott, P. Depledge, R. Faint, P. Mistry, and P. Charlton J. Med. Chem. 47 2004 1339 1350
-
(2004)
J. Med. Chem.
, vol.47
, pp. 1339-1350
-
-
Wang, S.1
Wan, N.C.2
Harrison, J.3
Miller, W.4
Chuckowree, I.5
Sohal, S.6
Hancox, T.C.7
Baker, S.8
Folkes, A.9
Wilson, F.10
Thompson, D.11
Cocks, S.12
Farmer, H.13
Boyce, A.14
Freathy, C.15
Broadbridge, J.16
Scott, J.17
Depledge, P.18
Faint, R.19
Mistry, P.20
Charlton, P.21
more..
-
67
-
-
0029075872
-
-
C.K. Osborne, E.B. H-Coronado, S.G. Hilsenbeck, B.L. McCue, A.E. Wakeling, R.A. McClelland, D.L. Manning, and R.L. Nicholson J. Natl. Cancer Inst. 87 1995 746 750
-
(1995)
J. Natl. Cancer Inst.
, vol.87
, pp. 746-750
-
-
Osborne, C.K.1
H-Coronado, E.B.2
Hilsenbeck, S.G.3
McCue, B.L.4
Wakeling, A.E.5
McClelland, R.A.6
Manning, D.L.7
Nicholson, R.L.8
-
71
-
-
1642487666
-
-
T. Konno, T. Daitoh, A. Noiri, J. Chae, T. Ishihara, and H. Yamanaka Org. Lett. 6 2004 933 936
-
(2004)
Org. Lett.
, vol.6
, pp. 933-936
-
-
Konno, T.1
Daitoh, T.2
Noiri, A.3
Chae, J.4
Ishihara, T.5
Yamanaka, H.6
-
72
-
-
13844269367
-
-
H. Liu, J. Liu, R.B. van Breemen, G.R.J. Thatcher, and J.L. Bolton Chem. Res. Toxicol. 18 2005 162 173
-
(2005)
Chem. Res. Toxicol.
, vol.18
, pp. 162-173
-
-
Liu, H.1
Liu, J.2
Van Breemen, R.B.3
Thatcher, G.R.J.4
Bolton, J.L.5
-
77
-
-
13244290109
-
-
J.F.R. Robertson, S.E. Come, S.E. Jones, L. Bex, M. Kaufmann, A. Markis, J.W.R. Nortier, K. Possinger, and L.E. Rutqvist Eur. J. Cancer 41 2005 346 356
-
(2005)
Eur. J. Cancer
, vol.41
, pp. 346-356
-
-
Robertson, J.F.R.1
Come, S.E.2
Jones, S.E.3
Bex, L.4
Kaufmann, M.5
Markis, A.6
Nortier, J.W.R.7
Possinger, K.8
Rutqvist, L.E.9
-
79
-
-
0038240962
-
-
L. Mauriac, J.E. Pippen, J.Q. Albano, S.Z. Gertler, and C.K. Osborne Eur. J. Cancer 39 2003 1228 1233
-
(2003)
Eur. J. Cancer
, vol.39
, pp. 1228-1233
-
-
Mauriac, L.1
Pippen, J.E.2
Albano, J.Q.3
Gertler, S.Z.4
Osborne, C.K.5
-
81
-
-
0029048255
-
-
P.V. de Velde, F. Nique, J. Bremaud, M.C. Hameau, D. Philibert, and G. Teutsch Ann. N.Y. Acad. Sci. 761 1995 164 175
-
(1995)
Ann. N.Y. Acad. Sci.
, vol.761
, pp. 164-175
-
-
De Velde, P.V.1
Nique, F.2
Bremaud, J.3
Hameau, M.C.4
Philibert, D.5
Teutsch, G.6
-
83
-
-
0037294086
-
-
J.C. Blazejewski, M.P. Wilmshurst, M.D. Popkin, C. Wakselman, G. Laurent, D. Nonclercq, A. Cleeren, Y. Ma, H.S. Seo, and G. Leclercq Biorg. Med. Chem. 11 2003 335 345
-
(2003)
Biorg. Med. Chem.
, vol.11
, pp. 335-345
-
-
Blazejewski, J.C.1
Wilmshurst, M.P.2
Popkin, M.D.3
Wakselman, C.4
Laurent, G.5
Nonclercq, D.6
Cleeren, A.7
Ma, Y.8
Seo, H.S.9
Leclercq, G.10
-
84
-
-
0035154447
-
-
G. Giannoukos, D. Szapary, C.L. Smith, J.E.W. Meeker, and S.S. Simons Jr. Mol. Endocrinol. 15 2001 255 270
-
(2001)
Mol. Endocrinol.
, vol.15
, pp. 255-270
-
-
Giannoukos, G.1
Szapary, D.2
Smith, C.L.3
Meeker, J.E.W.4
Simons Jr., S.S.5
-
85
-
-
0034727865
-
-
U. Fuhrmann, H.H. Stumpp, A. Cleve, G. Neef, W. Schwede, J. Hoffmann, K.H. Fritzemeter, and K. Chwalisz J. Med. Chem. 43 2000 5010
-
(2000)
J. Med. Chem.
, vol.43
, pp. 5010
-
-
Fuhrmann, U.1
Stumpp, H.H.2
Cleve, A.3
Neef, G.4
Schwede, W.5
Hoffmann, J.6
Fritzemeter, K.H.7
Chwalisz, K.8
-
96
-
-
0035939330
-
-
A.J. Barker, K.H. Gibson, W. Grundy, A.A. Godfrey, J.J. Barlow, M.P. Healy, J.R. Woodburn, S.E. Ashton, R.J. Curry, L. Scarlett, L. Henthorn, and L. Richards Biorg. Med. Chem. Lett. 11 2001 1911 1914
-
(2001)
Biorg. Med. Chem. Lett.
, vol.11
, pp. 1911-1914
-
-
Barker, A.J.1
Gibson, K.H.2
Grundy, W.3
Godfrey, A.A.4
Barlow, J.J.5
Healy, M.P.6
Woodburn, J.R.7
Ashton, S.E.8
Curry, R.J.9
Scarlett, L.10
Henthorn, L.11
Richards, L.12
-
97
-
-
22844452590
-
-
M.J. Alberti, E.P. auten, K.E. Lackey, O.B. McDonald, E.R. Wood, F. Preugschat, G.J. Cutler, L.K. Carson, W. Liu, and D.K. Jung Birog. Med. Chem. Lett. 15 2005 3778 3781
-
(2005)
Birog. Med. Chem. Lett.
, vol.15
, pp. 3778-3781
-
-
Alberti, M.J.1
Auten, E.P.2
Lackey, K.E.3
McDonald, O.B.4
Wood, E.R.5
Preugschat, F.6
Cutler, G.J.7
Carson, L.K.8
Liu, W.9
Jung, D.K.10
-
99
-
-
20444427212
-
-
V. Aparna, G. Rambabu, S.K. Panigrahi, J.A.R.P. Sharma, and G.R. Desiraju J. Chem. Inf. Model. 45 2005 725 738
-
(2005)
J. Chem. Inf. Model.
, vol.45
, pp. 725-738
-
-
Aparna, V.1
Rambabu, G.2
Panigrahi, S.K.3
Sharma, J.A.R.P.4
Desiraju, G.R.5
-
101
-
-
0032984348
-
-
J.S. Sebolt-Leopold, D.T. Dudley, R. Herrera, K.V. Becelare, A. Wiland, R.C. Gowan, H. Tecle, S.D. Barrett, A. Bridges, S. Przybranowski, W.R. Leopold, and A.R. Saltiel Nat. Med. 5 1999 810 816
-
(1999)
Nat. Med.
, vol.5
, pp. 810-816
-
-
Sebolt-Leopold, J.S.1
Dudley, D.T.2
Herrera, R.3
Becelare, K.V.4
Wiland, A.5
Gowan, R.C.6
Tecle, H.7
Barrett, S.D.8
Bridges, A.9
Przybranowski, S.10
Leopold, W.R.11
Saltiel, A.R.12
-
102
-
-
0035253847
-
-
J.B. Smaill, H.D.H. Showalter, H. Zhou, A.J. Bridges, D.J. McNamara, D.W. Fry, J.M. Nelson, V. Sherwood, P.W. Vincent, and B.J. Roberts J. Med. Chem. 44 2001 429 440
-
(2001)
J. Med. Chem.
, vol.44
, pp. 429-440
-
-
Smaill, J.B.1
Showalter, H.D.H.2
Zhou, H.3
Bridges, A.J.4
McNamara, D.J.5
Fry, D.W.6
Nelson, J.M.7
Sherwood, V.8
Vincent, P.W.9
Roberts, B.J.10
-
103
-
-
24944486001
-
-
S. Campos, O. Hamid, M.V. Seiden, A. Oza, M. Plante, R.K. Potkul, P.F. Lenehan, E.P. Kaldjian, M.L. Varterasian, C. Jordan, C. Charbonneau, and H. Hirte J. Clin. Oncol. 23 2005 5597 5604
-
(2005)
J. Clin. Oncol.
, vol.23
, pp. 5597-5604
-
-
Campos, S.1
Hamid, O.2
Seiden, M.V.3
Oza, A.4
Plante, M.5
Potkul, R.K.6
Lenehan, P.F.7
Kaldjian, E.P.8
Varterasian, M.L.9
Jordan, C.10
Charbonneau, C.11
Hirte, H.12
-
104
-
-
0037152415
-
-
A. Wisner, M.B. Floyd, S.K. Rabindran, R. Nilakantan, L.M. Greenberger, R. Shen, Y.F. Wang, H.R. Tsou, and E.G.F.R. Synthesis Biorg. Med. Chem. Lett. 12 2002 2893 2897
-
(2002)
Biorg. Med. Chem. Lett.
, vol.12
, pp. 2893-2897
-
-
Wisner, A.1
Floyd, M.B.2
Rabindran, S.K.3
Nilakantan, R.4
Greenberger, L.M.5
Shen, R.6
Wang, Y.F.7
Tsou, H.R.8
Synthesis, E.G.F.R.9
-
108
-
-
0037137612
-
-
P.W. Manley, P. Furet, G. Bold, J. Bruggen, J. Mestan, T. Meyer, C.R. Schnell, and J. Wood J. Med. Chem. 45 2002 5687 5693
-
(2002)
J. Med. Chem.
, vol.45
, pp. 5687-5693
-
-
Manley, P.W.1
Furet, P.2
Bold, G.3
Bruggen, J.4
Mestan, J.5
Meyer, T.6
Schnell, C.R.7
Wood, J.8
-
109
-
-
20144375600
-
-
K. Kubo, T. Shimizu, S. Ohyama, H. Murooka, A. Iwai, K. Nakamura, K. Hasegawa, Y. Kobayashi, N. Takahashi, K. Takahashi, S. Kato, T. Izawa, and T. Isoe J. Med. Chem. 48 2005 1359 1366
-
(2005)
J. Med. Chem.
, vol.48
, pp. 1359-1366
-
-
Kubo, K.1
Shimizu, T.2
Ohyama, S.3
Murooka, H.4
Iwai, A.5
Nakamura, K.6
Hasegawa, K.7
Kobayashi, Y.8
Takahashi, N.9
Takahashi, K.10
Kato, S.11
Izawa, T.12
Isoe, T.13
-
110
-
-
20144376862
-
-
P.A. Harris, M. Cheung, R.N. Hunter III, M.L. Brown, J.M. Veal, R.T. Nolte, L. Wang, W. Liu, R.M. Crisby, J.H. Johnson, A.H. Epperly, R. Kumar, D.K. Luttrell, and J.A. Stafford J. Med. Chem. 48 2005 1610 1619
-
(2005)
J. Med. Chem.
, vol.48
, pp. 1610-1619
-
-
Harris, P.A.1
Cheung, M.2
Hunter III, R.N.3
Brown, M.L.4
Veal, J.M.5
Nolte, R.T.6
Wang, L.7
Liu, W.8
Crisby, R.M.9
Johnson, J.H.10
Epperly, A.H.11
Kumar, R.12
Luttrell, D.K.13
Stafford, J.A.14
-
111
-
-
25144461671
-
-
E.L. Piatnitski, M.A.J. Duncton, A.S. Kiselyov, R.K. Rouse, D. Sherman, D.L. Milligan, C. Balagtas, W.C. Wong, J. Kawakami, and J.F. Doody Biorg. Med. Chem. Lett. 15 2005 4696 4698
-
(2005)
Biorg. Med. Chem. Lett.
, vol.15
, pp. 4696-4698
-
-
Piatnitski, E.L.1
Duncton, M.A.J.2
Kiselyov, A.S.3
Rouse, R.K.4
Sherman, D.5
Milligan, D.L.6
Balagtas, C.7
Wong, W.C.8
Kawakami, J.9
Doody, J.F.10
-
112
-
-
4644359863
-
-
M.F. McCarty, J. Wey, O. Stoeltzing, W. Liu, F. Fan, C. Bucana, P.F. Mansfield, A.J. Ryan, and L.M. Ellis Mol. Cancer Ther. 3 2004 1041 1048
-
(2004)
Mol. Cancer Ther.
, vol.3
, pp. 1041-1048
-
-
McCarty, M.F.1
Wey, J.2
Stoeltzing, O.3
Liu, W.4
Fan, F.5
Bucana, C.6
Mansfield, P.F.7
Ryan, A.J.8
Ellis, L.M.9
-
114
-
-
10744227153
-
-
D.E. Gingrich, D.R. Reddy, M.A. Iqbal, J. Singh, L.D. Aimone, T.S. Angeles, M. Albom, S. Yang, M.A. Ator, S.L. Meyer, C. Robinson, B.A. Ruggeri, C.A. Dionne, J.L. Vaught, J.P. Mallamo, and R.L. Hudkins J. Med. Chem. 46 2003 5375 5388
-
(2003)
J. Med. Chem.
, vol.46
, pp. 5375-5388
-
-
Gingrich, D.E.1
Reddy, D.R.2
Iqbal, M.A.3
Singh, J.4
Aimone, L.D.5
Angeles, T.S.6
Albom, M.7
Yang, S.8
Ator, M.A.9
Meyer, S.L.10
Robinson, C.11
Ruggeri, B.A.12
Dionne, C.A.13
Vaught, J.L.14
Mallamo, J.P.15
Hudkins, R.L.16
-
115
-
-
3242806740
-
-
J.T. Hunt, T. Mitt, R. Borzilleri, J.G. Brown, J. Fargnoli, B. Fink, W.C. Han, S. Mortillo, G. Vite, B. Wautlet, T. Wong, C. Yu, X. Zheng, and R. Bhide J. Med. Chem. 27 2004 4054 4059
-
(2004)
J. Med. Chem.
, vol.27
, pp. 4054-4059
-
-
Hunt, J.T.1
Mitt, T.2
Borzilleri, R.3
Brown, J.G.4
Fargnoli, J.5
Fink, B.6
Han, W.C.7
Mortillo, S.8
Vite, G.9
Wautlet, B.10
Wong, T.11
Yu, C.12
Zheng, X.13
Bhide, R.14
-
116
-
-
25144513049
-
-
B.E. Fink, G.D. Vite, H. Mastalerz, J.F. Kadow, S.H. Kim, K.J. Leavitt, K. Du, D. Crews, T. Mitt, T.W. Wong, J.T. Hunt, D.M. Vyas, and J.S. Tokarski Biorg. Med. Chem. 15 2005 4774 4779
-
(2005)
Biorg. Med. Chem.
, vol.15
, pp. 4774-4779
-
-
Fink, B.E.1
Vite, G.D.2
Mastalerz, H.3
Kadow, J.F.4
Kim, S.H.5
Leavitt, K.J.6
Du, K.7
Crews, D.8
Mitt, T.9
Wong, T.W.10
Hunt, J.T.11
Vyas, D.M.12
Tokarski, J.S.13
-
117
-
-
20444385804
-
-
R.M. Borzilleri, X. Zheng, L. Qian, C. Ellis, Z. Cai, B.S. Wautlet, S. Mortillo, R. Jeyaseelan Sr., S.W. Kukrai, A. Fura, A. Kamath, V. Vyas, J.S. Tokaski, J.C. Barrish, J.T. Hunt, L.J. Lombardo, J. Farnoli, and R.S. Bhide J. Med. Chem. 48 2005 3991 4008
-
(2005)
J. Med. Chem.
, vol.48
, pp. 3991-4008
-
-
Borzilleri, R.M.1
Zheng, X.2
Qian, L.3
Ellis, C.4
Cai, Z.5
Wautlet, B.S.6
Mortillo, S.7
Jeyaseelan Sr., R.8
Kukrai, S.W.9
Fura, A.10
Kamath, A.11
Vyas, V.12
Tokaski, J.S.13
Barrish, J.C.14
Hunt, J.T.15
Lombardo, L.J.16
Farnoli, J.17
Bhide, R.S.18
-
118
-
-
4944227798
-
-
S. Emanuel, R.H. Gruninger, A.F. Pasquera, P.J. Connoly, J.A. Seamon, S. Hazel, R. Tominovich, B. Hollister, C. Napier, M.R. D'Andrea, M. Reuman, G. Bignan, R. Tuman, D. Johnson, D. Moffati, M. Batchelor, A. Foley, J. O'Connell, R. Allen, M. Perry, L. Jolliffe, and S.A. Middleton Mol. Pharmacol. 66 2004 635 647
-
(2004)
Mol. Pharmacol.
, vol.66
, pp. 635-647
-
-
Emanuel, S.1
Gruninger, R.H.2
Pasquera, A.F.3
Connoly, P.J.4
Seamon, J.A.5
Hazel, S.6
Tominovich, R.7
Hollister, B.8
Napier, C.9
D'Andrea, M.R.10
Reuman, M.11
Bignan, G.12
Tuman, R.13
Johnson, D.14
Moffati, D.15
Batchelor, M.16
Foley, A.17
O'Connell, J.18
Allen, R.19
Perry, M.20
Jolliffe, L.21
Middleton, S.A.22
more..
-
121
-
-
8844234957
-
-
V.A. Nair, S.M. Mustafa, M.L. Mohler, S.J. Fisher, J.T. Dalton, and D.D. Miller Tetrahedron Lett. 45 2004 9475 9477 (and references cited therein)
-
(2004)
Tetrahedron Lett.
, vol.45
, pp. 9475-9477
-
-
Nair, V.A.1
Mustafa, S.M.2
Mohler, M.L.3
Fisher, S.J.4
Dalton, J.T.5
Miller, D.D.6
-
122
-
-
0037038324
-
-
H. Ohtsu, Z. Xiao, J. Ishida, M. Nagai, H.K. Wang, H. Itokawa, C.Y. Su, C. Shih, T. Chiand, E. Chang, Y. Lee, M.Y. Tsai, C. Chang, and K.H. Lee J. Med. Chem. 45 2002 5037 5042 (and references cited therein)
-
(2002)
J. Med. Chem.
, vol.45
, pp. 5037-5042
-
-
Ohtsu, H.1
Xiao, Z.2
Ishida, J.3
Nagai, M.4
Wang, H.K.5
Itokawa, H.6
Su, C.Y.7
Shih, C.8
Chiand, T.9
Chang, E.10
Lee, Y.11
Tsai, M.Y.12
Chang, C.13
Lee, K.H.14
-
123
-
-
33645456701
-
-
M. Sani, F. Viani, M. Binda, N. Zaffaroni, and M. Zanda Lett. Org. Chem. 2 2005 447 449
-
(2005)
Lett. Org. Chem.
, vol.2
, pp. 447-449
-
-
Sani, M.1
Viani, F.2
Binda, M.3
Zaffaroni, N.4
Zanda, M.5
-
124
-
-
0035445644
-
-
M.R. Karagas, G.L. Cushing Jr., E.R. Greeberg, L.A. Mott, S.K. Spencer, and D.W. Nierenberg Br. J. Cancer 85 2001 683 686
-
(2001)
Br. J. Cancer
, vol.85
, pp. 683-686
-
-
Karagas, M.R.1
Cushing Jr., G.L.2
Greeberg, E.R.3
Mott, L.A.4
Spencer, S.K.5
Nierenberg, D.W.6
-
125
-
-
0347719371
-
-
H. Schacke, A. Schottelius, W.D. Docke, P. Strehlke, S. Jaroch, N. Schmees, H. Rehwinkel, H. Hennekes, and K. Asadullah Proc. Natl. Acad. Sci. U.S.A. 101 2004 227 232
-
(2004)
Proc. Natl. Acad. Sci. U.S.A.
, vol.101
, pp. 227-232
-
-
Schacke, H.1
Schottelius, A.2
Docke, W.D.3
Strehlke, P.4
Jaroch, S.5
Schmees, N.6
Rehwinkel, H.7
Hennekes, H.8
Asadullah, K.9
-
126
-
-
25144466090
-
-
R. Batageri, Y. Zhang, R.M. Zindell, D.K. Kuzmich, T.M. Kirrane, J. Bentzien, M. Cardozo, A.J. Capolino, T.N. Fadara, R.M. Nelson, Z. Paw, D.T. Shih, C.K. Shih, L.Z. Jelaska, G. Nabozny, and D.S. Thomson Biorg. Med. Chem. Lett. 15 2005 4761 4769
-
(2005)
Biorg. Med. Chem. Lett.
, vol.15
, pp. 4761-4769
-
-
Batageri, R.1
Zhang, Y.2
Zindell, R.M.3
Kuzmich, D.K.4
Kirrane, T.M.5
Bentzien, J.6
Cardozo, M.7
Capolino, A.J.8
Fadara, T.N.9
Nelson, R.M.10
Paw, Z.11
Shih, D.T.12
Shih, C.K.13
Jelaska, L.Z.14
Nabozny, G.15
Thomson, D.S.16
-
127
-
-
22244432464
-
-
M. Barker, M. Clackers, D.A. Demaine, D. Humphreys, M.J. Johnston, H.T. Jones, F. Pacquet, J.M. Pritchard, M. Salter, S.E. Shanahan, P.A. Skone, V.M. Vinader, I. Uings, I.M. McLay, and S.J.F. Macdonald J. Med. Chem. 48 2005 4507 4510 (and references cited therein)
-
(2005)
J. Med. Chem.
, vol.48
, pp. 4507-4510
-
-
Barker, M.1
Clackers, M.2
Demaine, D.A.3
Humphreys, D.4
Johnston, M.J.5
Jones, H.T.6
Pacquet, F.7
Pritchard, J.M.8
Salter, M.9
Shanahan, S.E.10
Skone, P.A.11
Vinader, V.M.12
Uings, I.13
McLay, I.M.14
MacDonald, S.J.F.15
-
129
-
-
0032573082
-
-
S.A. Peterson, T. Klabunde, H.A. Lashuel, H. Purkey, J.C. Sacchettini, and J.W. Kelly Proc. Natl. Acad. Sci. U.S.A. 95 1998 12956 12960
-
(1998)
Proc. Natl. Acad. Sci. U.S.A.
, vol.95
, pp. 12956-12960
-
-
Peterson, S.A.1
Klabunde, T.2
Lashuel, H.A.3
Purkey, H.4
Sacchettini, J.C.5
Kelly, J.W.6
-
131
-
-
26444568206
-
-
R.E. Armer, M.R. Ashton, E.A. Boyd, C.J. Brennan, F.A. Brookfield, L. Gazi, S.L. Gyles, P.A. Hay, M.G. Hunter, D. Middlemiss, M. Whittaker, L. Xue, and R. Pettipher J. Med. Chem. 48 2005 6174 6177
-
(2005)
J. Med. Chem.
, vol.48
, pp. 6174-6177
-
-
Armer, R.E.1
Ashton, M.R.2
Boyd, E.A.3
Brennan, C.J.4
Brookfield, F.A.5
Gazi, L.6
Gyles, S.L.7
Hay, P.A.8
Hunter, M.G.9
Middlemiss, D.10
Whittaker, M.11
Xue, L.12
Pettipher, R.13
-
135
-
-
14944371100
-
-
N.A. Nussmeier, A.A. Whelton, M.T. Brown, R.M. Langford, A. Hoeft, and J.L. Parlow N. Engl. J. Med. 352 2005 1081 1091
-
(2005)
N. Engl. J. Med.
, vol.352
, pp. 1081-1091
-
-
Nussmeier, N.A.1
Whelton, A.A.2
Brown, M.T.3
Langford, R.M.4
Hoeft, A.5
Parlow, J.L.6
-
136
-
-
13944253576
-
-
J.C. Mozziconacci, E. Arnoult, P. Bernard, Q.T. Do, C. Marot, and L.M. Allory J. Med. Chem. 48 2005 1055 1068
-
(2005)
J. Med. Chem.
, vol.48
, pp. 1055-1068
-
-
Mozziconacci, J.C.1
Arnoult, E.2
Bernard, P.3
Do, Q.T.4
Marot, C.5
Allory, L.M.6
-
139
-
-
1842628789
-
-
E.R. Lepper, S.S.W. Ng, M. Gütschow, M. Weiss, S. Hauschildt, T.K. Hecker, F.A. Luzzio, K. Eger, and W.D. Figg J. Med. Chem. 47 2004 2219 2227 (and references cited therein)
-
(2004)
J. Med. Chem.
, vol.47
, pp. 2219-2227
-
-
Lepper, E.R.1
Ng, S.S.W.2
Gütschow, M.3
Weiss, M.4
Hauschildt, S.5
Hecker, T.K.6
Luzzio, F.A.7
Eger, K.8
Figg, W.D.9
-
140
-
-
0001093384
-
-
Y. Takeuchi, T. Shiragami, K. Kimura, E. Suzuki, and N. Shibata Org. Lett. 1 1999 1571 1573
-
(1999)
Org. Lett.
, vol.1
, pp. 1571-1573
-
-
Takeuchi, Y.1
Shiragami, T.2
Kimura, K.3
Suzuki, E.4
Shibata, N.5
-
142
-
-
20244384283
-
-
A. de Dios, C. Shih, B.L. de Uralde, C. Sánchez, M. del Prado, L.M.M. Cabrejas, S. Pleite, J.B. Urgoiti, M.J. Lorite, C.R. Nevill Jr., R. Bonjoukhian, J. York, M. Veith, Y. Wang, N. Magnus, R.M. Campbell, B.D. Anderson, D.J. McCann, D.D. Giera, P.A. Lee, R.M. Schultz, L.C. Li, L.M. Johnson, and J.A. Wolos J. Med. Chem. 48 2005 2270 2273
-
(2005)
J. Med. Chem.
, vol.48
, pp. 2270-2273
-
-
De Dios, A.1
Shih, C.2
De Uralde, B.L.3
Sánchez, C.4
Del Prado, M.5
Cabrejas, L.M.M.6
Pleite, S.7
Urgoiti, J.B.8
Lorite, M.J.9
Nevill Jr., C.R.10
Bonjoukhian, R.11
York, J.12
Veith, M.13
Wang, Y.14
Magnus, N.15
Campbell, R.M.16
Anderson, B.D.17
McCann, D.J.18
Giera, D.D.19
Lee, P.A.20
Schultz, R.M.21
Li, L.C.22
Johnson, L.M.23
Wolos, J.A.24
more..
-
145
-
-
23944478339
-
-
O. El-Kabbani, V. Carbone, C. Darmanin, M. Oka, A. Mitschler, A. Podjarny, C.S. Briese, and R.P.T. Chung J. Med. Chem. 48 2005 5536 5542
-
(2005)
J. Med. Chem.
, vol.48
, pp. 5536-5542
-
-
El-Kabbani, O.1
Carbone, V.2
Darmanin, C.3
Oka, M.4
Mitschler, A.5
Podjarny, A.6
Briese, C.S.7
Chung, R.P.T.8
-
147
-
-
13944276311
-
-
J.W.F. Whitehead, G.P. Lee, P. Gharagozloo, P. Hofer, A. Gehrig, P. Wintergerst, D. Symth, W. McCoull, M. Hachicha, A. Patel, and D.J. Kyle J. Med. Chem. 48 2005 1237 1243
-
(2005)
J. Med. Chem.
, vol.48
, pp. 1237-1243
-
-
Whitehead, J.W.F.1
Lee, G.P.2
Gharagozloo, P.3
Hofer, P.4
Gehrig, A.5
Wintergerst, P.6
Symth, D.7
McCoull, W.8
Hachicha, M.9
Patel, A.10
Kyle, D.J.11
-
148
-
-
0035254533
-
-
S.M. Thacher, J. Vasudevan, K.Y. Tsang, S. Nagpal, and R.A.S. Chandraratna J. Med. Chem. 44 2001 281 297
-
(2001)
J. Med. Chem.
, vol.44
, pp. 281-297
-
-
Thacher, S.M.1
Vasudevan, J.2
Tsang, K.Y.3
Nagpal, S.4
Chandraratna, R.A.S.5
-
150
-
-
22844449890
-
-
Z. Guo, D. Wu, Y.F. Zhu, F.C. Tucci, C.F. Regan, M.W. Rowbottom, R.S. Struthers, Q. Xie, S. Reijmers, S.K. Sullivan, Y. Sai, and C. Chen Biorg. Med. Chem. Lett. 15 2005 3685 3690
-
(2005)
Biorg. Med. Chem. Lett.
, vol.15
, pp. 3685-3690
-
-
Guo, Z.1
Wu, D.2
Zhu, Y.F.3
Tucci, F.C.4
Regan, C.F.5
Rowbottom, M.W.6
Struthers, R.S.7
Xie, Q.8
Reijmers, S.9
Sullivan, S.K.10
Sai, Y.11
Chen, C.12
-
153
-
-
0242443308
-
-
M. Kunkel, G.J. Forster, T.E. Reichert, J.-H. Jeong, P. Benz, P. Bartenstein, W. Wagner, and T.L. Whiteside Cancer 98 2003 2257 2265
-
(2003)
Cancer
, vol.98
, pp. 2257-2265
-
-
Kunkel, M.1
Forster, G.J.2
Reichert, T.E.3
Jeong, J.-H.4
Benz, P.5
Bartenstein, P.6
Wagner, W.7
Whiteside, T.L.8
-
156
-
-
0034667846
-
-
N. Avril, C.A. Rosé, M. Schelling, J. Dose, W. Kuhn, S. Bense, W. Weber, S. Ziegler, H. Graeff, and M. Schwaiger J. Clin. Oncol. 18 2000 3495 3502
-
(2000)
J. Clin. Oncol.
, vol.18
, pp. 3495-3502
-
-
Avril, N.1
Rosé, C.A.2
Schelling, M.3
Dose, J.4
Kuhn, W.5
Bense, S.6
Weber, W.7
Ziegler, S.8
Graeff, H.9
Schwaiger, M.10
-
157
-
-
25144508684
-
-
T. Toyokuni, J.S.D. Kumar, J.C. Walsh, A. Shapiro, J.J. Talley, M.E. Phelps, H.R. Herschman, J.R. Barrio, and N. Satyamurthy Biorg. Med. Chem. Lett. 15 2005 4699 4702
-
(2005)
Biorg. Med. Chem. Lett.
, vol.15
, pp. 4699-4702
-
-
Toyokuni, T.1
Kumar, J.S.D.2
Walsh, J.C.3
Shapiro, A.4
Talley, J.J.5
Phelps, M.E.6
Herschman, H.R.7
Barrio, J.R.8
Satyamurthy, N.9
-
160
-
-
25844485927
-
-
O. Jacobson, Y. Bechor, A. Icar, N. Novak, A. Birman, H. Marom, L. Fadeeva, E. Golan, I. Leibovitch, M. Gutman, E.E. Sapir, R. Chisin, M. Gozin, and E. Mishani Biorg. Med. Chem. 13 2005 6195 6205
-
(2005)
Biorg. Med. Chem.
, vol.13
, pp. 6195-6205
-
-
Jacobson, O.1
Bechor, Y.2
Icar, A.3
Novak, N.4
Birman, A.5
Marom, H.6
Fadeeva, L.7
Golan, E.8
Leibovitch, I.9
Gutman, M.10
Sapir, E.E.11
Chisin, R.12
Gozin, M.13
Mishani, E.14
-
161
-
-
0344120151
-
-
L. Martarello, C. Schaffrath, H. Deng, A.D. Gee, A. Lockhart, and D. O'Hagan J. Label. Compd. Radiopharm. 46 2003 1181 1189
-
(2003)
J. Label. Compd. Radiopharm.
, vol.46
, pp. 1181-1189
-
-
Martarello, L.1
Schaffrath, C.2
Deng, H.3
Gee, A.D.4
Lockhart, A.5
O'Hagan, D.6
-
162
-
-
33645460289
-
-
H. Deng, S.L. Cobb, A.D. Gee, A. Lockhart, L. Martarello, R.P. McGlinchey, D. O'Hagan, and M. Onega Chem. Commun. 2006 652 654
-
(2006)
Chem. Commun.
, pp. 652-654
-
-
Deng, H.1
Cobb, S.L.2
Gee, A.D.3
Lockhart, A.4
Martarello, L.5
McGlinchey, R.P.6
O'Hagan, D.7
Onega, M.8
-
163
-
-
1142310932
-
-
C. Dong, F. Lu-Huang, H. Deng, C. Schaffrath, J.B. Spencer, D. O'Hagan, and J.H. Naismith Nature 427 2004 561 565
-
(2004)
Nature
, vol.427
, pp. 561-565
-
-
Dong, C.1
Lu-Huang, F.2
Deng, H.3
Schaffrath, C.4
Spencer, J.B.5
O'Hagan, D.6
Naismith, J.H.7
-
164
-
-
1542286627
-
-
W. Cui, P. Otten, Y. Li, K.S. Koeneman, J. Yu, and R.P. Mason Magn. Resonance Med. 51 2004 616 620
-
(2004)
Magn. Resonance Med.
, vol.51
, pp. 616-620
-
-
Cui, W.1
Otten, P.2
Li, Y.3
Koeneman, K.S.4
Yu, J.5
Mason, R.P.6
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