Structure-activity relationships of 1,3,5-triazine-2,4,6-triones as human gonadotropin-releasing hormone receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 16, 2005, Pages 3685-3690

  Guo, Zhiqiang ^a   Wu, Dongpei ^a   Zhu, Yun Fei ^a   Tucci, Fabio C ^a   Regan, Collin F ^a   Rowbottom, Martin W ^a   Struthers, R Scott ^a   Xie, Qiu ^a   Reijmers, Shelby ^a   Sullivan, Susan K ^a   Sai, Yang ^a   Chen, Chen ^a  

^a NEUROCRINE BIOSCIENCES INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CYANURIC ACID; GONADORELIN ANTAGONIST;

ARTICLE; CONTROLLED STUDY; DRUG PENETRATION; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STABILITY; DRUG SYNTHESIS; EMBRYO; HUMAN; HUMAN CELL; STRUCTURE ACTIVITY RELATION;

DRUG EVALUATION, PRECLINICAL; HUMANS; MOLECULAR STRUCTURE; RECEPTORS, LHRH; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZINES;

EID: 22844449890     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.05.038     Document Type: Article

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