The heptahelical domain of GABAB2 is activated directly by CGP7930, a positive allosteric modulator of the GABAB receptor

Journal of Biological Chemistry

Volumn 279, Issue 28, 2004, Pages 29085-29091

  Binet, Virginie ^a   Brajon, Carole ^a   Le Corre, Laurent ^b   Acher, Francine ^b   Pin, Jean Philippe ^a   Prézeau, Laurent ^a,c  

^a INSERM   (France)

^b CNRS   (France)

^c INSTITUT DE GÉNOMIQUE FONCTIONNELLE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

BIOCHEMISTRY; BRAIN; CELLS; MOLECULAR STRUCTURE; PROTEINS;

AMINOBUTYRIC ACID; HOMOLOGY;

ORGANIC ACIDS;

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID B RECEPTOR STIMULATING AGENT; 4 AMINOBUTYRIC ACID B1 RECEPTOR; 4 AMINOBUTYRIC ACID B2 RECEPTOR; 4 AMINOBUTYRIC ACID B2 RECEPTOR STIMULATING AGENT; CGP 7930; G PROTEIN COUPLED RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; RECEPTOR; RECEPTOR SUBUNIT; RHODOPSIN; RHODOPSIN LIKE RECEPTOR; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; CELL SURFACE; CONCENTRATION RESPONSE; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; EXTRACELLULAR DOMAIN; HEPTAHELICAL DOMAIN; HUMAN; HUMAN CELL; MODULATION; PRIORITY JOURNAL; PROTEIN DOMAIN; RECEPTOR BINDING; RECEPTOR UPREGULATION; SEQUENCE HOMOLOGY;

EID: 3142685557     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.M400930200     Document Type: Article

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