Molecular Determinants Involved in the Allosteric Control of Agonist Affinity in the GABAB Receptor by the GABAB2 Subunit

Journal of Biological Chemistry

Volumn 279, Issue 16, 2004, Pages 15824-15830

  Liu, Jianfeng ^a,c   Maurel, Damien ^a,b   Etzol, Sébastien ^a   Brabet, Isabelle ^a   Ansanay, Hervé ^b   Pin, Jean Philippe ^a   Rondard, Philippe ^a  

^a INSTITUT DE GÉNOMIQUE FONCTIONNELLE   (France)

^b CIS Bio International   (France)

^c HUAZHONG UNIVERSITY OF SCIENCE AND TECHNOLOGY   (China)

Author keywords

[No Author keywords available]

Indexed keywords

ENERGY TRANSFER; FLUORESCENCE; OLIGOMERS; PROTEINS;

ALLOSTERIC CONTROL; HEPTAHELICAL DOMAIN (HD);

BIOCHEMISTRY;

4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID B RECEPTOR STIMULATING AGENT; 4 AMINOBUTYRIC ACID B1 RECEPTOR; 4 AMINOBUTYRIC ACID B2 RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; RECEPTOR SUBUNIT; UNCLASSIFIED DRUG;

ALLOSTERISM; ANIMAL CELL; ARTICLE; CARBOXY TERMINAL SEQUENCE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; EMBRYO; FLUORESCENCE RESONANCE ENERGY TRANSFER; HUMAN; HUMAN CELL; MOLECULAR BIOLOGY; MOLECULAR DYNAMICS; MOLECULAR INTERACTION; NONHUMAN; OLIGOMERIZATION; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN FUNCTION; PROTEIN PROTEIN INTERACTION; PROTEIN STRUCTURE;

ALLOSTERIC REGULATION; BINDING SITES; CELL LINE; GABA AGONISTS; HUMANS; MODELS, MOLECULAR; PROTEIN SUBUNITS; RECEPTORS, GABA-B; SIGNAL TRANSDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP;

ANIMALIA; DIONAEA;

EID: 1942469528     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.M313639200     Document Type: Article

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