Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors

Proceedings of the National Academy of Sciences of the United States of America

Volumn 101, Issue 1, 2004, Pages 378-383

  Goudett, Cyril ^a   Gaven, Florence ^a   Kniazeff, Julie ^a   Vol, Claire ^a   Liu, Jiangfeng ^a   Cohen Gonsaud, Martin ^a   Acher, Francine ^a   Prézeau, Laurent ^a   Pin, Jean Philippe ^a  

^a CNRS   (France)

Author keywords

Activation mechanism; Allostery; G protein coupled receptor; Inverse agonism; Modulator

Indexed keywords

2 METHYL 6 (PHENYLETHYNYL)PYRIDINE; 3,3' DIFLUOROBENZALDAZINE; FLUOROBENZENE; G PROTEIN COUPLED RECEPTOR; METABOTROPIC RECEPTOR 5; RECEPTOR; RHODOPSIN LIKE RECEPTOR; UNCLASSIFIED DRUG;

AGONIST; ALLOSTERISM; ARTICLE; CONTROLLED STUDY; HUMAN; HUMAN CELL; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN DOMAIN; RECEPTOR BINDING; REGULATORY MECHANISM;

ALLOSTERIC REGULATION; ANIMALS; CELL LINE; CELL MEMBRANE; HUMANS; HYDRAZINES; KINETICS; MODELS, MOLECULAR; PEPTIDE FRAGMENTS; PROTEIN STRUCTURE, TERTIARY; PYRIDINES; RATS; RECEPTORS, METABOTROPIC GLUTAMATE; RECOMBINANT PROTEINS; RHODOPSIN; SEQUENCE DELETION;

DIONAEA;

EID: 0346458626     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.0304699101     Document Type: Article

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