Activation mechanism of the heterodimeric GABA B receptor

Biochemical Pharmacology

Volumn 68, Issue 8, 2004, Pages 1565-1572

  Pin, Jean Philippe ^a   Kniazeff, Julie ^a   Binet, Virginie ^a   Liu, Jianfeng ^a   Maurel, Damien ^a,c   Galvez, Thierry ^a   Duthey, Béatrice ^a   Havlickova, Michaela ^b   Blahos, Jaroslav ^b   Prézeau, Laurent ^a   Rondard, Philippe ^a  

^a Laboratory of Functional Genomic   (France)

^b INSTITUTE OF MATHEMATICS   (Czech Republic)

^c CIS Bio International   (France)

Author keywords

Activation; Allosteric regulator; Baclofen; Dimerization; G protein coupled receptors; GABA B receptor

Indexed keywords

4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID B RECEPTOR STIMULATING AGENT; CGP 7930; G PROTEIN COUPLED RECEPTOR; RECEPTOR SUBUNIT;

ALLOSTERISM; AMINO ACID SEQUENCE; ARTICLE; BINDING AFFINITY; CIS ISOMER; DIMERIZATION; DRUG RECEPTOR BINDING; HUMAN; MOLECULAR CLONING; MOLECULAR RECOGNITION; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN FUNCTION; SIGNAL TRANSDUCTION; TRANS ISOMER;

ALLOSTERIC REGULATION; ANIMALS; BACLOFEN; DIMERIZATION; GABA AGONISTS; GAMMA-AMINOBUTYRIC ACID; GTP-BINDING PROTEINS; HUMANS; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; PROTEIN SUBUNITS; RECEPTORS, G-PROTEIN-COUPLED; RECEPTORS, GABA-B;

EID: 4644296105     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bcp.2004.06.035     Document Type: Article

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