Corticotropin releasing hormone - A GPCR drug target

Current Drug Targets

Volumn 8, Issue 1, 2007, Pages 105-115

  Hemley, C F ^a   McCluskey, A ^b   Keller, P A ^a  

^a UNIVERSITY OF WOLLONGONG   (Australia)

^b UNIVERSITY OF NEWCASTLE   (Australia)

Author keywords

Corticotrophin Releasing Hormone; Drug design; GPCR receptor

Indexed keywords

3 (6 DIMETHYLAMINO 4 METHYL 3 PYRIDINYL) 7 DIPROPYLAMINO 2,5 DIMETHYLPYRAZOLO[1,5 A]PYRIMIDINE; AMINO ACID; ANTIDEPRESSANT AGENT; ANXIOLYTIC AGENT; ASTRESSIN; BINDING PROTEIN; CORTICOTROPIN RELEASING FACTOR; CORTICOTROPIN RELEASING FACTOR AGONIST; CORTICOTROPIN RELEASING FACTOR ANTAGONIST; CORTICOTROPIN RELEASING FACTOR BINDING PROTEIN; CORTICOTROPIN RELEASING FACTOR RECEPTOR 1; CORTICOTROPIN RELEASING FACTOR RECEPTOR 2; CORTICOTROPIN RELEASING FACTOR RECEPTOR 3; G PROTEIN COUPLED RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; HORMONE RECEPTOR; LIGAND; NBI 34041; NBI 37582; PEPTIDE DERIVATIVE; PYRAZOLONE DERIVATIVE; RHODOPSIN; SAUVAGINE; SB 723620; UNCLASSIFIED DRUG; UNINDEXED DRUG; UROCORTIN; UROCORTIN I; UROCORTIN II; UROCORTIN III; UROTENSIN;

ALZHEIMER DISEASE; ANXIETY DISORDER; BINDING AFFINITY; BRAIN EDEMA; BRAIN ISCHEMIA; CLINICAL TRIAL; CRYSTALLIZATION; DEPRESSION; DRUG DESIGN; DRUG MEGADOSE; DRUG STRUCTURE; DRUG TARGETING; HUMAN; LIVER TOXICITY; NONHUMAN; PAIN; PREMATURITY; PROTEIN FUNCTION; PROTEIN LOCALIZATION; RECEPTOR BINDING; RECEPTOR INTRINSIC ACTIVITY; REVIEW; SIGNAL TRANSDUCTION;

AMINO ACID SEQUENCE; ANIMALS; CORTICOTROPIN-RELEASING HORMONE; DRUG DELIVERY SYSTEMS; HUMANS; MOLECULAR SEQUENCE DATA; RECEPTORS, CORTICOTROPIN-RELEASING HORMONE; RECEPTORS, G-PROTEIN-COUPLED;

EID: 33846002760     PISSN: 13894501     EISSN: None     Source Type: Journal    
DOI: 10.2174/138945007779315542     Document Type: Review

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