CP-154,526: A potent and selective nonpeptide antagonist of corticotropin releasing factor receptors

Proceedings of the National Academy of Sciences of the United States of America

Volumn 93, Issue 19, 1996, Pages 10477-10482

  Schulz, David W ^a   Mansbach, Robert S ^a   Sprouse, Jeffrey ^a   Braselton, John P ^a   Collins, Judy ^a   Corman, Michael ^a   Dunaiskis, Audrey ^a   Faraci, Steve ^a   Schmidt, Anne W ^a   Seeger, Thomas ^a   Seymour, Patricia ^a   Tingley III, F David ^a   Winston, Elizabeth N ^a   Chen, Yuhpyng L ^a   Heym, James ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ADENYLATE CYCLASE; BUTYL[2,5 DIMETHYL 7 (2,4,6 TRIMETHYLPHENYL) 7H PYRROLO[2,3 D]PYRIMIDIN 4 YL]ETHYLAMINE; CORTICOTROPIN; CORTICOTROPIN RELEASING FACTOR RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; ENZYME ACTIVATION; ENZYME ACTIVITY; IMMUNOREACTIVITY; LOCUS CERULEUS; MELANCHOLIA; NEUROMODULATION; NORADRENERGIC SYSTEM; PRIORITY JOURNAL; RECEPTOR BINDING;

ACOUSTIC STIMULATION; ADENYLATE CYCLASE; ADRENOCORTICOTROPIC HORMONE; ANIMALS; BINDING, COMPETITIVE; CALLITHRIX; CELL LINE; CELL MEMBRANE; CEREBRAL CORTEX; CEREBRAL VENTRICLES; CORTICOTROPIN-RELEASING HORMONE; DOGS; GUINEA PIGS; HUMANS; INJECTIONS, INTRAVENTRICULAR; KINETICS; LOCUS COERULEUS; MALE; NEURONS; PITUITARY GLAND; PYRIMIDINES; PYRROLES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, CORTICOTROPIN-RELEASING HORMONE; STARTLE REACTION;

EID: 0013522651     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.93.19.10477     Document Type: Article

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