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Volumn 10, Issue 1, 2002, Pages 175-183

CRHR1 Receptor binding and lipophilicity of pyrrolopyrimidines, potential nonpeptide corticotropin-releasing hormone type 1 receptor antagonists

(13) Hsin, Ling Wei a Tian, Xinrong a Webster, Elizabeth L b,c Coop, Andrew d Caldwell, Timothy M a Jacobson, Arthur E a Chrousos, George P c Gold, Philip W b Habib, Kamal E b Ayala, Alejandro b Eckelman, William C e Contoreggi, Carlo f Rice, Kenner C a

a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES (United States)

b NATIONAL INSTITUTE OF MENTAL HEALTH (United States)

c EUNICE KENNEDY SHRIVER NATIONAL INSTITUTE OF CHILD HEALTH AND HUMAN DEVELOPMENT (United States)

d UNIVERSITY OF MARYLAND SCHOOL OF PHARMACY (United States)

e NATIONAL INSTITUTES OF HEALTH (United States)

f NATIONAL INSTITUTE ON DRUG ABUSE (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTALARMIN; CORTICOTROPIN RELEASING FACTOR; CORTICOTROPIN RELEASING FACTOR ANTAGONIST; DIMETHYL SULFOXIDE; HYDROXYL GROUP; PYRROLOPYRIMIDINE DERIVATIVE; CORTICOTROPIN RELEASING FACTOR RECEPTOR; PYRIMIDINE DERIVATIVE; PYRROLE DERIVATIVE; RECEPTORS, CORTICOTROPIN RELEASING HORMONE;

ARTICLE; CONTROLLED STUDY; DRUG DEVELOPMENT; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; LIPOPHILICITY; NONHUMAN; ANIMAL; CHEMISTRY; MALE; MASS SPECTROMETRY; METABOLISM; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PROTEIN BINDING; RAT; RAT STRAIN;

ANIMAL; MAGNETIC RESONANCE SPECTROSCOPY; MALE; PROTEIN BINDING; PYRIMIDINES; PYRROLES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, CORTICOTROPIN-RELEASING HORMONE; SPECTRUM ANALYSIS, MASS;

EID: 0036006471 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00261-9 Document Type: Article

Times cited : (38)

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