-
1
-
-
0011235592
-
-
R. Neier, Ed.; Thieme Verlag: Stuttgart
-
Stanovnik, B.; Svete, J. In: Science of Synthesis, R. Neier, Ed.; Thieme Verlag: Stuttgart, 2002; Vol. 12, pp. 15-225.
-
(2002)
Science of Synthesis
, vol.12
, pp. 15-225
-
-
Stanovnik, B.1
Svete, J.2
-
2
-
-
0039539863
-
-
Schaumann, E, Ed.; Thieme Verlag
-
Kirschke, K. In: Houben-Weyl, Methoden der organischen Chemie,; Schaumann, E, Ed.; Thieme Verlag, 1994, Vol. E8b, 399-763.
-
(1994)
Houben-Weyl, Methoden Der Organischen Chemie
, vol.E8b
, pp. 399-763
-
-
Kirschke, K.1
-
3
-
-
0000756640
-
-
D. H. R. Barton, W. D. Ollis, Eds.; Pergamon: Oxford
-
Grimmett, M.R. In: Comprehensive Organic Chemistry, D. H. R. Barton, W. D. Ollis, Eds.; Pergamon: Oxford, 1979, 4, 357-410.
-
(1979)
Comprehensive Organic Chemistry
, vol.4
, pp. 357-410
-
-
Grimmett, M.R.1
-
4
-
-
0004246795
-
-
R. C. Elderfield, Ed.; Wiley: New York
-
Jacobs, T.L. In: Heterocyclic Compounds, R. C. Elderfield, Ed.; Wiley: New York 1957, 5, 45-162.
-
(1957)
Heterocyclic Compounds
, vol.5
, pp. 45-162
-
-
Jacobs, T.L.1
-
6
-
-
0003593749
-
-
Interscience: New York
-
Behr, L.C.; Fusco, R.; Jarboe, C.H. In: The Chemistry of Heterocyclic Compounds, Interscience: New York, 1967, vol. 22, pp. 10-64.
-
(1967)
The Chemistry of Heterocyclic Compounds
, vol.22
, pp. 10-64
-
-
Behr, L.C.1
Fusco, R.2
Jarboe, C.H.3
-
7
-
-
84943407995
-
-
A. R. Katritzky, C. W. Rees, Eds.; Pergamon: Oxford
-
Elguero, J. In: Comprehensive Heterocyclic Chemistry, A. R. Katritzky, C. W. Rees, Eds.; Pergamon: Oxford 1984, vol. 5, pp. 167-303.
-
(1984)
Comprehensive Heterocyclic Chemistry
, vol.5
, pp. 167-303
-
-
Elguero, J.1
-
8
-
-
84944033746
-
-
A. R. Katritzky, E. F. V. Scriven, Eds.; Elsevier: Oxford
-
Elguero, J. In: Comprehensive Heterocyclic Chemistry II, A. R. Katritzky, E. F. V. Scriven, Eds.; Elsevier: Oxford 1996, vol. 3, pp. 1-75.
-
(1996)
Comprehensive Heterocyclic Chemistry II
, vol.3
, pp. 1-75
-
-
Elguero, J.1
-
9
-
-
0032950304
-
Synthesis of pyrazoles and condensed pyrazoles
-
Makino, K.; Kim, H.S.; Kurasawa, Y. Synthesis of pyrazoles and condensed pyrazoles. J. Heterocycl. Chem., 1999, 36(2), 321-332.
-
(1999)
J. Heterocycl. Chem
, vol.36
, Issue.2
, pp. 321-332
-
-
Makino, K.1
Kim, H.S.2
Kurasawa, Y.3
-
10
-
-
1542607035
-
Synthesis of pyrazoles
-
Makino, K.; Kim, H.S.; Kurasawa, Y. Synthesis of pyrazoles. J. Heterocycl. Chem., 1998, 35(3), 489-497.
-
(1998)
J. Heterocycl. Chem
, vol.35
, Issue.3
, pp. 489-497
-
-
Makino, K.1
Kim, H.S.2
Kurasawa, Y.3
-
11
-
-
0029819305
-
Ring transformation of 5-acylpyrimidines and 5-acyluracils into pyrazoles with hydrazines in acidic medium
-
Takagi, K.; Hubert-Habart, M. Ring transformation of 5-acylpyrimidines and 5-acyluracils into pyrazoles with hydrazines in acidic medium. J. Heterocycl. Chem., 1996, 33(4),1003-1015.
-
(1996)
J. Heterocycl. Chem
, vol.33
, Issue.4
, pp. 1003-1015
-
-
Takagi, K.1
Hubert-Habart, M.2
-
12
-
-
84948499677
-
Recent developments in the synthesis of pyrazole derivatives
-
Elnagdi, M.H.; Elgemeie, G.E.H.; Abd-Elaal, F. A.-E. Recent developments in the synthesis of pyrazole derivatives. Heterocycles, 1985, 23(12), 3121-3153.
-
(1985)
Heterocycles
, vol.23
, Issue.12
, pp. 3121-3153
-
-
Elnagdi, M.H.1
Elgemeie, G.E.H.2
Abd-Elaal F.A.-E3
-
13
-
-
33645784098
-
Stereoselective cycloadditions of nitrilimines as a source of enantiopure heterocycles
-
Molteni, G. stereoselective cycloadditions of nitrilimines as a source of enantiopure heterocycles. Heterocycles, 2005, 65(10), 2513-2537.
-
(2005)
Heterocycles
, vol.65
, Issue.10
, pp. 2513-2537
-
-
Molteni, G.1
-
14
-
-
0842289719
-
Scorpionates: Genesis, milestones, prognosis
-
Trofimenko, S. Scorpionates: genesis, milestones, prognosis. Polyhedron, 2004, 23(2-3), 197-203.
-
(2004)
Polyhedron
, vol.23
, Issue.2-3
, pp. 197-203
-
-
Trofimenko, S.1
-
15
-
-
0034799031
-
Coordination and supramolecular chemistry of multinucleating ligands containing two or more pyrazolylpyridine 'arms'
-
Ward, M.D.; McCleverty, J.A.; Jeffery, J.C. Coordination and supramolecular chemistry of multinucleating ligands containing two or more pyrazolylpyridine 'arms'. Coord. Chem. Rev., 2001, 222(1), 251-272.
-
(2001)
Coord. Chem. Rev
, vol.222
, Issue.1
, pp. 251-272
-
-
Ward, M.D.1
McCleverty, J.A.2
Jeffery, J.C.3
-
16
-
-
0033803029
-
Coordination chemistry with pyrazole-based chelating ligands: Molecular structural aspects
-
Mukherjee, R. Coordination chemistry with pyrazole-based chelating ligands: molecular structural aspects. Coord. Chem. Rev., 2000, 203(1), 151-218.
-
(2000)
Coord. Chem. Rev
, vol.203
, Issue.1
, pp. 151-218
-
-
Mukherjee, R.1
-
17
-
-
0034749037
-
Progress in pyrazole chemistry
-
Sadimenko, A.P. Progress in pyrazole chemistry. Adv. Heterocycl. Chem., 2001, 80, 157-240.
-
(2001)
Adv. Heterocycl. Chem
, vol.80
, pp. 157-240
-
-
Sadimenko, A.P.1
-
18
-
-
0036096076
-
Synthesis and properties of acetylenic derivatives of pyrazoles
-
Vasilevsky, S.F.; Tretyakov, E.V.; Elguero, J. Synthesis and properties of acetylenic derivatives of pyrazoles. Adv. Heterocycl. Chem., 2002, 82, 1-99.
-
(2002)
Adv. Heterocycl. Chem
, vol.82
, pp. 1-99
-
-
Vasilevsky, S.F.1
Tretyakov, E.V.2
Elguero, J.3
-
19
-
-
33746494445
-
Cross-Coupling Reactions on Azoles with Two and More Heteroatoms
-
Schnürch, M.; Flasik, R.; Khan, A.F.; Spina, M.; Mihovilovic, M.D.; Stanetty, P. Cross-Coupling Reactions on Azoles with Two and More Heteroatoms. Eur. J. Org. Chem., 2006, (15), 3283-3307.
-
(2006)
Eur. J. Org. Chem
, vol.15
, pp. 3283-3307
-
-
Schnürch, M.1
Flasik, R.2
Khan, A.F.3
Spina, M.4
Mihovilovic, M.D.5
Stanetty, P.6
-
20
-
-
0036736760
-
Unsaturated O- and N-heterocycles from carbohydrate feedstocks
-
Lichtenthaler, F.W. Unsaturated O- and N-heterocycles from carbohydrate feedstocks. Acc. Chem. Res., 2002, 35, 728-737.
-
(2002)
Acc. Chem. Res
, vol.35
, pp. 728-737
-
-
Lichtenthaler, F.W.1
-
21
-
-
0346394029
-
Structural revision in pyrazole chemistry
-
Kumar, D.; Singh, S.P. Structural revision in pyrazole chemistry. Heterocycles, 2004, 63(1), 145-173.
-
(2004)
Heterocycles
, vol.63
, Issue.1
, pp. 145-173
-
-
Kumar, D.1
Singh, S.P.2
-
22
-
-
0034759408
-
Pyrazol-3-ones part 1: Synthesis and applications
-
Varvounis, G.; Fiamegos, Y.; Pilidis, G. Pyrazol-3-ones part 1: Synthesis and applications. Adv. Heterocycl. Chem., 2001, 80, 73-156.
-
(2001)
Adv. Heterocycl. Chem
, vol.80
, pp. 73-156
-
-
Varvounis, G.1
Fiamegos, Y.2
Pilidis, G.3
-
23
-
-
11144220008
-
Pyrazol-3-ones. Part II: Reactions of the ring atoms
-
Varvounis, G.; Fiamegos, Y.; Pilidis, G. Pyrazol-3-ones. Part II: Reactions of the Ring Atoms. Adv. Heterocycl. Chem., 2004, 87, 141-272.
-
(2004)
Adv. Heterocycl. Chem
, vol.87
, pp. 141-272
-
-
Varvounis, G.1
Fiamegos, Y.2
Pilidis, G.3
-
24
-
-
37549069310
-
Pyrazol-3-ones. Part III: Reactivity of the ring substituents
-
Varvounis, G.; Fiamegos, Y.; Pilidis, G. Pyrazol-3-ones. Part III: Reactivity of the Ring Substituents. Adv. Heterocycl. Chem., 2007, 95, 27-141.
-
(2007)
Adv. Heterocycl. Chem
, vol.95
, pp. 27-141
-
-
Varvounis, G.1
Fiamegos, Y.2
Pilidis, G.3
-
25
-
-
33746556850
-
The calculated enthalpies of the nine pyrazole anions, cations, and radicals: A comparison with experiment
-
Alkorta, I.; Elguero, J. The calculated enthalpies of the nine pyrazole anions, cations, and radicals: a comparison with experiment. Tetrahedron, 2006, 62, 8683-8686.
-
(2006)
Tetrahedron
, vol.62
, pp. 8683-8686
-
-
Alkorta, I.1
Elguero, J.2
-
26
-
-
33746331066
-
Thermochemical Studies of Pyrazolide
-
Gianola, A.J.; Ichino, T.; Kato, S.; Bierbaum, V.M.; Lineberger, W.C. Thermochemical Studies of Pyrazolide. J. Phys. Chem. A, 2006, 110(27), 8457-8466.
-
(2006)
J. Phys. Chem. A
, vol.110
, Issue.27
, pp. 8457-8466
-
-
Gianola, A.J.1
Ichino, T.2
Kato, S.3
Bierbaum, V.M.4
Lineberger, W.C.5
-
27
-
-
0345415478
-
Lithium-pyrazole-3,4,5-tricarbonitrile: Ion Pairing and Lithium Ion Affinity Studies
-
Markusson, H.; Béranger, S.; Johansson, P.; Armand, M.; Jacobsson, P. Lithium-pyrazole-3,4,5-tricarbonitrile: Ion Pairing and Lithium Ion Affinity Studies. J. Phys. Chem. A, 2003, 107, 10177-10183.
-
(2003)
J. Phys. Chem. A
, vol.107
, pp. 10177-10183
-
-
Markusson, H.1
Béranger, S.2
Johansson, P.3
Armand, M.4
Jacobsson, P.5
-
28
-
-
0031541387
-
Substituent effects on the 15N NMR Parameters of Azoles
-
Claramunt, R.M.; Sanz, D.; López, C.; Jiménez, J.A.; Jimeno, M.L.; Elguero, J.; Fruchier, A. Substituent effects on the 15N NMR Parameters of Azoles. Magn. Reson. Chem., 1997, 35(1), 35-75.
-
(1997)
Magn. Reson. Chem
, vol.35
, Issue.1
, pp. 35-75
-
-
Claramunt, R.M.1
Sanz, D.2
López, C.3
Jiménez, J.A.4
Jimeno, M.L.5
Elguero, J.6
Fruchier, A.7
-
29
-
-
48549100882
-
13C and 15N NMR chemical shifts of 1-(2',4'-dinitrophenyl) and 1-(2',4',6;-trinitrophenyl) pyrazoles in the solid state and in solution
-
García, M.A.; Claramunt, R.M.; Elguero, J. 13C and 15N NMR chemical shifts of 1-(2',4'-dinitrophenyl) and 1-(2',4',6;-trinitrophenyl) pyrazoles in the solid state and in solution. Magn. Reson. Chem., 2008, 46, 697-700.
-
(2008)
Magn. Reson. Chem
, vol.46
, pp. 697-700
-
-
García, M.A.1
Claramunt, R.M.2
Elguero, J.3
-
30
-
-
33646345854
-
1H, 13C and 15N NMR study in solution and in the solid state of six N-substituted pyrazoles and indazoles
-
Claramunt, R.M.; Santa María, M.D.; Sanz, D.; Alkorta, I.; Elguero, J. A 1H, 13C and 15N NMR study in solution and in the solid state of six N-substituted pyrazoles and indazoles. Magn. Reson. Chem., 2006, 44(5), 566-570.
-
(2006)
Magn. Reson. Chem
, vol.44
, Issue.5
, pp. 566-570
-
-
Claramunt, R.M.1
Santa, M.M.D.2
Sanz, D.3
Alkorta, I.4
Elguero, J.A.5
-
31
-
-
51449086400
-
1H, 13C NMR, X-ray and conformational studies of new 1-alkyl-3-benzoyl-pyrazole and 1-alkyl-3-benzoyl-pyrazoline derivatives
-
López-Cara, L.C.; Carrión, M.D.; Camacho, M.E.; Gallo, M.A.; Espinosa, A.; Choquesillo-Lazarte, D.; Gonzalez-Pérez, J.M.; Guadix, A.E. 1H, 13C NMR, X-ray and conformational studies of new 1-alkyl-3-benzoyl-pyrazole and 1-alkyl-3-benzoyl-pyrazoline derivatives. Magn. Reson. Chem., 2008, 46, 878-885.
-
(2008)
Magn. Reson. Chem
, vol.46
, pp. 878-885
-
-
López-Cara, L.C.1
Carrión, M.D.2
Camacho, M.E.3
Gallo, M.A.4
Espinosa, A.5
Choquesillo-Lazarte, D.6
Gonzalez-Pérez, J.M.7
Guadix, A.E.8
-
32
-
-
75149166575
-
A theoretical comparison of the chemical shifts of three related heterocycles: 1 H-pyrazoles, 1H-1,2,4-triazoles and 1H-1,2,4-diazaphospholes
-
Alkorta, I.; Blanco, F.; Elguero, J. A theoretical comparison of the chemical shifts of three related heterocycles: 1 H-pyrazoles, 1H-1,2,4-triazoles and 1H-1,2,4-diazaphospholes. J. Mol. Struct. THEOCHEM, 2010, 942(1-3), 1-6.
-
(2010)
J. Mol. Struct. THEOCHEM
, vol.942
, Issue.1-3
, pp. 1-6
-
-
Alkorta, I.1
Blanco, F.2
Elguero, J.3
-
33
-
-
0035821428
-
A complete model for the prediction of 1H- and 13C-NMR chemical shifts and torsional angles in phenylsubstituted pyrazoles
-
Carrillo, J.R.; Cossío, F.P.; Díaz-Ortíz, A.; Gómez-Escalonilla, M.J.; de la Hoz, A.; Lecea, B.; Moreno, A.; Prieto, P. A complete model for the prediction of 1H- and 13C-NMR chemical shifts and torsional angles in phenylsubstituted pyrazoles. Tetrahedron, 2001, 57(19), 4179-4187.
-
(2001)
Tetrahedron
, vol.57
, Issue.19
, pp. 4179-4187
-
-
Carrillo, J.R.1
Cossío, F.P.2
Díaz-Ortíz, A.3
Gómez-Escalonilla, M.J.4
de la, H.A.5
Lecea, B.6
Moreno, A.7
Prieto, P.8
-
34
-
-
33846428817
-
Characterization of peptide-pyrazole interactions in solution by low-temperature NMR studies
-
Wang, W.; Weisz, K. characterization of peptide-pyrazole interactions in solution by low-temperature NMR studies. Chem. Eur. J., 2007, 13, 854-861.
-
(2007)
Chem. Eur. J
, vol.13
, pp. 854-861
-
-
Wang, W.1
Weisz, K.2
-
35
-
-
0036396046
-
Polymorphism vs. desmotropy: The cases of 3-Phenyl- and 5-Phenyl- 1Hpyrazoles and 3-Phenyl-1H-indazole
-
García, M.A.; López, C.; Claramunt, R.M.; Kenz, A.; Pierrot, M., Elguero, J. Polymorphism vs. desmotropy: The cases of 3-Phenyl- and 5-Phenyl- 1Hpyrazoles and 3-Phenyl-1H-indazole. Helv. Chim. Acta, 2002, 85(9), 2763-2776.
-
(2002)
Helv. Chim. Acta
, vol.85
, Issue.9
, pp. 2763-2776
-
-
García, M.A.1
López, C.2
Claramunt, R.M.3
Kenz, A.4
Pierrot, M.5
Elguero, J.6
-
36
-
-
0033857116
-
The tautomerism of heterocycles: Five-membered rings with two or more heteroatoms
-
Minkin, V.I.; Garnovskii, A.D.; Elguero, J.; Katritzky, A.R.; Denisko, O.V. The tautomerism of heterocycles: Five-membered rings with two or more heteroatoms. Adv. Heterocycl. Chem., 2000, 76, 157-323.
-
(2000)
Adv. Heterocycl. Chem
, vol.76
, pp. 157-323
-
-
Minkin, V.I.1
Garnovskii, A.D.2
Elguero, J.3
Katritzky, A.R.4
Denisko, O.V.5
-
37
-
-
0003313815
-
-
Academic Press:, New York
-
J. Elguero, C. Marzin, A. R. Katritzky, P. Linda, Adv. Heterocycl. Chem., Suppl. 1, Academic Press:, New York 1976.
-
(1976)
Adv. Heterocycl. Chem
, Issue.SUPPL. 1
-
-
Elguero, J.1
Marzin, C.2
Katritzky, A.R.3
Linda, P.4
-
38
-
-
0030853511
-
Structure and tautomerism of 3(5)-amino-5(3)-arylpyrazoles in the solid state and in solution
-
Puello, J.Q.; Obanto, B.I.; Foces-Foces, C.; Infantes, L.; Claramunt, R.-M.; Cabildo, P.; Jimenes, J.A.; Elguero, J. Structure and tautomerism of 3(5)-amino-5(3)-arylpyrazoles in the solid state and in solution: An X-ray and NMR study. Tetrahedron, 1997, 53(31), 10783-10802.
-
(1997)
An X-ray and NMR Study. Tetrahedron
, vol.53
, Issue.31
, pp. 10783-10802
-
-
Puello, J.Q.1
Obanto, B.I.2
Foces-Foces, C.3
Infantes, L.4
Claramunt, R.-M.5
Cabildo, P.6
Jimenes, J.A.7
Elguero, J.8
-
39
-
-
0032793816
-
Aminopyrazoles and their conjugated acids. An X-ray study of 3,5-dimethyl- 4-aminopyrazole and the picrate of 3(5)-aminopyrazole
-
Infantes, L.; Foces-Foces, C.; Claramunt, R.-M.; Lopes, C.; Elguero, J. Aminopyrazoles and their conjugated acids. An X-ray study of 3,5-dimethyl- 4-aminopyrazole and the picrate of 3(5)-aminopyrazole. J. Heterocyl. Chem., 1999, 36(3), 595-600.
-
(1999)
J. Heterocyl. Chem
, vol.36
, Issue.3
, pp. 595-600
-
-
Infantes, L.1
Foces-Foces, C.2
Claramunt, R.-M.3
Lopes, C.4
Elguero, J.5
-
40
-
-
0037454715
-
The structure of the agrochemical fungicidal 4-chloro-3-(3,5-dichlorophenyl)-1H-pyrazole (RPA 406194) and related compounds
-
Vors, J.-P.; Gerbaud, V.; Gabas, N.; Canselier, J.P.; Jagerovic, N.; Jimenoc, M.L.; Elguero, J. The structure of the agrochemical fungicidal 4-chloro-3-(3,5-dichlorophenyl)-1H-pyrazole (RPA 406194) and related compounds. Tetrahedron, 2003, 59(4), 555-560.
-
(2003)
Tetrahedron
, vol.59
, Issue.4
, pp. 555-560
-
-
Vors, J.-P.1
Gerbaud, V.2
Gabas, N.3
Canselier, J.P.4
Jagerovic, N.5
Jimenoc, M.L.6
Elguero, J.7
-
41
-
-
40649101845
-
A molecular balance to measure the strength of N-H π hydrogen bonds based on the tautomeric equilibria of C-benzylphenyl substituted NH-pyrazoles
-
Cornago, P.; Claramunt, R.M.; Bouissane, L.; Elguero, J. A molecular balance to measure the strength of N-H π hydrogen bonds based on the tautomeric equilibria of C-benzylphenyl substituted NH-pyrazoles. Tetrahedron, 2008, 64, 3667-3673.
-
(2008)
Tetrahedron
, vol.64
, pp. 3667-3673
-
-
Cornago, P.1
Claramunt, R.M.2
Bouissane, L.3
Elguero, J.4
-
42
-
-
34447102569
-
Structure and tautomerism of 4-bromo substituted 1H-pyrazoles
-
Trofimenko, S.; Yap, G.A.P.; Jove, F.A.; Claramunt, R.M.; García, M.Á.; Santa Maria, M.D.; Alkorta, I.; Elguero, J. Structure and tautomerism of 4-bromo substituted 1H-pyrazoles. Tetrahedron, 2007, 63(34), 8104-8111.
-
(2007)
Tetrahedron
, vol.63
, Issue.34
, pp. 8104-8111
-
-
Trofimenko, S.1
Yap, G.A.P.2
Jove, F.A.3
Claramunt, R.M.4
García, M.A.5
Santa, M.D.6
Alkorta, I.7
Elguero, J.8
-
43
-
-
19544363799
-
Obrazovanie nesimmetrichnyh 2- (diacilmetilen)-2,3-digidro-1H-benzimidazolov pri acidolize 1-benzoil-2-(bbenzoiloksi- b-fenilvinil)-1H-benzimidazola
-
Dzvinchuk, I.B.; Lozinskii, M.O. Obrazovanie nesimmetrichnyh 2- (diacilmetilen)-2,3-digidro-1H-benzimidazolov pri acidolize 1-benzoil-2-(bbenzoiloksi- b-fenilvinil)-1H-benzimidazola. Khim. Geterotsikl. Soedin., 2001, 606-612;
-
(2001)
Khim. Geterotsikl. Soedin
, pp. 606-612
-
-
Dzvinchuk, I.B.1
Lozinskii, M.O.2
-
44
-
-
0345977281
-
Formation of Unsymmetrical 2-(Diacylmethylene)-2,3- dihydro-1H-benzimidazoles During Acidolysis of 1-Benzoyl-2-(β- benzoyloxy- β-phenylvinyl)-1H-benzimidazole
-
Formation of Unsymmetrical 2-(Diacylmethylene)-2,3- dihydro-1H-benzimidazoles During Acidolysis of 1-Benzoyl-2-(β- benzoyloxy- β-phenylvinyl)-1H-benzimidazole. Chem. Heterocyclic Comp., 2001, 37(5), 554-559.
-
(2001)
Chem. Heterocyclic Comp
, vol.37
, Issue.5
, pp. 554-559
-
-
-
45
-
-
55149117850
-
Sintez i tautomeriya 2-[3(5)- aril(metil)pirazol-4-il]-1-benzimidazolov
-
Dzvinchuk, I.B.; Lozinskii, M.O. Sintez i tautomeriya 2-[3(5)-aril(metil)pirazol-4-il]-1-benzimidazolov. Khim. Geterotsikl. Soedin., 2006, 1370-1378;
-
(2006)
Khim. Geterotsikl. Soedin
, pp. 1370-1378
-
-
Dzvinchuk, I.B.1
Lozinskii, M.O.2
-
46
-
-
33845510685
-
Synthesis and tautomerism of 2-[3(5)-aryl(methyl)pyrazol-4-yl]- 1-benzimidazoles
-
Synthesis and tautomerism of 2-[3(5)-aryl(methyl)pyrazol-4-yl]- 1-benzimidazoles. Chem. Heterocycl. Comp., 2006, 42(9), 1190-1196.
-
(2006)
Chem. Heterocycl. Comp
, vol.42
, Issue.9
, pp. 1190-1196
-
-
-
47
-
-
33750486809
-
The structure of pyrazoles in the solid state: A combined cpmas, Nmr, and crystallographic study
-
Claramunt, R.M.; Cornago, P.; Torres, V.; Pinilla, E.; Torres, M.R.; Samat, A.; Lokshin, V.; Valés, M.; Elguero, J. the structure of pyrazoles in the solid state: a combined cpmas, Nmr, and crystallographic study. J. Org. Chem., 2006, 71, 6881-6891.
-
(2006)
J. Org. Chem
, vol.71
, pp. 6881-6891
-
-
Claramunt, R.M.1
Cornago, P.2
Torres, V.3
Pinilla, E.4
Torres, M.R.5
Samat, A.6
Lokshin, V.7
Valés, M.8
Elguero, J.9
-
48
-
-
33845379599
-
Dynamic intermolecular tautomerism of 3,5-dimethylpyrazole in the solid state by carbon- 13 CP/MAS NMR spectroscopy and x-ray crystallography
-
Baldy, A.; Elguero, J.; Faure, R.; Pierrot, M.; Vincent, E.-J. Dynamic intermolecular tautomerism of 3,5-dimethylpyrazole in the solid state by carbon- 13 CP/MAS NMR spectroscopy and x-ray crystallography. J. Am. Chem. Soc., 1985, 107(18), 5290-5291.
-
(1985)
J. Am. Chem. Soc
, vol.107
, Issue.18
, pp. 5290-5291
-
-
Baldy, A.1
Elguero, J.2
Faure, R.3
Pierrot, M.4
Vincent, E.-J.5
-
49
-
-
0034815821
-
A solid-state NMR, x-ray diffraction, and ab initio computational study of hydrogen-bond structure and dynamics of pyrazole-4-carboxylic acid chains
-
Foces-Foces, C.; Echevarría, A.; Jagerovic, N.; Alkorta, I.; Elguero, J.; Langer, U.; Klein, O.; Minguet-Bonvehí, M.; Limbach, H.-H. a solid-state NMR, x-ray diffraction, and ab initio computational study of hydrogen-bond structure and dynamics of pyrazole-4-carboxylic acid chains. J. Am. Chem. Soc., 2001, 123(32), 7898-7906.
-
(2001)
J. Am. Chem. Soc
, vol.123
, Issue.32
, pp. 7898-7906
-
-
Foces-Foces, C.1
Echevarría, A.2
Jagerovic, N.3
Alkorta, I.4
Elguero, J.5
Langer, U.6
Klein, O.7
Minguet-Bonvehí, M.8
Limbach, H.-H.9
-
50
-
-
1442275753
-
Kinetic hydrogen/ deuterium isotope effects in multiple proton transfer reactions
-
Limbach, H.-H.; Klein, O.; López del Amo, J.M.; Elguero, J. Kinetic hydrogen/ deuterium isotope effects in multiple proton transfer reactions. Z. Phys. Chem., 2004, 218(1), 17-49.
-
(2004)
Z. Phys. Chem
, vol.218
, Issue.1
, pp. 17-49
-
-
Limbach, H.-H.1
Klein, O.2
López del Amo, J.M.3
Elguero, J.4
-
51
-
-
33644644738
-
Pyrazoles as molecular probes to study the properties of co-crystals by solid state NMR spectroscopy
-
López, C.; Claramunt, R.M.; García, M.A.; Elguero, J. Pyrazoles as molecular probes to study the properties of co-crystals by solid state NMR spectroscopy. Cent. Eur. J. Chem., 2004, 2(4), 660-671.
-
(2004)
Cent. Eur. J. Chem
, vol.2
, Issue.4
, pp. 660-671
-
-
López, C.1
Claramunt, R.M.2
García, M.A.3
Elguero, J.4
-
52
-
-
46249113822
-
Proton transfer in C -halogen pyrazole cyclamers. A theoretical study
-
Alkorta, I.; Blanco, F.; Elguero, J. Proton transfer in C -halogen pyrazole cyclamers. A theoretical study. Struct. Chem., 2008, 19, 191-198.
-
(2008)
Struct. Chem
, vol.19
, pp. 191-198
-
-
Alkorta, I.1
Blanco, F.2
Elguero, J.3
-
53
-
-
33644913976
-
Double proton transfer reactions with plateau-like transition state regions: Pyrazole-trifluoroacetic acid clusters
-
Schweiger, S.; Rauhut, G. double proton transfer reactions with plateau-like transition state regions: pyrazole-trifluoroacetic acid clusters. J. Phys. Chem. A, 2006, 110, 2816-2820.
-
(2006)
J. Phys. Chem. A
, vol.110
, pp. 2816-2820
-
-
Schweiger, S.1
Rauhut, G.2
-
54
-
-
0042233915
-
Excited-state intramolecular proton transfer in five-membered hydrogen-bonding systems: 2-pyridyl pyrazoles
-
Yu, W.S.; Cheng, C.-C.; Cheng, Y.-M.; Wu, P.-C.; Song, Y.H.; Chi, Y.; Chou, P.-T. excited-state intramolecular proton transfer in five-membered hydrogen-bonding systems: 2-pyridyl pyrazoles. J. Am. Chem. Soc., 2003, 125(36), 10800-10801.
-
(2003)
J. Am. Chem. Soc
, vol.125
, Issue.36
, pp. 10800-10801
-
-
Yu, W.S.1
Cheng, C.-C.2
Cheng, Y.-M.3
Wu, P.-C.4
Song, Y.H.5
Chi, Y.6
Chou, P.-T.7
-
55
-
-
39349106836
-
Retro-[3 + 2]-cycloaddition reactions in the decomposition of five-membered nitrogen-containing heterocycles
-
da Silva, G.; Bozzelli, J.W. retro-[3 + 2]-cycloaddition reactions in the decomposition of five-membered nitrogen-containing heterocycles. J. Org. Chem., 2008, 73, 1343-1353.
-
(2008)
J. Org. Chem
, vol.73
, pp. 1343-1353
-
-
da Silva, G.1
Bozzelli, J.W.2
-
56
-
-
17744362499
-
Role of conformation and electronic structure in the chemistry of ground and excited state o-pyrazolylphenylnitrenes
-
Carra, C.; Bally, T.; Albini, A. role of conformation and electronic structure in the chemistry of ground and excited state o-pyrazolylphenylnitrenes. J. Am. Chem. Soc., 2005, 127, 5552-5562.
-
(2005)
J. Am. Chem. Soc
, vol.127
, pp. 5552-5562
-
-
Carra, C.1
Bally, T.2
Albini, A.3
-
57
-
-
0035804939
-
Flash vacuum pyrolysis over solid catalysts. 1. pyrazoles over zeolites
-
Moyano, E.L.; Yranzo, G.I. flash vacuum pyrolysis over solid catalysts. 1. pyrazoles over zeolites. J. Org. Chem., 2001, 66, 2943-2947.
-
(2001)
J. Org. Chem
, vol.66
, pp. 2943-2947
-
-
Moyano, E.L.1
Yranzo, G.I.2
-
58
-
-
0037111682
-
Flash vacuum pyrolysis over solid catalysts. 2. pyrazoles over hydrotalcites
-
Moyano, E.L.; del Arco, M.; Rives, V.; Yranzo, G.I. Flash vacuum pyrolysis over solid catalysts. 2. pyrazoles over hydrotalcites. J. Org. Chem., 2002, 67, 8147-8150.
-
(2002)
J. Org. Chem
, vol.67
, pp. 8147-8150
-
-
Moyano, E.L.1
del Arco, M.2
Rives, V.3
Yranzo, G.I.4
-
59
-
-
0036712012
-
Switchable reactivity: The site-selective functionalization of trifluoromethyl-substituted pyrazoles
-
Schlosser, M.; Volle, J.-N.; Leroux, F.; Schenk, K. Switchable reactivity: the site-selective functionalization of trifluoromethyl-substituted pyrazoles. Eur. J. Org. Chem., 2002, (17), 2913-2920.
-
(2002)
Eur. J. Org. Chem
, vol.17
, pp. 2913-2920
-
-
Schlosser, M.1
Volle, J.-N.2
Leroux, F.3
Schenk, K.4
-
60
-
-
0037696879
-
New pyrazoliumcarboxylates as structural analogues of the pseudo-cross-conjugated betainic alkaloid nigellicine
-
Schmidt, A.; Habeck, T.; Kindermann, M.K.; Nieger, M. new pyrazoliumcarboxylates as structural analogues of the pseudo-cross-conjugated betainic alkaloid nigellicine. J. Org. Chem., 2003, 68(15), 5977-5982.
-
(2003)
J. Org. Chem
, vol.68
, Issue.15
, pp. 5977-5982
-
-
Schmidt, A.1
Habeck, T.2
Kindermann, M.K.3
Nieger, M.4
-
61
-
-
19844383213
-
Nucleophilic carbenes of pyrazoles starting from pseudo-cross-conjugated mesomeric betaines
-
Schmidt, A.; Habeck, T. nucleophilic carbenes of pyrazoles starting from pseudo-cross-conjugated mesomeric betaines. Lett. Org. Chem., 2005, 2(1), 37-39.
-
(2005)
Lett. Org. Chem
, vol.2
, Issue.1
, pp. 37-39
-
-
Schmidt, A.1
Habeck, T.2
-
62
-
-
79958226857
-
Funktionalisierte 4-aminochinoline durch umlagerung von n-heterocyclischen carbenen des pyrazols
-
Schmidt, A.; Münster, N.; Dreger, A. funktionalisierte 4-aminochinoline durch umlagerung von n-heterocyclischen carbenen des pyrazols. Angew. Chem., 2010, 122(15), 2851-2854;
-
(2010)
Angew. Chem
, vol.122
, Issue.15
, pp. 2851-2854
-
-
Schmidt, A.1
Münster, N.2
Dreger, A.3
-
63
-
-
77950504117
-
Functionalized 4-aminoquinolines by rearrangement of pyrazole N-heterocyclic carbenes
-
Functionalized 4-aminoquinolines by rearrangement of pyrazole N-heterocyclic carbenes. Angew. Chem. Int. Ed., 2010, 49(15), 2790-2793.
-
(2010)
Angew. Chem. Int. Ed
, vol.49
, Issue.15
, pp. 2790-2793
-
-
-
64
-
-
77954970942
-
Rearrangements of n-heterocyclic carbenes of pyrazole to 4- aminoquinolines and benzoquinolines
-
Dreger, A.; Cisneros Camuña, R.; Münster, N.; Rokob, T.A.; Pápai, I.; Schmidt, A. rearrangements of n-heterocyclic carbenes of pyrazole to 4- aminoquinolines and benzoquinolines. Eur. J. Org. Chem., 2010, (22), 4296-4305.
-
(2010)
Eur. J. Org. Chem
, vol.22
, pp. 4296-4305
-
-
Dreger, A.1
Cisneros, C.R.2
Münster, N.3
Rokob, T.A.4
Pápai, I.5
Schmidt, A.6
-
65
-
-
55149119722
-
A theoretical insight into the reaction mechanism of photochemical transposition from pyrazole to imidazole
-
Su, M.-D. A theoretical insight into the reaction mechanism of photochemical transposition from pyrazole to imidazole. J. Phys. Chem. A, 2008, 112(41), 10420-10428.
-
(2008)
J. Phys. Chem. A
, vol.112
, Issue.41
, pp. 10420-10428
-
-
Su, M.-D.1
-
66
-
-
23944509573
-
Synthesis of new 3h-pyrazoles and cyclopropenyl alcohols directly from propargyl alcohols
-
Hamdi, N.; Dixneuf, P.H.; Khemiss, A. synthesis of new 3h-pyrazoles and cyclopropenyl alcohols directly from propargyl alcohols. Eur. J. Org. Chem., 2005, (16), 3526-3529.
-
(2005)
Eur. J. Org. Chem
, vol.16
, pp. 3526-3529
-
-
Hamdi, N.1
Dixneuf, P.H.2
Khemiss, A.3
-
67
-
-
0009401381
-
Withasomnine. A pyrazole alkaloid from Withania somnifera Dun
-
Schröter, H.B.; Neumann, D.; Katritzky, A.R.; Swinbourne, F.J. Withasomnine. A pyrazole alkaloid from Withania somnifera Dun. Tetrahedron, 1966, 22(8), 2895-2897.
-
(1966)
Tetrahedron
, vol.22
, Issue.8
, pp. 2895-2897
-
-
Schröter, H.B.1
Neumann, D.2
Katritzky, A.R.3
Swinbourne, F.J.4
-
68
-
-
0037013971
-
Radical cyclisation onto pyrazoles: Synthesis of withasomnine
-
Allin, S.M.; Barton, W.R.S.; Bowman, W.R.; McInally, T. Radical cyclisation onto pyrazoles: synthesis of withasomnine. Tetrahedron Lett., 2002, 43, 4191-4193.
-
(2002)
Tetrahedron Lett
, vol.43
, pp. 4191-4193
-
-
Allin, S.M.1
Barton, W.R.S.2
Bowman, W.R.3
McInally, T.4
-
69
-
-
0028001924
-
Pyrazole alkaloids from Newbouldia laevis
-
Adesanya, S.A.; Nia, R.; Fontaine, C.; Païs, M. Pyrazole alkaloids from Newbouldia laevis. Phytochemistry, 1994, 35(4), 1053-1055.
-
(1994)
Phytochemistry
, vol.35
, Issue.4
, pp. 1053-1055
-
-
Adesanya, S.A.1
Nia, R.2
Fontaine, C.3
Païs, M.4
-
70
-
-
0031985265
-
New pyrazole alkaloids from the root bark of Newbouldia laevis
-
Aladesanmi, A.J.; Nia, R.; Nahrstedt, A. New pyrazole alkaloids from the root bark of Newbouldia laevis. Planta Med., 1998, 64, 90-91.
-
(1998)
Planta Med
, vol.64
, pp. 90-91
-
-
Aladesanmi, A.J.1
Nia, R.2
Nahrstedt, A.3
-
71
-
-
39149100002
-
Constituents of the stem bark of Discopodium penninervium and their LTB4 and COX-1 and -2 inhibitory activities
-
Wube, A.A.; Wenzig, E.-M.; Gibbons, S.; Asres, K.; Bauer, R.; Bucar, F. Constituents of the stem bark of Discopodium penninervium and their LTB4 and COX-1 and -2 inhibitory activities. Phytochemistry, 2008, 69, 982-987.
-
(2008)
Phytochemistry
, vol.69
, pp. 982-987
-
-
Wube, A.A.1
Wenzig, E.-M.2
Gibbons, S.3
Asres, K.4
Bauer, R.5
Bucar, F.6
-
72
-
-
0009357016
-
Pyrazole alkaloids from Elytraria acaulis
-
Ravikanth, V.; Ramesh, P.; Diwan, P.V.; Venkateswarlu, Y. Pyrazole alkaloids from Elytraria acaulis. Biochem. Sys. Ecol., 2001, 29, 753-754.
-
(2001)
Biochem. Sys. Ecol
, vol.29
, pp. 753-754
-
-
Ravikanth, V.1
Ramesh, P.2
Diwan, P.V.3
Venkateswarlu, Y.4
-
73
-
-
0542371982
-
Heteroaromatic acid from marine sponge Suberites vestigium
-
Mishra, P.D.; Wahidullah, S.; Kamat, S.Y. A heteroaromatic acid from marine sponge Suberites vestigium. Indian J. Chem., Sect. B, 1998, 37B(2), 199-200.
-
(1998)
Indian J. Chem., Sect. B
, vol.37 B
, Issue.2
, pp. 199-200
-
-
Mishra, P.D.1
Wahidullah, S.2
Kamat, S.Y.A.3
-
74
-
-
0030796455
-
Secondary metabolites from the sponge tedania anhelans: Isolation and characterization of two novel pyrazole acids and other metabolites
-
Parameswaran, P.S.; Naik, C.G.; Hegde, V.R. secondary metabolites from the sponge tedania anhelans: isolation and characterization of two novel pyrazole acids and other metabolites. J. Nat. Prod., 1997, 60(8), 802-803.
-
(1997)
J. Nat. Prod
, vol.60
, Issue.8
, pp. 802-803
-
-
Parameswaran, P.S.1
Naik, C.G.2
Hegde, V.R.3
-
75
-
-
0038203630
-
New manzamine alkaloids with activity against infectious and tropical parasitic diseases from an indonesian sponge
-
Rao, K.V.; Santarsiero, B.D.; Mesecar, A.D.; Schinazi, R.F.; Tekwani, B.L. Hamann, M.T.; new manzamine alkaloids with activity against infectious and tropical parasitic diseases from an indonesian sponge. J. Nat. Prod., 2003, 66, 823-828.
-
(2003)
J. Nat. Prod
, vol.66
, pp. 823-828
-
-
Rao, K.V.1
Santarsiero, B.D.2
Mesecar, A.D.3
Schinazi, R.F.4
Tekwani, B.L.5
Hamann, M.T.6
-
76
-
-
0001221337
-
The synthesis of L-α-amino- β- (pyrazolyl-N)-propionic acid in Citrullus vulgaris
-
Sugimoto, N.; Watanabe, H.; Ide, A. The synthesis of L-α-amino- β- (pyrazolyl-N)-propionic acid in Citrullus vulgaris. Tetrahedron, 1960, 11(4), 231-233.
-
(1960)
Tetrahedron
, vol.11
, Issue.4
, pp. 231-233
-
-
Sugimoto, N.1
Watanabe, H.2
Ide, A.3
-
77
-
-
51149219272
-
C-Nucleoside studies. Part 14. A new synthesis of pyrazofurin
-
Buchanan, J.G.; Stobie, A.; Wightman, R.H. C-Nucleoside studies. Part 14. A new synthesis of pyrazofurin. J. Chem. Soc., Perkin Trans. 1, 1981, (8), 2374-2378.
-
(1981)
J. Chem. Soc. Perkin Trans
, vol.1
, Issue.8
, pp. 2374-2378
-
-
Buchanan, J.G.1
Stobie, A.2
Wightman, R.H.3
-
78
-
-
33750865454
-
The chemistry of c-nucleosides and their analogs i: C-nucleosides of hetero monocyclic bases
-
Shaban, M.A.E.; Nasr, A.Z. the chemistry of c-nucleosides and their analogs i: c-nucleosides of hetero monocyclic bases. Adv. Heterocycl. Chem., 1997, 68, 223-432.
-
(1997)
Adv. Heterocycl. Chem
, vol.68
, pp. 223-432
-
-
Shaban, M.A.E.1
Nasr, A.Z.2
-
79
-
-
0015928319
-
Isolation and characterization of an α-Cnucleoside antibiotic related to pyrazomycin
-
Gutowski, G.E.; Chaney, M.O.; Jones, N.D.; Hamill, R.L.; Davis, F.A.; Miller, R.D. Pyrazomycin B: Isolation and characterization of an α-Cnucleoside antibiotic related to pyrazomycin. Biochem. Biophys. Res. Commun., 1973, 51(2), 312-317.
-
(1973)
Biochem. Biophys. Res. Commun
, vol.51
, Issue.2
, pp. 312-317
-
-
Gutowski, G.E.1
Chaney, M.O.2
Jones, N.D.3
Hamill, R.L.4
Davis, F.A.5
Miller, R.D.6
Pyrazomycin, B.7
-
80
-
-
36549013145
-
Pyrazole chemistry in crop protection
-
Lamberth, C. Pyrazole chemistry in crop protection. Heterocycles, 2007, 71(7), 1467-1502.
-
(2007)
Heterocycles
, vol.71
, Issue.7
, pp. 1467-1502
-
-
Lamberth, C.1
-
81
-
-
42249084709
-
Antifungal and antimycobacterial activity of 1-(3,5-diaryl-4,5-dihydro-1Hpyrazol-4-yl)-1H-imidazole derivatives
-
Zampieri, D.; Mamolo, M.G.; Laurini, E.; Scialino, G.; Banfi, E.; Vio, L. Antifungal and antimycobacterial activity of 1-(3,5-diaryl-4,5-dihydro-1Hpyrazol-4-yl)-1H-imidazole derivatives. Bioorg. Med. Chem., 2008, 16, 4516-4522.
-
(2008)
Bioorg. Med. Chem
, vol.16
, pp. 4516-4522
-
-
Zampieri, D.1
Mamolo, M.G.2
Laurini, E.3
Scialino, G.4
Banfi, E.5
Vio, L.6
-
82
-
-
0028172369
-
Inhibition by SK&F 96365 of Ca2+ current, IL-2 production and activation in T lymphocytes
-
Chung, S.C.; McDonald, T.V.; Gardner, P. Inhibition by SK&F 96365 of Ca2+ current, IL-2 production and activation in T lymphocytes. Br. J. Pharmacol., 1994, 113(3), 861-868.
-
(1994)
Br. J. Pharmacol
, vol.113
, Issue.3
, pp. 861-868
-
-
Chung, S.C.1
McDonald, T.V.2
Gardner, P.3
-
83
-
-
27944489028
-
Novel 1,3- dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine derivatives as high affinity and selective A2B adenosine receptor antagonists
-
Elzein, E.; Kalla, R.; Li, X.; Perry, T.; Parchill, E.; Palle, V.; Varkhedkar, V.; Gimbel, A.; Zeng, D.; Lustig, D.; Leung, K.; Zablocki, J. Novel 1,3- dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine derivatives as high affinity and selective A2B adenosine receptor antagonists. Bioorg. Med. Chem. Lett., 2006, 16, 302-306.
-
(2006)
Bioorg. Med. Chem. Lett
, vol.16
, pp. 302-306
-
-
Elzein, E.1
Kalla, R.2
Li, X.3
Perry, T.4
Parchill, E.5
Palle, V.6
Varkhedkar, V.7
Gimbel, A.8
Zeng, D.9
Lustig, D.10
Leung, K.11
Zablocki, J.12
-
84
-
-
33645665682
-
Discovery of 4-{4-[3-(Pyridin-2-yl)-1H-pyrazol-4-yl] pyridin-2-yl}-N-(tetrahydro-2H- pyran-4-yl) benzamide (GW788388): A potent, selective, and orally active transforming growth factor- β Type I receptor inhibitor
-
Gellibert, F.; de Gouville, A.-C.; Woolven, J.; Mathews, N.; Nguyen, V.-L.; Bertho-Ruault, C.; Patikis, A.; Grygielko, E.T.; Laping, N.J.; Huet, S. Discovery of 4-{4-[3-(Pyridin-2-yl)-1H-pyrazol-4-yl] pyridin-2-yl}-N-(tetrahydro-2H- pyran-4-yl) benzamide (GW788388): A potent, selective, and orally active transforming growth factor- β Type I receptor inhibitor. J. Med. Chem., 2006, 49, 2210-2221.
-
(2006)
J. Med. Chem
, vol.49
, pp. 2210-2221
-
-
Gellibert, F.1
de Gouville, A.-C.2
Woolven, J.3
Mathews, N.4
Nguyen, V.-L.5
Bertho-Ruault, C.6
Patikis, A.7
Grygielko, E.T.8
Laping, N.J.9
Huet, S.10
-
85
-
-
38949111028
-
Selective, high affinity A2B adenosine receptor antagonists: N-1 monosubstituted 8-(pyrazol-4-yl)xanthines
-
Kalla, R.V.; Elzein, E.; Perry, T.; Li, X.; Gimbel, A.; Yang, M.; Zeng, D.; Zablocki, J. Selective, high affinity A2B adenosine receptor antagonists: N-1 monosubstituted 8-(pyrazol-4-yl)xanthines. Bioorg. Med. Chem. Lett., 2008, 18, 1397-1401.
-
(2008)
Bioorg. Med. Chem. Lett
, vol.18
, pp. 1397-1401
-
-
Kalla, R.V.1
Elzein, E.2
Perry, T.3
Li, X.4
Gimbel, A.5
Yang, M.6
Zeng, D.7
Zablocki, J.8
-
86
-
-
41849134287
-
5-tert-Butyl-N-pyrazol-4-yl-4,5,6,7-tetrahydrobenzo[d]isoxazole- 3-carboxamide derivatives as novel potent inhibitors of Mycobacterium tuberculosis pantothenate synthetase: Initiating a quest for New antitubercular drugs
-
Velaparthi, S.; Brunsteiner, M.; Uddin, R.; Wan, B.; Franzblau, S.G.; Petukhov, P.A. 5-tert-Butyl-N-pyrazol-4-yl-4,5,6,7-tetrahydrobenzo[d]isoxazole- 3-carboxamide derivatives as novel potent inhibitors of Mycobacterium tuberculosis pantothenate synthetase: Initiating a quest for New antitubercular drugs. J. Med. Chem., 2008, 51, 1999-2002.
-
(2008)
J. Med. Chem
, vol.51
, pp. 1999-2002
-
-
Velaparthi, S.1
Brunsteiner, M.2
Uddin, R.3
Wan, B.4
Franzblau, S.G.5
Petukhov, P.A.6
-
87
-
-
36148964016
-
Synthesis and evaluation of antiparasitic activities of new 4-[5-(4- Phenoxyphenyl)-2H-pyrazol-3-yl] morpholine derivatives
-
Kuettel, S.; Zambon, A.; Kaiser, M.; Brun, R.; Scapozza, L.; Perozzo, R. synthesis and evaluation of antiparasitic activities of new 4-[5-(4- Phenoxyphenyl)-2H-pyrazol-3-yl] morpholine derivatives. J. Med. Chem., 2007, 50, 5833-5839.
-
(2007)
J. Med. Chem
, vol.50
, pp. 5833-5839
-
-
Kuettel, S.1
Zambon, A.2
Kaiser, M.3
Brun, R.4
Scapozza, L.5
Perozzo, R.6
-
88
-
-
35848942839
-
Structure-based design of (5- Arylamino-2H-pyrazol-3-yl)-biphenyl-2',4'-diols as novel and potent Human CHK1 inhibitors
-
Teng, M.; Zhu, J.; Johnson, M.D.; Chen, P.; Kornmann, J.; Chen, E.; Blasina, A.; Register, J.; Anderes, K.; Rogers, C.; Deng, Y.; Ninkovic, S.; Grant, S.; Hu, Q.; Lundgren, K.; Peng, Z.; Kania, R.S. Structure-based design of (5- Arylamino-2H-pyrazol-3-yl)-biphenyl-2',4'-diols as novel and potent Human CHK1 inhibitors. J. Med. Chem., 2007, 50, 5253-5256.
-
(2007)
J. Med. Chem
, vol.50
, pp. 5253-5256
-
-
Teng, M.1
Zhu, J.2
Johnson, M.D.3
Chen, P.4
Kornmann, J.5
Chen, E.6
Blasina, A.7
Register, J.8
Anderes, K.9
Rogers, C.10
Deng, Y.11
Ninkovic, S.12
Grant, S.13
Hu, Q.14
Lundgren, K.15
Peng, Z.16
Kania, R.S.17
-
89
-
-
13444266910
-
Synthesis and biological evaluation of the 1,5-Diarylpyrazole class of cyclooxygenase-2 inhibitors: Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1- yl]benzenesulfonamide (SC-58635, Celecoxib)
-
Penning, T.D.; Talley, J.J.; Bertenshaw, S.R.; Carter, J.S.; Collins, P.W.; Doctor, S.; Graneto, M.J.; Lee, L.F.; Malecha, J.W.; Mirashiro, J.M.; Rogers, R.S.; Rogier, D.J.; Yu, S.S.; Anderson, G.D.; Burton, E.G.; Cogburn, J.N.; Gregory, S.A.; Koboldt, C.M.; Perkins, W.E.; Seibert, K.; Veenhuizen, A.M.; Zhang, Y.Y.; Isakson, P.C. Synthesis and biological evaluation of the 1,5-Diarylpyrazole class of cyclooxygenase-2 inhibitors: identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1- yl]benzenesulfonamide (SC-58635, Celecoxib). J. Med. Chem., 1997, 40(9), 1347-1365.
-
(1997)
J. Med. Chem
, vol.40
, Issue.9
, pp. 1347-1365
-
-
Penning, T.D.1
Talley, J.J.2
Bertenshaw, S.R.3
Carter, J.S.4
Collins, P.W.5
Doctor, S.6
Graneto, M.J.7
Lee, L.F.8
Malecha, J.W.9
Mirashiro, J.M.10
Rogers, R.S.11
Rogier, D.J.12
Yu, S.S.13
Anderson, G.D.14
Burton, E.G.15
Cogburn, J.N.16
Gregory, S.A.17
Koboldt, C.M.18
Perkins, W.E.19
Seibert, K.20
Veenhuizen, A.M.21
Zhang, Y.Y.22
Isakson, P.C.23
more..
-
91
-
-
33750522014
-
Identification of 2-hydroxymethyl-4-[5-(4-methoxyphenyl)-3-trifluoromethyl-pyrazol-1-yl]-N-propionylbenzenesulfonamide sodium as a potential COX-2 inhibitor for oral and parenteral administration
-
Singh, S.K.; Vobbalareddy, S.; Kalleda, S.R.; Casturi, S.R.; Datla, S.R.; Mamidi, R.N.V.S.; Mullangi, R.; Ramanujam, R.; Yeleswarapu, K.R.; Iqbal, J. Identification of 2-hydroxymethyl-4-[5-(4-methoxyphenyl)-3-trifluoromethyl-pyrazol-1-yl]-N-propionylbenzenesulfonamide sodium as a potential COX-2 inhibitor for oral and parenteral administration. Bioorg. Med. Chem., 2006, 14, 8626-8634.
-
(2006)
Bioorg. Med. Chem
, vol.14
, pp. 8626-8634
-
-
Singh, S.K.1
Vobbalareddy, S.2
Kalleda, S.R.3
Casturi, S.R.4
Datla, S.R.5
Mamidi, R.N.V.S.6
Mullangi, R.7
Ramanujam, R.8
Yeleswarapu, K.R.9
Iqbal, J.10
-
92
-
-
33847783301
-
Synthesis and in vivo evaluation of [18F]-4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1Hpyrazol- 1-yl] benzenesulfonamide as a PET imaging probe for COX-2 expression
-
Prabhakaran, J.; Underwood, M.D.; Parsey, V.R.; Arango, V.; Majo, V.J.; Simpson, N.R.; Van Heertum, R.; Mann, J.J.; Kumar, J.S.D. Synthesis and in vivo evaluation of [18F]-4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1Hpyrazol- 1-yl] benzenesulfonamide as a PET imaging probe for COX-2 expression. Bioorg. Med. Chem., 2007, 15, 1802-1807.
-
(2007)
Bioorg. Med. Chem
, vol.15
, pp. 1802-1807
-
-
Prabhakaran, J.1
Underwood, M.D.2
Parsey, V.R.3
Arango, V.4
Majo, V.J.5
Simpson, N.R.6
van Heertum, R.7
Mann, J.J.8
Kumar, J.S.D.9
-
93
-
-
11144354316
-
Synthesis and selective cyclooxygenase-2 inhibitory activity of a series of novel, nitric oxide donor-containing pyrazoles
-
Ranatunge, R.R.; Augustyniak, M.; Bandarage, U.K.; Earl, R.A.; Ellis, J.L.; Garvey, D.S.; Janero, D.R.; Letts, L.G.; Martino, A.M.; Murty, M.G.; Richardson, S.K.; Schroeder, J.D.; Shumway, M.J.; Tam, S.W.; Trocha, M.; Young, D.V. Synthesis and selective cyclooxygenase-2 inhibitory activity of a series of novel, nitric oxide donor-containing pyrazoles. J. Med. Chem., 2004, 47(9), 2180-2193.
-
(2004)
J. Med. Chem
, vol.47
, Issue.9
, pp. 2180-2193
-
-
Ranatunge, R.R.1
Augustyniak, M.2
Bandarage, U.K.3
Earl, R.A.4
Ellis, J.L.5
Garvey, D.S.6
Janero, D.R.7
Letts, L.G.8
Martino, A.M.9
Murty, M.G.10
Richardson, S.K.11
Schroeder, J.D.12
Shumway, M.J.13
Tam, S.W.14
Trocha, M.15
Young, D.V.16
-
94
-
-
52949112645
-
Regioselective preparation of N-methylpyrazole derivative
-
Profeta, R.; Mattioli, M.; Micheli, F.; Piga, E.; Spada, S.; Tarsi, L.; Andreotti, D. Regioselective preparation of N-methylpyrazole derivative. Synlett, 2008, (15), 2283-2286.
-
(2008)
Synlett
, vol.15
, pp. 2283-2286
-
-
Profeta, R.1
Mattioli, M.2
Micheli, F.3
Piga, E.4
Spada, S.5
Tarsi, L.6
Andreotti, D.7
-
95
-
-
33646821317
-
Novel potent and selective calcium-release-activated calcium (CRAC) channel inhibitors. Part 1: Synthesis and inhibitory activity of 5-(1-methyl-3-trifluoromethyl-1Hpyrazol-5-yl)-2-thiophenecarboxamides
-
Yonetoku, Y.; Kubota, H.; Okamoto, Y.; Toyoshima, A.; Funatsu, M.; Ishikawa, J.; Takeuchi, M.; Ohta, M.; Tsukamoto, S.-I. Novel potent and selective calcium-release-activated calcium (CRAC) channel inhibitors. Part 1: Synthesis and inhibitory activity of 5-(1-methyl-3-trifluoromethyl-1Hpyrazol-5-yl)-2-thiophenecarboxamides. Bioorg. Med. Chem., 2006, 14, 4750-4760.
-
(2006)
Bioorg. Med. Chem
, vol.14
, pp. 4750-4760
-
-
Yonetoku, Y.1
Kubota, H.2
Okamoto, Y.3
Toyoshima, A.4
Funatsu, M.5
Ishikawa, J.6
Takeuchi, M.7
Ohta, M.8
Tsukamoto, S.-I.9
-
96
-
-
33846039221
-
Identification and optimisation of a series of substituted 5-(1H-pyrazol-3-yl)-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors
-
Price, S.; Bordogna, W.; Bull, R.J.; Clark, D.E.; Crackett, P.H.; Dyke, H.J.; Gill, M.; Harris, N.V.; Gorski, J.; Lloyd, J.; Lockey, P.M.; Mullet, J.; Roach, A.G.; Roussel, F.; White, A.B. Identification and optimisation of a series of substituted 5-(1H-pyrazol-3-yl)-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors. Bioorg. Med. Chem. Lett., 2007, 17, 370-375.
-
(2007)
Bioorg. Med. Chem. Lett
, vol.17
, pp. 370-375
-
-
Price, S.1
Bordogna, W.2
Bull, R.J.3
Clark, D.E.4
Crackett, P.H.5
Dyke, H.J.6
Gill, M.7
Harris, N.V.8
Gorski, J.9
Lloyd, J.10
Lockey, P.M.11
Mullet, J.12
Roach, A.G.13
Roussel, F.14
White, A.B.15
-
97
-
-
48849095518
-
Potent and selective pyrazole-based inhibitors of B-Raf kinase
-
Hansen, J.D.; Grina, J.; Newhouse, B.; Welch, M.; Topalov, G.; Littman, N.; Callejo, M.; Gloor, S.; Martinson, M.; Laird, E.; Brandhuber, B.J.; Vigers, G.; Morales, T.; Woessner, R.; Randolph, N.; Lyssikatos, J.; Olivero, A. Potent and selective pyrazole-based inhibitors of B-Raf kinase. Bioorg. Med. Chem. Lett., 2008, 18, 4692-4695.
-
(2008)
Bioorg. Med. Chem. Lett
, vol.18
, pp. 4692-4695
-
-
Hansen, J.D.1
Grina, J.2
Newhouse, B.3
Welch, M.4
Topalov, G.5
Littman, N.6
Callejo, M.7
Gloor, S.8
Martinson, M.9
Laird, E.10
Brandhuber, B.J.11
Vigers, G.12
Morales, T.13
Woessner, R.14
Randolph, N.15
Lyssikatos, J.16
Olivero, A.17
-
98
-
-
47349110358
-
Synthesis and discovery of autophagy inducers for A549 and H460 lung cancer cells, novel 1-(2'-hydroxy-3'-aroxypropyl)-3-aryl-1H-pyrazole-5- carbohydrazide derivatives
-
Fan, C.-D.; Zhao, B.-X.; Wie, F.; Zhang, G.-H.; Dong, W.-L.; Miao, J.-Y. Synthesis and discovery of autophagy inducers for A549 and H460 lung cancer cells, novel 1-(2'-hydroxy-3'-aroxypropyl)-3-aryl-1H-pyrazole-5- carbohydrazide derivatives. Bioorg. Med. Chem. Lett., 2008, 18, 3860-3864.
-
(2008)
Bioorg. Med. Chem. Lett
, vol.18
, pp. 3860-3864
-
-
Fan, C.-D.1
Zhao, B.-X.2
Wie, F.3
Zhang, G.-H.4
Dong, W.-L.5
Miao, J.-Y.6
-
99
-
-
47149102125
-
Discovery of brain penetrant, soluble, pyrazole amide EP1 receptor antagonists
-
Hall, A.; Billinton, A.; Bristow, A.K.; Brown, S.H.; Chowdhury, A.; Cutler, L.; Giblin, G.M.P.; Goldsmith, P.; Hayhow, T.G.; Kilford, I.R.; Naylor, A.; Passingham, B.; Rawlings, D.A. Discovery of brain penetrant, soluble, pyrazole amide EP1 receptor antagonists. Bioorg. Med. Chem. Lett., 2008, 18, 4027-4032.
-
(2008)
Bioorg. Med. Chem. Lett
, vol.18
, pp. 4027-4032
-
-
Hall, A.1
Billinton, A.2
Bristow, A.K.3
Brown, S.H.4
Chowdhury, A.5
Cutler, L.6
Giblin, G.M.P.7
Goldsmith, P.8
Hayhow, T.G.9
Kilford, I.R.10
Naylor, A.11
Passingham, B.12
Rawlings, D.A.13
-
100
-
-
47849115661
-
Pyrazole inhibitors of coactivator associated arginine methyltransferase 1 (CARM1)
-
Purandare, A.V.; Chen, Z.; Huynh, T.; Pang, S.; Geng, J.; Vaccaro, W.; Poss, M.A.; Oconnell, J.; Nowak, K.; Jayaraman, L. Pyrazole inhibitors of coactivator associated arginine methyltransferase 1 (CARM1). Bioorg. Med. Chem. Lett., 2008, 18, 4438-4441.
-
(2008)
Bioorg. Med. Chem. Lett
, vol.18
, pp. 4438-4441
-
-
Purandare, A.V.1
Chen, Z.2
Huynh, T.3
Pang, S.4
Geng, J.5
Vaccaro, W.6
Poss, M.A.7
Oconnell, J.8
Nowak, K.9
Jayaraman, L.10
-
101
-
-
48149103866
-
Convenient access to 1,3,4-trisubstituted pyrazoles carrying 5-nitrothiophene moiety via 1,3-dipolar cycloaddition of sydnones with acetylenic ketones and their antimicrobial evaluation
-
Rai, N.S.; Kalluraya, B.; Lingappa, B.; Shenoy, S.; Puranic, V.G. Convenient access to 1,3,4-trisubstituted pyrazoles carrying 5-nitrothiophene moiety via 1,3-dipolar cycloaddition of sydnones with acetylenic ketones and their antimicrobial evaluation. Eur. J. Med. Chem., 2008, 43, 1715-1720.
-
(2008)
Eur. J. Med. Chem
, vol.43
, pp. 1715-1720
-
-
Rai, N.S.1
Kalluraya, B.2
Lingappa, B.3
Shenoy, S.4
Puranic, V.G.5
-
102
-
-
33745143300
-
N-Acylated sulfonamide sodium salt: A prodrug of choice for the bifunctional 2-hydroxymethyl-4-(5- phenyl-3-trifluoromethyl-pyrazol-1-yl) benzenesulfonamide class of COX-2 inhibitors
-
Singh, S.K.; Vobbalareddy, S.; Kalleda, S.R.; Casturi, S.R.; Mullangi, R.; Ramanujam, R.; Yeleswarapu, K.R.; Iqbal, J. N-Acylated sulfonamide sodium salt: A prodrug of choice for the bifunctional 2-hydroxymethyl-4-(5- phenyl-3-trifluoromethyl-pyrazol-1-yl) benzenesulfonamide class of COX-2 inhibitors. Bioorg. Med. Chem. Lett., 2006, 16, 3921-3926.
-
(2006)
Bioorg. Med. Chem. Lett
, vol.16
, pp. 3921-3926
-
-
Singh, S.K.1
Vobbalareddy, S.2
Kalleda, S.R.3
Casturi, S.R.4
Mullangi, R.5
Ramanujam, R.6
Yeleswarapu, K.R.7
Iqbal, J.8
-
103
-
-
8644252687
-
Discovery of positive allosteric modulators for the metabotropic glutamate Receptor Subtype 5 from a Series of N-(1,3-Diphenyl-1H- pyrazol-5-yl)benzamides that potentiate receptor function in vivo
-
Lindsley, C.W.; Wisnoski, D.D.; Duggan, M.E.; Leister, W.H.; Hartman, G.D.; Huff, J.R.; Williams, D.L.; ÓBrien, J.A.; Lemaire, W.; Sur, C. Discovery of positive allosteric modulators for the metabotropic glutamate Receptor Subtype 5 from a Series of N-(1,3-Diphenyl-1H- pyrazol-5-yl)benzamides that potentiate receptor function in vivo. J. Med. Chem., 2004, 47(24), 5825-5828.
-
(2004)
J. Med. Chem
, vol.47
, Issue.24
, pp. 5825-5828
-
-
Lindsley, C.W.1
Wisnoski, D.D.2
Duggan, M.E.3
Leister, W.H.4
Hartman, G.D.5
Huff, J.R.6
Williams, D.L.7
ÓBrien, J.A.8
Lemaire, W.9
Sur, C.10
-
104
-
-
20144381462
-
A novel selective positive allosteric modulator of metabotropic glutamate receptor subtype 5 has in vivo activity and antipsychotic-like effects in rat behavioral models
-
Kinney, G.G.; ÓBrien, J.A.; Lemaire, W.; Burno, M.; Bickel, D.J.; Clements, M.K.; Chen, T.-B.; Wisnoski, D.D.; Lindsley, C.W.; Tiller, R.P.; Smith, S.; Jacobson, M.A.; Sur, C.; Duggan, M.E.; Petitbone, D.J.; Conn, P.J.; Williams, D.L. a novel selective positive allosteric modulator of metabotropic glutamate receptor subtype 5 has in vivo activity and antipsychotic-like effects in rat behavioral models. J. Pharmacol. Exp. Ther., 2005, 313(1), 199-206.
-
(2005)
J. Pharmacol. Exp. Ther
, vol.313
, Issue.1
, pp. 199-206
-
-
Kinney, G.G.1
ÓBrien, J.A.2
Lemaire, W.3
Burno, M.4
Bickel, D.J.5
Clements, M.K.6
Chen, T.-B.7
Wisnoski, D.D.8
Lindsley, C.W.9
Tiller, R.P.10
Smith, S.11
Jacobson, M.A.12
Sur, C.13
Duggan, M.E.14
Petitbone, D.J.15
Conn, P.J.16
Williams, D.L.17
-
105
-
-
33744801125
-
Substituent effects of N-(1,3- diphenyl-1H-pyrazol-5-yl)benzamides on positive allosteric modulation of the metabotropic glutamate-5 receptor in rat cortical astrocytes
-
de Paulis, T.; Hemstapat, K.; Chen, Y.; Zhang, Y.; Saleh, S.; Alagille, D.; Baldwin, R.M.; Tamagnan, G.D.; Conn, P.J. Substituent effects of N-(1,3- diphenyl-1H-pyrazol-5-yl)benzamides on positive allosteric modulation of the metabotropic glutamate-5 receptor in rat cortical astrocytes. J. Med. Chem., 2006, 49, 3332-3344.
-
(2006)
J. Med. Chem
, vol.49
, pp. 3332-3344
-
-
de Paulis, T.1
Hemstapat, K.2
Chen, Y.3
Zhang, Y.4
Saleh, S.5
Alagille, D.6
Baldwin, R.M.7
Tamagnan, G.D.8
Conn, P.J.9
-
106
-
-
40749109749
-
1,3-Dipropyl-8-(1- phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists
-
Tabrizi, M.A.; Baraldi, P.G.; Preti, D.; Romagnoli, R.; Saponaro, G.; Baraldi, S.; Moorman, A.R.; Zaid, A.N.; Varani, K.; Borea, P.A. 1,3-Dipropyl-8-(1- phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists. Bioorg. Med. Chem., 2008, 16, 2419-2430.
-
(2008)
Bioorg. Med. Chem
, vol.16
, pp. 2419-2430
-
-
Tabrizi, M.A.1
Baraldi, P.G.2
Preti, D.3
Romagnoli, R.4
Saponaro, G.5
Baraldi, S.6
Moorman, A.R.7
Zaid, A.N.8
Varani, K.9
Borea, P.A.10
-
107
-
-
37049038205
-
Development of a scalable synthesis of gsk183390a, a ppar α/γ agonist
-
Oh, L.M.; Wang, H.; Shilcrat, S.C.; Herrmann, R.E.; Patience, D.B.; Spoors, P.G.; Sisko, J. development of a scalable synthesis of gsk183390a, a ppar α/γ agonist. Org. Proc. Res. Dev., 2007, 11, 1032-1042.
-
(2007)
Org. Proc. Res. Dev
, vol.11
, pp. 1032-1042
-
-
Oh, L.M.1
Wang, H.2
Shilcrat, S.C.3
Herrmann, R.E.4
Patience, D.B.5
Spoors, P.G.6
Sisko, J.7
-
108
-
-
29544446323
-
Antimalarial activity of 4-(5-trifluoromethyl-1H-pyrazol-1-yl)-chloroquine analogues
-
Cunico, W.; Cechinel, C.A.; Bonacorso, H.G.; Martins, M.A.P.; Zanatta, N.; de Souza, M.V.N.; Freitas, I.O.; Soares, R.P.P.; Krettli, A.U. Antimalarial activity of 4-(5-trifluoromethyl-1H-pyrazol-1-yl)-chloroquine analogues. Bioorg. Med. Chem. Lett., 2006, 16, 649-653.
-
(2006)
Bioorg. Med. Chem. Lett
, vol.16
, pp. 649-653
-
-
Cunico, W.1
Cechinel, C.A.2
Bonacorso, H.G.3
Martins, M.A.P.4
Zanatta, N.5
de Souza, M.V.N.6
Freitas, I.O.7
Soares, R.P.P.8
Krettli, A.U.9
-
109
-
-
33846896972
-
5-((1H-Pyrazol-4-yl)methylene)-2- thioxothiazolidin-4-one inhibitors of ADAMTS-5
-
Gilbert, A.M.; Bursavich, M.G.; Lombardi, S.; Georgiadis, K.E.; Reifenberg, E.; Flannery, C.R.; Morris, E.A. 5-((1H-Pyrazol-4-yl)methylene)-2- thioxothiazolidin-4-one inhibitors of ADAMTS-5. Bioorg. Med. Chem. Lett., 2007, 17, 1189-1192.
-
(2007)
Bioorg. Med. Chem. Lett
, vol.17
, pp. 1189-1192
-
-
Gilbert, A.M.1
Bursavich, M.G.2
Lombardi, S.3
Georgiadis, K.E.4
Reifenberg, E.5
Flannery, C.R.6
Morris, E.A.7
-
110
-
-
48449100032
-
Synthesis and antiviral evaluation of some new pyrazole and fused pyrazolopyrimidine derivatives
-
Rashad, A.E.; Hegab, M.I.; Abdel-Megeid, R.E.; Micky, J.A.; Abdel- Megeid, F.M.E. Synthesis and antiviral evaluation of some new pyrazole and fused pyrazolopyrimidine derivatives. Bioorg. Med. Chem., 2008, 16, 7102-7106.
-
(2008)
Bioorg. Med. Chem
, vol.16
, pp. 7102-7106
-
-
Rashad, A.E.1
Hegab, M.I.2
Abdel-Megeid, R.E.3
Micky, J.A.4
Abdel-Megeid, F.M.E.5
-
111
-
-
33644883681
-
Discovery of S-[5-Amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(2,3- dihydroxypropoxy)phenyl]methanone (RO3201195), an orally bioavailable and highly selective Inhibitor of p38 Map Kinase
-
Goldstein, D.M.; Alfredson, T.; Bertrand, J.; Browner, M.F.; Clifford, K.; Dalrymple, S.A.; Dunn, J.; Freire-Moar, J.; Harris, S.; Labadie, S.S.; La Fargue, J.; Lapierre, J.M.; Larrabee, S.; Li, F.; Papp, E.; McWeeney, D.; Ramesha, C.; Roberts, R.; Rotstein, D.; Pablo, B.S.; Sjogren, E.B.; So, O.-Y.; Talamas, F.X.; Tao, W.; Trejo, A.; Villasenor, A.; Welch, M.; Welch, T.; Weller, P.; Whiteley, P.E.; Young, K.; Zipfel, S. Discovery of S-[5-Amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(2,3- dihydroxypropoxy)phenyl]methanone (RO3201195), an orally bioavailable and highly selective Inhibitor of p38 Map Kinase. J. Med. Chem., 2006, 49, 1562-1575.
-
(2006)
J. Med. Chem
, vol.49
, pp. 1562-1575
-
-
Goldstein, D.M.1
Alfredson, T.2
Bertrand, J.3
Browner, M.F.4
Clifford, K.5
Dalrymple, S.A.6
Dunn, J.7
Freire-Moar, J.8
Harris, S.9
Labadie, S.S.10
la Fargue, J.11
Lapierre, J.M.12
Larrabee, S.13
Li, F.14
Papp, E.15
McWeeney, D.16
Ramesha, C.17
Roberts, R.18
Rotstein, D.19
Pablo, B.S.20
Sjogren, E.B.21
So, O.-Y.22
Talamas, F.X.23
Tao, W.24
Trejo, A.25
Villasenor, A.26
Welch, M.27
Welch, T.28
Weller, P.29
Whiteley, P.E.30
Young, K.31
Zipfel, S.32
more..
-
112
-
-
44849132107
-
Diazen-1-ium- 1,2-diolated nitric oxide donor ester prodrugs of 1-(4- methanesulfonylphenyl)-5-aryl-1H-pyrazol-3-carboxylic acids: Synthesis, nitric oxide release studies and anti-inflammatory activities
-
Abdellatif, K.R.A.; Chowdhury, M.A.; Dong, Y.; Knaus, E.E. Diazen-1-ium- 1,2-diolated nitric oxide donor ester prodrugs of 1-(4- methanesulfonylphenyl)-5-aryl-1H-pyrazol-3-carboxylic acids: Synthesis, nitric oxide release studies and anti-inflammatory activities. Bioorg. Med. Chem., 2008, 16, 6528-6534.
-
(2008)
Bioorg. Med. Chem
, vol.16
, pp. 6528-6534
-
-
Abdellatif, K.R.A.1
Chowdhury, M.A.2
Dong, Y.3
Knaus, E.E.4
-
113
-
-
48949115102
-
Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide (SR141716) a potent CB1 receptor antagonist
-
Srivastava, B.K.; Soni, R.; Patel, J.Z.; Jha, S.; Shedage, S.A.; Gandhi, N.; Sairam, K.V.V.M.; Pawar, V.; Sadhwani, N.; Mitra, P.; Jain, M.R.; Patel, P.R. Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide (SR141716) a potent CB1 receptor antagonist. Bioorg. Med. Chem. Lett., 2008, 18, 3882-3886.
-
(2008)
Bioorg. Med. Chem. Lett
, vol.18
, pp. 3882-3886
-
-
Srivastava, B.K.1
Soni, R.2
Patel, J.Z.3
Jha, S.4
Shedage, S.A.5
Gandhi, N.6
Sairam, K.V.V.M.7
Pawar, V.8
Sadhwani, N.9
Mitra, P.10
Jain, M.R.11
Patel, P.R.12
-
114
-
-
20144379406
-
Bioisosteric replacements of the pyrazole moiety of rimonabant: Synthesis, biological properties, and molecular modeling investigations of thiazoles, triazoles, and imidazoles as potent and selective cb1 cannabinoid receptor antagonists
-
Lange, J.H.M.; van Stuivenberg, H.H.; Coolen, H.K.A.C.; Adolfs, T.J.P.; McCreary, A.C.; Keizer, H.G.; Wals, H.C.; Veerman, W.; Borst, A.J.M.; de Looff, W.; Verveer, P.C.; Kruse, C.G. bioisosteric replacements of the pyrazole moiety of rimonabant: synthesis, biological properties, and molecular modeling investigations of thiazoles, triazoles, and imidazoles as potent and selective cb1 cannabinoid receptor antagonists. J. Med. Chem., 2005, 48, 1823-1838.
-
(2005)
J. Med. Chem
, vol.48
, pp. 1823-1838
-
-
Lange, J.H.M.1
van Stuivenberg, H.H.2
Coolen, H.K.A.C.3
Adolfs, T.J.P.4
McCreary, A.C.5
Keizer, H.G.6
Wals, H.C.7
Veerman, W.8
Borst, A.J.M.9
de Looff, W.10
Verveer, P.C.11
Kruse, C.G.12
-
115
-
-
33746693727
-
Phototransformation of the insecticide fipronil: Identification of novel photoproducts and evidence for an alternative pathway of photodegradation
-
Raveton, M.; Aajoud, A.; Willison, J.C.; Aouadi, H.; Tissut, M.; Ravanel, P. phototransformation of the insecticide fipronil: identification of novel photoproducts and evidence for an alternative pathway of photodegradation. Environ. Sci. Technol., 2006, 40, 4151-4157.
-
(2006)
Environ. Sci. Technol
, vol.40
, pp. 4151-4157
-
-
Raveton, M.1
Aajoud, A.2
Willison, J.C.3
Aouadi, H.4
Tissut, M.5
Ravanel, P.6
-
116
-
-
0033784992
-
Elucidation of Fipronil Photodegradation pathways
-
Ngim, K.K.; Mabury, S.A.; Crosby, D.G. Elucidation of Fipronil Photodegradation pathways. J. Agric. Food Chem., 2000, 48, 4661-4665.
-
(2000)
J. Agric. Food Chem
, vol.48
, pp. 4661-4665
-
-
Ngim, K.K.1
Mabury, S.A.2
Crosby, D.G.3
-
117
-
-
43449106481
-
Improved regioselectivity in pyrazole formation through the use of fluorinated alcohols as solvents: Synthesis and biological activity of fluorinated tebufenpyrad analogs
-
Fustero, S.; Román, R.; Sanz-Cervera, J.F.; Simón-Fuentes, A.; Cuñat, A.C.; Villanova, S.; Murguía, M. improved regioselectivity in pyrazole formation through the use of fluorinated alcohols as solvents: synthesis and biological activity of fluorinated tebufenpyrad analogs. J. Org. Chem., 2008, 73, 3523-3529.
-
(2008)
J. Org. Chem
, vol.73
, pp. 3523-3529
-
-
Fustero, S.1
Román, R.2
Sanz-Cervera, J.F.3
Simón-Fuentes, A.4
Cuñat, A.C.5
Villanova, S.6
Murguía, M.7
-
118
-
-
0033666768
-
Metabolism of Furametpyr. 1. identification of metabolites and in vitro biotransformation in rats and humans
-
Nagahori, H.; Yoshino, H.; Tomigahara, Y.; Isobe, N.; Kaneko, H.; Nakatsuka, I. Metabolism of Furametpyr. 1. identification of metabolites and in vitro biotransformation in rats and humans. J. Agric. Food Chem., 2000, 48, 5754-5759.
-
(2000)
J. Agric. Food Chem
, vol.48
, pp. 5754-5759
-
-
Nagahori, H.1
Yoshino, H.2
Tomigahara, Y.3
Isobe, N.4
Kaneko, H.5
Nakatsuka, I.6
-
119
-
-
20444415984
-
Identification of antitumor activity of pyrazole oxime ethers
-
Park, H.-J.; Lee, K.; Park, S.-J.; Ahn, B.; Lee, J.-C.; Cho, H.Y.; Lee, K.-I. Identification of antitumor activity of pyrazole oxime ethers. Bioorg. Med. Chem. Lett., 2005, 15, 3307-3312.
-
(2005)
Bioorg. Med. Chem. Lett
, vol.15
, pp. 3307-3312
-
-
Park, H.-J.1
Lee, K.2
Park, S.-J.3
Ahn, B.4
Lee, J.-C.5
Cho, H.Y.6
Lee, K.-I.7
-
120
-
-
37849017426
-
Substituted pyrazoles as hepatoselective HMG-CoA reductase inhibitors: Discovery of (3R,5R)-7-[2-(4-Fluoro-phenyl)-4-isopropyl-5-(4-methyl-benzylcarbamoyl)-2H-pyrazol-3-yl]-3,5- dihydroxyheptanoic Acid (PF-3052334) as a Candidate for the Treatment of Hypercholesterolemia
-
Pfefferkorn, J.A.; Choi, C.; Larsen, S.D.; Auerbach, B.; Hutchings, R.; Park, W.; Askew, A.; Dillon, L.; Hanselman, J.C.; Lin, Z.; Lu, G.H.; Robertson, A.; Sekerke, C.; Harris, M.S.; Pavlovsky, A.; Bainbridge, G.; Caspers, N.; Kowala, M., Tait, B. D. Substituted pyrazoles as hepatoselective HMG-CoA reductase inhibitors: discovery of (3R,5R)-7-[2-(4-Fluoro-phenyl)-4-isopropyl-5-(4-methyl-benzylcarbamoyl)-2H-pyrazol-3-yl]-3,5- dihydroxyheptanoic Acid (PF-3052334) as a Candidate for the Treatment of Hypercholesterolemia. J. Med. Chem., 2008, 51, 31-45.
-
(2008)
J. Med. Chem
, vol.51
, pp. 31-45
-
-
Pfefferkorn, J.A.1
Choi, C.2
Larsen, S.D.3
Auerbach, B.4
Hutchings, R.5
Park, W.6
Askew, A.7
Dillon, L.8
Hanselman, J.C.9
Lin, Z.10
Lu, G.H.11
Robertson, A.12
Sekerke, C.13
Harris, M.S.14
Pavlovsky, A.15
Bainbridge, G.16
Caspers, N.17
Kowala, M.18
Tait, B.D.19
-
121
-
-
4143078217
-
A study on the synthesis and photophysical performances of some pyrazole and triazole fluorescent brightening agents
-
Wang, X.; Li, W.; Zhang, X.-H.; Liu, D.-Z.; Zhou, X.-Q. A study on the synthesis and photophysical performances of some pyrazole and triazole fluorescent brightening agents. Dyes Pig., 2005, 64(2), 141-146.
-
(2005)
Dyes Pig
, vol.64
, Issue.2
, pp. 141-146
-
-
Wang, X.1
Li, W.2
Zhang, X.-H.3
Liu, D.-Z.4
Zhou, X.-Q.5
-
122
-
-
0038729126
-
Photoinduced electron transfer reactions of 3H-Pyrazole derivatives. Formation of solvent adduct by specific sensitizer
-
Karatsu, T.; Shiochi, N.; Aono, T.; Miyagawa, N.; Kitamura, A. Photoinduced electron transfer reactions of 3H-Pyrazole derivatives. Formation of solvent adduct by specific sensitizer. Bull. Chem. Soc. Jpn., 2003, 76(6), 1227-1231.
-
(2003)
Bull. Chem. Soc. Jpn
, vol.76
, Issue.6
, pp. 1227-1231
-
-
Karatsu, T.1
Shiochi, N.2
Aono, T.3
Miyagawa, N.4
Kitamura, A.5
-
123
-
-
3042567398
-
Photoinduced electron transfer reactions of 3,3-Dialkylated 4,5-diphenyl-3H-pyrazoles: A new route to the formation of the solvent adducts
-
Yen, Y.-P.; Huang, T.-M.; Tseng, Y.-P.; Lin, H.-Y.; Lai, C.-C. Photoinduced electron transfer reactions of 3,3-Dialkylated 4,5-diphenyl-3H-pyrazoles: A new route to the formation of the solvent adducts. J. Chin. Chem. Soc., 2004, 51(2), 393-398.
-
(2004)
J. Chin. Chem. Soc
, vol.51
, Issue.2
, pp. 393-398
-
-
Yen, Y.-P.1
Huang, T.-M.2
Tseng, Y.-P.3
Lin, H.-Y.4
Lai, C.-C.5
-
124
-
-
33746611878
-
Syntheses and properties of new photochromic diarylethene derivatives having a pyrazole unit
-
Pu, S.; Yang, T.; Xu, J.; Chen, B. Syntheses and properties of new photochromic diarylethene derivatives having a pyrazole unit. Tetrahedron Lett., 2006, 47(36), 6473-6477.
-
(2006)
Tetrahedron Lett
, vol.47
, Issue.36
, pp. 6473-6477
-
-
Pu, S.1
Yang, T.2
Xu, J.3
Chen, B.4
-
125
-
-
35048850347
-
Synthesis and Solid-State Photochromism of 1,3-Diphenyl-4- (2-chlorobenzal)-5-hydroxypyrazole 4- methylthiosemicarbazone
-
Guo, J.; Liu, L.; Liu, G.; Jia, D.; Xie, X. Synthesis and Solid-State Photochromism of 1,3-Diphenyl-4- (2-chlorobenzal)-5-hydroxypyrazole 4- methylthiosemicarbazone. Org. Lett., 2007, 9(20), 3989-3992.
-
(2007)
Org. Lett
, vol.9
, Issue.20
, pp. 3989-3992
-
-
Guo, J.1
Liu, L.2
Liu, G.3
Jia, D.4
Xie, X.5
-
126
-
-
11844287668
-
Phosphorescent organogels via "Metallophilic" interactions for reversible RGB-color switching
-
Kishimura, A.; Yamashita, T.; Aida, T. Phosphorescent organogels via "Metallophilic" interactions for reversible RGB-color switching. J. Am. Chem. Soc., 2005, 127, 179-183.
-
(2005)
J. Am. Chem. Soc
, vol.127
, pp. 179-183
-
-
Kishimura, A.1
Yamashita, T.2
Aida, T.3
-
127
-
-
48849102030
-
Blueemitting cationic iridium complexes with 2-(1H-Pyrazol-1-yl)pyridine as the ancillary ligand for efficient light-emitting electrochemical cells
-
He, L.; Duan, L.; Qiao, J.; Wang, R.; Wei, P.; Wang, L.; Qiu, Y. Blueemitting cationic iridium complexes with 2-(1H-Pyrazol-1-yl)pyridine as the ancillary ligand for efficient light-emitting electrochemical cells. Adv. Funct. Mater., 2008, 18, 2123-2131.
-
(2008)
Adv. Funct. Mater
, vol.18
, pp. 2123-2131
-
-
He, L.1
Duan, L.2
Qiao, J.3
Wang, R.4
Wei, P.5
Wang, L.6
Qiu, Y.7
-
128
-
-
33745684776
-
New Efficient bluegreenish electroluminescent materials of 1,3,4-Oxadiazole-based pyrazole DERIVATIVES
-
Chang, E.-M.; Lin, C.J.; Wong, F.F.; Yeh, M.-Y. New Efficient bluegreenish electroluminescent materials of 1,3,4-Oxadiazole-based pyrazole DERIVATIVES. Heterocycles, 2006, 68(4), 733-748.
-
(2006)
Heterocycles
, vol.68
, Issue.4
, pp. 733-748
-
-
Chang, E.-M.1
Lin, C.J.2
Wong, F.F.3
Yeh, M.-Y.4
-
129
-
-
0035208217
-
Difunctional pyrazole derivatives - key compounds en route to multidentate pyrazolate ligands
-
Röder, J.C.; Meyer, F.; Konrad, M.; Sandhöfner, S.; Kaifer, E.; Pritzkow, H. Difunctional pyrazole derivatives - key compounds en route to multidentate pyrazolate ligands. Eur. J. Org. Chem., 2001, (23), 4479-4487.
-
(2001)
Eur. J. Org. Chem
, vol.23
, pp. 4479-4487
-
-
Röder, J.C.1
Meyer, F.2
Konrad, M.3
Sandhöfner, S.4
Kaifer, E.5
Pritzkow, H.6
-
130
-
-
53849090649
-
Manganese(II) coordination polymer with ditopic bis(pyrazol-1-yl)borate bridges
-
Morawitz, T.; Bolte, M.; Lerner, H.-W.; Wagner, M. A manganese(II) coordination polymer with ditopic bis(pyrazol-1-yl)borate bridges. Z. Anorg. Allg. Chem., 2008, 634, 1409-1414.
-
(2008)
Z. Anorg. Allg. Chem
, vol.634
, pp. 1409-1414
-
-
Morawitz, T.1
Bolte, M.2
Lerner, H.-W.3
Wagner, M.A.4
-
131
-
-
33947402170
-
Anion doping as a probe of cooperativity in the molecular spin-crossover compound [FeL2][BF4]2 (L = 2,6-di{pyrazol-1-yl}pyridine)
-
Carbonera, C.; Kilner, C.A.; Létard, J.-F.; Halcrow, M.A. Anion doping as a probe of cooperativity in the molecular spin-crossover compound [FeL2][BF4]2 (L = 2,6-di{pyrazol-1-yl}pyridine). J. Chem. Soc., Dalton Trans., 2007, 1284-1292.
-
(2007)
J. Chem. Soc., Dalton Trans
, pp. 1284-1292
-
-
Carbonera, C.1
Kilner, C.A.2
Létard, J.-F.3
Halcrow, M.A.4
-
132
-
-
46149089610
-
Selective extraction, separation and speciation of iron in different samples using 4-acetyl-5-methyl-1-phenyl-1H-pyrazole-3- carboxylic acid
-
Saçmaci, Ş.; Kartal, Ş. Selective extraction, separation and speciation of iron in different samples using 4-acetyl-5-methyl-1-phenyl-1H-pyrazole-3- carboxylic acid. Anal. Chim. Acta, 2008, 623, 46-52.
-
(2008)
Anal. Chim. Acta
, vol.623
, pp. 46-52
-
-
Saçmaci, S.1
Kartal, S.2
-
133
-
-
51549114661
-
Redox-Active p-Quinone-Based Bis(pyrazol-1-yl)methane Ligands: Synthesis and Coordination Behaviour
-
Scheuermann, S.; Kretz, T.; Vitze, H.; Bats, J.W.; Bolte, M.; Lerner, H.-W.; Wagner, M. Redox-Active p-Quinone-Based Bis(pyrazol-1-yl)methane Ligands: Synthesis and Coordination Behaviour. Chem. Eur. J., 2008, 14(8), 2590-2601.
-
(2008)
Chem. Eur. J
, vol.14
, Issue.8
, pp. 2590-2601
-
-
Scheuermann, S.1
Kretz, T.2
Vitze, H.3
Bats, J.W.4
Bolte, M.5
Lerner, H.-W.6
Wagner, M.7
-
134
-
-
12344310469
-
Multifunctional high-spin biradical pyrazolylbipyridine-bisnitronylnitroxide
-
Zoppellaro, G.; Enkelmann, V.; Geies, A.; Baumgarten, M. A Multifunctional high-spin biradical pyrazolylbipyridine-bisnitronylnitroxide. Org. Lett., 2004, 6(26), 4929-4932.
-
(2004)
Org. Lett
, vol.6
, Issue.26
, pp. 4929-4932
-
-
Zoppellaro, G.1
Enkelmann, V.2
Geies, A.3
Baumgarten, M.A.4
-
135
-
-
4544220557
-
2,6- Bis(pyrazolyl)pyridine functionalised with two nitronylnitroxide and iminonitroxide radicals
-
Zoppellaro, G.; Geies, A.; Enkelmann, V.; Baumgarten, M. 2,6- Bis(pyrazolyl)pyridine functionalised with two nitronylnitroxide and iminonitroxide radicals. Eur. J. Org. Chem., 2004, (11), 2367-2374.
-
(2004)
Eur. J. Org. Chem
, Issue.11
, pp. 2367-2374
-
-
Zoppellaro, G.1
Geies, A.2
Enkelmann, V.3
Baumgarten, M.4
-
136
-
-
53849098580
-
Schiff Base macrocycles containing pyrroles and pyrazoles
-
Katsiaouni, S.; Dechert, S.; Briñas, R.P.; Brückner, C.; Meyer, F. Schiff Base macrocycles containing pyrroles and pyrazoles. Chem. Eur. J., 2008, 14, 4823-4835.
-
(2008)
Chem. Eur. J
, vol.14
, pp. 4823-4835
-
-
Katsiaouni, S.1
Dechert, S.2
Briñas, R.P.3
Brückner, C.4
Meyer, F.5
-
137
-
-
33846610111
-
Synthesis and characterization of pyrazolyl-functionalized imidazolium-based ionic liquids and hemilabile (carbene)palladium(ii) complex catalyzed heck reaction
-
Wang, R.; Zeng, Z.; Twamley, B.; Piekarski, M.M.; Shreeve, J.M. synthesis and characterization of pyrazolyl-functionalized imidazolium-based ionic liquids and hemilabile (carbene)palladium(ii) complex catalyzed heck reaction. Eur. J. Org. Chem., 2007, (4), 655-661.
-
(2007)
Eur. J. Org. Chem
, Issue.4
, pp. 655-661
-
-
Wang, R.1
Zeng, Z.2
Twamley, B.3
Piekarski, M.M.4
Shreeve, J.M.5
-
138
-
-
24944570649
-
New Pyrazolino- and Pyrrolidino[60]fullerenes with Transition-Metal Chelating Pyridine Substituents: Synthesis and Complexation to Ru(II)
-
Modin, J.; Johansson, H.; Grennberg, H. New Pyrazolino- and Pyrrolidino[60]fullerenes with Transition-Metal Chelating Pyridine Substituents: Synthesis and Complexation to Ru(II). Org. Lett., 2005, 7(18), 3977-3979.
-
(2005)
Org. Lett
, vol.7
, Issue.18
, pp. 3977-3979
-
-
Modin, J.1
Johansson, H.2
Grennberg, H.3
-
139
-
-
66249139887
-
MTO/H2O2/Pyrazole-Mediated NOxidation of meso-Tetraarylporphyrins and -chlorins, and S-Oxidation of a meso-Tetraaryldithiaporphyrin and -chlorin
-
Banerjee, S.; Zeller, M.; Brückner, C. MTO/H2O2/Pyrazole-Mediated NOxidation of meso-Tetraarylporphyrins and -chlorins, and S-Oxidation of a meso-Tetraaryldithiaporphyrin and -chlorin. J. Org. Chem., 2009, 74(11), 4283-4288.
-
(2009)
J. Org. Chem
, vol.74
, Issue.11
, pp. 4283-4288
-
-
Banerjee, S.1
Zeller, M.2
Brückner, C.3
-
140
-
-
0033565013
-
Role of Aggregates in Claisen acylation reactions of imidazole, Pyrazole, and Thioesters with Lithium Enolates in THF
-
Streitwieser, A.; Leung, S.S.-W.; Kim, Y.-J. Role of Aggregates in Claisen acylation reactions of imidazole, Pyrazole, and Thioesters with Lithium Enolates in THF. Org. Lett., 1999, 1(1), 145-147.
-
(1999)
Org. Lett
, vol.1
, Issue.1
, pp. 145-147
-
-
Streitwieser, A.1
Leung, S.S.-W.2
Kim, Y.-J.3
-
141
-
-
18244398634
-
Enantioselective Enol lactone synthesis under double catalytic conditions
-
Itoh, K.; Hasegawa, M.; Tanaka, J.; Kanemasa, S. Enantioselective Enol lactone synthesis under double catalytic conditions. Org. Lett., 2005, 7(6), 979-981.
-
(2005)
Org. Lett
, vol.7
, Issue.6
, pp. 979-981
-
-
Itoh, K.1
Hasegawa, M.2
Tanaka, J.3
Kanemasa, S.4
-
142
-
-
0035954866
-
Efficient introduction of protected guanidines in BOC solid phase peptide synthesis
-
Zhang, Y.; Kennan, A.J. Efficient introduction of protected guanidines in BOC solid phase peptide synthesis. Org. Lett., 2001, 3(15), 2341-2344.
-
(2001)
Org. Lett
, vol.3
, Issue.15
, pp. 2341-2344
-
-
Zhang, Y.1
Kennan, A.J.2
-
143
-
-
18544410293
-
Optimisation of the Synthesis of guanidines from amines via nitroguanidines Using 3,5-Dimethyl-N-nitro-1Hpyrazole-1-carboxamidine
-
Castillo-Meléndez, J.A.; Golding, B.T. Optimisation of the Synthesis of guanidines from amines via nitroguanidines Using 3,5-Dimethyl-N-nitro-1Hpyrazole-1-carboxamidine. Synthesis, 2004, (10), 1655-1663.
-
(2004)
Synthesis
, vol.10
, pp. 1655-1663
-
-
Castillo-Meléndez, J.A.1
Golding, B.T.2
-
144
-
-
8144231437
-
3(5)-(2-Hydroxyphenyl)-5(3)-styrylpyrazoles: Synthesis and Diels-Alder Transformations
-
Silva, V.L.M.; Silva, A.M.S.; Pinto, D.C. G.A.; Cavaleiro, J.A.S.; Elguero, J. 3(5)-(2-Hydroxyphenyl)-5(3)-styrylpyrazoles: Synthesis and Diels-Alder Transformations. Eur. J. Org. Chem., 2004, (21), 4348-4356.
-
(2004)
Eur. J. Org. Chem
, vol.21
, pp. 4348-4356
-
-
Silva, V.L.M.1
Silva, A.M.S.2
Pinto, D.C.G.A.3
Cavaleiro, J.A.S.4
Elguero, J.5
-
145
-
-
0037327598
-
New bis(chalcones) and their transformation into Bis(pyrazoline) and bis(pyrazole) derivatives
-
Pinto, D.C.G.A.; Silva, A.M.S.; Cavaleiro, J.A.S.; Elguero, J. New bis(chalcones) and their transformation into Bis(pyrazoline) and bis(pyrazole) derivatives. Eur. J. Org. Chem., 2003, (4), 747-755.
-
(2003)
Eur. J. Org. Chem
, vol.4
, pp. 747-755
-
-
Pinto, D.C.G.A.1
Silva, A.M.S.2
Cavaleiro, J.A.S.3
Elguero, J.4
-
146
-
-
0043287135
-
Oligo(1,4-phenylenepyrazole-3,5-diyl)s
-
Meier, H.; Hormaza, A. Oligo(1,4-phenylenepyrazole-3,5-diyl)s. Eur. J. Org. Chem., 2003, (17), 3372-3377.
-
(2003)
Eur. J. Org. Chem
, vol.17
, pp. 3372-3377
-
-
Meier, H.1
Hormaza, A.2
-
147
-
-
35948963968
-
SmCl3-Catalyzed C-Acylation of 1,3-Dicarbonyl compounds and malononitrile
-
Shen, Q.; Huang, W.; Wang, J.; Zhou, X. SmCl3-Catalyzed C-Acylation of 1,3-Dicarbonyl compounds and malononitrile. Org. Lett., 2007, 9(22), 4491-4494.
-
(2007)
Org. Lett
, vol.9
, Issue.22
, pp. 4491-4494
-
-
Shen, Q.1
Huang, W.2
Wang, J.3
Zhou, X.4
-
148
-
-
33744477678
-
Three-Component, one-pot reaction for the combinatorial synthesis of 1,3,4-substituted pyrazoles
-
Xie, F.; Cheng, G.; Hu, Y. Three-Component, one-pot reaction for the combinatorial synthesis of 1,3,4-substituted pyrazoles. J. Comb. Chem., 2006, 8, 286-288.
-
(2006)
J. Comb. Chem
, vol.8
, pp. 286-288
-
-
Xie, F.1
Cheng, G.2
Hu, Y.3
-
149
-
-
12344281353
-
Synthesis of Pyrazolyl-2-pyrazolines by Treatment of 3-(3-Aryl-3-oxopropenyl)chromen-4-ones with hydrazine and their oxidation to Bis(pyrazoles)
-
Lévai, A.; Silva, A.M.S.; Pinto, D.C.G.A.; Cavaleiro, J.A.S.; Alkorta, I.; Elguero, J.; Jekö, J. Synthesis of Pyrazolyl-2-pyrazolines by Treatment of 3-(3-Aryl-3-oxopropenyl)chromen-4-ones with hydrazine and their oxidation to Bis(pyrazoles). Eur. J. Org. Chem., 2004, (22), 4672-4679.
-
(2004)
Eur. J. Org. Chem
, vol.22
, pp. 4672-4679
-
-
Lévai, A.1
Silva, A.M.S.2
Pinto, D.C.G.A.3
Cavaleiro, J.A.S.4
Alkorta, I.5
Elguero, J.6
Jekö, J.7
-
150
-
-
0036859230
-
3-Aroyl-5-hydroxyflavones: Synthesis and transformation into aroylpyrazoles
-
Pinto, D.C.G.A.; Silva, A.M.S.; Almeida, L.M.P.M.; Cavaleiro, J.A.S; Elguero J. 3-Aroyl-5-hydroxyflavones: synthesis and transformation into aroylpyrazoles. Eur. J. Org. Chem., 2002, (22), 3807-3815.
-
(2002)
Eur. J. Org. Chem
, vol.22
, pp. 3807-3815
-
-
Pinto, D.C.G.A.1
Silva, A.M.S.2
Almeida, L.M.P.M.3
Cavaleiro, J.A.S.4
Elguero, J.5
-
151
-
-
84961980498
-
Synthesis of pyrazoles by treatment of 3-Benzylchromones, 3-Benzylflavones and their 4-Thio analogues with hydrazine
-
Lévai, A.; Silva, A.M.S.; Cavaleiro, J.A.S.; Alkorta, I.; Elguero, J.; Jekö, J. Synthesis of pyrazoles by treatment of 3-Benzylchromones, 3-Benzylflavones and their 4-Thio analogues with hydrazine. Eur. J. Org. Chem., 2006, (12), 2825-2832.
-
(2006)
Eur. J. Org. Chem
, vol.12
, pp. 2825-2832
-
-
Lévai, A.1
Silva, A.M.S.2
Cavaleiro, J.A.S.3
Alkorta, I.4
Elguero, J.5
Jekö, J.6
-
152
-
-
0034365633
-
Syntheses of Pyrazole Iso-C-nucleosides
-
Michalik, D.; Peseke, K. Syntheses of Pyrazole Iso-C-nucleosides. J. Carbohydr Chem., 2000, 19(8), 1049-1057.
-
(2000)
J. Carbohydr Chem
, vol.19
, Issue.8
, pp. 1049-1057
-
-
Michalik, D.1
Peseke, K.2
-
153
-
-
0035850191
-
Synthesis of derivatives of C-nucleoside analogues using 'push-pull' functionalized monosaccharides
-
Michalik, D.; Feist, H.; Peseke, K. Synthesis of derivatives of C-nucleoside analogues using 'push-pull' functionalized monosaccharides. Carbohydr Res., 2001, 333, 197-201.
-
(2001)
Carbohydr Res
, vol.333
, pp. 197-201
-
-
Michalik, D.1
Feist, H.2
Peseke, K.3
-
154
-
-
32244449191
-
Regioselective synthesis of 4-(2-alkyl-5-methyl-2H-pyrazol-3-yl)- piperidines
-
Dirat, O.; Clipson, A.; Elliot, J.M.; Garrett, S.; Jones, A.B.; Reader, M.; Shaw, D. Regioselective synthesis of 4-(2-alkyl-5-methyl-2H-pyrazol-3-yl)- piperidines. Tetrahedron Lett., 2006, 47, 1729-1731.
-
(2006)
Tetrahedron Lett
, vol.47
, pp. 1729-1731
-
-
Dirat, O.1
Clipson, A.2
Elliot, J.M.3
Garrett, S.4
Jones, A.B.5
Reader, M.6
Shaw, D.7
-
155
-
-
19944402969
-
New hydroxy-pyrazoline intermediates, subtle regioselectivity and relative reaction rate variations observed during acid catalyzed and neutral pyrazole cyclization
-
Norris, T.; Colon-Cruz, R.; Ripin, D.H.B. New hydroxy-pyrazoline intermediates, subtle regioselectivity and relative reaction rate variations observed during acid catalyzed and neutral pyrazole cyclization. Org. Biomol. Chem., 2005, 3, 1844-1849.
-
(2005)
Org. Biomol. Chem
, vol.3
, pp. 1844-1849
-
-
Norris, T.1
Colon-Cruz, R.2
Ripin, D.H.B.3
-
156
-
-
0033803272
-
The reaction between hydrazines and-dicarbonyl compounds: Proposal for a mechanism
-
Elguero, J.; Rozas, I.; Singh, S.P.; Kumar, D.; Batra, H.; Naithani, R. The reaction between hydrazines and-dicarbonyl compounds: proposal for a mechanism. Can. J. Chem., 2000, 78(8), 1109-1120.
-
(2000)
Can. J. Chem
, vol.78
, Issue.8
, pp. 1109-1120
-
-
Elguero, J.1
Rozas, I.2
Singh, S.P.3
Kumar, D.4
Batra, H.5
Naithani, R.6
-
157
-
-
37049090641
-
Mechanisms of heterocycle ring formation. Part 5. A carbon-13 nuclear magnetic resonance study of pyrazolinone synthesis by the reaction of-ketoesters with substituted hydrazine
-
Katritzky, A.R.; Barczynski, P.; Ostercamp, D.L. Mechanisms of heterocycle ring formation. Part 5. A carbon-13 nuclear magnetic resonance study of pyrazolinone synthesis by the reaction of-ketoesters with substituted hydrazines. J. Chem. Soc., Perkin Trans. II, 1987, (8), 969-975.
-
(1987)
J. Chem. Soc., Perkin Trans
, vol.II
, Issue.8
, pp. 969-975
-
-
Katritzky, A.R.1
Barczynski, P.2
Ostercamp, D.L.3
-
158
-
-
33747409049
-
The reaction of aryl and heteroarylhydrazines with aryl-trifluoromethyl-diketones
-
Singh, S.P.; Kumar, V.; Aggarwal, R.; Elguero, J. The reaction of aryl and heteroarylhydrazines with aryl-trifluoromethyl-diketones. J. Heterocycl. Chem., 2006, 43(4), 1003-1014.
-
(2006)
J. Heterocycl. Chem
, vol.43
, Issue.4
, pp. 1003-1014
-
-
Singh, S.P.1
Kumar, V.2
Aggarwal, R.3
Elguero, J.4
-
159
-
-
33644889440
-
Regioselectivity in the formation of norbornene-fused pyrazoles: Preparation of 1- substituted derivatives of 4,5,6,7-tetrahydro-1H-4,7-methanoindazole
-
Fernández, F.; Caamaño, O.; García, M.D.; Alkorta, I.; Elguero, J. Regioselectivity in the formation of norbornene-fused pyrazoles: preparation of 1- substituted derivatives of 4,5,6,7-tetrahydro-1H-4,7-methanoindazole. Tetrahedron, 2006, 62, 3362-3369.
-
(2006)
Tetrahedron
, vol.62
, pp. 3362-3369
-
-
Fernández, F.1
Caamaño, O.2
García, M.D.3
Alkorta, I.4
Elguero, J.5
-
160
-
-
45749090163
-
Pyrazole formation: Examination of kinetics, substituent effects, and mechanistic pathways
-
Sloop, J.C.; Lechner, B.; Washington, G.; Bumgardner, C.L.; Loehle, W.D.; Creasy, W. Pyrazole formation: examination of kinetics, substituent effects, and mechanistic pathways. Int. J. Chem. Kin., 2008, 40, 370-383.
-
(2008)
Int. J. Chem. Kin
, vol.40
, pp. 370-383
-
-
Sloop, J.C.1
Lechner, B.2
Washington, G.3
Bumgardner, C.L.4
Loehle, W.D.5
Creasy, W.6
-
161
-
-
0000808376
-
Rearrangements and cyclization-XVII: Mechanism of the formation of 1,2-azoles in reactions of 1,1-diacyclopropanes with hydrazine and hydroxylamine derivatives
-
Zefirov, N.S.; Kozhushkov, S.I.; Kuznetsova, T.S.; Ershov, B.A.; Selivanov, S.I. Rearrangements and cyclization-XVII: Mechanism of the formation of 1,2-azoles in reactions of 1,1-diacyclopropanes with hydrazine and hydroxylamine derivatives. Tetrahedron, 1986, 42(2), 709-713.
-
(1986)
Tetrahedron
, vol.42
, Issue.2
, pp. 709-713
-
-
Zefirov, N.S.1
Kozhushkov, S.I.2
Kuznetsova, T.S.3
Ershov, B.A.4
Selivanov, S.I.5
-
162
-
-
0002650309
-
Isolation of dihydroxypyrazolidine and 5-hydroxy- 2-pyrazoline intermediates in the synthesis of pyrazoles from-diketones and hydrazine
-
Elguero, J.; Yranzo, G.I. Isolation of dihydroxypyrazolidine and 5-hydroxy- 2-pyrazoline intermediates in the synthesis of pyrazoles from-diketones and hydrazine. J. Chem. Res. Synopses, 1990, (4), 120-121.
-
(1990)
J. Chem. Res. Synopses
, vol.4
, pp. 120-121
-
-
Elguero, J.1
Yranzo, G.I.2
-
163
-
-
0242487852
-
1,1,1- Trichloro-4,4-diethoxy-3-buten-2-one and its trichloroacetylacetate derivatives: Synthesis and applications in regiospecific preparation of azoles
-
Martins, M.A.P.; Pereira, C.M.P.; Zimmermann, N.E.K.; Moura, S. Sinhorin, A.P.; Cunico, W.; Zanatta, N.; Bonacorso, H.G.; Flores, A.C.F. 1,1,1- Trichloro-4,4-diethoxy-3-buten-2-one and its trichloroacetylacetate derivatives: synthesis and applications in regiospecific preparation of azoles. Synthesis, 2003, (15), 2353-2357.
-
(2003)
Synthesis
, vol.15
, pp. 2353-2357
-
-
Martins, M.A.P.1
Pereira, C.M.P.2
Zimmermann, N.E.K.3
Moura, S.4
Sinhorin, A.P.5
Cunico, W.6
Zanatta, N.7
Bonacorso, H.G.8
Flores, A.C.F.9
-
164
-
-
0034627385
-
Synthesis of 3- trialkylsilyl pyrazoles from β-oxo acylsilane
-
Gérard, S.; Plantier-Royon, R.; Nuzillard, J.-M.; Portella, C. Synthesis of 3- trialkylsilyl pyrazoles from β-oxo acylsilanes. Tetrahedron Lett., 2000, 41(50), 9791-9795.
-
(2000)
Tetrahedron Lett
, vol.41
, Issue.50
, pp. 9791-9979
-
-
Gérard, S.1
Plantier-Royon, R.2
Nuzillard, J.-M.3
Portella, C.4
-
165
-
-
33746402789
-
Synthesis of new trifluoromethyl-containing 1-(3,5- dialkyl-4-hydroxybenzyl)-pyrazole and -pyrazol-5-one deriatives and their corresponding aroxyls
-
Dinoiu, V.; Lü, J.-M. Synthesis of new trifluoromethyl-containing 1-(3,5- dialkyl-4-hydroxybenzyl)-pyrazole and -pyrazol-5-one deriatives and their corresponding aroxyls. J. Serb. Chem. Soc., 2006, 71(4), 323-330.
-
(2006)
J. Serb. Chem. Soc
, vol.71
, Issue.4
, pp. 323-330
-
-
Dinoiu, V.1
Lü, J.-M.2
-
166
-
-
56249118348
-
An improved preparation of 3- alkoxypyrazoles
-
Guillou, S.; Bonhomme, F.J.; Janin, Y.L. An improved preparation of 3- alkoxypyrazoles. Synthesis, 2008, (21), 3504-3508.
-
(2008)
Synthesis
, vol.21
, pp. 3504-3508
-
-
Guillou, S.1
Bonhomme, F.J.2
Janin, Y.L.3
-
167
-
-
2542589435
-
Fully automated Polymer-Assisted synthesis of 1,5-Biaryl pyrazoles
-
Vickerstaffe, E.; Warrington, B.H.; Ladlow, M.; Ley, S.V. Fully automated Polymer-Assisted synthesis of 1,5-Biaryl pyrazoles. J. Comb. Chem., 2004, 6, 332-339.
-
(2004)
J. Comb. Chem
, vol.6
, pp. 332-339
-
-
Vickerstaffe, E.1
Warrington, B.H.2
Ladlow, M.3
Ley, S.V.4
-
168
-
-
0037319206
-
Microwave-assisted solution-phase synthesis of 1,4,5-Trisubstituted pyrazoles
-
Giacomelli, G.; Porcheddu, A.; Salaris, M.; Taddei, M. Microwave-assisted solution-phase synthesis of 1,4,5-Trisubstituted pyrazoles. Eur. J. Org. Chem., 2003, (3), 537-541.
-
(2003)
Eur. J. Org. Chem
, vol.3
, pp. 537-541
-
-
Giacomelli, G.1
Porcheddu, A.2
Salaris, M.3
Taddei, M.4
-
169
-
-
1942521608
-
Regioselective rapid analogue syntheses of 1-methyl-3,5-diarylpyrazoles via palladium-catalysed coupling to 3(5)- pyrazolyl nonaflates
-
Bourrain, S.; Ridgill, M.; Collins, I. Regioselective rapid analogue syntheses of 1-methyl-3,5-diarylpyrazoles via palladium-catalysed coupling to 3(5)- pyrazolyl nonaflates. Synlett, 2004, (5), 795-798.
-
(2004)
Synlett
, vol.5
, pp. 795-798
-
-
Bourrain, S.1
Ridgill, M.2
Collins, I.3
-
170
-
-
33746105769
-
1,3-Diketones from acid chlorides and Ketones: A rapid and general one-pot synthesis of pyrazoles
-
Heller, S.T.; Natarajan, S.R. 1,3-Diketones from acid chlorides and Ketones: A rapid and general one-pot synthesis of pyrazoles. Org. Lett., 2006, 8(13), 2675-2678.
-
(2006)
Org. Lett
, vol.8
, Issue.13
, pp. 2675-2678
-
-
Heller, S.T.1
Natarajan, S.R.2
-
171
-
-
48349083015
-
Synthesis of derivatives of pyrazole with chiral substituents at the nitrogen atom
-
Kurkin, A.V.; Utkina, A.A.; Yurovskaya, M.A. Synthesis of derivatives of pyrazole with chiral substituents at the nitrogen atom. Chem. Heterocycl. Comp., 2008, 44(1), 106-108.
-
(2008)
Chem. Heterocycl. Comp
, vol.44
, Issue.1
, pp. 106-108
-
-
Kurkin, A.V.1
Utkina, A.A.2
Yurovskaya, M.A.3
-
172
-
-
0034618340
-
Versatile and efficient solid-phase syntheses of pyrazoles and isoxazoles
-
Shen, D.-M; Shu, M.; Chapman, K.T. Versatile and efficient solid-phase syntheses of pyrazoles and isoxazoles. Org. Lett., 2000, 2(18), 2789-2792.
-
(2000)
Org. Lett
, vol.2
, Issue.18
, pp. 2789-2792
-
-
Shen, D.-M.1
Shu, M.2
Chapman, K.T.3
-
173
-
-
57649126101
-
One-pot synthesis of trifluoromethyl-containing pyrazoles via sequential yb(pfo)3-catalyzed three-component reaction and ibx-mediated oxidation
-
Shen, L.; Zhang, J.; Cao, S.; Yu, J.; Liu, N.; Wu, J.; Qian, X. one-pot synthesis of trifluoromethyl-containing pyrazoles via sequential yb(pfo)3-catalyzed three-component reaction and ibx-mediated oxidation. Synlett, 2008, (19), 3058-3062.
-
(2008)
Synlett
, vol.19
, pp. 3058-3062
-
-
Shen, L.1
Zhang, J.2
Cao, S.3
Yu, J.4
Liu, N.5
Wu, J.6
Qian, X.7
-
174
-
-
45749146306
-
Ytterbium(III) Perfluorooctanoate catalyzed one-pot, three-component synthesis of fully substituted pyrazoles under solvent-free conditions
-
Shen, L.; Cao, S.; Liu, N.; Wu, J.; Zhu, L.; Qian, X. Ytterbium(III) Perfluorooctanoate catalyzed one-pot, three-component synthesis of fully substituted pyrazoles under solvent-free conditions. Synlett, 2008, (9), 1341-1344.
-
(2008)
Synlett
, vol.9
, pp. 1341-1344
-
-
Shen, L.1
Cao, S.2
Liu, N.3
Wu, J.4
Zhu, L.5
Qian, X.6
-
175
-
-
28844481893
-
Layered zirconium sulfophenyl phosphonate as heterogeneous catalyst in the synthesis of pyrazoles and 4,5,6,7-Tetrahydro-1(2)Hindazoles
-
Curini, M.; Rosati, O.; Campagna, V.; Montanari, F.; Cravotto, G.; Boccalini, M. Layered zirconium sulfophenyl phosphonate as heterogeneous catalyst in the synthesis of pyrazoles and 4,5,6,7-Tetrahydro-1(2)Hindazoles. Synlett, 2005, (19), 2927-2930.
-
(2005)
Synlett
, vol.19
, pp. 2927-2930
-
-
Curini, M.1
Rosati, O.2
Campagna, V.3
Montanari, F.4
Cravotto, G.5
Boccalini, M.6
-
176
-
-
77955361025
-
The preparation of substituted pyrazoles from-Dibromo-enones by a Tandem Condensation/Suzuki-Miyaura cross-coupling Process
-
Beltrán-Rodil, S.; Edwards, M.G.; Pugh, D.S.; Reid, M.; Taylor, R.J.K. The preparation of substituted pyrazoles from-Dibromo-enones by a Tandem Condensation/Suzuki-Miyaura cross-coupling Process. Synlett, 2010, (4), 602-606.
-
(2010)
Synlett
, vol.4
, pp. 602-606
-
-
Beltrán-Rodil, S.1
Edwards, M.G.2
Pugh, D.S.3
Reid, M.4
Taylor, R.J.K.5
-
177
-
-
33745612700
-
A general method for the preparation of 3-acyl-4- cyano-5-amino-pyrazoles
-
Ge, M.; Cline, E.; Yang, L. A general method for the preparation of 3-acyl-4- cyano-5-amino-pyrazoles. Tetrahedron Lett., 2006, 47(32), 5797-5799.
-
(2006)
Tetrahedron Lett
, vol.47
, Issue.32
, pp. 5797-5799
-
-
Ge, M.1
Cline, E.2
Yang, L.3
-
178
-
-
0035148326
-
Microwave Assisted Synthesis of 1-Aryl-3-dimethylaminoprop-2-enones: A Simple and Rapid Access to 3(5)-Arylpyrazoles
-
Pleier, A.-K.; Glas, H.; Grosche, M.; Sirsch, P.; Thiel, W.R. Microwave Assisted Synthesis of 1-Aryl-3-dimethylaminoprop-2-enones: A Simple and Rapid Access to 3(5)-Arylpyrazoles. Synthesis, 2001, (1), 55-62.
-
(2001)
Synthesis
, vol.1
, pp. 55-62
-
-
Pleier, A.-K.1
Glas, H.2
Grosche, M.3
Sirsch, P.4
Thiel, W.R.5
-
179
-
-
3142775570
-
Montmorillonite KSF clay-promoted synthesis of enantiomerically pure 5- substituted pyrazoles from 2,3-dihydro-4H-pyran-4-ones
-
Yadav, J.S.; Subba Reddy, B.V.; Srinivas, M.; Prabhakar, A.; Jagadeesh, B. Montmorillonite KSF clay-promoted synthesis of enantiomerically pure 5- substituted pyrazoles from 2,3-dihydro-4H-pyran-4-ones. Tetrahedron Lett., 2004, 45(31), 6033-6036.
-
(2004)
Tetrahedron Lett
, vol.45
, Issue.31
, pp. 6033-6036
-
-
Yadav, J.S.1
Subba, R.B.V.2
Srinivas, M.3
Prabhakar, A.4
Jagadeesh, B.5
-
180
-
-
5644285399
-
Rapid and efficient synthesis of optically active pyrazoles under solvent-free conditions
-
Yadav, J.S.; Reddy, B.V.S.; Satheesh, G.; Naga Lakshmi, P.; Kiran Kumarb, S.; Kunwar, A.C. Rapid and efficient synthesis of optically active pyrazoles under solvent-free conditions. Tetrahedron Lett., 2004, 45(46), 8587-8590.
-
(2004)
Tetrahedron Lett
, vol.45
, Issue.46
, pp. 8587-8590
-
-
Yadav, J.S.1
Reddy, B.V.S.2
Satheesh, G.3
Naga, L.P.4
Kiran, K.S.5
Kunwar, A.C.6
-
181
-
-
0035812782
-
Regioselective synthesis of polysubstituted pyrazoles and isoxazoles
-
Katritzky, A.R.; Wang, M.; Zhang, S.; Voronkov, M.V.; Steel, P.J. Regioselective synthesis of polysubstituted pyrazoles and isoxazoles. J. Org. Chem., 2001, 66, 6787-6791.
-
(2001)
J. Org. Chem
, vol.66
, pp. 6787-6791
-
-
Katritzky, A.R.1
Wang, M.2
Zhang, S.3
Voronkov, M.V.4
Steel, P.J.5
-
182
-
-
28044473878
-
Regioselective Synthesis of 1-Aryl-3,4-substituted/annulated-5-(methylthio)pyrazoles and 1- Aryl-3-(methylthio)-4,5-substituted/annulated Pyrazoles
-
Peruncheralathan, S.; Khan, T.A.; Ila, H.; Junjappa, H. Regioselective Synthesis of 1-Aryl-3,4-substituted/annulated-5-(methylthio)pyrazoles and 1- Aryl-3-(methylthio)-4,5-substituted/annulated Pyrazoles. J. Org. Chem., 2005, 70, 10030-10035.
-
(2005)
J. Org. Chem
, vol.70
, pp. 10030-10035
-
-
Peruncheralathan, S.1
Khan, T.A.2
Ila, H.3
Junjappa, H.4
-
183
-
-
27744591612
-
Highly regioselective synthesis of 1-Aryl-3 (or 5)-alkyl/aryl-5 (or 3)-(N-cycloamino)pyrazoles
-
Peruncheralathan, S.; Yadav, A.K.; Ila, H.; Junjappa, H. Highly regioselective synthesis of 1-Aryl-3 (or 5)-alkyl/aryl-5 (or 3)-(N-cycloamino)pyrazoles. J. Org. Chem., 2005, 70, 9644-9647.
-
(2005)
J. Org. Chem
, vol.70
, pp. 9644-9647
-
-
Peruncheralathan, S.1
Yadav, A.K.2
Ila, H.3
Junjappa, H.4
-
184
-
-
2542609193
-
Hydroxyalkynyl Ketones as useful scaffolds for the preparation of combinatorial libraries of furans, isoxazoles and pyrazoles
-
Sauers, R.R.; van Arnum, S.D. -Hydroxyalkynyl Ketones as useful scaffolds for the preparation of combinatorial libraries of furans, isoxazoles and pyrazoles. J. Comb. Chem., 2004, 6, 350-355.
-
(2004)
J. Comb. Chem
, vol.6
, pp. 350-355
-
-
Sauers, R.R.1
van Arnum, S.D.2
-
185
-
-
28244440942
-
Synthesis of substituted 1-C-Phenyl-D-tetritols and 1-C-(1H-Pyrazol-4-yl)- D-tetritols by ring transformation of 2-Formylglycals
-
Montero, A.; Michalik, M.; Feist, H.; Reinke, H.; Rudloff, I.; Peseke, K. Synthesis of substituted 1-C-Phenyl-D-tetritols and 1-C-(1H-Pyrazol-4-yl)- D-tetritols by ring transformation of 2-Formylglycals. J. Carbohydr. Chem., 2004, 23(5), 313-324.
-
(2004)
J. Carbohydr. Chem
, vol.23
, Issue.5
, pp. 313-324
-
-
Montero, A.1
Michalik, M.2
Feist, H.3
Reinke, H.4
Rudloff, I.5
Peseke, K.6
-
186
-
-
46749133810
-
An improved synthesis of pyrimidine- and pyrazole-based acyclo-C-nucleosides as carbohybrids
-
Sagar, R.; Kim, M.-J.; Park, S.B. An improved synthesis of pyrimidine- and pyrazole-based acyclo-C-nucleosides as carbohybrids. Tetrahedron Lett., 2008, 49, 5080-5083.
-
(2008)
Tetrahedron Lett
, vol.49
, pp. 5080-5083
-
-
Sagar, R.1
Kim, M.-J.2
Park, S.B.3
-
187
-
-
0035136831
-
Efficient synthesis of 4-Fluoro-5-(perfluoroalkyl)pyrazoles from organofluorosilicon building blocks
-
Bouillon, J.P.; Didier, B.; Dondy, B.; Doussot, P.; Plantier-Royon, R.; Portella, C. Efficient synthesis of 4-Fluoro-5-(perfluoroalkyl)pyrazoles from organofluorosilicon building blocks. Eur. J. Org. Chem., 2001, (1), 187-192.
-
(2001)
Eur. J. Org. Chem
, vol.1
, pp. 187-192
-
-
Bouillon, J.P.1
Didier, B.2
Dondy, B.3
Doussot, P.4
Plantier-Royon, R.5
Portella, C.6
-
188
-
-
34347344028
-
Synthesis of Pyrazoles by a one-pot tandem cyclization-dehydrogenation approach on Pd/C/K- 10 catalyst
-
Landge, S.M.; Schmidt, A.; Outerbridge, V.; Török, B. Synthesis of Pyrazoles by a one-pot tandem cyclization-dehydrogenation approach on Pd/C/K- 10 catalyst. Synlett, 2007, (10), 1600-1604.
-
(2007)
Synlett
, vol.10
, pp. 1600-1604
-
-
Landge, S.M.1
Schmidt, A.2
Outerbridge, V.3
Török, B.4
-
189
-
-
33646797446
-
Palladium-catalyzed C-N bond formation: Synthesis of 1-aryl-1H-pyrazoles from β-bromovinyl aldehydes and arylhydrazines
-
Cho, C.S.; Patel, D.P. Palladium-catalyzed C-N bond formation: synthesis of 1-aryl-1H-pyrazoles from β-bromovinyl aldehydes and arylhydrazines. Tetrahedron, 2006, 62(26), 6388-6391.
-
(2006)
Tetrahedron
, vol.62
, Issue.26
, pp. 6388-6391
-
-
Cho, C.S.1
Patel, D.P.2
-
190
-
-
14644442895
-
Synthesis of 5- Hydroxy- and 5-Amino-1-tosyl-5-phenyl-3-(2-arylvinyl)-4,5--dihydropyrazoles
-
Kuźmenok, N.M.; Kovaĺchuk, T.A.; Zvonok, A.M. Synthesis of 5- Hydroxy- and 5-Amino-1-tosyl-5-phenyl-3-(2-arylvinyl)-4,5--dihydropyrazoles. Synlett, 2005, (3), 485-486.
-
(2005)
Synlett
, vol.3
, pp. 485-486
-
-
Kuźmenok, N.M.1
Kovaĺchuk, T.A.2
Zvonok, A.3
-
191
-
-
70350510129
-
The chemistry of-ditosyloxyketones: New and convenient route for the synthesis of 1,4,5-trisubstituted pyrazoles from-chalcone ditosylates
-
Prakash, O.; Sharma, D.; Kamal, R.; Kumar, R.; Nair, R.R. The chemistry of-ditosyloxyketones: new and convenient route for the synthesis of 1,4,5-trisubstituted pyrazoles from-chalcone ditosylates. Tetrahedron, 2009, 65(49), 10175-10181.
-
(2009)
Tetrahedron
, vol.65
, Issue.49
, pp. 10175-10181
-
-
Prakash, O.1
Sharma, D.2
Kamal, R.3
Kumar, R.4
Nair, R.R.5
-
192
-
-
28844457259
-
Facile preparation of allyl amines and pyrazoles by hydrazinolysis of 2-ketoaziridines
-
Chen, G.; Sasaki, M.; Yudin, A.K. Facile preparation of allyl amines and pyrazoles by hydrazinolysis of 2-ketoaziridines. Tetrahedron Lett., 2006, 47(3), 255-259.
-
(2006)
Tetrahedron Lett
, vol.47
, Issue.3
, pp. 255-259
-
-
Chen, G.1
Sasaki, M.2
Yudin, A.K.3
-
193
-
-
0035251041
-
Scope and limitations in the regioselective synthesis of 1,3,5- trisubstituted pyrazoles from -Amino Enones and hydrazine derivatives. 13C-chemical shift prediction rules for 1,3,5-Trisubstituted pyrazoles
-
Alberola, A.; Calvo Bleye, L.; González-Ortega, A.; Sábada, M.L.; Sañudo, M.C. Scope and limitations in the regioselective synthesis of 1,3,5- trisubstituted pyrazoles from -Amino Enones and hydrazine derivatives. 13C-chemical shift prediction rules for 1,3,5-Trisubstituted pyrazoles. Heterocycles, 2001, 55(2), 331-351.
-
(2001)
Heterocycles
, vol.55
, Issue.2
, pp. 331-351
-
-
Alberola, A.1
Calvo, B.L.2
González-Ortega, A.3
Sábada, M.L.4
Sañudo, M.C.5
-
194
-
-
28844470382
-
Silylated-enaminones as precursors in the regioselective synthesis of silyl pyrazoles
-
Calle, M.; Calvo, L.A.; González-Ortega, A.; González-Nogal, A.M. Silylated-enaminones as precursors in the regioselective synthesis of silyl pyrazoles. Tetrahedron, 2006, 62, 611-618.
-
(2006)
Tetrahedron
, vol.62
, pp. 611-618
-
-
Calle, M.1
Calvo, L.A.2
González-Ortega, A.3
González-Nogal, A.M.4
-
195
-
-
27644584128
-
A convenient approach to the synthesis of -heterocyclic amino acids from carboxy lactams through ring-chain transformation; part 1: Synthesis of (2s)-/(2r)-2- amino-4-(1-aryl-/1,5-diaryl-1h-pyrazol-3-yl)butyric acid
-
Singh, R.K.; Sinha, N.; Jain, S.; Salman, M.; Naqvi, F.; Anand, N. a convenient approach to the synthesis of -heterocyclic amino acids from carboxy lactams through ring-chain transformation; part 1: synthesis of (2s)-/(2r)-2- amino-4-(1-aryl-/1,5-diaryl-1h-pyrazol-3-yl)butyric acid. Synthesis, 2005, (16), 2765-2771.
-
(2005)
Synthesis
, vol.16
, pp. 2765-2771
-
-
Singh, R.K.1
Sinha, N.2
Jain, S.3
Salman, M.4
Naqvi, F.5
Anand, N.6
-
196
-
-
27644552250
-
Expeditious Solidphase synthesis of pyrazoledicarboxylic acid derivatives by functionalization of resin-bound cyanoformate
-
Morelli, C.F.; Saladino, A.; Speranza, G.; Manitto, P. Expeditious Solidphase synthesis of pyrazoledicarboxylic acid derivatives by functionalization of resin-bound cyanoformate. Eur. J. Org. Chem., 2005, (21), 4621-4627.
-
(2005)
Eur. J. Org. Chem
, vol.21
, pp. 4621-4627
-
-
Morelli, C.F.1
Saladino, A.2
Speranza, G.3
Manitto, P.4
-
197
-
-
0141742132
-
Toward safer methodologies for the synthesis of polyheterocyclic systems: Intramolecular arylation of arenes under mizoroki-heck reaction conditions
-
Hernández, S.; SanMartin, R.; Tellitu, I.; Domínguez, E. Toward safer methodologies for the synthesis of polyheterocyclic systems: intramolecular arylation of arenes under mizoroki heck reaction conditions. Org. Lett., 2003, 5(7), 1095-1098.
-
(2003)
Org. Lett
, vol.5
, Issue.7
, pp. 1095-1098
-
-
Hernández, S.1
Sanmartin, R.2
Tellitu, I.3
Domínguez, E.4
-
198
-
-
33746868887
-
Synthesis of N-Methoxy-N-methyl-?-enaminoketoesters: New synthetic precursors for the regioselective synthesis of heterocyclic compounds
-
Persson, T.; Nielsen, J. Synthesis of N-Methoxy-N-methyl-?-enaminoketoesters: new synthetic precursors for the regioselective synthesis of heterocyclic compounds. Org. Lett., 2006, 8(15), 3219-3222.
-
(2006)
Org. Lett
, vol.8
, Issue.15
, pp. 3219-3222
-
-
Persson, T.1
Nielsen, J.2
-
199
-
-
51549101998
-
Room temperature ICl-Induced Dehydration/ Iodination of 1-Acyl-5-hydroxy-4,5-dihydro-1H-pyrazoles. A selective route to substituted 1-Acyl-4-iodo-1H-pyrazoles
-
Waldo, J.P.; Mehta, S.; Larock, R.C. Room temperature ICl-Induced Dehydration/ Iodination of 1-Acyl-5-hydroxy-4,5-dihydro-1H-pyrazoles. A selective route to substituted 1-Acyl-4-iodo-1H-pyrazoles. J. Org. Chem., 2008, 73, 6666-6670.
-
(2008)
J. Org. Chem
, vol.73
, pp. 6666-6670
-
-
Waldo, J.P.1
Mehta, S.2
Larock, R.C.3
-
200
-
-
0142027266
-
Synthesis of multi-substituted pyrazoles utilizing the N-Alkylated 3- Hydroxy-3-propargyl- or allenylisoindolines
-
Choi, Y.H.; Kim, K.S.; Lee, S.; Jeong, T.-S.; Lee, H.-Y.; Kim, Y.H.; Lee, W.S. Synthesis of multi-substituted pyrazoles utilizing the N-Alkylated 3- Hydroxy-3-propargyl- or allenylisoindolines. Heterocycles, 2003, 60(11), 2499-2510.
-
(2003)
Heterocycles
, vol.60
, Issue.11
, pp. 2499-2510
-
-
Choi, Y.H.1
Kim, K.S.2
Lee, S.3
Jeong, T.-S.4
Lee, H.-Y.5
Kim, Y.H.6
Lee, W.S.7
-
201
-
-
0037463787
-
Practical routes to diacetylenic ketones and their application for the preparation of alkynyl substituted pyridines, pyrimidines and pyrazoles
-
Adamo, M.F.A.; Adlington, R.M.; Baldwin, J.E.; Pritchard, G.J.; Rathmella, R.E. Practical routes to diacetylenic ketones and their application for the preparation of alkynyl substituted pyridines, pyrimidines and pyrazoles. Tetrahedron, 2003, 59(13), 2197-2205.
-
(2003)
Tetrahedron
, vol.59
, Issue.13
, pp. 2197-2205
-
-
Adamo, M.F.A.1
Adlington, R.M.2
Baldwin, J.E.3
Pritchard, G.J.4
Rathmella, R.E.5
-
202
-
-
26444497881
-
One-pot construction of pyrazoles and isoxazoles with Palladium-Catalyzed four-component coupling
-
Ahmed, M.S.M.; Kobayashi, K.; Mori, A. One-pot construction of pyrazoles and isoxazoles with Palladium-Catalyzed four-component coupling. Org. Lett., 2005, 7(20), 4487-4489.
-
(2005)
Org. Lett
, vol.7
, Issue.20
, pp. 4487-4489
-
-
Ahmed, M.S.M.1
Kobayashi, K.2
Mori, A.3
-
203
-
-
38849143259
-
One-pot four-component reaction for the generation of pyrazoles and pyrimidines
-
Stonehouse, J.P.; Chekmarev, D.S.; Ivanova, N.V.; Lang, S.; Pairaudeau, G.; Smith, N.; Stocks, M.J.; Sviridov, S.I.; Utkina, L.M. one-pot four-component reaction for the generation of pyrazoles and pyrimidines. Synlett, 2008, (1), 100-104.
-
(2008)
Synlett
, vol.1
, pp. 100-104
-
-
Stonehouse, J.P.1
Chekmarev, D.S.2
Ivanova, N.V.3
Lang, S.4
Pairaudeau, G.5
Smith, N.6
Stocks, M.J.7
Sviridov, S.I.8
Utkina, L.M.9
-
204
-
-
52249112156
-
Regioselective three-component synthesis of highly fluorescent 1,3,5-Trisubstituted pyrazoles
-
Willy, B.; Müller, T.J.J. Regioselective three-component synthesis of highly fluorescent 1,3,5-Trisubstituted pyrazoles. Eur. J. Org. Chem., 2008, (24), 4157-4168.
-
(2008)
Eur. J. Org. Chem
, vol.24
, pp. 4157-4168
-
-
Willy, B.1
Müller, T.J.J.2
-
205
-
-
43349104749
-
Onepot three-component synthesis of pyrazoles through a tandem couplingcyclocondensation sequence
-
Liu, H.-L.; Jiang, H.-F.; Zhang, M.; Yao, W.-J.; Zhu, Q.-H.; Tang, Z. Onepot three-component synthesis of pyrazoles through a tandem couplingcyclocondensation sequence. Tetrahedron Lett., 2008, 49, 3805-3809.
-
(2008)
Tetrahedron Lett
, vol.49
, pp. 3805-3809
-
-
Liu, H.-L.1
Jiang, H.-F.2
Zhang, M.3
Yao, W.-J.4
Zhu, Q.-H.5
Tang, Z.6
-
206
-
-
33947729953
-
Regioselective microwave-assisted synthesis of substituted pyrazoles from ethynyl ketones
-
Bagley, M.C.; Lubinu, M.C.; Mason, C. Regioselective microwave-assisted synthesis of substituted pyrazoles from ethynyl ketones. Synlett, 2007, (5), 704-708.
-
(2007)
Synlett
, vol.5
, pp. 704-708
-
-
Bagley, M.C.1
Lubinu, M.C.2
Mason, C.3
-
207
-
-
58149341296
-
A novel one-pot, threecomponent synthesis of dialkyl 5-(alkylamino)-1-aryl-1h-pyrazole-3,4-dicarboxylates
-
Adib, M.; Mohammadi, B.; Reza Bijanzadeh, H. A novel one-pot, threecomponent synthesis of dialkyl 5-(alkylamino)-1-aryl-1h-pyrazole-3,4-dicarboxylates. Synlett, 2008, (20), 3180-3182.
-
(2008)
Synlett
, vol.20
, pp. 3180-3182
-
-
Adib, M.1
Mohammadi, B.2
Reza, B.H.3
-
208
-
-
35848958616
-
Palladium-catalyzed alkynylcarbonylation of Aryl Iodides with the use of Mo(CO)6 in the presence of tBu3P ligand
-
Iizuka, M.; Kondo, Y. Palladium-catalyzed alkynylcarbonylation of Aryl Iodides with the use of Mo(CO)6 in the presence of tBu3P ligand. Eur. J. Org. Chem., 2007, (31), 5180-5182.
-
(2007)
Eur. J. Org. Chem
, vol.31
, pp. 5180-5182
-
-
Iizuka, M.1
Kondo, Y.2
-
209
-
-
48849090860
-
Zinc-Catalyzed synthesis of pyrazolines and pyrazoles via hydrohydrazination
-
Alex, K.; Tillack, A.; Schwarz, N.; Beller, M. Zinc-Catalyzed synthesis of pyrazolines and pyrazoles via hydrohydrazination. Org. Lett., 2008, 10(12), 2377-2379.
-
(2008)
Org. Lett
, vol.10
, Issue.12
, pp. 2377-2379
-
-
Alex, K.1
Tillack, A.2
Schwarz, N.3
Beller, M.4
-
210
-
-
52749097629
-
A convenient synthesis of novel 7- phosphonylbenzyl-2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]- pyrimidine derivatives
-
Xiao, L.-X.; Li, K.; Meng, L.; Shi, D.-Q. A convenient synthesis of novel 7- phosphonylbenzyl-2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]- pyrimidine derivatives. Heteroatom Chem., 2008, 19(6), 634-638.
-
(2008)
Heteroatom Chem
, vol.19
, Issue.6
, pp. 634-638
-
-
Xiao, L.-X.1
Li, K.2
Meng, L.3
Shi, D.-Q.4
-
211
-
-
13544271031
-
Solid-phase synthesis of 5-amino-1-(Substituted Thiocarbamoyl)pyrazole and 1,2,4- triazole derivatives via dithiocarbazate linker
-
Hwang, J.Y.; Choi, H.-S.; Lee, D.-H.; Yoo, S.-E.; Gong, Y.D. Solid-phase synthesis of 5-amino-1-(Substituted Thiocarbamoyl)pyrazole and 1,2,4- triazole derivatives via dithiocarbazate linker. J. Comb. Chem., 2005, 7, 136-141.
-
(2005)
J. Comb. Chem
, vol.7
, pp. 136-141
-
-
Hwang, J.Y.1
Choi, H.-S.2
Lee, D.-H.3
Yoo, S.-E.4
Gong, Y.D.5
-
212
-
-
34250342161
-
Two new syntheses of a 4-aminopyrazole: Condensation of an N-substituted vinamidinium salt with a functionalized hydrazine
-
Hill, G.B.; Mortlock, A.A. Two new syntheses of a 4-aminopyrazole: condensation of an N-substituted vinamidinium salt with a functionalized hydrazine. Synthesis, 2007, (11), 1697-1701.
-
(2007)
Synthesis
, vol.11
, pp. 1697-1701
-
-
Hill, G.B.1
Mortlock, A.A.2
-
213
-
-
18444398039
-
The application of vinylogous iminium salt derivatives to the regiocontrolled preparation of heterocyclic appended pyrazoles
-
Gupton, J.T.; Clough, S.C.; Miller, R.B.; Norwood, B.K.; Hickenboth, C.R.; Chertudi, I.B.; Cutro, S.R.; Petrich, S.A.; Hicks, F.A.; Wilkinson, D.R.; Sikorski, J.A. The application of vinylogous iminium salt derivatives to the regiocontrolled preparation of heterocyclic appended pyrazoles. Tetrahedron, 2002, 58(27), 5467-5474.
-
(2002)
Tetrahedron
, vol.58
, Issue.27
, pp. 5467-5474
-
-
Gupton, J.T.1
Clough, S.C.2
Miller, R.B.3
Norwood, B.K.4
Hickenboth, C.R.5
Chertudi, I.B.6
Cutro, S.R.7
Petrich, S.A.8
Hicks, F.A.9
Wilkinson, D.R.10
Sikorski, J.A.11
-
214
-
-
31144467616
-
Aqueous N-Heterocyclization of primary amines and hydrazines with dihalides: Microwave-assisted syntheses of Nazacycloalkanes, isoindole, pyrazole, pyrazolidine, and phthalazine derivatives
-
Ju, Y.; Varma, R.S. Aqueous N-Heterocyclization of primary amines and hydrazines with dihalides: microwave-assisted syntheses of Nazacycloalkanes, isoindole, pyrazole, pyrazolidine, and phthalazine derivatives. J. Org. Chem., 2006, 71, 135-141.
-
(2006)
J. Org. Chem
, vol.71
, pp. 135-141
-
-
Ju, Y.1
Varma, R.S.2
-
215
-
-
0033020246
-
Tosylhydrazono phosphonates in organic synthesis. An Unambiguous entry to polysubstituted pyrazoles
-
Almirante, N.; Benicchio, A.; Cerri, A.; Fedrizzi, G.; Marazzi, G.; Santagostino, M.-Tosylhydrazono phosphonates in organic synthesis. An Unambiguous entry to polysubstituted pyrazoles. Synlett, 1999, (3), 299-302.
-
(1999)
Synlett
, vol.3
, pp. 299-302
-
-
Almirante, N.1
Benicchio, A.2
Cerri, A.3
Fedrizzi, G.4
Marazzi, G.5
Santagostino, M.6
-
216
-
-
0034029615
-
A New Straightforward Formation of aminopyrazoles from isocyanides
-
Atlan, V.; Buron, C.; El Kaïm, L. A New Straightforward Formation of aminopyrazoles from isocyanides. Synlett, 2000, (4), 489-490.
-
(2000)
Synlett
, vol.4
, pp. 489-490
-
-
Atlan, V.1
Buron, C.2
El Kaïm, L.3
-
217
-
-
33745386374
-
A concise synthesis of Trifluoromethyl-substituted 4-aryloxy pyrazoles
-
Jones, L.H.; Mowbray, C. A concise synthesis of Trifluoromethyl-substituted 4-aryloxy pyrazoles. Synlett, 2006, (9), 1404-1406.
-
(2006)
Synlett
, vol.9
, pp. 1404-1406
-
-
Jones, L.H.1
Mowbray, C.2
-
218
-
-
0034008049
-
Trichloroacylhydrazones: New straightforward preparation of pyrazoles from keto esters
-
El Kaim, L.; Lacroix, S. Trichloroacylhydrazones: New straightforward preparation of pyrazoles from keto esters. Synlett, 2000, (3), 353-354.
-
(2000)
Synlett
, vol.3
, pp. 353-354
-
-
El Kaim, L.1
Lacroix, S.2
-
219
-
-
33747214078
-
Reaction of N-Monosubstituted hydrazones with Nitroolefins: A novel regioselective pyrazole synthesis
-
Deng, X.; Mani, N.S. Reaction of N-Monosubstituted hydrazones with Nitroolefins: A novel regioselective pyrazole synthesis. Org. Lett., 2006, 8(16), 3505-3508.
-
(2006)
Org. Lett
, vol.8
, Issue.16
, pp. 3505-3508
-
-
Deng, X.1
Mani, N.S.2
-
220
-
-
41849086318
-
Regioselective Synthesis of 1,3,5-Tri- and 1,3,4,5- Tetrasubstituted Pyrazoles from N-arylhydrazones and nitroolefins
-
Deng, X.; Mani, N.S. Regioselective Synthesis of 1,3,5-Tri- and 1,3,4,5- Tetrasubstituted Pyrazoles from N-arylhydrazones and nitroolefins. J. Org. Chem., 2008, 73, 2412-2415.
-
(2008)
J. Org. Chem
, vol.73
, pp. 2412-2415
-
-
Deng, X.1
Mani, N.S.2
-
221
-
-
8744252642
-
A mild procedure for the preparation of 3-Aryl-4-formylpyrazoles
-
De Luca, L.; Giacomelli, G.; Masala, S.; Porcheddu, A. A mild procedure for the preparation of 3-Aryl-4-formylpyrazoles. Synlett, 2004, (13), 2299-2302.
-
(2004)
Synlett
, vol.13
, pp. 2299-2302
-
-
de Luca, L.1
Giacomelli, G.2
Masala, S.3
Porcheddu, A.4
-
222
-
-
38349141840
-
Synthesis of pyrazole- 3-carboxylates and pyrazole-1,5-dicarboxylates by one-pot cyclization of hydrazone dianions with diethyl oxalate
-
Dang, T.T.; Dang, T.T.; Fischer, C.; Görls, H.; Langer, P. Synthesis of pyrazole- 3-carboxylates and pyrazole-1,5-dicarboxylates by one-pot cyclization of hydrazone dianions with diethyl oxalate. Tetrahedron, 2008, 64(9), 2207-2215.
-
(2008)
Tetrahedron
, vol.64
, Issue.9
, pp. 2207-2215
-
-
Dang, T.T.1
Dang, T.T.2
Fischer, C.3
Görls, H.4
Langer, P.5
-
223
-
-
34247097022
-
One-pot synthesis of pyrazole-5- carboxylates by cyclization of hydrazone 1,4-dianions with diethyl oxalate
-
Dang, T. T.; Dang, T.T.; Langer, P. One-pot synthesis of pyrazole-5- carboxylates by cyclization of hydrazone 1,4-dianions with diethyl oxalate. Tetrahedron Lett., 2007, 48(20), 3591-3593.
-
(2007)
Tetrahedron Lett
, vol.48
, Issue.20
, pp. 3591-3593
-
-
Dang, T.T.1
Dang, T.T.2
Langer, P.3
-
224
-
-
0036843335
-
Coupling of Heteroaryldiazonium tetrafluoroborates with 1,3-dicarbonyl compounds-regioselective synthesis of Alkyl 1-Heteroaryl-4-hydroxy-1H-pyrazole-3-carboxylates
-
Renik, S.; Svete, J.; Stanovnik, B. Coupling of Heteroaryldiazonium tetrafluoroborates with 1,3-dicarbonyl compounds-regioselective synthesis of Alkyl 1-Heteroaryl-4-hydroxy-1H-pyrazole-3-carboxylates. Heterocycles, 2002, 57(11), 2091-2106.
-
(2002)
Heterocycles
, vol.57
, Issue.11
, pp. 2091-2106
-
-
Renik, S.1
Svete, J.2
Stanovnik, B.3
-
225
-
-
0037711833
-
Synthesis of aminopyrazoles from-Oxoketene O,NAcetals using montmorillonite k-10/ultrasound
-
Braibante, M.E.F.; Braibante, H.T.S.; da Roza, J.K.; Henriques, D.M.; de Carvalho Tavares, L. Synthesis of aminopyrazoles from-Oxoketene O,NAcetals using montmorillonite k-10/ultrasound. Synthesis, 2003, (8), 1160-1162.
-
(2003)
Synthesis
, vol.8
, pp. 1160-1162
-
-
Braibante, M.E.F.1
Braibante, H.T.S.2
da Roza, J.K.3
Henriques, D.M.4
de Carvalho, T.L.5
-
226
-
-
34548335098
-
Efficient regiocontrolled synthesis and antimicrobial activity of pyrazoles
-
Braibante, M.E.F.; Braibante, H.T.S.; de Carvalho Tavares, L.; Rohte, S.F.; Costa, C.C.; Morel, A.F.; Stüker, C.Z.; Burrow, R.A. Efficient regiocontrolled synthesis and antimicrobial activity of pyrazoles. Synthesis, 2007, (16), 2485-2490.
-
(2007)
Synthesis
, vol.16
, pp. 2485-2490
-
-
Braibante, M.E.F.1
Braibante, H.T.S.2
de Carvalho, T.L.3
Rohte, S.F.4
Costa, C.C.5
Morel, A.F.6
Stüker, C.Z.7
Burrow, R.A.8
-
227
-
-
47049104389
-
Flexible protocol for the Chemo- and regioselective building of pyrroles and pyrazoles by Reactions of Danishefsky's Dienes with 1,2-Diaza-1,3-butadienes
-
Attanasi, O.A.; Favi, G.; Filippone, P.; Giorgi, G.; Mantellini, F.; Moscatelli, G.; Spinelli, D. flexible protocol for the Chemo- and regioselective building of pyrroles and pyrazoles by Reactions of Danishefsky's Dienes with 1,2-Diaza-1,3-butadienes. Org. Lett., 2008, 10(10), 1983-1986.
-
(2008)
Org. Lett
, vol.10
, Issue.10
, pp. 1983-1986
-
-
Attanasi, O.A.1
Favi, G.2
Filippone, P.3
Giorgi, G.4
Mantellini, F.5
Moscatelli, G.6
Spinelli, D.7
-
228
-
-
45549094745
-
Base-Mediated reaction of hydrazones and nitroolefins with a reversed regioselectivity: A novel synthesis of 1,3,4-Trisubstituted Pyrazoles
-
Deng, X.; Mani, N.S. Base-Mediated reaction of hydrazones and nitroolefins with a reversed regioselectivity: A novel synthesis of 1,3,4-Trisubstituted Pyrazoles. Org. Lett., 2008, 10(6), 1307-1310.
-
(2008)
Org. Lett
, vol.10
, Issue.6
, pp. 1307-1310
-
-
Deng, X.1
Mani, N.S.2
-
229
-
-
45149147297
-
Silver(I)-Catalyzed Facile synthesis of pyrazoles From Propargyl N-Sulfonylhydrazones
-
Lee, Y.T.; Chung, Y.K. Silver(I)-Catalyzed Facile synthesis of pyrazoles From Propargyl N-Sulfonylhydrazones. J. Org. Chem., 2008, 73(12), 4698- 4701.
-
(2008)
J. Org. Chem
, vol.73
, Issue.12
, pp. 4698-4701
-
-
Lee, Y.T.1
Chung, Y.K.2
-
230
-
-
45149100137
-
Simple approach to some N-(5-Hydroxy- 1-phenyl-1H-pyrazol-4-yl)benzamides
-
Čuček, K.; Golobi A.; Verek, B. Simple approach to some N-(5-Hydroxy- 1-phenyl-1H-pyrazol-4-yl)benzamides. Heterocycles, 2007, 73(1), 555-566.
-
(2007)
Heterocycles
, vol.73
, Issue.1
, pp. 555-566
-
-
Čuček, K.1
Golobi, A.2
Verek, B.3
-
231
-
-
29744448555
-
Preparation and reactions of 3-phosphinyl-1-aza-1,3-butadienes. Synthesis of phosphorylated pyridine and pyrazole derivatives
-
Palacios, F.; Aparicio, D.; López, Y.; de los Santos, J.M.; Ezpeleta, J.M. Preparation and reactions of 3-phosphinyl-1-aza-1,3-butadienes. Synthesis of phosphorylated pyridine and pyrazole derivatives. Tetrahedron, 2006, 62, 1095-1101.
-
(2006)
Tetrahedron
, vol.62
, pp. 1095-1101
-
-
Palacios, F.1
Aparicio, D.2
López, Y.3
de los Santos, J.M.4
Ezpeleta, J.M.5
-
232
-
-
46149089401
-
A facile and convenient approach to the synthesis of 3,5-diaryl-1H-pyrazoles
-
Nikpour, F.; Beigvand, M. A facile and convenient approach to the synthesis of 3,5-diaryl-1H-pyrazoles. Monatsh. Chem., 2008, 139, 821-824.
-
(2008)
Monatsh. Chem
, vol.139
, pp. 821-824
-
-
Nikpour, F.1
Beigvand, M.2
-
233
-
-
41649099221
-
Expedient synthesis of pyrazoles substituted with amino, hydroxyl and thioamide groups
-
Trofimov, B.A.; Mal'kina, A.G.; Borisova, A.P.; Nosyreva, V.V.; Shemyakina, O.A.; Kazheva, O.N.; Shilov, G.V.; Dyachenko, O.A. Expedient synthesis of pyrazoles substituted with amino, hydroxyl and thioamide groups. Tetrahedron Lett., 2008, 49(19), 3104-3107.
-
(2008)
Tetrahedron Lett
, vol.49
, Issue.19
, pp. 3104-3107
-
-
Trofimov, B.A.1
Mal'kina, A.G.2
Borisova, A.P.3
Nosyreva, V.V.4
Shemyakina, O.A.5
Kazheva, O.N.6
Shilov, G.V.7
Dyachenko, O.A.8
-
234
-
-
40849096351
-
Efficient Syntheses of Some Versatile 3,5-Bifunctional Pyrazole building blocks
-
Sachse, A.; Penkova, L.; Noël, G.; Dechert, S.; Varzatskii, O.A.; Fritsky, I.O.; Meyer, F. Efficient Syntheses of Some Versatile 3,5-Bifunctional Pyrazole building blocks. Synthesis, 2008, (5), 800-806.
-
(2008)
Synthesis
, vol.5
, pp. 800-806
-
-
Sachse, A.1
Penkova, L.2
Noël, G.3
Dechert, S.4
Varzatskii, O.A.5
Fritsky, I.O.6
Meyer, F.7
-
235
-
-
45249111549
-
Facile and straightforward method leading to substituted 4-Amino-1-arylpyrazoles
-
Šimnek, P.; Svobodová, M.; Bertolasi, V.; Macháček, V. Facile and straightforward method leading to substituted 4-Amino-1-arylpyrazoles. Synthesis, 2008, (11), 1761-1766.
-
(2008)
Synthesis
, vol.11
, pp. 1761-1766
-
-
Šimnek, P.1
Svobodová, M.2
Bertolasi, V.3
Macháček, V.4
-
236
-
-
0037074195
-
Synthesis and biological evaluation of new pyrazole- and tetrazole- related C-nucleosides with modified sugar moieties
-
Popsavin, M.; Torovi, L.; Spai, S.; Stankov, S.; Kapor, A.; Tomi, Z.; Popsavin, V. Synthesis and biological evaluation of new pyrazole- and tetrazole- related C-nucleosides with modified sugar moieties. Tetrahedron, 2002, 58, 569-580.
-
(2002)
Tetrahedron
, vol.58
, pp. 569-580
-
-
Popsavin, M.1
Torovi, L.2
Spai, S.3
Stankov, S.4
Kapor, A.5
Tomi, Z.6
Popsavin, V.7
-
237
-
-
57149131220
-
A novel synthesis of 1,3,5- trisubstituted pyrazoles through a spiro-pyrazoline intermediate via a tandem 1,3-dipolar cycloaddition/elimination
-
Dadiboyena, S.; Valente, E.J.; Hamme II, A.T. A novel synthesis of 1,3,5- trisubstituted pyrazoles through a spiro-pyrazoline intermediate via a tandem 1,3-dipolar cycloaddition/elimination. Tetrahedron Lett., 2009, 50, 291-294.
-
(2009)
Tetrahedron Lett
, vol.50
, pp. 291-294
-
-
Dadiboyena, S.1
Valente, E.J.2
Hamme II, A.T.3
-
238
-
-
34848859255
-
Synthesis of pentafluorosulfanylpyrazole and pentafluorosulfanyl-1,2,3- triazole and Their derivatives as Energetic materials by click chemistry
-
Ye, C.; Gard, G.L.; Winter, R.W.; Syvret, R.G.; Twamley, B.; Shreeve, J.M. Synthesis of pentafluorosulfanylpyrazole and pentafluorosulfanyl-1,2,3- triazole and Their derivatives as Energetic materials by click chemistry. Org. Lett., 2007, 9(19), 3841-3844.
-
(2007)
Org. Lett
, vol.9
, Issue.19
, pp. 3841-3844
-
-
Ye, C.1
Gard, G.L.2
Winter, R.W.3
Syvret, R.G.4
Twamley, B.5
Shreeve, J.M.6
-
239
-
-
0037533016
-
Novel one-pot method for the preparation of pyrazoles by 1,3-Dipolar cycloadditions of diazo compounds generated in situ
-
Aggarwal, V.K.; de Vicente, J.; Bonnert, R.V. A Novel one-pot method for the preparation of pyrazoles by 1,3-Dipolar cycloadditions of diazo compounds generated in situ. J. Org. Chem., 2003, 68, 5381-5383.
-
(2003)
J. Org. Chem
, vol.68
, pp. 5381-5383
-
-
Aggarwal, V.K.1
de Vicente, J.2
Bonnert, R.V.A.3
-
240
-
-
70149100867
-
New one-pot synthesis of pyrazole-5-carboxylates by 1,3-dipole cycloadditions of ethyl diazoacetate with-methylene carbonyl compounds
-
Gioiello, A.; Khamidullina, A.; Fulco, M.C.; Venturoni, F.; Zlotsky, S.; Pellicciari, R. New one-pot synthesis of pyrazole-5-carboxylates by 1,3-dipole cycloadditions of ethyl diazoacetate with-methylene carbonyl compounds. Tetrahedron Lett., 2009, 50(44), 5978-5980.
-
(2009)
Tetrahedron Lett
, vol.50
, Issue.44
, pp. 5978-5980
-
-
Gioiello, A.1
Khamidullina, A.2
Fulco, M.C.3
Venturoni, F.4
Zlotsky, S.5
Pellicciari, R.6
-
241
-
-
34248586827
-
A regioselective route to 5-substituted pyrazole- and pyrazoline-3-phosphonic acids and esters
-
Conti, P.; Pinto, A.; Tamborini, L.; Rizzo, V.; De Micheli, C. A regioselective route to 5-substituted pyrazole- and pyrazoline-3-phosphonic acids and esters. Tetrahedron, 2007, 63(25), 5554-5560.
-
(2007)
Tetrahedron
, vol.63
, Issue.25
, pp. 5554-5560
-
-
Conti, P.1
Pinto, A.2
Tamborini, L.3
Rizzo, V.4
de Micheli, C.5
-
242
-
-
0037429086
-
Nitrilimine cycloaddition to 4- (pyrazol-5-yl)carbonyl-2-azetidinone and 4-(pyrazol-4-yl)carbonyl-2-azetidinone
-
Del Buttero, P.; Moltenia, G.; Pilatib, T. Nitrilimine cycloaddition to 4- (pyrazol-5-yl)carbonyl-2-azetidinone and 4-(pyrazol-4-yl)carbonyl-2- azetidinone. Tetrahedron Lett., 2003, 44, 1425-1427.
-
(2003)
Tetrahedron Lett
, vol.44
, pp. 1425-1427
-
-
Del Buttero, P.1
Moltenia, G.2
Pilatib, T.3
-
243
-
-
74749088348
-
Synthesis of novel pyrazoles via [2+3]-dipolar cycloaddition using alkyne surrogates
-
Dadiboyena, S.; Valente, E.J.; Hamme II, A.T. Synthesis of novel pyrazoles via [2+3]-dipolar cycloaddition using alkyne surrogates. Tetrahedron Lett., 2010, 51(9), 1341-1343.
-
(2010)
Tetrahedron Lett
, vol.51
, Issue.9
, pp. 1341-1343
-
-
Dadiboyena, S.1
Valente, E.J.2
Hamme II, A.T.3
-
244
-
-
36448943266
-
An efficient synthesis of 2- Diazo-2-(trimethylsilyl)ethanols and their application to pyrazole synthesis
-
Hari, Y.; Tsuchida, S.; Sone, R.; Aoyama, T. An efficient synthesis of 2- Diazo-2-(trimethylsilyl)ethanols and their application to pyrazole synthesis. Synthesis, 2007, (21), 3371-3375.
-
(2007)
Synthesis
, Issue.21
, pp. 3371-3375
-
-
Hari, Y.1
Tsuchida, S.2
Sone, R.3
Aoyama, T.4
-
245
-
-
33947609921
-
Base-Mediated reaction of the Bestmann Ohira reagent with nitroalkenes for the Regioselective synthesis of phosphonylpyrazoles
-
Muruganantham, R.; Mobin, S.M.; Namboothiri, I.N.N. Base-Mediated reaction of the Bestmann Ohira reagent with nitroalkenes for the Regioselective synthesis of phosphonylpyrazoles. Org. Lett., 2007, 9(6), 1125-1128.
-
(2007)
Org. Lett
, vol.9
, Issue.6
, pp. 1125-1128
-
-
Muruganantham, R.1
Mobin, S.M.2
Namboothiri, I.N.N.3
-
246
-
-
33745725835
-
Novel synthesis of highly functionalized pyrazolines and pyrazoles by triphenylphosphine-mediated reaction of dialkyl azodicarboxylate with allenic esters
-
Nair, V.; Biju, A.T.; Mohanan, K.; Suresh, E. Novel synthesis of highly functionalized pyrazolines and pyrazoles by triphenylphosphine-mediated reaction of dialkyl azodicarboxylate with allenic esters. Org. Lett., 2006, 8(11), 2213-2216.
-
(2006)
Org. Lett
, vol.8
, Issue.11
, pp. 2213-2216
-
-
Nair, V.1
Biju, A.T.2
Mohanan, K.3
Suresh, E.4
-
247
-
-
53849083120
-
Allenylphosphonates-useful precursors of pyrazoles and 1,2,3-Triazoles
-
Chakravarty, M.; Kumar, N.N.B.; Sajna, K.V.; Swamy, K.C.K. Allenylphosphonates-useful precursors of pyrazoles and 1,2,3-Triazoles. Eur. J. Org. Chem., 2008, (26), 4500-4510.
-
(2008)
Eur. J. Org. Chem
, vol.26
, pp. 4500-4510
-
-
Chakravarty, M.1
Kumar, N.N.B.2
Sajna, K.V.3
Swamy, K.C.K.4
-
248
-
-
33751213878
-
Microwave-assisted synthesis of pyrazoles by 1,3-Dipolar cycloaddition of diazo compounds to acetylene derivatives
-
Zrinski, I.; Juribasic, M.; Eckert-Maksic, M. Microwave-assisted synthesis of pyrazoles by 1,3-Dipolar cycloaddition of diazo compounds to acetylene derivatives. Heterocycles, 2006, 68(9), 1961-1967.
-
(2006)
Heterocycles
, vol.68
, Issue.9
, pp. 1961-1967
-
-
Zrinski, I.1
Juribasic, M.2
Eckert-Maksic, M.3
-
249
-
-
63649120694
-
1,3-Dipolar cycloaddition of diazoacetate compounds to terminal alkynes promoted by Zn(OTf)2: An efficient way to the preparation of pyrazoles
-
He, S.; Chen, L.; Niu, Y.-N.; Wu, L.-Y.; Liang, Y.-M. 1,3-Dipolar cycloaddition of diazoacetate compounds to terminal alkynes promoted by Zn(OTf)2: an efficient way to the preparation of pyrazoles. Tetrahedron Lett., 2009, 50(20), 2443-2445.
-
(2009)
Tetrahedron Lett
, vol.50
, Issue.20
, pp. 2443-2445
-
-
He, S.1
Chen, L.2
Niu, Y.-N.3
Wu, L.-Y.4
Liang, Y.-M.5
-
250
-
-
66149125218
-
One-pot synthesis of Narylpyrazoles from arylhalides
-
Gerstenberger, B.S.; Rauckhorst, M.R.; Starr, J.T. One-pot synthesis of Narylpyrazoles from arylhalides. Org. Lett., 2009, 11(10), 2097-2100.
-
(2009)
Org. Lett
, vol.11
, Issue.10
, pp. 2097-2100
-
-
Gerstenberger, B.S.1
Rauckhorst, M.R.2
Starr, J.T.3
-
251
-
-
77951554730
-
A sydnone cycloaddition route to pyrazole boronic esters
-
Browne, D.L.; Helm, M.D.; Plant, A.; Harrity, J.P.A. A sydnone cycloaddition route to pyrazole boronic esters. Angew. Chem., 2007, 119(45), 8810-8812;
-
(2007)
Angew. Chem
, vol.119
, Issue.45
, pp. 8810-8812
-
-
Browne, D.L.1
Helm, M.D.2
Plant, A.3
Harrity, J.P.A.4
-
252
-
-
36549038697
-
A sydnone cycloaddition route to pyrazole boronic esters
-
A sydnone cycloaddition route to pyrazole boronic esters. Angew. Chem. Int. Ed., 2007, 46, 8656-8658.
-
(2007)
Angew. Chem. Int. Ed
, vol.46
, pp. 8656-8658
-
-
-
253
-
-
33645759529
-
Convenient and Efficient synthesis of pyrazole-Based DHODase inhibitors from 3- Aryl-4-cyanosydnone
-
Chang, E.-M.; Chen, T.-H.; Wong, F.F.; Chang, E.-C.; Yeh, M.-Y. Convenient and Efficient synthesis of pyrazole-Based DHODase inhibitors from 3- Aryl-4-cyanosydnone. Synlett, 2006, (6), 901-904.
-
(2006)
Synlett
, vol.6
, pp. 901-904
-
-
Chang, E.-M.1
Chen, T.-H.2
Wong, F.F.3
Chang, E.-C.4
Yeh, M.-Y.5
-
254
-
-
71749097873
-
Recent developments in the chemistry of sydnones
-
Browne, D.L.; Harrity, J.P.A. Recent developments in the chemistry of sydnones. Tetrahedron, 2010, 66(3), 553-568.
-
(2010)
Tetrahedron
, vol.66
, Issue.3
, pp. 553-568
-
-
Browne, D.L.1
Harrity, J.P.A.2
-
255
-
-
33745852809
-
Regioselectivity in 1,3-Dipolar Cycloaddition of 3-(4-Ethoxyphenyl)-4-cyanosydnone with propargylic esters
-
Chang, E.-M.; Wong, F.F.; Chen, T.-H.; Chiang, K.-C.; Yeh, M.-Y. Regioselectivity in 1,3-Dipolar Cycloaddition of 3-(4-Ethoxyphenyl)-4-cyanosydnone with propargylic esters. Heterocycles, 2006, 68(5), 1007-1015.
-
(2006)
Heterocycles
, vol.68
, Issue.5
, pp. 1007-1015
-
-
Chang, E.-M.1
Wong, F.F.2
Chen, T.-H.3
Chiang, K.-C.4
Yeh, M.-Y.5
-
256
-
-
58149305979
-
Cross coupling of Bromo sydnones: Development of a Flexible Route toward Functionalized pyrazoles
-
Browne, D.L.; Taylor, J.B.; Plant, A.; Harrity, J.P.A. Cross coupling of Bromo sydnones: development of a Flexible Route toward Functionalized pyrazoles. J. Org. Chem., 2009, 74, 396-400.
-
(2009)
J. Org. Chem
, vol.74
, pp. 396-400
-
-
Browne, D.L.1
Taylor, J.B.2
Plant, A.3
Harrity, J.P.A.4
-
257
-
-
66149124436
-
Solid-Phase synthesis of amino acid derived N-Unsubstituted pyrazoles via sydnones
-
Harju, K.; Vesterinen, J.; Yli-Kauhaluoma, J. Solid-Phase synthesis of amino acid derived N-Unsubstituted pyrazoles via sydnones. Org. Lett., 2009, 11(10), 2219-2221.
-
(2009)
Org. Lett
, vol.11
, Issue.10
, pp. 2219-2221
-
-
Harju, K.1
Vesterinen, J.2
Yli-Kauhaluoma, J.3
-
258
-
-
0034620920
-
Facile synthesis of pyrazoles and pyrroles via thermolysis of tetrazolo[1,5-b]pyridazines, tetrazolo[1,5-a]pyrimidines and tetrazolo[1,5-a]pyridines
-
Simoni, D.; Rondanin, R.; Furnò, G.; Aiello, E.; Invidiata, F.P. Facile synthesis of pyrazoles and pyrroles via thermolysis of tetrazolo[1,5-b]pyridazines, tetrazolo[1,5-a]pyrimidines and tetrazolo[1,5-a]pyridines. Tetrahedron Lett., 2000, 41(15), 2699-2703.
-
(2000)
Tetrahedron Lett
, vol.41
, Issue.15
, pp. 2699-2703
-
-
Simoni, D.1
Rondanin, R.2
Furnò, G.3
Aiello, E.4
Invidiata, F.P.5
-
259
-
-
85196231603
-
-
Shablykin, O.V.; Brovarets, V.S.; Rusanov, E.B.; Drach, B.S. Zhur. Obsh. Khim. 2008, 78, 674;
-
(2008)
Zhur. Obsh. Khim
, vol.78
, pp. 674
-
-
Shablykin, O.V.1
Brovarets, V.S.2
Rusanov, E.B.3
Drach, B.S.4
-
260
-
-
44349113673
-
Three ways of reactions of 5-(3,5-dimethyl-1 H - pyrazol-1-yl)-2-phenyl-1,3-oxazole-4-carbonitrile and its analogs with nitrogen- containing bases
-
Three ways of reactions of 5-(3,5-dimethyl-1 H - pyrazol-1-yl)-2-phenyl-1,3-oxazole-4-carbonitrile and its analogs with nitrogen- containing bases. Russ. J. Gen. Chem., 2008, 78(4), 655.
-
(2008)
Russ. J. Gen. Chem
, vol.78
, Issue.4
, pp. 674
-
-
-
261
-
-
14844350074
-
Oxaziridine-mediated amination of primary amines: Scope and application to a one-pot pyrazole synthesis
-
Armstrong, A.; Jones, L.H.; Knight, J.D.; Kelsey, R.D. Oxaziridine-mediated amination of primary amines: Scope and application to a one-pot pyrazole synthesis. Org. Lett., 2005, 7(4), 713-716.
-
(2005)
Org. Lett
, vol.7
, Issue.4
, pp. 713-716
-
-
Armstrong, A.1
Jones, L.H.2
Knight, J.D.3
Kelsey, R.D.4
-
262
-
-
26844581526
-
A Novel Route to Fully Substituted 1H-Pyrazoles
-
Suen, Y.F.; Hope, H.; Nantz, M.H.; Haddadin, M.J.; Kurth, M.J. A Novel Route to Fully Substituted 1H-Pyrazoles. J. Org. Chem., 2005, 70, 8468-8471.
-
(2005)
J. Org. Chem
, vol.70
, pp. 8468-8471
-
-
Suen, Y.F.1
Hope, H.2
Nantz, M.H.3
Haddadin, M.J.4
Kurth, M.J.5
-
263
-
-
48849112035
-
Efficient and divergent synthesis of fully substituted 1H-Pyrazoles and isoxazoles from cyclopropyl oximes
-
Wang, K.; Xiang, D.; Liu, J.; Pan, W.; Dong, D. Efficient and divergent synthesis of fully substituted 1H-Pyrazoles and isoxazoles from cyclopropyl oximes. Org. Lett., 2008, 10(9), 1691-1694.
-
(2008)
Org. Lett
, vol.10
, Issue.9
, pp. 1691-1694
-
-
Wang, K.1
Xiang, D.2
Liu, J.3
Pan, W.4
Dong, D.5
-
264
-
-
0038765391
-
An Alternative Route for Carboni Lindsey Reaction: N,N Cycloaddition of an Alkene to s-Tetrazine
-
Zhou, X.; Kovalev (the late), E.G.; Klug, J.T.; Khodorkovsky, V. An Alternative Route for Carboni Lindsey Reaction: N,N Cycloaddition of an Alkene to s-Tetrazine. Org. Lett., 2001, 3(11), 1725-1727.
-
(2001)
Org. Lett
, vol.3
, Issue.11
, pp. 1725-1727
-
-
Zhou, X.1
Kovalev, E.G.2
Klug, J.T.3
Khodorkovsky, V.4
-
265
-
-
67650541096
-
The conversion of isothiazoles into pyrazoles using hydrazine
-
Ioannidou, H.A.; Koutentis, P.A. The conversion of isothiazoles into pyrazoles using hydrazine. Tetrahedron, 2009, 65(34), 7023-7037.
-
(2009)
Tetrahedron
, vol.65
, Issue.34
, pp. 7023-7037
-
-
Ioannidou, H.A.1
Koutentis, P.A.2
-
266
-
-
35348998945
-
Straightforward transformation of isoxazoles into pyrazoles: Renewed and improved
-
Sviridov, S.I.; Vasil'ev, A.A.; Shorshnev, S.V. Straightforward transformation of isoxazoles into pyrazoles: renewed and improved. Tetrahedron, 2007, 63(49), 12195-12201.
-
(2007)
Tetrahedron
, vol.63
, Issue.49
, pp. 12195-12201
-
-
Sviridov, S.I.1
Vasil'ev, A.A.2
Shorshnev, S.V.3
-
267
-
-
55149083190
-
2-(Pirazol-4-il)-5-fenil- 1,3,4-tiadiazoly
-
Shokol, T.V.; Semenyuchenko, V.V.; Khilya, V.P. 2-(Pirazol-4-il)-5-fenil- 1,3,4-tiadiazoly. Khim. Geterotsikl. Soedin., 2005, 5, 781-788;
-
(2005)
Khim. Geterotsikl. Soedin
, vol.5
, pp. 781-788
-
-
Shokol, T.V.1
Semenyuchenko, V.V.2
Khilya, V.P.3
-
268
-
-
24644451095
-
5-Phenyl-2- (pyrazol-4-yl)-1,3,4-thiadiazoles
-
5-Phenyl-2- (pyrazol-4-yl)-1,3,4-thiadiazoles. Chem. Heterocycl. Comp. 2005, 41(5), 673-678.
-
(2005)
Chem. Heterocycl. Comp
, vol.41
, Issue.5
, pp. 673-678
-
-
-
269
-
-
33750623389
-
Domino Cu-catalyzed C-N coupling/ hydroamidation: A highly efficient synthesis of nitrogen heterocycles
-
Martín, R.; Rivero, M.R.; Buchwald, S.L. Domino Cu-catalyzed C-N coupling/ hydroamidation: a highly efficient synthesis of nitrogen heterocycles. Angew. Chem. Int. Ed., 2006, 45, 7079-7082.
-
(2006)
Angew. Chem. Int. Ed
, vol.45
, pp. 7079-7082
-
-
Martín, R.1
Rivero, M.R.2
Buchwald, S.L.3
-
270
-
-
51149116300
-
A Regiospecific Approach to N-Alkylpyrazoles and the derived N-oxides using 5-endo-dig cyclisations of alkynyl nitrosamines
-
Hayes, S.J.; Knight, D.W.; ÓHalloran, M.; Pickering, S.R. A Regiospecific Approach to N-Alkylpyrazoles and the derived N-oxides using 5-endo-dig cyclisations of alkynyl nitrosamines. Synlett, 2008, (14), 2188-2190.
-
(2008)
Synlett
, vol.14
, pp. 2188-2190
-
-
Hayes, S.J.1
Knight, D.W.2
ÓHalloran, M.3
Pickering, S.R.4
-
271
-
-
0037882618
-
Oxidative Aromatization of 1,3,5-trisubstituted pyrazolines and hantzsch 1,4-dihydropyridines by Pd/C in acetic acid
-
Nakamichi, N.; Kawashita, Y.; Hayashi, M. Oxidative Aromatization of 1,3,5-trisubstituted pyrazolines and hantzsch 1,4-dihydropyridines by Pd/C in acetic acid. Org. Lett., 2002, 4(22), 3955-3957.
-
(2002)
Org. Lett
, vol.4
, Issue.22
, pp. 3955-3957
-
-
Nakamichi, N.1
Kawashita, Y.2
Hayashi, M.3
-
272
-
-
43849088792
-
Silica Sulfuric Acid-Activated Poly-1,3,-dichloro-5-methyl-5(4'-vinylphenyl)hydantoin (PDCVH) as an Effective reagent for oxidation of 1,3,5-trisubstituted 2-pyrazolines both under microwave irradiation and thermal condition
-
Azarifar, D.; Maleki, B.; Setayeshnazar, M. Silica Sulfuric Acid-Activated Poly-1,3,-dichloro-5-methyl-5(4'-vinylphenyl)hydantoin (PDCVH) as an Effective reagent for oxidation of 1,3,5-trisubstituted 2-pyrazolines both under microwave irradiation and thermal condition. Heterocycles, 2008, 75(3), 669-673.
-
(2008)
Heterocycles
, vol.75
, Issue.3
, pp. 669-673
-
-
Azarifar, D.1
Maleki, B.2
Setayeshnazar, M.3
-
273
-
-
33746013175
-
Microwave-promoted aromatization of 1,3,5- trisubstituted 4,5-Dihydro-1H-pyrazoles by calcium hypochlorite under Solvent- free Conditions
-
Azarifar, D.; Gharshasbi, A. Microwave-promoted aromatization of 1,3,5- trisubstituted 4,5-Dihydro-1H-pyrazoles by calcium hypochlorite under Solvent- free Conditions. Heterocycles, 2006, 68(6), 1209-1215.
-
(2006)
Heterocycles
, vol.68
, Issue.6
, pp. 1209-1215
-
-
Azarifar, D.1
Gharshasbi, A.2
-
274
-
-
26044462279
-
Microwave-assisted aromatization of 1,3,5- trisubstituted 2-pyrazolines by silica-supported N-bromosuccinimide as a useful reagent under solvent free 'dry' condition
-
Azarifar, D.; Maleki, B. microwave-assisted aromatization of 1,3,5- trisubstituted 2-pyrazolines by silica-supported N-bromosuccinimide as a useful reagent under solvent free 'dry' condition. Heterocycles, 2005, 65(4), 865-870.
-
(2005)
Heterocycles
, vol.65
, Issue.4
, pp. 865-870
-
-
Azarifar, D.1
Maleki, B.2
-
275
-
-
2542504592
-
Activated carbon-promoted oxidative aromatization of hantzsch 1,4-dihydropyridines and 1,3,5- trisubstituted pyrazolines using molecular oxygen
-
Nakamichi, N.; Kawashita, Y.; Hayashi, M. activated carbon-promoted oxidative aromatization of hantzsch 1,4-dihydropyridines and 1,3,5- trisubstituted pyrazolines using molecular oxygen. Synthesis, 2004, (7), 1015-1020.
-
(2004)
Synthesis
, vol.7
, pp. 1015-1020
-
-
Nakamichi, N.1
Kawashita, Y.2
Hayashi, M.3
-
276
-
-
0037711699
-
Zr(NO3)4: A versatile oxidizing agent for aromatization of hantzsch 1,4-dihydropyridines and 1,3,5-trisubstituted pyrazolines
-
Sabitha, G.; Kiran Kumar Reddy, G.S.; Srinivas Reddy, C.; Fatima, N.; Yadav, J.S. Zr(NO3)4: a versatile oxidizing agent for aromatization of hantzsch 1,4-dihydropyridines and 1,3,5-trisubstituted pyrazolines. Synthesis, 2003, (8), 1267-1271.
-
(2003)
Synthesis
, vol.8
, pp. 1267-1271
-
-
Sabitha, G.1
Kiran, K.R.G.S.2
Srinivas, R.C.3
Fatima, N.4
Yadav, J.S.5
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