Antifungal and antimycobacterial activity of 1-(3,5-diaryl-4,5-dihydro-1H-pyrazol-4-yl)-1H-imidazole derivatives

Bioorganic and Medicinal Chemistry

Volumn 16, Issue 8, 2008, Pages 4516-4522

  Zampieri, Daniele ^a   Mamolo, Maria Grazia ^a   Laurini, Erik ^a   Scialino, Giuditta ^a   Banfi, Elena ^a   Vio, Luciano ^a  

^a UNIVERSITY OF TRIESTE   (Italy)

Author keywords

1 (3,5 Diaryl 4,5 dihydro 1H pyrazol 4 yl) 1H imidazole derivatives; Antifungal and antimycobacterial activity

Indexed keywords

(4,5 DIHYDRO 1,3,5 TRIPHENYL 1H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 (3,5 BIS (2,4 DICHLOROPHENYL) 4,5 DIHYDRO 1 (4 FLUOROPHENYL) 1 H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 (3,5 BIS (4 BROMOPHENYL) 4,5 DIHYDRO 1 (4 FLUOROPHENYL) 1H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 (4,5 DIHYDRO 3,5 DIPHENYL 1 (4 FLUOROPHENYL) 1H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 (4,5 DIHYDRO 3,5 DIPHENYL 1,1 METHYL 1H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 (4,5 DIHYDRO 3,5 DIPHENYL 1H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 [3,4 BIS (4 BROMOPHENYL) 4,5 DIHYDRO 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [3,5 BIS (2,4 DICHLOROPHENYL) 4,5 DIHYDRO 1 METHYL 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [3,5 BIS (2,4 DICHLOROPHENYL) 4,5 DIHYDRO 1 PHENYL 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [3,5 BIS (2,4 DICHLOROPHENYL) 4,5 DIHYDRO 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [3,5 BIS (4 BROMOPHENYL) (4,5 DIHYDRO 1 METHYL 1H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 [3,5 BIS (4 BROMOPHENYL) 4,5 DIHYDRO 1 PHENYL 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [3,5 BIS (4 CHLOROPHENYL) (4,5 DIHYDRO 1 METHYL 1H PYRAZOL 4 YL) 1H IMIDAZOLE; 1 [3,5 BIS (4 CHLOROPHENYL) 4,5 DIHYDRO 1 PHENYL 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [3,5 BIS (4 CHLORPHENYL) 4,5 DIHYDRO 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [4,5 DIHYDRO 1 (4 FLUOROPHENYL) 3,5 BIS (4 METHYLPHENYL) 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [4,5 DIHYDRO 1 METHYL 3,5 BIS (4 METHYL PHENYL) 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [4,5 DIHYDRO 3,5 BIS (4 METHYL PHENYL) 1 PHENYL 1H PYRAZOL 4 YL] 1H IMIDAZOLE; 1 [4,5 DIHYDRO 3,5 BIS (4 METHYLPHENYL) 1H PYRAZOL 4 YL] 1H IMIDAZOLE; IMIDAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; MYCOBACTERIUM TUBERCULOSIS;

ANTI-BACTERIAL AGENTS; ANTIFUNGAL AGENTS; CANDIDA ALBICANS; HYDROGEN; IMIDAZOLES; MAGNETIC RESONANCE SPECTROSCOPY; MOLECULAR STRUCTURE; MYCOBACTERIUM TUBERCULOSIS; PYRAZOLES; STRUCTURE-ACTIVITY RELATIONSHIP;

CANDIDA ALBICANS;

EID: 42249084709     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2008.02.055     Document Type: Article

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