Activation of HIF-prolyl hydroxylases by R59949, an inhibitor of the diacylglycerol kinase

Journal of Biological Chemistry

Volumn 280, Issue 25, 2005, Pages 24238-24244

  Temes, Elisa ^a   Martín Puig, Silvia ^a   Acosta Iborra, Bárbara ^a   Castellanos, Maria C ^a   Feijoo Cuaresma, Mónica ^a   Olmos, Gemma ^a,b   Aragonés, Julián ^a,c   Landazuri, Manuel O ^a  

^a UNIVERSIDAD AUTÓNOMA DE MADRID   (Spain)

^b UNIVERSITY OF ALCALÁ   (Spain)

^c DEPARTMENT OF PLANT SYSTEMS BIOLOGY   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

ACTIVATION ANALYSIS; BIOCHEMISTRY; CELLS; DIMERS; ENZYME INHIBITION; OXYGEN;

CELLULAR ADAPTATION; HYPOXIA-INDUCIBLE FACTORS (HIF); PROLYL;

ENZYME KINETICS;

3 [2 [4 (4,4' DIFLUOROBENZHYDRYLIDENE)PIPERIDINO]ETHYL] 2,3 DIHYDRO 2 THIOXO 4(1H) QUINAZOLINONE; DIACYLGLYCEROL KINASE INHIBITOR; HYPOXIA INDUCIBLE FACTOR 1ALPHA; HYPOXIA INDUCIBLE FACTOR 2ALPHA; MESSENGER RNA; OXYGEN; PROCOLLAGEN PROLINE 2 OXOGLUTARATE 4 DIOXYGENASE; TRANSCRIPTION FACTOR; VON HIPPEL LINDAU PROTEIN;

ARTICLE; CELL FUNCTION; CONTROLLED STUDY; DRUG ACTIVATION; DRUG EFFECT; ENZYME ACTIVITY; HUMAN; HUMAN CELL; HYPOXIA; IMMUNOPRECIPITATION; IN VITRO STUDY; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN PROCESSING; PROTEIN PROTEIN INTERACTION; PROTEIN TARGETING;

CELL LINE; DIACYLGLYCEROL KINASE; ENZYME ACTIVATION; ENZYME INHIBITORS; HUMANS; IMMUNOPRECIPITATION; PIPERIDINES; PROCOLLAGEN-PROLINE DIOXYGENASE; QUINAZOLINES; QUINAZOLINONES; RNA, MESSENGER; TUMOR SUPPRESSOR PROTEINS; UBIQUITIN-PROTEIN LIGASES; VON HIPPEL-LINDAU TUMOR SUPPRESSOR PROTEIN;

EID: 21244492413     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.M414694200     Document Type: Article

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