Analogues of dealanylalahopcin are inhibitors of human HIF prolyl hydroxylases

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 8, 2003, Pages 1451-1454

  Schlemminger, Imre ^a   Mole, David R ^b   McNeill, Luke A ^a   Dhanda, Anupma ^a   Hewitson, Kirsty S ^a   Tian, Ya Min ^b   Ratcliffe, Peter J ^b   Pugh, Christopher W ^b   Schofield, Christopher J ^a  

^a UNIVERSITY OF OXFORD   (United Kingdom)

^b UNIVERSITY OF OXFORD   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 OXOGLUTARIC ACID; DEALANYLALAHOPCIN DERIVATIVE; ENZYME INHIBITOR; HYDROXAMIC ACID; HYPOXIA INDUCIBLE FACTOR 1ALPHA; OXYGENASE; PROCOLLAGEN PROLINE 2 OXOGLUTARATE 4 DIOXYGENASE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL ASSAY; DRUG ACTIVITY; DRUG BINDING SITE; DRUG INHIBITION; DRUG SCREENING; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME SUBSTRATE; HYDROPHOBICITY; IC 50; IRON CHELATION; NONHUMAN; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY;

EID: 0037451821     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00149-5     Document Type: Article

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