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BRISTOL-MYERS SQUIBB CO (Priestley ES, Decicco CP, Hudyma TW, Zheng X): Compounds useful for treating hepatitis C virus. WO-03026587 (2003).
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BRISTOL-MYERS SQUIBB CO (Priestley ES, Decicco CP, Hudyma TW, Zheng X): Compounds useful for treating hepatitis C virus. WO-03026587 (2003).
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83
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68549127750
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NEOGENESIS PHARMACEUTICALS INC (Shipps GW Jr, Rosner KE, Popovici-Muller J, Deng Y, Wang T, Curran PJ): Novel pyrazolo[1,5 a]pyrimidine compounds useful as inhibitors of hepatitis C virus replication. WO-03101993 (2003).
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NEOGENESIS PHARMACEUTICALS INC (Shipps GW Jr, Rosner KE, Popovici-Muller J, Deng Y, Wang T, Curran PJ): Novel pyrazolo[1,5 a]pyrimidine compounds useful as inhibitors of hepatitis C virus replication. WO-03101993 (2003).
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84
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68549091650
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BOEHRINGER INGELHEIM CANADA LTD (Beaulieu PL, Fazal G, Goulet S, Kukolj G, Poirier M, Tsantrizos YS): Novel azaheterocyclic amides or thioamide viral replication inhibitors. WO-03007945 (2003).
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BOEHRINGER INGELHEIM CANADA LTD (Beaulieu PL, Fazal G, Goulet S, Kukolj G, Poirier M, Tsantrizos YS): Novel azaheterocyclic amides or thioamide viral replication inhibitors. WO-03007945 (2003).
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85
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68549106815
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SMITHKLINE BEECHAM CORP (Dhanak D, Kaura AC, Shaw A): Novel quinolinone inhibitors of hepatitis C virus. WO-00185172 (2001).
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SMITHKLINE BEECHAM CORP (Dhanak D, Kaura AC, Shaw A): Novel quinolinone inhibitors of hepatitis C virus. WO-00185172 (2001).
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86
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68549114396
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Darcy MG, Dhanak D, Duffy KJ, Erickson GA, Fitch DM, Gates
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AT, Johnston VK, Sarisky RT, Sharp MJ, Shaw AN et al, Novel antiviral 1,2,4-benzothiadiazine 1,1-dioxide derivatives. WO-02098424 2002
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SMITHKLINE BEECHAM CORP (Chai D, Darcy MG, Dhanak D, Duffy KJ, Erickson GA, Fitch DM, Gates AT, Johnston VK, Sarisky RT, Sharp MJ, Shaw AN et al): Novel antiviral 1,2,4-benzothiadiazine 1,1-dioxide derivatives. WO-02098424 (2002).
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87
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68549141024
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SMITHKLINE BEECHAM CORP (Darcy MG, Dhanak D, Duffy KJ, Fitch DM, Sarisky RT, Shaw AN, Tedesco R, Zimmerman MN): Novel nitrogen heterocycle compounds useful for the treatment of RNA virus infection, hepatitis C virus infection, hepatocellular carcinoma and liver fibrosis. WO-03059356 (2003).
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SMITHKLINE BEECHAM CORP (Darcy MG, Dhanak D, Duffy KJ, Fitch DM, Sarisky RT, Shaw AN, Tedesco R, Zimmerman MN): Novel nitrogen heterocycle compounds useful for the treatment of RNA virus infection, hepatitis C virus infection, hepatocellular carcinoma and liver fibrosis. WO-03059356 (2003).
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88
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68549121777
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SMITHKLINE BEECHAM CORP (Dhanak D, Duffy KJ, Sarisky RT, Shaw AN, Tedesco R): Novel anti-infectives. WO-03037262 (2003).
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SMITHKLINE BEECHAM CORP (Dhanak D, Duffy KJ, Sarisky RT, Shaw AN, Tedesco R): Novel anti-infectives. WO-03037262 (2003).
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89
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68549127751
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SMITHKLINE BEECHAM CORP (Duffy KJ, Evans KA, Fitch DM, Gates AT, Johnston VK, Sarisky RT): Novel 4-hydroxy-3-(1,1-dioxo-1,4-dihydrobenzo[1,2,4]thiadiazin-3-yl)-1, 5-dihydropyrrol-2-one derivatives useful for treating hepatitis C virus infection. WO-03099801 (2003).
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SMITHKLINE BEECHAM CORP (Duffy KJ, Evans KA, Fitch DM, Gates AT, Johnston VK, Sarisky RT): Novel 4-hydroxy-3-(1,1-dioxo-1,4-dihydrobenzo[1,2,4]thiadiazin-3-yl)-1, 5-dihydropyrrol-2-one derivatives useful for treating hepatitis C virus infection. WO-03099801 (2003).
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90
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-
68549105107
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SHIRE BIOCHEM INC (Chan CKL, Bidard J, Das SK, Pereira OZ, Shuttleworth S, Siddiqui MA, Wang W): Novel biaryl compounds useful for the treatment of flavivirus infections. WO-02100846 (2002).
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SHIRE BIOCHEM INC (Chan CKL, Bidard J, Das SK, Pereira OZ, Shuttleworth S, Siddiqui MA, Wang W): Novel biaryl compounds useful for the treatment of flavivirus infections. WO-02100846 (2002).
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91
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68549131539
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SHIRE BIOCHEM INC (Chan CKL, Bidard J, Das SK, Nguyen BN, Pereira OZ, Reddy TJ, Siddiqui MA, Wang W, Yannopoulos C): Novel substituted thiophene compounds useful for the treatment of flavirus infections. WO-02100851 (2002).
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SHIRE BIOCHEM INC (Chan CKL, Bidard J, Das SK, Nguyen BN, Pereira OZ, Reddy TJ, Siddiqui MA, Wang W, Yannopoulos C): Novel substituted thiophene compounds useful for the treatment of flavirus infections. WO-02100851 (2002).
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92
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68549121779
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SHIRE BIOCHEM INC (Kong LCC, Siddiqui MA): Thiazole derivatives and their use for the treatment or prevention of Flavivirus infections. EP-01321463 (2003).
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SHIRE BIOCHEM INC (Kong LCC, Siddiqui MA): Thiazole derivatives and their use for the treatment or prevention of Flavivirus infections. EP-01321463 (2003).
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93
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68549114397
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AGOURON PHARMACEUTICALS INC (Love RA, Yu X, Diehl W, Hickey MJ, Parge HE, Gao J, Fuhrman S): Hepatitis C virus (HCV) NS5B RNA polymerase and mutants thereof. EP-01256628 (2002).
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AGOURON PHARMACEUTICALS INC (Love RA, Yu X, Diehl W, Hickey MJ, Parge HE, Gao J, Fuhrman S): Hepatitis C virus (HCV) NS5B RNA polymerase and mutants thereof. EP-01256628 (2002).
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94
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68549127753
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PFIZER INC (Gonzalez J, Borchardt AJ, Dragovich PS, Jewell TM, Linton MA, Zhou R, Li H, Tatlock JH, Abreo MA, Prins TJ): Use of pyranone derivatives as inhibitors of hepatitis C virus RNA-dependent RNA polymerase. WO-03095441 (2003).
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PFIZER INC (Gonzalez J, Borchardt AJ, Dragovich PS, Jewell TM, Linton MA, Zhou R, Li H, Tatlock JH, Abreo MA, Prins TJ): Use of pyranone derivatives as inhibitors of hepatitis C virus RNA-dependent RNA polymerase. WO-03095441 (2003).
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95
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68549106818
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PFIZER INC (Borchardt AJ, Goble MP): Novel pyranone and pyrandiones useful as HCV polymerase inhibitors for treating hepatitis C virus infection. WO-03082848 (2003).
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PFIZER INC (Borchardt AJ, Goble MP): Novel pyranone and pyrandiones useful as HCV polymerase inhibitors for treating hepatitis C virus infection. WO-03082848 (2003).
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96
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68549098789
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WYETH/VIROPHARMA INC (Gopalsamy A, Collette MS, Ellingboe JW, Laporte MG, Mansour TS, Burns CJ, Park K, Condon SM): The use of pyranoindole derivatives as hepatitis C polymerase inhibitors. WO-03099275 (2003).
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WYETH/VIROPHARMA INC (Gopalsamy A, Collette MS, Ellingboe JW, Laporte MG, Mansour TS, Burns CJ, Park K, Condon SM): The use of pyranoindole derivatives as hepatitis C polymerase inhibitors. WO-03099275 (2003).
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97
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68549134209
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WYETH/VIROPHARMA INC (Gopalsamy A, Ellingboe JW, Mansour TS): Novel (R)-enantiomers of pyranoindole compounds useful for treating hepatitis C viral infection. WO-03099824 (2003).
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WYETH/VIROPHARMA INC (Gopalsamy A, Ellingboe JW, Mansour TS): Novel (R)-enantiomers of pyranoindole compounds useful for treating hepatitis C viral infection. WO-03099824 (2003).
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98
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68549139126
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B&C BIOPHARM (Kim J-W, Lee S-W, Lee G-H, Han J-J, Park S-J, Park E-Y, Shin J-C, Novel 6-(4-substituted-anilino)pyrimidine derivatives useful for the treatment of HCV infection. WO-03084953 2003
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B&C BIOPHARM (Kim J-W, Lee S-W, Lee G-H, Han J-J, Park S-J, Park E-Y, Shin J-C): Novel 6-(4-substituted-anilino)pyrimidine derivatives useful for the treatment of HCV infection. WO-03084953 (2003).
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99
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68549119728
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FUJISAWA PHARMACEUTICAL CO LTD (Inoue T, Maki K, Hatakenaka K, Yamagishi Y): Novel compositions comprising fused benzene compounds useful as RNA-dependent RNA polymerase inhibitors for treating viral infections. WO-03082265 (2003).
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FUJISAWA PHARMACEUTICAL CO LTD (Inoue T, Maki K, Hatakenaka K, Yamagishi Y): Novel compositions comprising fused benzene compounds useful as RNA-dependent RNA polymerase inhibitors for treating viral infections. WO-03082265 (2003).
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100
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-
68549089777
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DONG WHA P ARM IND CO LTD (Yoon S-J, Lee S-W, Lee J-S, Kim N-D, Lee G-H, Lee H-D, Kim J-W, Park S-J, Park H-J): 6-Methylnicotinamide derivatives as antiviral agents. WO-00178648 (2003).
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DONG WHA P ARM IND CO LTD (Yoon S-J, Lee S-W, Lee J-S, Kim N-D, Lee G-H, Lee H-D, Kim J-W, Park S-J, Park H-J): 6-Methylnicotinamide derivatives as antiviral agents. WO-00178648 (2003).
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-
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101
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-
68549089776
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DONG WHA PHARM IND CO LTD (Chung Y-H, Lee C-W, Yang W-Y, Lee H-D, Park W-J, Chang Y-Y, Lee J-S): Novel 2,4-difluorobenzamide derivatives as antiviral agents for treating HBV and HCV infections. WO-03002518 (2003).
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DONG WHA PHARM IND CO LTD (Chung Y-H, Lee C-W, Yang W-Y, Lee H-D, Park W-J, Chang Y-Y, Lee J-S): Novel 2,4-difluorobenzamide derivatives as antiviral agents for treating HBV and HCV infections. WO-03002518 (2003).
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102
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68549089775
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DONG WHA PHARM IND CO LTD (Chung Y-H, Lee C-W, Yang W-Y, Lee H-D, Park W-J, Chang Y-Y, Lee J-S): Methoxy-1,3,5-triazine derivatives with activity against HBV and HCV polymerases. WO-02079187 (2002).
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DONG WHA PHARM IND CO LTD (Chung Y-H, Lee C-W, Yang W-Y, Lee H-D, Park W-J, Chang Y-Y, Lee J-S): Methoxy-1,3,5-triazine derivatives with activity against HBV and HCV polymerases. WO-02079187 (2002).
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103
-
-
68549139127
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SMITHKLINE BEECHAM CORP (Dhanak D, Carr T): Novel heterocyclic compounds for the treatment of hepatitis C viral infection. WO-00185720 (2001).
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SMITHKLINE BEECHAM CORP (Dhanak D, Carr T): Novel heterocyclic compounds for the treatment of hepatitis C viral infection. WO-00185720 (2001).
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104
-
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68549108626
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GLAXO WELLCOME PLC (Bravi G, Goodland HS, Haigh D, Hartley CD, Lovegrove VLH, Shah P, Slater MJ): 4-(5-Membered)-heteroaryl acyl pyrrolidine derivatives as HCV inhibitors. WO-03037894 (2003).
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GLAXO WELLCOME PLC (Bravi G, Goodland HS, Haigh D, Hartley CD, Lovegrove VLH, Shah P, Slater MJ): 4-(5-Membered)-heteroaryl acyl pyrrolidine derivatives as HCV inhibitors. WO-03037894 (2003).
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-
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105
-
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68549114398
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GLAXO WELLCOME PLC (Bravi G, Guidetti R, Haigh D, Hartley CD, Howes PD, Jackson DL, Lovegrove VLH, Shah P, Slater MJ, Wareing KJ): 4-(6-Membered)-heteroaryl acyl pyrrolidine derivatives as HCV inhibitors. WO-03037895 (2003).
-
GLAXO WELLCOME PLC (Bravi G, Guidetti R, Haigh D, Hartley CD, Howes PD, Jackson DL, Lovegrove VLH, Shah P, Slater MJ, Wareing KJ): 4-(6-Membered)-heteroaryl acyl pyrrolidine derivatives as HCV inhibitors. WO-03037895 (2003).
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-
-
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106
-
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68549126126
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GLAXO WELLCOME PLC (Slater MJ, Howes PD): Novel acyl bicyclic pyrrole derivative RNA-dependent RNA polymerase inhibitors useful for treating viral infections. WO-03097646 (2003).
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GLAXO WELLCOME PLC (Slater MJ, Howes PD): Novel acyl bicyclic pyrrole derivative RNA-dependent RNA polymerase inhibitors useful for treating viral infections. WO-03097646 (2003).
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107
-
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68549086116
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GLAXO WELLCOME P LC (Bravi G, Howes PD, Lovegrove VLH, Shah P, Slater MJ): Acyl dihydro pyrrole derivatives as HCV inhibitors. WO-03037893 (2003).
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GLAXO WELLCOME P LC (Bravi G, Howes PD, Lovegrove VLH, Shah P, Slater MJ): Acyl dihydro pyrrole derivatives as HCV inhibitors. WO-03037893 (2003).
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108
-
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68549121778
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GLAXO WELLCOME PLC (Burton G, Goodland HS, Haigh D, Kiesow TJ, Ku TW, Slater MJ): Novel 4-cyanopyrrolidine-2-carboxylic acid derivatives and their use as NS5B polymerase inhibitors for the treatment of viral infections, especially HCV infection. WO-2004009543 (2004).
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GLAXO WELLCOME PLC (Burton G, Goodland HS, Haigh D, Kiesow TJ, Ku TW, Slater MJ): Novel 4-cyanopyrrolidine-2-carboxylic acid derivatives and their use as NS5B polymerase inhibitors for the treatment of viral infections, especially HCV infection. WO-2004009543 (2004).
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109
-
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68549095234
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PHARMACIA & UPJOHN CO (Battistini C, Casuscelli F, Kelly RC, Maggiora LL, Mitchell MA, Piutti C, Reding MT, Novel substituted diphenylamine derivatives useful for the treatment of HCV infection. WO-2004002940 2004
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PHARMACIA & UPJOHN CO (Battistini C, Casuscelli F, Kelly RC, Maggiora LL, Mitchell MA, Piutti C, Reding MT): Novel substituted diphenylamine derivatives useful for the treatment of HCV infection. WO-2004002940 (2004).
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110
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68549093481
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PHARMACIA & UPJOHN CO (Finzel BC, Funk LA, Kelly RC, Reding MT, Wicnienski NA, Novel substituted 2-aminobenzamide derivatives as inhibitors of viral RNA-dependent RNA polymerase useful for treating viral infections. WO-2004002944 2004
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PHARMACIA & UPJOHN CO (Finzel BC, Funk LA, Kelly RC, Reding MT, Wicnienski NA): Novel substituted 2-aminobenzamide derivatives as inhibitors of viral RNA-dependent RNA polymerase useful for treating viral infections. WO-2004002944 (2004).
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-
-
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111
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68549137536
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PHARMACIA & UPJOHN CO (Gao H, Greene ML, Gross RJ, Nugent RA, Pfefferkorn J, Novel amine substituted acrylic acid compounds useful for the treatment of viral infection, hepatitis and hepatitis C virus infection. WO-2004002977 2004
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PHARMACIA & UPJOHN CO (Gao H, Greene ML, Gross RJ, Nugent RA, Pfefferkorn J): Novel amine substituted acrylic acid compounds useful for the treatment of viral infection, hepatitis and hepatitis C virus infection. WO-2004002977 (2004).
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112
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68549119727
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RIGEL PHARMACEUTICALS INC (Singh R, Goff D, Lu H, Issankani SD, Sun T): Novel hydrated p-toluenesulfonate salt of 5-[4-[2-(N-methyl-N-(2-pyridyl)amino) ethoxy]benzyl]thiazolidine-2,4-dione. WO-03040112 (2003).
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RIGEL PHARMACEUTICALS INC (Singh R, Goff D, Lu H, Issankani SD, Sun T): Novel hydrated p-toluenesulfonate salt of 5-[4-[2-(N-methyl-N-(2-pyridyl)amino) ethoxy]benzyl]thiazolidine-2,4-dione. WO-03040112 (2003).
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-
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113
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68549106817
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RIGEL PHARMACEUTICALS INC (Singh R, Goff D, Partridge J): Novel pyridyl-substituted heterocycles, useful for treating or preventing hepatitis C virus infection. WO-2004018463 (2004).
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RIGEL PHARMACEUTICALS INC (Singh R, Goff D, Partridge J): Novel pyridyl-substituted heterocycles, useful for treating or preventing hepatitis C virus infection. WO-2004018463 (2004).
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