-
1
-
-
85004871005
-
-
Barany, G., Merrifield, R.B. Solid-phase peptide synthesis. In: The Peptides, Vol. 2. Gross, E., Meienhofer, J. (Eds.). Academic Press: New York 1979,1 -284.
-
(1979)
Solid-phase Peptide Synthesis. In: the Peptides, Vol. 2. Gross, E., Meienhofer, J. (Eds.). Academic Press: New York
, pp. 1-284
-
-
Barany, G.1
Merrifield, R.B.2
-
3
-
-
0027591808
-
-
Danishevsky, S.J., McClure, K.F., Randolph, J.T., Ruggeri, R.B. A strategy for the solid phase synthesis of oligosaccharides. Science 1993, 260:1307-9.
-
(1993)
A Strategy for the Solid Phase Synthesis of Oligosaccharides. Science
, vol.260
, pp. 1307-1309
-
-
Danishevsky, S.J.1
McClure, K.F.2
Randolph, J.T.3
Ruggeri, R.B.4
-
5
-
-
0003834870
-
-
Fields, G.B., Tian, Z., Barany, G. Principles and practice of solidphase peptide synthesis. In: Synthetic Peptides: A User's Guide. Grant, G.A. (Ed.). W.H. Freeman: New York 1992, 77-183.
-
(1992)
Principles and Practice of Solidphase Peptide Synthesis. In: Synthetic Peptides: a User's Guide. Grant, G.A. (Ed.). W.H. Freeman: New York
, pp. 77-183
-
-
Fields, G.B.1
Tian, Z.2
Barany, G.3
-
7
-
-
1542440857
-
-
Barany, G., Albericio, F., Kates, S.A., Kempe, M. Polymer preprints. Am Chem Soc Div Polym Chem 1997, in press.
-
(1997)
Polymer Preprints. Am Chem Soc Div Polym Chem
-
-
Barany, G.1
Albericio, F.2
Kates, S.A.3
Kempe, M.4
-
9
-
-
33745579755
-
-
b Szostak, J. Ed. Chem Rev 1997, 97: 347-509. Additionally, the journal Molecular Diversity contains relevant articles in combinatorial chemistry.
-
The design, synthesis, evaluation and decoding of small-molecule combinatorial libraries has recently been reviewed. See: a) Czarnik, A. Ed. Ace Chem Res 1996,29:111 -70. b) Szostak, J. Ed. Chem Rev 1997, 97: 347-509. Additionally, the journal Molecular Diversity contains relevant articles in combinatorial chemistry.
-
(1996)
The Design, Synthesis, Evaluation and Decoding of Small-molecule Combinatorial Libraries Has Recently Been Reviewed. See: A Czarnik, A. Ed. Ace Chem Res
, vol.29
, pp. 111-170
-
-
-
13
-
-
0027202613
-
-
DeWitt, S.H., Kiely, U.S., Stankovic, C.J., Schroeder, M.C., Cody, D.M.R., Pavia, M.R. "Diversomers": An approach to nonpep-tide, nonoligomeric chemical diversity. Proc Natl Acad Sei USA 1993,90:6909-13.
-
(1993)
"Diversomers": An Approach to Nonpep-tide, Nonoligomeric Chemical Diversity. Proc Natl Acad Sei USA
, vol.90
, pp. 6909-6913
-
-
Dewitt, S.H.1
Kiely, U.S.2
Stankovic, C.J.3
Schroeder, M.C.4
Cody, D.M.R.5
Pavia, M.R.6
-
14
-
-
0028151071
-
-
Kurth, M.J., Randall, L.A.A., Chen, C., Melander, C., Miller, R.B. Library-based lead compound discovery: Antioxidants by an analogous synthesis/deconvolutive assay strategy. J Org Chem 1994, 59: 5862-4.
-
(1994)
Library-based Lead Compound Discovery: Antioxidants by An Analogous Synthesis/deconvolutive Assay Strategy. J Org Chem
, vol.59
, pp. 5862-5864
-
-
Kurth, M.J.1
Randall, L.A.A.2
Chen, C.3
Melander, C.4
Miller, R.B.5
-
15
-
-
0031040133
-
-
Obrecht, D., Abrecht, C., Grieder, A. et al. A novel and efficient approach for the combinatorial synthesis of structurally diverse pyrimidines on solid support. Helv Chim Acta 1997, 80: 65-72.
-
(1997)
A Novel and Efficient Approach for the Combinatorial Synthesis of Structurally Diverse Pyrimidines on Solid Support. Helv Chim Acta
, vol.80
, pp. 65-72
-
-
Obrecht, D.1
Abrecht, C.2
Grieder, A.3
-
16
-
-
0029883736
-
-
Kobayashi, S., Hachiya, I., Suzuki, S., Morowaki, M. Polymersupportedsilyl enol ethers. Synthesis and reactions with imines for the preparation of an amino alcohol library. Tetrahedron Lett 1996, 37:2809-12.
-
(1996)
Polymersupportedsilyl Enol Ethers. Synthesis and Reactions with Imines for the Preparation of An Amino Alcohol Library. Tetrahedron Lett
, vol.37
, pp. 2809-2812
-
-
Kobayashi, S.1
Hachiya, I.2
Suzuki, S.3
Morowaki, M.4
-
17
-
-
0030605818
-
-
Kobayashi, S., Hachiya, I., Yasuda, M. Aldol reaction on solid phase. Sc(OTf)3-catalyzed aldol reactions of polymer-supported silyl enol ethers with aldehydes. Tetrahedron Lett 1996, 37: 5569-72.
-
(1996)
Aldol Reaction on Solid Phase. Sc(OTf)3-catalyzed Aldol Reactions of Polymer-supported Silyl Enol Ethers with Aldehydes. Tetrahedron Lett
, vol.37
, pp. 5569-5572
-
-
Kobayashi, S.1
Hachiya, I.2
Yasuda, M.3
-
19
-
-
0031562046
-
-
Sylvain, C., Wagner, A., Mioskowski, C. Ozone: A versatile reagent for solid phase synthesis. Tetrahedron Lett 1997, 38: 1043-4.
-
(1997)
Ozone: a Versatile Reagent for Solid Phase Synthesis. Tetrahedron Lett
, vol.38
, pp. 1043-1044
-
-
Sylvain, C.1
Wagner, A.2
Mioskowski, C.3
-
21
-
-
3242702692
-
-
Ruhland, T., Kunzer, H. Structurally diverse 2,6-disubstituted quinoline derivatives by solid-phase synthesis. Tetrahedron Lett 1996,37:2757-60.
-
(1996)
Structurally Diverse 2,6-disubstituted Quinoline Derivatives by Solid-phase Synthesis. Tetrahedron Lett
, vol.37
, pp. 2757-2760
-
-
Ruhland, T.1
Kunzer, H.2
-
24
-
-
33947092534
-
-
Mitchell, A.R., Kent, S.B.H., Engelhard, M., Merrifield, R.B. A new synthetic route to tert-butyloxycarbonylaminoacyl-4-(oxymethyl)phenylacetamidomethyl-resin, an improved support for solidphase peptide synthesis. J Org Chem 1978, 43: 2845-52.
-
(1978)
A New Synthetic Route to Tert-butyloxycarbonylaminoacyl-4-(oxymethyl)phenylacetamidomethyl-resin, An Improved Support for Solidphase Peptide Synthesis. J Org Chem
, vol.43
, pp. 2845-2852
-
-
Mitchell, A.R.1
Kent, S.B.H.2
Engelhard, M.3
Merrifield, R.B.4
-
28
-
-
0030600160
-
-
Buckman, B.O., Mohan, R. Solid-phase synthesis of 1,3-dia/kyl quinazoline-2,4-diones. Tetrahedron Lett 1996, 37:4439-42.
-
(1996)
Solid-phase Synthesis of 1,3-dia/kyl Quinazoline-2,4-diones. Tetrahedron Lett
, vol.37
, pp. 4439-4442
-
-
Buckman, B.O.1
Mohan, R.2
-
30
-
-
0029918554
-
-
Barn, D.R., Morphy, J.R., Rees, D.C. Synthesis of an array of amides by aluminium chloride assisted cleavage of resin-bound esters. Tetrahedron Lett 1996, 37: 3213-6.
-
(1996)
Synthesis of An Array of Amides by Aluminium Chloride Assisted Cleavage of Resin-bound Esters. Tetrahedron Lett
, vol.37
, pp. 3213-3216
-
-
Barn, D.R.1
Morphy, J.R.2
Rees, D.C.3
-
31
-
-
0028053596
-
-
Yu, K.-L., Deshpande, M.S., Vyas, D.M. Heck reactions in solid phase synthesis. Tetrahedron Lett 1994, 35: 8919-22.
-
(1994)
Heck Reactions in Solid Phase Synthesis. Tetrahedron Lett
, vol.35
, pp. 8919-8922
-
-
Yu, K.-L.1
Deshpande, M.S.2
Vyas, D.M.3
-
32
-
-
0001644755
-
-
Guiles, J.W., Johnson, S.J., Murray, W.V. Solid-phase Suzuki coupling for C-C bond formation. J Org Chem 1996, 61: 5169-71.
-
(1996)
Solid-phase Suzuki Coupling for C-C Bond Formation. J Org Chem
, vol.61
, pp. 5169-5171
-
-
Guiles, J.W.1
Johnson, S.J.2
Murray, W.V.3
-
33
-
-
0030063277
-
-
Strocker, A.M., Keating, T.A., Tempest, P.A., Armstrong, R.W. Use of a convertible isocyanide for generation of Ugi reaction derivatives on solid support: Synthesis of a-acylaminoesters and pyrroles. Tetrahedron Lett 1996, 37:1149-52.
-
(1996)
Use of a Convertible Isocyanide for Generation of Ugi Reaction Derivatives on Solid Support: Synthesis of A-acylaminoesters and Pyrroles. Tetrahedron Lett
, vol.37
, pp. 1149-1152
-
-
Strocker, A.M.1
Keating, T.A.2
Tempest, P.A.3
Armstrong, R.W.4
-
34
-
-
0029940759
-
-
Mjalli, M., Sarshar, S., Baiga, T.J. Solid phase synthesis of pyrroles derived from a four component condensation. Tetrahedron Lett 1996, 37:2943-6.
-
(1996)
Solid Phase Synthesis of Pyrroles Derived from a Four Component Condensation. Tetrahedron Lett
, vol.37
, pp. 2943-2946
-
-
Mjalli, M.1
Sarshar, S.2
Baiga, T.J.3
-
35
-
-
0030059786
-
-
Zhang, C.Z., Moran, E.J., Woiwode, T.F., Short, K.M., Mjalli, MM.Synthesisoftetrasubstitutedimidazolesviaa-(N-acyl-N-alkylamino)-ß- ketoamides on Wang resin. Tetrahedron Lett 1996, 37: 751-4.
-
(1996)
Synthesisoftetrasubstitutedimidazolesviaa-(N-acyl-N-alkylamino)-ß- ketoamides on Wang Resin. Tetrahedron Lett
, vol.37
, pp. 751-754
-
-
Zhang, C.Z.1
Moran, E.J.2
Woiwode, T.F.3
Short, K.M.4
Mjalli, M.M.5
-
38
-
-
0141856793
-
-
MacDonald, A.A., DeWitt, S.H., Hogan, E.M., Ramage, R. A solid phase approach to quinolones using the Diversomer technology. Tetrahedron Lett 1996, 37: 4815-8.
-
(1996)
A Solid Phase Approach to Quinolones Using the Diversomer Technology. Tetrahedron Lett
, vol.37
, pp. 4815-4818
-
-
MacDonald, A.A.1
Dewitt, S.H.2
Hogan, E.M.3
Ramage, R.4
-
40
-
-
0030569368
-
-
Mayer, J. P., Zhang, J., Bjergarde, K. et al. Solid-phase synthesis of 1,4-benzodiazepine-2,5-diones. Tetrahedron Lett 1996, 37: 8081-4.
-
(1996)
Solid-phase Synthesis of 1,4-benzodiazepine-2,5-diones. Tetrahedron Lett
, vol.37
, pp. 8081-8084
-
-
Mayer, J.P.1
Zhang, J.2
Bjergarde, K.3
-
41
-
-
0029944026
-
-
Hamper, B.C., Dukesherer, D.R., South, M.S. Solid-phase synthesis of proline analogs via a three component 1,3-dipolar cycloaddition. Tetrahedron Lett 1996,37: 3671-4.
-
(1996)
Solid-phase Synthesis of Proline Analogs Via a Three Component 1,3-dipolar Cycloaddition. Tetrahedron Lett
, vol.37
, pp. 3671-3674
-
-
Hamper, B.C.1
Dukesherer, D.R.2
South, M.S.3
-
42
-
-
45549111520
-
-
Mergler, M., Tanner, R., Gosteli, J., Grogg, P. Peptide synthesis by a combination of solid-phase and solution methods. I: A new very acid-labile anchor group for the solid-phase synthesis of fully protected peptide fragments. Tetrahedron Lett 1988,29:4005-8.
-
(1988)
Peptide Synthesis by a Combination of Solid-phase and Solution Methods. I: a New Very Acid-labile Anchor Group for the Solid-phase Synthesis of Fully Protected Peptide Fragments. Tetrahedron Lett
, vol.29
, pp. 4005-4008
-
-
Mergler, M.1
Tanner, R.2
Gosteli, J.3
Grogg, P.4
-
44
-
-
0029042575
-
-
Murphy, M.M., Schullek, J.R., Gordon, E.M., Gallop, M.A. Combinatorial organic synthesis of highly functional/zed pyrrolidines: Identification of a potent angiotensin converting enzyme inhibitor from a mercaptoacyl proline library. J Am Chem Soc 1995, 117: 7029-30.
-
(1995)
Combinatorial Organic Synthesis of Highly Functional/zed Pyrrolidines: Identification of a Potent Angiotensin Converting Enzyme Inhibitor from a Mercaptoacyl Proline Library. J Am Chem Soc
, vol.117
, pp. 7029-7030
-
-
Murphy, M.M.1
Schullek, J.R.2
Gordon, E.M.3
Gallop, M.A.4
-
45
-
-
0030200397
-
-
Gordeev, M.F., Patel, D.V., Wu, J., Gordon, E.M. Approaches to combinatorial synthesis of heterocycles: Solid phase synthesis of pyridines and pyrido[2,3-d]pyrimidines. Tetrahedron Lett 1996, 36:4643-6.
-
(1996)
Approaches to Combinatorial Synthesis of Heterocycles: Solid Phase Synthesis of Pyridines and Pyrido[2,3-d]pyrimidines. Tetrahedron Lett
, vol.36
, pp. 4643-4646
-
-
Gordeev, M.F.1
Patel, D.V.2
Wu, J.3
Gordon, E.M.4
-
46
-
-
0031562439
-
-
Gordeev, M.F., Patel, D.V., Hui, H.C., Gordon, E.M. A general and efficient solid phase synthesis of quinazoline-2,4-diones. Tetrahedron Lett 1997, 38:1729-32.
-
(1997)
A General and Efficient Solid Phase Synthesis of Quinazoline-2,4-diones. Tetrahedron Lett
, vol.38
, pp. 1729-1732
-
-
Gordeev, M.F.1
Patel, D.V.2
Hui, H.C.3
Gordon, E.M.4
-
47
-
-
0031575621
-
-
Routledge, A., Abell, C., Balasubramanian, S. The use of a dithiane protected benzoin photolabile safety catch linker for solid-phase synthesis. Tetrahedron Lett 1997, 38:1227-30.
-
(1997)
The Use of a Dithiane Protected Benzoin Photolabile Safety Catch Linker for Solid-phase Synthesis. Tetrahedron Lett
, vol.38
, pp. 1227-1230
-
-
Routledge, A.1
Abell, C.2
Balasubramanian, S.3
-
48
-
-
37049077100
-
-
Akaji, K., Kiso, Y., Carpino, L.A. Fmoc-based solid-phase peptide synthesis using a new t-alcohol type 4-(r,r-dimethyl-1'hydmxypropyl)phenoxyacetyl handle (DHPP)-resin (Fmoc=9-fluorenyloxycarbonyl). J Chem Soc Chem Commun 1990, 584-6.
-
(1990)
Fmoc-based Solid-phase Peptide Synthesis Using a New T-alcohol Type 4-(r,r-dimethyl-1'hydmxypropyl)phenoxyacetyl Handle (DHPP)-resin (Fmoc=9-fluorenyloxycarbonyl). J Chem Soc Chem Commun
, pp. 584-586
-
-
Akaji, K.1
Kiso, Y.2
Carpino, L.A.3
-
49
-
-
0030975349
-
-
Blackburn, C., Pingali, A., Kehoe, T., Herman, L.W., Wang, H., Kates, S.A. Libraries of angiotensin converting enzyme inhibitors: Solid-phase synthesis and affinity selection. Biorg Med Chem Lett 1997,7:823-6.
-
(1997)
Libraries of Angiotensin Converting Enzyme Inhibitors: Solid-phase Synthesis and Affinity Selection. Biorg Med Chem Lett
, vol.7
, pp. 823-826
-
-
Blackburn, C.1
Pingali, A.2
Kehoe, T.3
Herman, L.W.4
Wang, H.5
Kates, S.A.6
-
52
-
-
0029891295
-
-
Mohan, R., Chou, Y.-L., Morrissey, M.M. Pictet-Spenglerreaction on solid support: Synthesis of 1,2,3,4-tetrahydro-ß-carboline libraries. Tetrahedron Lett 1996, 37: 3963-6.
-
(1996)
Pictet-Spenglerreaction on Solid Support: Synthesis of 1,2,3,4-tetrahydro-ß-carboline Libraries. Tetrahedron Lett
, vol.37
, pp. 3963-3966
-
-
Mohan, R.1
Chou, Y.-L.2
Morrissey, M.M.3
-
58
-
-
0029092629
-
-
Wang, G.T., Li, S., Wideburg, N., Krafft, G.A., Kempf, D.J. Synthetic chemical diversity: Solid phase synthesis of libraries of 2 symmetric inhibitors of HIV protease containing diaminodiol and diaminoalcohol cores. J Med Chem 1995, 38: 2995-3002.
-
(1995)
Synthetic Chemical Diversity: Solid Phase Synthesis of Libraries of 2 Symmetric Inhibitors of HIV Protease Containing Diaminodiol and Diaminoalcohol Cores. J Med Chem
, vol.38
, pp. 2995-3002
-
-
Wang, G.T.1
Li, S.2
Wideburg, N.3
Krafft, G.A.4
Kempf, D.J.5
-
59
-
-
0031575632
-
-
Yoo, S., Seo, J., Kyu-yang, Y., Gong, Y. Solid-phase synthesis ofbiphenyltetrazole derivatives. Tetrahedron Lett 1997,38:1203-6.
-
(1997)
Solid-phase Synthesis Ofbiphenyltetrazole Derivatives. Tetrahedron Lett
, vol.38
, pp. 1203-1206
-
-
Yoo, S.1
Seo, J.2
Kyu-yang, Y.3
Gong, Y.4
-
62
-
-
0031562077
-
-
Nefzi, A., Ostrech, J.M., Meyer. J.P., Houghten, R.A. Solidphase synthesis of heterocyclic compounds from linear peptides: Cyclic ureas and thioureas. Tetrahedron Lett 1997,38: 931-4.
-
(1997)
Solidphase Synthesis of Heterocyclic Compounds from Linear Peptides: Cyclic Ureas and Thioureas. Tetrahedron Lett
, vol.38
, pp. 931-934
-
-
Nefzi, A.1
Ostrech, J.M.2
Meyer, J.P.3
Houghten, R.A.4
-
63
-
-
0025032015
-
-
Albericio, F., Kneib-Cordonier, N., Biancalana, S. et al. Preparation and application of the 5-(4-(9-fluorenylmethoxycarbonyl)aminomethyl-3,5-dimethoxyphenoxy)- valericacid(PAL) handle forthe solid-phase synthesis of C-terminal peptide amides under mild conditions. J Org Chem 1990, 55: 3730-43.
-
(1990)
Preparation and Application of the 5-(4-(9-fluorenylmethoxycarbonyl)aminomethyl-3,5-dimethoxyphenoxy)- valericacid(PAL) Handle Forthe Solid-phase Synthesis of C-terminal Peptide Amides under Mild Conditions. J Org Chem
, vol.55
, pp. 3730-3743
-
-
Albericio, F.1
Kneib-Cordonier, N.2
Biancalana, S.3
-
64
-
-
0027279553
-
-
Kates, S.A., Daniels, S.B., Albericio, F. Automatedallyl cleavage for continuous-flow synthesis of cyclic and branched peptides. Anal Biochem 1993, 212: 303-10.
-
(1993)
Automatedallyl Cleavage for Continuous-flow Synthesis of Cyclic and Branched Peptides. Anal Biochem
, vol.212
, pp. 303-310
-
-
Kates, S.A.1
Daniels, S.B.2
Albericio, F.3
-
65
-
-
33745524373
-
-
Blackburn, C., Herman, L.W., Sole, N.A., Triolo, S.A., Kates, S.A. Reagents for solid-phase and small molecule combinatorial synthesis. So/id-phase synthesis: Developing small molecule libraries. (Feb 1-2, San Diego) 1996, Poster presentation.
-
(1996)
Reagents for Solid-phase and Small Molecule Combinatorial Synthesis. So/id-phase Synthesis: Developing Small Molecule Libraries. (Feb 1-2, San Diego)
-
-
Blackburn, C.1
Herman, L.W.2
Sole, N.A.3
Triolo, S.A.4
Kates, S.A.5
-
66
-
-
0007404508
-
-
Larhed, M., Lindeberg, G., Halberg, A. Rapid microwave-assisted Suzuki coup/ing on solid-phase. Tetrahedron Lett 1996,37: 8219-22.
-
(1996)
Rapid Microwave-assisted Suzuki Coup/ing on Solid-phase. Tetrahedron Lett
, vol.37
, pp. 8219-8222
-
-
Larhed, M.1
Lindeberg, G.2
Halberg, A.3
-
67
-
-
0000908874
-
-
Zuckermann, R.N., Kerr, Ü.M., Kent, S.B.H., Moos, W.H. Efficient method for the preparation of peptoids [oligofN-substituted glycines)] by submonomer solid-phase synthesis. J Am Chem Soc 1992,114:10646-7.
-
(1992)
Efficient Method for the Preparation of Peptoids [OligofN-substituted Glycines] by Submonomer Solid-phase Synthesis. J Am Chem Soc
, vol.114
, pp. 10646-10647
-
-
Zuckermann, R.N.1
Kerr, Ü.M.2
Kent, S.B.H.3
Moos, W.H.4
-
68
-
-
0028033882
-
-
Miller, S.M., Simon, R.J., Ng, S., Zuckerman, R.N., Kerr, J.M., Moos, W.H. Proteolyticstudies of homologouspeptide andN-substituted glycine peptoid oligomers. Bio Med Chem Lett 1994, 4: 2657-62.
-
(1994)
Proteolyticstudies of Homologouspeptide AndN-substituted Glycine Peptoid Oligomers. Bio Med Chem Lett
, vol.4
, pp. 2657-2662
-
-
Miller, S.M.1
Simon, R.J.2
Ng, S.3
Zuckerman, R.N.4
Kerr, J.M.5
Moos, W.H.6
-
73
-
-
15844401384
-
-
Kim, J.-M., Bi, Y., Paikoff, S.R., Schultz, P.G. The solid phase synthesis of oligoureas. Tetrahedron Lett 1996,37: 5305-8.
-
(1996)
The Solid Phase Synthesis of Oligoureas. Tetrahedron Lett
, vol.37
, pp. 5305-5308
-
-
Kim, J.-M.1
Bi, Y.2
Paikoff, S.R.3
Schultz, P.G.4
-
74
-
-
0030570917
-
-
Paikoff, S.J., Wilson, T.E., Cho, C.Y. et al. The solid-phase synthesis of N-alkylcarbamate oligomers. Tetrahedron Lett 1996,37: 5653-6.
-
(1996)
The Solid-phase Synthesis of N-alkylcarbamate Oligomers. Tetrahedron Lett
, vol.37
, pp. 5653-5656
-
-
Paikoff, S.J.1
Wilson, T.E.2
Cho, C.Y.3
-
77
-
-
0028850379
-
-
Cao, X., Moran, E.J., Siev, D., Lio, A., Ohasi, C., Mjalli, A.M.M. Synthesis of NH-acyl-a-aminoamldes on Rink resin: Inhibitors of the hematopoietic protein tyrosine phosphatase (HePTP). Bioorg Med Chem Lett 1995, 5: 2953-8.
-
(1995)
Synthesis of NH-acyl-a-aminoamldes on Rink Resin: Inhibitors of the Hematopoietic Protein Tyrosine Phosphatase (HePTP). Bioorg Med Chem Lett
, vol.5
, pp. 2953-2958
-
-
Cao, X.1
Moran, E.J.2
Siev, D.3
Lio, A.4
Ohasi, C.5
Mjalli, A.M.M.6
-
81
-
-
0030021771
-
-
Beaver, K.A., Siegmund, A.C., Spear, K.L. Application of the sulfonamide functional group as an anchor for solid phase organic synthesis. Tetrahedron Lett 1996, 37:1145-8.
-
(1996)
Application of the Sulfonamide Functional Group As An Anchor for Solid Phase Organic Synthesis. Tetrahedron Lett
, vol.37
, pp. 1145-1148
-
-
Beaver, K.A.1
Siegmund, A.C.2
Spear, K.L.3
-
83
-
-
0029812374
-
-
Han, Y, Bontems, S.L., Hegyes, P. et al. Preparation and applications ofxanthenylamide (XAL) handles for solid-phase synthesis of C-terminal peptide amides under particularly mild conditions. J Org Chem 1996, 61: 6326.
-
(1996)
Preparation and Applications Ofxanthenylamide (XAL) Handles for Solid-phase Synthesis of C-terminal Peptide Amides under Particularly Mild Conditions. J Org Chem
, vol.61
, pp. 6326
-
-
Han, Y.1
Bontems, S.L.2
Hegyes, P.3
-
86
-
-
0028109561
-
-
Pâtek, M., Drake, B., Lebl, M. All-cis cyclopentane scaffolding for combinatorial solid phase synthesis of small non-peptide compounds. Tetrahedron Lett 1994, 35: 9169-72.
-
(1994)
All-cis Cyclopentane Scaffolding for Combinatorial Solid Phase Synthesis of Small Non-peptide Compounds. Tetrahedron Lett
, vol.35
, pp. 9169-9172
-
-
Pâtek, M.1
Drake, B.2
Lebl, M.3
-
87
-
-
37049133408
-
-
Kenner, G.W., McDermott, J.R., Sheppard, R.C. The safety catch principle in solid-phase peptide synthesis. J Chem Soc Chem Commun 1971, 636-7.
-
(1971)
The Safety Catch Principle in Solid-phase Peptide Synthesis. J Chem Soc Chem Commun
, pp. 636-637
-
-
Kenner, G.W.1
McDermott, J.R.2
Sheppard, R.C.3
-
90
-
-
84985272116
-
-
Barlos, K., Gatos, D., Kallitsis, J., Papaioannou, D., Sotiriou, P. Anwendung von 4-polystyryltriphenylmethylchlorid zur synthese vonpeptiden und aminosäure-derivaten. Liebigs Ann Chem 1988, 1079-81.
-
(1988)
Anwendung Von 4-polystyryltriphenylmethylchlorid Zur Synthese Vonpeptiden und Aminosäure-derivaten. Liebigs Ann Chem
, pp. 1079-1081
-
-
Barlos, K.1
Gatos, D.2
Kallitsis, J.3
Papaioannou, D.4
Sotiriou, P.5
-
91
-
-
0000121634
-
-
Fyles, T.M., Leznoff, C.C., Weatherston, J. Bifunctionalizedresins. Applications to the synthesis of insect sex attractants. Can J Chem 1978, 56:1031-41.
-
(1978)
Bifunctionalizedresins. Applications to the Synthesis of Insect Sex Attractants. Can J Chem
, vol.56
, pp. 1031-1041
-
-
Fyles, T.M.1
Leznoff, C.C.2
Weatherston, J.3
-
92
-
-
3743084024
-
-
Chen, C., Randall, L.A.A., Miller, R.B., Jones, A.D., Kurth, M.J. "Analogous" organic synthesis ofsmall-compound libraries: Validation of combinatorial chemistry in small-molecule synthesis. JAm Chem Soc 1994;116:2661-2.
-
(1994)
"Analogous" Organic Synthesis Ofsmall-compound Libraries: Validation of Combinatorial Chemistry in Small-molecule Synthesis. JAm Chem Soc
, vol.116
, pp. 2661-2662
-
-
Chen, C.1
Randall, L.A.A.2
Miller, R.B.3
Jones, A.D.4
Kurth, M.J.5
-
93
-
-
37049078898
-
-
Egner, B.J., Cardno, N., Bradley, M. Linkers for combinatorial chemistry and reaction analysis using solid phase in situ mass spectrometry. J Chem Soc Chem Commun 1995, 2163-4.
-
(1995)
Linkers for Combinatorial Chemistry and Reaction Analysis Using Solid Phase in Situ Mass Spectrometry. J Chem Soc Chem Commun
, pp. 2163-2164
-
-
Egner, B.J.1
Cardno, N.2
Bradley, M.3
-
96
-
-
0030034999
-
-
Dressman, B.A., Spangle, L.A., Kaldor, S.W. Solid phase synthesis ofhydantolns using a carbamate linker and a novel cyclization/cleavage step. Tetrahedron Lett 1996, 37: 9337-40.
-
(1996)
Solid Phase Synthesis Ofhydantolns Using a Carbamate Linker and a Novel Cyclization/cleavage Step. Tetrahedron Lett
, vol.37
, pp. 9337-9340
-
-
Dressman, B.A.1
Spangle, L.A.2
Kaldor, S.W.3
-
97
-
-
0030599228
-
-
Gouilleux, L., Fehrentz, J.-A., Winternitz, F., Martinez, J. Solid phase synthesis of chiral3-substitutedquinazo/ine-2,4-diones. Tetrahedron Lett 1996, 37: 7031-4.
-
(1996)
Solid Phase Synthesis of Chiral3-substitutedquinazo/ine-2,4-diones. Tetrahedron Lett
, vol.37
, pp. 7031-7034
-
-
Gouilleux, L.1
Fehrentz, J.-A.2
Winternitz, F.3
Martinez, J.4
-
98
-
-
0029013332
-
-
Baldwin, J.J., Burbaum, J.J., Henderson, I., Ohtmeyer, M.H.J. Synthesis of a small molecule combinatorial library encoded with molecular tags. J Am Chem Soc 1995,117:5588-9.
-
(1995)
Synthesis of a Small Molecule Combinatorial Library Encoded with Molecular Tags. J Am Chem Soc
, vol.117
, pp. 5588-5589
-
-
Baldwin, J.J.1
Burbaum, J.J.2
Henderson, I.3
Ohtmeyer, M.H.J.4
-
99
-
-
0027104788
-
-
Beebe, X., Schore, N.E., Kurth, M.J. Polymer-supported syntheses of 2,5-disubstituted tetrahydrofurans. J Am Chem Soc 1992,114:10061-2.
-
(1992)
Polymer-supported Syntheses of 2,5-disubstituted Tetrahydrofurans. J Am Chem Soc
, vol.114
, pp. 10061-10062
-
-
Beebe, X.1
Schore, N.E.2
Kurth, M.J.3
-
100
-
-
0002469361
-
-
Jensen, K.J., Songster, M.F., Vágner, J., Alsina, J., Albericio, F., Barany, G. A novel handle approach for solid phase peptide synthesis: Backbone amide linker (BAL) anchoring. In: Peptides Chemistry and Biology. Proceedings of the Fourteenth American Peptide Symposium. Kaumaya, P.T.P., Hodges, R.S. (Eds.). Mayflower Worldwide Ltd.: Birmingham 1996, 30-2.
-
(1996)
A Novel Handle Approach for Solid Phase Peptide Synthesis: Backbone Amide Linker (BAL) Anchoring. In: Peptides Chemistry and Biology. Proceedings of the Fourteenth American Peptide Symposium. Kaumaya, P.T.P., Hodges, R.S. (Eds.). Mayflower Worldwide Ltd.: Birmingham
, pp. 30-32
-
-
Jensen, K.J.1
Songster, M.F.2
Vágner, J.3
Alsina, J.4
Albericio, F.5
Barany, G.6
-
101
-
-
0029128552
-
-
Boojamra, C.G., Burow, K., Ellman, J.A. An expedient and high-yielding method for the solid-phase synthesis of diverse 1,4-benzodiazepine-2,5-diones. J Org Chem 1995, 60: 5742-3.
-
(1995)
An Expedient and High-yielding Method for the Solid-phase Synthesis of Diverse 1,4-benzodiazepine-2,5-diones. J Org Chem
, vol.60
, pp. 5742-5743
-
-
Boojamra, C.G.1
Burow, K.2
Ellman, J.A.3
-
102
-
-
0031575637
-
-
Gray, N.S., Kwon, S., Schultz, P.G. Combinatorial synthesis of 2,9-substitutedpurines. Tetrahedron Lett 1997, 38:1161-4.
-
(1997)
Combinatorial Synthesis of 2,9-substitutedpurines. Tetrahedron Lett
, vol.38
, pp. 1161-1164
-
-
Gray, N.S.1
Kwon, S.2
Schultz, P.G.3
-
104
-
-
0029361890
-
-
Meyers, H.V., Diiley, G.J., Durgin, T.L. et al. Multiple simultaneous synthesis of phenolic libraries. Mol Diversity 1995,1:13-20.
-
(1995)
Multiple Simultaneous Synthesis of Phenolic Libraries. Mol Diversity
, vol.1
, pp. 13-20
-
-
Meyers, H.V.1
Diiley, G.J.2
Durgin, T.L.3
-
105
-
-
0030569267
-
-
Panek, J.S., Zhu; B. Synthesis of aromatic 1,2-diazines by inverse electron demand Diels-Alder reaction of polymer-supported 1,2,4,5-triazines. Tetrahedron Lett 1996, 37: 8151-4.
-
(1996)
Synthesis of Aromatic 1,2-diazines by Inverse Electron Demand Diels-Alder Reaction of Polymer-supported 1,2,4,5-triazines. Tetrahedron Lett
, vol.37
, pp. 8151-8154
-
-
Panek, J.S.1
Zhu, B.2
-
106
-
-
0029991217
-
-
Morphy, J.R., Rankovic, Z., Rees, D.C. A novel strategy for solid-phase synthesis. Tetrahedron Lett 1996, 37: 3209-12.
-
(1996)
A Novel Strategy for Solid-phase Synthesis. Tetrahedron Lett
, vol.37
, pp. 3209-3212
-
-
Morphy, J.R.1
Rankovic, Z.2
Rees, D.C.3
-
107
-
-
0013249477
-
-
Chenera, B., Finkelstein, J.A., Veber, D.F. Protodetachable arylsilane polymer linkages for use in solid phase organic synthesis. J Am Chem Soc 1995,117:11999-2000.
-
(1995)
Protodetachable Arylsilane Polymer Linkages for Use in Solid Phase Organic Synthesis. J Am Chem Soc
, vol.117
, pp. 11999-12000
-
-
Chenera, B.1
Finkelstein, J.A.2
Veber, D.F.3
-
110
-
-
0029865824
-
-
Han, Y., Walker, S.D., Young, R.N. Silicon directed ipso-substitution ol'polymer-bound'arylsilanes: Preparation ofbiaryls via the Suzuki cross-coupling reaction. Tetrahedron Lett 1996,37:2703-6.
-
(1996)
Silicon Directed Ipso-substitution Ol'polymer-bound'arylsilanes: Preparation Ofbiaryls Via the Suzuki Cross-coupling Reaction. Tetrahedron Lett
, vol.37
, pp. 2703-2706
-
-
Han, Y.1
Walker, S.D.2
Young, R.N.3
-
111
-
-
0030607141
-
-
Kaldor, S.W., Siegel, M.G., Fritz, J.E., Dressman, B.A., Hahn, P.J. Use of solid supported nucleophiles and electrophiles for the purification of non-peptide small molecule libraries. Tetrahedron Lett 1996, 37:7193-6.
-
(1996)
Use of Solid Supported Nucleophiles and Electrophiles for the Purification of Non-peptide Small Molecule Libraries. Tetrahedron Lett
, vol.37
, pp. 7193-7196
-
-
Kaldor, S.W.1
Siegel, M.G.2
Fritz, J.E.3
Dressman, B.A.4
Hahn, P.J.5
-
112
-
-
0027500111
-
-
Lebl, M., Pâtek, M., Kocis, P. et al. Multiple release ofequimolar amounts ofpeptides from a polymeric carrier using orthogonal linkage-cleavage chemistry. Int J Pept Protein Res 1993,41:201-3.
-
(1993)
Multiple Release Ofequimolar Amounts Ofpeptides from a Polymeric Carrier Using Orthogonal Linkage-cleavage Chemistry. Int J Pept Protein Res
, vol.41
, pp. 201-203
-
-
Lebl, M.1
Pâtek, M.2
Kocis, P.3
-
113
-
-
0027367140
-
-
Kocis, P., Krchnak, V., Lebl, M. Symmetrical structure allowing the selective multiple release of a defined quantity ofpeptide from a single bead of polymeric support. Tetrahedron Lett 1993, 34: 7251-2.
-
(1993)
Symmetrical Structure Allowing the Selective Multiple Release of a Defined Quantity Ofpeptide from a Single Bead of Polymeric Support. Tetrahedron Lett
, vol.34
, pp. 7251-7252
-
-
Kocis, P.1
Krchnak, V.2
Lebl, M.3
-
114
-
-
0027142990
-
-
Salmon, S.E., Lam, K.S., Lebl, M. et al. Discovery ol biologically active peptides in random libraries: Solution-phase testing after staged orthogonal release from resin beads. Proc Natl Acad Sei USA 1993, 90:11708-12.
-
(1993)
Discovery Ol Biologically Active Peptides in Random Libraries: Solution-phase Testing after Staged Orthogonal Release from Resin Beads. Proc Natl Acad Sei USA
, vol.90
, pp. 11708-11712
-
-
Salmon, S.E.1
Lam, K.S.2
Lebl, M.3
-
115
-
-
0030603050
-
-
Seneci, P., Sizemore, C., Islam, K., Kocis, P. Combinatorial chemistry and natural products. Teicoplanin aglycone as a molecular scaffold for solid phase synthesis of combinatorial libraries. Tetrahedron Lett 1996, 37: 6319-22.
-
(1996)
Combinatorial Chemistry and Natural Products. Teicoplanin Aglycone As a Molecular Scaffold for Solid Phase Synthesis of Combinatorial Libraries. Tetrahedron Lett
, vol.37
, pp. 6319-6322
-
-
Seneci, P.1
Sizemore, C.2
Islam, K.3
Kocis, P.4
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