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0028243847
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85047670016
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For example, see: Bray, A. M.; Chiefari, D. S.; Valerio, R. M.; Maeji, N. J. Tetrahedron Lett. 1995, 35, 5081.
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0342285879
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Patent Fr. 1,384,209 Jan. 4
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(a) 2-Pyridylisocyanide: Ugi, I.; Fetzer, U.; Unterstenhoefer, G.; Behrenz, W.; Frohberger, P. E.; Scheinpflug, H. Patent Fr. 1,384,209 Jan. 4, 1965; Chem. Abstr. 1965, 63, 6924e.
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Scheinpflug, H.6
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17
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84917967252
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(a) 2-Pyridylisocyanide: Ugi, I.; Fetzer, U.; Unterstenhoefer, G.; Behrenz, W.; Frohberger, P. E.; Scheinpflug, H. Patent Fr. 1,384,209 Jan. 4, 1965; Chem. Abstr. 1965, 63, 6924e.
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18
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0001223891
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(b) Phenylisocyanide: Walborsky, H. M.; Ronman, P. J. Org. Chem. 1978, 43, 731. Both isocyanides are prepared in one step from commercially available formamides.
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Walborsky, H.M.1
Ronman, P.2
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19
-
-
85030188681
-
-
note
-
Calculation based upon commercially available 1° amines, aldehydes, carboxylic acids and alkynes contained in the ACD database, MDL Information Systems. Traditionally, N-acyl-N-alkyl-a-amino amides have been prepared on solid suport via reductive amination of an a-amino acid with an aldehyde followed by acylation of the resulting 2° amine. Since a limited number of a-amino acids are commercially available, this approach drastically reduces the final library size.
-
-
-
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25
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33845551642
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and references therein
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Flynn, D. L.; Zelle, R. E.; Grieco, P. A. J. Org. Chem. 1983, 48, 2424, and references therein.
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Flynn, D.L.1
Zelle, R.E.2
Grieco, P.A.3
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26
-
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85030189246
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-
note
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2NH. These results as well as subsequent functional transformations of these intermediates will be reported shortly.
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-
-
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28
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0011267872
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(a) Knorr, R.; Trzeciak, A.; Bannwarth, W.; Gillessen, D. Tetrahedron Lett. 1987, 30, 1927.
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Knorr, R.1
Trzeciak, A.2
Bannwarth, W.3
Gillessen, D.4
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30
-
-
85030197643
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-
note
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13C NMR and high resolution MS.
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