A General and Expedient Method for the Solid-Phase Synthesis of Structurally Diverse 1-Phenylpyrazolone Derivatives

Synlett

Volumn 1996, Issue 7, 1996, Pages 667-668

  Tietze, Lutz F ^a   Steinmetz, Adrian ^a  

^a UNIVERSITY OF GÖTTINGEN   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0001791986     PISSN: 09365214     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-1996-5548     Document Type: Article

References (27)

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16. Selected new publications on combinatorial chemistry: a) Ley, S. V.; Mynett, D. M.; Koot, W.-J. Synlett 1995, 1017-1020. b) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937-940. c) Marzinzik, A. L.; Felder, E. R. Tetrahedron Lett. 1996, 37, 1003-1006. d) Zhang, C.; Moran, E. J.; Woiwode, T. F.; Short, K. M.; Mjalli, A. M. M. Tetrahedron Lett. 1996, 37, 751-754.
17. Selected new publications on combinatorial chemistry: a) Ley, S. V.; Mynett, D. M.; Koot, W.-J. Synlett 1995, 1017-1020. b) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937-940. c) Marzinzik, A. L.; Felder, E. R. Tetrahedron Lett. 1996, 37, 1003-1006. d) Zhang, C.; Moran, E. J.; Woiwode, T. F.; Short, K. M.; Mjalli, A. M. M. Tetrahedron Lett. 1996, 37, 751-754.
18. Selected new publications on combinatorial chemistry: a) Ley, S. V.; Mynett, D. M.; Koot, W.-J. Synlett 1995, 1017-1020. b) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937-940. c) Marzinzik, A. L.; Felder, E. R. Tetrahedron Lett. 1996, 37, 1003-1006. d) Zhang, C.; Moran, E. J.; Woiwode, T. F.; Short, K. M.; Mjalli, A. M. M. Tetrahedron Lett. 1996, 37, 751-754.
19. Selected new publications on combinatorial chemistry: a) Ley, S. V.; Mynett, D. M.; Koot, W.-J. Synlett 1995, 1017-1020. b) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937-940. c) Marzinzik, A. L.; Felder, E. R. Tetrahedron Lett. 1996, 37, 1003-1006. d) Zhang, C.; Moran, E. J.; Woiwode, T. F.; Short, K. M.; Mjalli, A. M. M. Tetrahedron Lett. 1996, 37, 751-754.
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22. Polymer-bound Li-enolates: a) Backes, B. J.; Ellman, J. A. J. Am. Chem. Soc. 1994, 116, 11171-11172. b) Moon, H. S.; Schore, N. E.; Kurth, M. J. Tetrahedron Lett. 1994, 35, 8915-8918. c) Moon, H. S.; Schore, N. E.; Kurth, M. J. J. Org. Chem. 1992, 57, 6088-6089. d) Worste, P. M.; McArthur, C. R.; Leznoff, C. C. Angew. Chem. 1979, 91, 255; Angew. Chem. Int. Ed. Engl. 1979, 18, 221-222.
23. Polymer-bound Li-enolates: a) Backes, B. J.; Ellman, J. A. J. Am. Chem. Soc. 1994, 116, 11171-11172. b) Moon, H. S.; Schore, N. E.; Kurth, M. J. Tetrahedron Lett. 1994, 35, 8915-8918. c) Moon, H. S.; Schore, N. E.; Kurth, M. J. J. Org. Chem. 1992, 57, 6088-6089. d) Worste, P. M.; McArthur, C. R.; Leznoff, C. C. Angew. Chem. 1979, 91, 255; Angew. Chem. Int. Ed. Engl. 1979, 18, 221-222.
24. Polymer-bound Li-enolates: a) Backes, B. J.; Ellman, J. A. J. Am. Chem. Soc. 1994, 116, 11171-11172. b) Moon, H. S.; Schore, N. E.; Kurth, M. J. Tetrahedron Lett. 1994, 35, 8915-8918. c) Moon, H. S.; Schore, N. E.; Kurth, M. J. J. Org. Chem. 1992, 57, 6088-6089. d) Worste, P. M.; McArthur, C. R.; Leznoff, C. C. Angew. Chem. 1979, 91, 255; Angew. Chem. Int. Ed. Engl. 1979, 18, 221-222.
25. Polymer-bound Li-enolates: a) Backes, B. J.; Ellman, J. A. J. Am. Chem. Soc. 1994, 116, 11171-11172. b) Moon, H. S.; Schore, N. E.; Kurth, M. J. Tetrahedron Lett. 1994, 35, 8915-8918. c) Moon, H. S.; Schore, N. E.; Kurth, M. J. J. Org. Chem. 1992, 57, 6088-6089. d) Worste, P. M.; McArthur, C. R.; Leznoff, C. C. Angew. Chem. 1979, 91, 255; Angew. Chem. Int. Ed. Engl. 1979, 18, 221-222.
26. Huckin, S. N.; Weiler, L. J. Am. Chem. Soc. 1974, 96, 1082-1087.
27. All compounds were completely characterized.