-
1
-
-
2042437650
-
-
E. S. Lander, L. M. Linton, B. Birren, C. Nusbaum, M. C. Zody,Baldwin, K. Devon, K. Dewar, M. Doyle, W. Fitz-Hugh et al., Nature 2001, 409, 860-921.
-
(2001)
Nature
, vol.409
, pp. 860-921
-
-
Lander, E.S.1
Linton, L.M.2
Birren, B.3
Nusbaum, C.4
Zody, M.C.5
Baldwin, J.6
Devon, K.7
Dewar, K.8
Doyle, M.9
Fitz-Hugh, W.10
-
2
-
-
0035895505
-
-
J. C. Venter, M. D. Adams, E. W. Myers, P. W. Li, R. J. Mural, G. G. Sutton, H. O. Smith, M. Yandell, C. A. Evans, R. A. Holt et al., Science 2001, 291, 1304-1341.
-
(2001)
Science
, vol.291
, pp. 1304-1341
-
-
Venter, J.C.1
Adams, M.D.2
Myers, E.W.3
Li, P.W.4
Mural, R.J.5
Sutton, G.G.6
Smith, H.O.7
Yandell, M.8
Evans, C.A.9
Holt, R.A.10
-
9
-
-
0037032835
-
-
G. Manning, D. B. Whyte, R. Martinez, T. Hunter, S. Sudar-sanam, Science 2002, 298, 1912-1934.
-
(2002)
Science
, vol.298
, pp. 1912-1934
-
-
Manning, G.1
Whyte, D.B.2
Martinez, R.3
Hunter, T.4
Sudar-sanam, S.5
-
10
-
-
0034788453
-
-
P. Traxler, G. Bold, E. Buchdunger, G. Caravatti, P. Furet, P. Manley, T. O'Reilly,J. Wood,J. Zimmermann, Med. Res. Rev. 2001, 21, 499-512.
-
(2001)
Med. Res. Rev.
, vol.21
, pp. 499-512
-
-
Traxler, P.1
Bold, G.2
Buchdunger, E.3
Caravatti, G.4
Furet, P.5
Manley, P.6
O'Reilly, T.7
Wood, J.8
Zimmermann, J.9
-
12
-
-
0035990893
-
-
D. Fabbro, S. Ruetz, E. Buchdunger, S. W. Cowan-Jacob, G. Fendrich, J. Liebetanz,J. Mestan, T. O'Reilly, P. Traxler, B. Chaudhuri, H. Fretz, J. Zimmermann, T. Meyer, G. Caravatti, P. Furet, P. W. Manley, Pharm. Thera- peutics 2002, 93, 79-98.
-
(2002)
Pharm. Thera- peutics
, vol.93
, pp. 79-98
-
-
Fabbro, D.1
Ruetz, S.2
Buchdunger, E.3
Cowan-Jacob, S.W.4
Fendrich, G.5
Liebetanz, J.6
Mestan, J.7
O'Reilly, T.8
Traxler, P.9
Chaudhuri, B.10
Fretz, H.11
Zimmermann, J.12
Meyer, T.13
Caravatti, G.14
Furet, P.15
Manley, P.W.16
-
13
-
-
0036635291
-
-
R. Capdeville, E. Buchdunger, J. Zimmermann, A. Matter, Nat. Rev.Drug Discov. 2002, 1, 493-502.
-
(2002)
Nat. Rev.Drug Discov.
, vol.1
, pp. 493-502
-
-
Capdeville, R.1
Buchdunger, E.2
Zimmermann, J.3
Matter, A.4
-
14
-
-
0038678969
-
-
M. Mushin,J. Graham, P. Kirkpatrick, Nat. Rev. Drug Discov. 2003, 2, 515-516.
-
(2003)
Nat. Rev. Drug Discov.
, vol.2
, pp. 515-516
-
-
Mushin, M.1
Graham, J.2
Kirkpatrick, P.3
-
15
-
-
1642401467
-
-
G. M. Mine, Annu. Rep. Med. Chem.2003, 38, 383-396 (see also http://www.phrma.org/).
-
(2003)
Annu. Rep. Med. Chem
, vol.38
, pp. 383-396
-
-
Mine, G.M.1
-
19
-
-
0028605318
-
-
J. C. Lee,J. T. Laydon, P. C. McDonnell, T. F. Gallagher, S. Kumar, D. Green, D. McNulty, M. J. Blumenthal,J. R. Keys, S. WLa. ndvatter,J. E. Strickler, M. M. McLaughlin,I. R. Siemens, S. M. Fisher, G. P. Livi,J. R. White, J. L. Adams, P. R. Young, Nature 1994, 372, 739-746.
-
(1994)
Nature
, vol.372
, pp. 739-746
-
-
Lee, J.C.1
Laydon, J.T.2
McDonnell, P.C.3
Gallagher, T.F.4
Kumar, S.5
Green, D.6
McNulty, D.7
Blumenthal, M.J.8
Keys, J.R.9
WLandvatter, S.10
Strickler, J.E.11
McLaughlin, M.M.12
Siemens, I.R.13
Fisher, S.M.14
Livi, G.P.15
White, J.R.16
Adams, J.L.17
Young, P.R.18
-
22
-
-
0034616930
-
-
T. R. Hughes, M. J. Marton, A. R. Jones, C. J. Roberts, R. Stoughton, C. D. Armour, H. A. Bennett, E. Coffey, H. Dai, Y. D. He, M. J. Kidd, A. M. King, M. R. Meyer, D. Slade, P. Y. Lum, S. B. Stepaniants, D. D. Shoemaker, D. Gachotte, K. Chakraburtty, J. Simon, M. Bard, S. H. Friend, Cell 2000, 102, 109-126.
-
(2000)
Cell
, vol.102
, pp. 109-126
-
-
Hughes, T.R.1
Marton, M.J.2
Jones, A.R.3
Roberts, C.J.4
Stoughton, R.5
Armour, C.D.6
Bennett, H.A.7
Coffey, E.8
Dai, H.9
He, Y.10
Kidd, D.M.J.11
King, A.M.12
Meyer, M.R.13
Slade, D.14
Lum, P.Y.15
Stepaniants, S.B.16
Shoemaker, D.D.17
Gachotte, D.18
Chakraburtty, K.19
Simon, J.20
Bard, M.21
Friend, S.H.22
more..
-
23
-
-
0032563315
-
-
N. S. Gray, L. Wodicka, A. M. Thunnissen, T. C. Norman, S. Kwon, F. H. Espinoza, D. O. Morgan, G. Barnes, S. LeClerc, L. Meijer, S. H. Kim, D. J. Lockhart, P. G. Schultz, Science 1998, 281, 533-538.
-
(1998)
Science
, vol.281
, pp. 533-538
-
-
Gray, N.S.1
Wodicka, L.2
Thunnissen, A.M.3
Norman, T.C.4
Kwon, S.5
Espinoza, F.H.6
Morgan, D.O.7
Barnes, G.8
LeClerc, S.9
Meijer, L.10
Kim, S.H.11
Lockhart, D.J.12
Schultz, P.G.13
-
24
-
-
0033592983
-
-
J. S. Hardwick, F. G. Kuruvilla, J. K. Tong, A. F. Shamji, S. L. Schreiber, Proc. Natl. Acad. Sci.USA 1999, 96, 14866-14870.
-
(1999)
Proc. Natl. Acad. Sci.USA
, vol.96
, pp. 14866-14870
-
-
Hardwick, J.S.1
Kuruvilla, F.G.2
Tong, J.K.3
Shamji, A.F.4
Schreiber, S.L.5
-
25
-
-
0034649569
-
-
A. F. Shamji, F. G. Kuruvilla, S. L. Schreiber, Curr. Biol. 2000, 10, 1574-1581.
-
(2000)
Curr. Biol.
, vol.10
, pp. 1574-1581
-
-
Shamji, A.F.1
Kuruvilla, F.G.2
Schreiber, S.L.3
-
26
-
-
0035671295
-
-
N. Custodia, S. J. Won, A. Novillo, M. Wieland, C. Li,I. P. Callard, Ann. N Y Acad. Sci. 2001, 948, 32-42.
-
(2001)
Ann. N Y Acad. Sci.
, vol.948
, pp. 32-42
-
-
Custodia, N.1
Won, S.J.2
Novillo, A.3
Wieland, M.4
Li, C.5
Callard, I.P.6
-
27
-
-
0037967631
-
-
G. Le Goff, S. Boundy, P. J. Daborn, J. L. Yen, L. Sofer, R. Lind, C. Sabourault, L. Madi-Ravazzi, R. H. ffrench Constant,Insect Biochem. Mol. Biol. 2003, 33, 701-708.
-
(2003)
Insect Biochem. Mol. Biol.
, vol.33
, pp. 701-708
-
-
Le Goff, G.1
Boundy, S.2
Daborn, P.J.3
Yen, J.L.4
Sofer, L.5
Lind, R.6
Sabourault, C.7
Madi-Ravazzi, L.8
Ffrench Constant, R.H.9
-
28
-
-
0344010927
-
-
P. R. Hoyt, M. J. Doktycz, K. L. Beattie, M. S. Greeley Jr., Ecotoxicology 2003, 12, 469-474.
-
(2003)
Ecotoxicology
, vol.12
, pp. 469-474
-
-
Hoyt, P.R.1
Doktycz, M.J.2
Beattie, K.L.3
Greeley, M.S.4
-
29
-
-
0035816183
-
-
F. W. Frueh, K. C. Hayashibara, P. O. Brown, J. P. Whitlock Jr., Toxicol.Lett. 2001, 122, 189-203.
-
(2001)
Toxicol.Lett.
, vol.122
, pp. 189-203
-
-
Frueh, F.W.1
Hayashibara, K.C.2
Brown, P.O.3
Whitlock, J.P.4
-
31
-
-
0038273551
-
-
L. J. Browne, L. M. Furness, G. Natsoulis, C. Pearson, K. Jarnagin, Targets 2002, 1, 59-65.
-
(2002)
Targets
, vol.1
, pp. 59-65
-
-
Browne, L.J.1
Furness, L.M.2
Natsoulis, G.3
Pearson, C.4
Jarnagin, K.5
-
32
-
-
0035845531
-
-
J. E. Staunton, D. K. Slonim, H. A. Coller, P. Tamayo, M. J. Angelo, J. Park, U. Scherf,J. K. Lee, W. O. Reinhold,J. N. Weinstein, J. P. Mesirov, E. S. Lander, T. R. Golub, Proc. Natl. Acad. Sci. USA 2001, 98, 10787-10792.
-
(2001)
Proc. Natl. Acad. Sci. USA
, vol.98
, pp. 10787-10792
-
-
Staunton, J.E.1
Slonim, D.K.2
Coller, H.A.3
Tamayo, P.4
Angelo, M.J5
Park, J.6
Scherf, U.7
Lee, J.K.8
Reinhold, W.O.9
Weinstein, J.N.10
Mesirov, J.P.11
Lander, E.S.12
Golub, T.R.13
-
34
-
-
0033874150
-
-
A. C. Bishop, O. Buzko, S. Heyeck-Dumas, I. Jung, B. Kraybill, Y. Liu, K. Shah, S. Ulrich, L. Witucki, F. Yang, C. Zhang, K. M. Shokat, Annu. Rev. Biophys. Biomol. Struct. 2000, 29, 577-606.
-
(2000)
Annu. Rev. Biophys. Biomol. Struct.
, vol.29
, pp. 577-606
-
-
Bishop, A.C.1
Buzko, O.2
Heyeck-Dumas, S.3
Jung, I.4
Kraybill, B.5
Liu, Y.6
Shah, K.7
Ulrich, S.8
Witucki, L.9
Yang, F.10
Zhang, C.11
Shokat, K.M.12
-
37
-
-
0035312350
-
-
A. C. Bishop, O. Buzko, K. M. Shokat, Trends Cell Biol. 2001, 11, 167-172.
-
(2001)
Trends Cell Biol.
, vol.11
, pp. 167-172
-
-
Bishop, A.C.1
Buzko, O.2
Shokat, K.M.3
-
38
-
-
0034699382
-
-
A. C. Bishop, J. A. Ubersax, D. T. Petsch, D. P. Matheos, N. S. Gray,J. Blethrow, E. Shimizu,J. Z. Tsien, P. G. Schultz, M. D. Rose,J. L. Wood, D. O. Morgan, K. M. Shokat, Nature 2000, 407, 395-401.
-
(2000)
Nature
, vol.407
, pp. 395-401
-
-
Bishop, A.C.1
Ubersax, J.A.2
Petsch, D.T.3
Matheos, D.P.4
Gray, N.S.5
Blethrow, J.6
Shimizu, E.7
Tsien, J.Z.8
Schultz, P.G.9
Rose, M.D.10
Wood, J.L.11
Morgan, D.O.12
Shokat, K.M.13
-
39
-
-
0035947671
-
-
H. Habelhah, K. Shah, L. Huang, A. L. Burlingame, K. M. Shokat, Z. Ronai, J. Biol. Chem. 2001, 276, 18090-18095.
-
(2001)
J. Biol. Chem.
, vol.276
, pp. 18090-18095
-
-
Habelhah, H.1
Shah, K.2
Huang, L.3
Burlingame, A.L.4
Shokat, K.M.5
Ronai, Z.6
-
41
-
-
0242300176
-
-
J. A. Ubersax, E. L. Woodbury, P. N. Quang, M. Paraz,J. D. Blethrow, K. Shah, K. M. Shokat, D. O. Morgat, Nature 2003, 425, 859-864.
-
(2003)
Nature
, vol.425
, pp. 859-864
-
-
Ubersax, J.A.1
Woodbury, E.L.2
Quang, P.N.3
Paraz, M.4
Blethrow, J.D.5
Shah, K.6
Shokat, K.M.7
Morgat, D.O.8
-
42
-
-
0038351827
-
-
S. T. Eblen, N. V. Kumar, K. Shah, M. J. Henderson, C. K. W. Watts, K. M. Shokat, M. J. Weber, J. Biol.Chem. 2003, 278, 14926-14935.
-
(2003)
J. Biol.Chem.
, vol.278
, pp. 14926-14935
-
-
Eblen, S.T.1
Kumar, N.V.2
Shah, K.3
Henderson, M.J.4
Watts, C.K.W.5
Shokat, K.M.6
Weber, M.J.7
-
43
-
-
0035940479
-
-
A. S. Carroll, A. C. Bishop, J. L. DeRisi, K. M. Shokat, E. K. O'Shea, Proc. Natl. Acad. Sci. USA 2001, 98, 12578-12583.
-
(2001)
Proc. Natl. Acad. Sci. USA
, vol.98
, pp. 12578-12583
-
-
Carroll, A.S.1
Bishop, A.C.2
DeRisi, J.L.3
Shokat, K.M.4
O'Shea, E.K.5
-
44
-
-
0142026209
-
-
S. Kumar, J. Boehm, J. C. Lee, Nat. Rev.Drug Discovery 2003, 2, 717-726.
-
(2003)
Nat. Rev.Drug Discovery
, vol.2
, pp. 717-726
-
-
Kumar, S.1
Boehm, J.2
Lee, J.C.3
-
45
-
-
12644277392
-
-
K. P. Wilson, P. G. McCaffrey, K. Hsiao, S. Pazhanisamy, V. Galullo, G. W. Bemis, M. J. Fitzgibbon, P. R. Caron, M. A. Murcko, M. S. S. Su, Chem. Biol. 1997, 4, 423-431.
-
(1997)
Chem. Biol.
, vol.4
, pp. 423-431
-
-
Wilson, K.P.1
McCaffrey, P.G.2
Hsiao, K.3
Pazhanisamy, S.4
Galullo, V.5
Bemis, G.W.6
Fitzgibbon, M.J.7
Caron, P.R.8
Murcko, M.A.9
Su, M.S.S.10
-
46
-
-
0030954172
-
-
L. Tong, S. Pav, D. M. White, S. Rogers, K. M. Crane, C. L. Cywin, M. L. Brown, C. A. Pargellis, Nat. Struct. Biol. 1997, 4, 311-316.
-
(1997)
Nat. Struct. Biol.
, vol.4
, pp. 311-316
-
-
Tong, L.1
Pav, S.2
White, D.M.3
Rogers, S.4
Crane, K.M.5
Cywin, C.L.6
Brown, M.L.7
Pargellis, C.A.8
-
47
-
-
0032102902
-
-
P. A. Eyers, M. Craxton, N. Morrice, P. Cohen, M. Goedert, Chem. Biol.1998, 5, 321-328.
-
(1998)
Chem. Biol.
, vol.5
, pp. 321-328
-
-
Eyers, P.A.1
Craxton, M.2
Morrice, N.3
Cohen, P.4
Goedert, M.5
-
48
-
-
10744227768
-
-
R. J. Gum, M. M. McLaughlin, S. Kumar, Z. Wang, M. J. Bower, J. C. Lee,J. L. Adams, G. P. Livi, E. J. Goldsmith, P. R. Young,J. Biol.Chem. 1998, 273, 15605-15610.
-
(1998)
J. Biol.Chem.
, vol.273
, pp. 15605-15610
-
-
Gum, R.J.1
McLaughlin, M.M.2
Kumar, S.3
Wang, Z.4
Bower, M.J.5
Lee, J.C.6
Adams, J.L.7
Livi, G.P.8
Goldsmith, E.J.9
Young, P.R.10
-
49
-
-
0031793432
-
-
T. Fox, J. T. Coll, X. Xie, P. J. Ford, U. A. Germann, M. D. Porter, S. Pahzanisamy, M. A. Fleming, V. Galullo, M. S. S. Su, K. P. Wilson, Protein Sci. 1998, 7, 2249-2255.
-
(1998)
Protein Sci.
, vol.7
, pp. 2249-2255
-
-
Fox, T.1
Coll, J.T.2
Xie, X.3
Ford, P.J.4
Germann, U.A.5
Porter, M.D.6
Pahzanisamy, S.7
Fleming, M.A.8
Galullo, V.9
Su, M.S.S.10
Wilson, K.P.11
-
50
-
-
0032901378
-
-
P. A. Eyers, P. van den Ijssel, R. A. Quinlan, M. Goedert, P. Cohen, FEBS Letters 1999, 451, 191-196.
-
(1999)
FEBS Letters
, vol.451
, pp. 191-196
-
-
Eyers, P.A.1
van den Ijssel, P.2
Quinlan, R.A.3
Goedert, M.4
Cohen, P.5
-
51
-
-
0037115644
-
-
P. La Rosee, A. S. Corbin, E. P. Stoff-regen, M. W. Deininger, B. J. Druker, Cancer Res. 2002, 62, 7149-7153.
-
(2002)
Cancer Res.
, vol.62
, pp. 7149-7153
-
-
La Rosee, P.1
Corbin, A.S.2
Stoff-regen, E.P.3
Deininger, M.W.4
Druker, B.J.5
-
52
-
-
0037674323
-
-
S. Blencke, A. Ullrich, H. Daub, J. Biol. Chem. 2003, 278, 15435-15440.
-
(2003)
J. Biol. Chem.
, vol.278
, pp. 15435-15440
-
-
Blencke, S.1
Ullrich, A.2
Daub, H.3
-
54
-
-
0034086397
-
-
M. Knockaert, N. Gray, E. Damiens, Y. T. Chang, P. Grellier, K. Grant, D. Fergusson, J. Mottram, M. Soete, J. F. Dubremetz, K. Le Roch, C. Doerig, P. Schultz, L. Meijer, Chem. Biol. 2000, 7, 411-422.
-
(2000)
Chem. Biol.
, vol.7
, pp. 411-422
-
-
Knockaert, M.1
Gray, N.2
Damiens, E.3
Chang, Y.T.4
Grellier, P.5
Grant, K.6
Fergusson, D.7
Mottram, J.8
Soete, M.9
Dubremetz, J.F.10
Le Roch, K.11
Doerig, C.12
Schultz, P.13
Meijer, L.14
-
55
-
-
0037067733
-
-
M. Knockaert, K. Wieking, S. Schmitt, M. Leost, K. M. Grant,J. C. Mottram, C. Kunick, L. Meijer, J. Biol. Chem.2002, 277, 25493-25501.
-
(2002)
J. Biol. Chem
, vol.277
, pp. 25493-25501
-
-
Knockaert, M.1
Wieking, K.2
Schmitt, S.3
Leost, M.4
Grant, K.M.5
Mottram, J.C.6
Kunick, C.7
Meijer, L.8
-
56
-
-
0036310685
-
-
L. M. Schang, A. Bantly, M. Knockaert, F. Shaheen, L. Meijer, M. H. Malim, N. S. Gray, P. A. Schaffer, J. Virol. 2002, 76, 7874-7882.
-
(2002)
J. Virol.
, vol.76
, pp. 7874-7882
-
-
Schang, L.M.1
Bantly, A.2
Knockaert, M.3
Shaheen, F.4
Meijer, L.5
Malim, M.H.6
Gray, N.S.7
Schaffer, P.A.8
-
57
-
-
9144219693
-
-
K. Godl,J. Wissing, A. Kurtenbach, P. Habenberger, S. Blencke, H. Gutbrod, K. Salassidis, M. Stein-Gerlach, A. Missio, M. Cotten, H. Daub, Proc. Natl. Acad.Sci. USA 2003, 100, 15434-15439.
-
(2003)
Proc. Natl. Acad.Sci. USA
, vol.100
, pp. 15434-15439
-
-
Godl, K.1
Wissing, J.2
Kurtenbach, A.3
Habenberger, P.4
Blencke, S.5
Gutbrod, H.6
Salassidis, K.7
Stein-Gerlach, M.8
Missio, A.9
Cotten, M.10
Daub, H.11
-
58
-
-
0036318795
-
-
H. Daub, S. Blencke, P. Habenberger, A. Kurtenbach, J. Dennenmoser,J. Wissing, A. Ullrich, M. Cotten, J. Virol. 2002, 76, 8124-8137.
-
(2002)
J. Virol
, vol.76
, pp. 8124-8137
-
-
Daub, H.1
Blencke, S.2
Habenberger, P.3
Kurtenbach, A.4
Dennenmoser, J.5
Wissing, J.6
Ullrich, A.7
Cotten, M.8
-
59
-
-
0034306450
-
-
S. P. Davies, H. Reddy, M. Caivano, P. Cohen, Biochem. J. 2000, 351, 95-105.
-
(2000)
Biochem. J.
, vol.351
, pp. 95-105
-
-
Davies, S.P1
Reddy, H.2
Caivano, M.3
Cohen, P.4
-
60
-
-
0037075549
-
-
A. I. Chin, P. W. Dempsey, K. Bruhn, J. F. Miller, Y. Xu, G. Cheng, Nature 2002, 416, 190-194.
-
(2002)
Nature
, vol.416
, pp. 190-194
-
-
Chin, A.I.1
Dempsey, P.W.2
Bruhn, K.3
Miller, J.F.4
Xu, Y.5
Cheng, G.6
-
61
-
-
0037075551
-
-
K. Kobayashi, N. Inohara, L. D. Hernandez,J. E. Galán, G. Núnez, C. A. Janeway, R. Medzhitov, R. A. Flavell, Nature 2002, 416, 194-199.
-
(2002)
Nature
, vol.416
, pp. 194-199
-
-
Kobayashi, K.1
Inohara, N.2
Hernandez, L.D.3
Galán, J.E.4
Núnez, G.5
Janeway, C.A.6
Medzhitov, R.7
Flavell, R.A.8
|