Effect of supercritical CO2 plasticization on the degradation and residual crystallinity of melt-extruded spironolactone

Polymers for Advanced Technologies

Volumn 25, Issue 10, 2014, Pages 1135-1144

  Vigh, Tamás ^a   Sauceau, Martial ^b   Fages, Jacques ^b   Rodier, Elisabeth ^b   Wagner, István ^a   Sóti, Péter L ^a   Marosi, György ^a   Nagy, Zsombor K ^a  

^a BUDAPEST UNIVERSITY OF TECHNOLOGY AND ECONOMICS   (Hungary)

^b UNIVERSITÉ DE TOULOUSE   (France)

Author keywords

Amorphization; Degradation; Foaming; Immediate release; Supercritical fluid extrusion

Indexed keywords

AMORPHIZATION; CARBON DIOXIDE; CRYSTALLINITY; DEGRADATION; DISPERSIONS; DRUG PRODUCTS; EFFLUENT TREATMENT; EXTRUSION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; MELT SPINNING; RUNWAY FOAMING; SCANNING ELECTRON MICROSCOPY; SUPERCRITICAL FLUIDS; TARGETED DRUG DELIVERY;

ACTIVE PHARMACEUTICAL INGREDIENTS; CHEMOMETRIC ANALYSIS; CONTINUOUS MANUFACTURING; EXTRUSION TEMPERATURES; HOMOGENEOUS STRUCTURE; IMMEDIATE RELEASE; PLASTICIZING EFFECTS; SUPERCRITICAL FLUID EXTRUSION;

CONTROLLED DRUG DELIVERY;

EID: 84927796237     PISSN: 10427147     EISSN: 10991581     Source Type: Journal    
DOI: 10.1002/pat.3367     Document Type: Article

References (55)

1. Z. K. Nagy, A. Balogh, B. Vajna, A. Farkas, G. Patyi, Á. Kramarics, G. Marosi, J. Pharm. Sci. 2012, 101, 322-332. DOI: 10.1002/jps.22731
2. M. M. Crowley, F. Zhang, M. A. Repka, S. Thumma, S. B. Upadhye, S. K. Battu, J. W. McGinity, C. Martin, Drug Dev. Ind. Pharm. 2007, 33, 909-926. DOI: 10.1080/03639040701498759
3. M. A. Repka, S. K. Battu, S. B. Upadhye, S. Thumma, M. M. Crowley, F. Zhang, C. Martin, J. W. McGinity, Drug Dev. Ind. Pharm. 2007, 33, 1043-1057. DOI: 10.1080/03639040701525627
4. Z. K. Nagy, K. Nyúl, I. Wagner, K. Molnár, G. Marosi, Express Polym. Lett. 2010, 4, 763-772. DOI: 10.3144/expresspolymlett.2010.92
5. P. Kocbek, S. Baumgartner, J. Kristl, Int. J. Pharm. 2006, 312, 179-86. DOI: 10.1016/j.ijpharm.2006.01.008
6. C. Mártha, L. Kürti, G. Farkas, O. Jójárt-Laczkovich, B. Szalontai, E. Glässer, M. A. Deli, P. Szabo-Revesz, Eur. Polym. J. 2013, 49, 2426-2432. DOI: 10.1016/j.eurpolymj.2013.03.006
7. U.S. Department of Health and Human Services, Food and Drug Administration, 2004, http://www.fda.gov/downloads/Drugs/Guidances/ucm070305.pdf Date accessed: 11-02-2014.
8. J. Breitenbach, Eur. J. Pharm. Biopharm. 2002, 54, 107-117. DOI: 10.1016/S0939-6411(02)00061-9
9. J. Breitenbach, Am. J. Drug Deliv. 2006, 4, 61-64. DOI: 10.2165/00137696-200604020-00001
10. B. Vajna, H. Pataki, Z. Nagy, I. Farkas, G. Marosi, Int. J. Pharm. 2011, 419, 107-113. DOI: 10.1016/j.ijpharm.2011.07.023
11. J. C. DiNunzio, C. Brough, J. R. Hughey, D. A. Miller, R. O. Williams III, J. W. McGinity, Eur. J. Pharm. Biopharm. 2010, 74, 340-351. DOI: 10.1016/j.ejpb.2009.09.007
12. J. E. Patterson, M. B. James, A. H. Forster, R. W. Lancaster, J. M. Butler, T. Rades, Int. J. Pharm. 2007, 336, 22-34. DOI: 10.1016/j.ijpharm.2006.11.030
13. J. R. Hughey, J. M. Keen, C. Brough, S. Saeger, J. W. McGinity, Int. J. Pharm. 2011, 419, 222-230. DOI: 10.1016/j.ijpharm.2011.08.007
14. E. Petritz, T. Tritthart, R. Wintersteiger, J. Biochem. Biophys. Methods 2006, 69, 101-112. DOI: 10.1016/j.jbbm.2006.03.007
15. A. Krupa, D. Majda, R. Jachowicz, W. Mozgawa, Thermochim. Acta 2010, 509, 12-17. DOI: 10.1016/j.tca.2010.05.009
16. F. Kayaci, Y. Ertas, T. Uyar, J. Agric. Food Chem. 2013, 61, 8156-8165. DOI: 10.1021/jf402923c
17. Z. K. Nagy, M. Sauceau, K. Nyúl, E. Rodier, B. Vajna, G. Marosi, J. Fages, Polym. Adv. Technol. 2012, 23, 909-918. DOI: 10.1002/pat.1991
18. S. Li, M. Xiao, Y. Guan, D. Wei, H. Xiao, A. Zheng, Eur. Polym. J. 2012, 48, 362-371. DOI: 10.1016/j.eurpolymj.2011.11.015
19. G. Verreck, A. Decorte, K. Heymans, J. Adriaensen, D. H. Liu, D. L. Tomasko, A. Arien, J. Peeters, G. Van den Mooter, M. E. Brewster, Int. J. Pharm. 2006, 327, 45-50. DOI: 10.1016/j.ijpharm.2006.07.024
20. A. Salerno, U. Clerici, C. Domingo, Eur. Polym. J. 2014, 51, 1-11. DOI: 10.1016/j.eurpolymj.2013.11.015
21. G. Bánsághi, E. Székely, D. M. Sevillano, Z. Juvancz, B. Simándi, J. Supercrit. Fluids 2012, 69, 113-116. DOI: 10.1016/j.supflu.2012.05.016
22. C. Ortuño, T. Duong, M. Balaban, J. Benedito, J. Supercrit. Fluids 2013, 82, 56-62. DOI: 10.1016/j.supflu.2013.06.005
23. S. S. H. Rizvi, S. J. Mulvaney, A. S. Sokhey, Trends Food Sci. Technol. 1995, 6, 232-240. DOI: 10.1016/S0924-2244(00)89084-6
24. M. Sauceau, J. Fages, A. Common, C. Nikitine, E. Rodier, Prog. Polym. Sci. 2011, 36, 749-766. DOI: 10.1016/j.progpolymsci.2010.12.004
25. G. Verreck, A. Decorte, K. Heymans, J. Adriaensen, D. Cleeren, A. Jacobs, D. H. Liu, D. L. Tomasko, A. Arien, J. Peeters, P. Rombaut, G. Van den Mooter, M. E. Brewster, Eur. J. Pharm. Sci. 2005, 26, 349-58. DOI: 10.1016/j.ejps.2005.07.006
26. G. Verreck, A. Decorte, K. Heymans, J. Adriaensen, D. Liu, D. L. Tomasko, A. Arien, J. Peeters, P. Rombaut, G. Van den Mooter, M. E. Brewster, J. Supercrit. Fluids 2007, 40, 153-162. DOI: 10.1016/j.supflu.2006.05.005
27. G. Verreck, A. Decorte, H. Li, D. Tomasko, A. Arien, J. Peeters, P. Rombaut, G. Van den Mooter, M. E. Brewster, J. Supercrit. Fluids 2006, 38, 383-391. DOI: 10.1016/j.supflu.2005.11.022
28. A. Dolenc, J. Kristl, S. Baumgartner, O. Planinsek, Int. J. Pharm. 2009, 376, 204-12. DOI: 10.1016/j.ijpharm.2009.04.038
29. C. Nikitine, E. Rodier, M. Sauceau, J.-J. Letourneau, J. Fages, J. Appl. Polym. Sci. 2010, 115, 981-990. DOI: 10.1002/app.31031
30. M. D. Hargreaves, N. A. Macleod, M. R. Smith, D. Andrews, S. V. Hammond, P. Matousek, J. Pharm. Biomed. Anal. 2011, 54, 463-468. DOI: 10.1016/j.jpba.2010.09.015
31. A. Aina, M. D. Hargreaves, P. Matousek, J. C. Burley, Analyst 2010, 135, 2328-2333. DOI: 10.1039/c0an00352b
32. S. Šašić, S. Mehrens, Anal. Chem. 2011, 84, 1019-1025. DOI: 10.1021/ac202396u
33. A. Heinz, M. Savolainen, T. Rades, C. J. Strachan, Eur. J. Pharm. Sci. 2007, 32, 182-192. DOI: 10.1016/j.ejps.2007.07.003
34. Z. Német, G. C. Kis, G. Pokol, Á. Demeter, J. Pharm. Biomed. Anal. 2009, 49, 338-346. DOI: 10.1016/j.jpba.2008.11.033
35. L. Nørgaard, M. T. Hahn, L. B. Knudsen, I. A. Farhat, S. B. Engelsen, Int. Dairy J. 2005, 15, 1261-1270. DOI: 10.1016/j.idairyj.2004.12.009
36. E. Widjaja, P. Kanaujia, G. Lau, W. K. Ng, M. Garland, C. Saal, A. Hanefeld, M. Fischbach, M. Maio, R. B. H. Tan, Eur. J. Pharm. Sci. 2011, 42, 45-54. DOI: 10.1016/j.ejps.2010.10.004
37. K. Nakamoto, T. Urasaki, S. Hondo, N. Murahashi, E. Yonemochi, K. Terada, J. Pharm. Biomed. Anal. 2013, 75, 105-111. DOI: 10.1016/j.jpba.2012.11.020
38. H. Pataki, I. Markovits, B. Vajna, Z. K. Nagy, G. Marosi, Cryst. Growth Des. 2012, 12, 5621-5628. DOI: 10.1021/cg301135z
39. H. Pataki, I. Csontos, Z. K. Nagy, B. Vajna, M. Molnar, L. Katona, G. Marosi, Org. Process Res. Dev. 2013, 17, 493-499. DOI: 10.1021/op300062t
40. T. Seki, J. Mochida, M. Okamoto, O. Hosoya, K. Juni, K. Morimoto, Chem. Pharm. Bull. 2003, 51, 734-736. DOI: 10.1248/cpb.51.734
41. J. L. Sutter, E. P. K. Lau, In: Anal. Profiles Drug Subst., Vol. 4 (Ed.: F. Klaus ), Academic Press, London, 1975, pp.431-451.
42. M. Sauceau, C. Nikitine, E. Rodier, J. Fages, J. Supercrit. Fluids 2007, 43, 367-373. DOI: 10.1016/j.supflu.2007.05.014
43. National Institute of Standards and Technology, http://webbook.nist.gov/chemistry/ Date accessed: 05/02/2014.
44. R. Span, W. Wagner, J. Phys. Chem. Ref. Data 1996, 25, 1509-1596. DOI: 10.1063/1.555991
45. M. Fukuda, N. A. Peppas, J. W. McGinity, J. Control. Release 2006, 115, 121-129. DOI: 10.1016/j.jconrel.2006.07.018
46. D. W. Van Krevelen, Properties of polymers: their correlation with chemical structure, their numerical estimation and prediction from additive group contributions, Elsevier, Amsterdam, 1997.
47. H. E. Naguib, C. B. Park, U. Panzer, N. Reichelt, Polym. Eng. Sci. 2002, 42, 1481-1492. DOI: 10.1002/pen.11045
48. C. B. Park, A. H. Behravesh, R. D. Venter, Polym. Eng. Sci. 1998, 38, 1812-1823. DOI: 10.1002/pen.10351
49. W. Wang, A. H. Barber, J. Polym. Sci. Part B Polym. Phys. 2012, 50, 546-551. DOI: 10.1002/polb.23030
50. M. Fejos, K. Molnár, J. Karger-Kocsis, Materials (Basel). 2013, 6, 4489-4504. DOI: 10.3390/ma6104489
51. K. Y. Cho, S. S. H. Rizvi, Food Res. Int. 2009, 42, 603-611. DOI: 10.1016/j.foodres.2008.12.015
52. G. Verreck, I. Chun, J. Rosenblatt, J. Peeters, A. Van Dijck, J. Mensch, M. Noppe, M. E. Brewster, J. Control. Release 2003, 92, 349-360. DOI: 10.1016/S0168-3659(03)00342-0
53. M. Poostforush, H. Azizi, eXPRESS Polym. Lett. 2014, 8, 293-299. DOI: 10.3144/expresspolymlett.2014.32
54. T. Vigh, T. Horváthová, A. Balogh, P. L. Sóti, G. Drávavölgyi, Z. K. Nagy, G. Marosi, Eur. J. Pharm. Sci. 2013, 49, 595-602. DOI: 10.1016/j.ejps.2013.04.034
55. O. Rajabi, F. Tayyari, R. Salari, S. F. Tayyari, J. Mol. Struct. 2008, 878, 78-83. DOI: 10.1016/j.molstruc.2007.07.043