Development of a universal radioactive DNA methyltransferase inhibition test for high-throughput screening and mechanistic studies

Nucleic Acids Research

Volumn 41, Issue 19, 2013, Pages

  Gros, Christina ^a   Chauvigné, Laura ^a   Poulet, Anaïs ^a   Menon, Yoann ^a   Ausseil, Frédéric ^a   Dufau, Isabelle ^a   Arimondo, Paola B ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

DNA METHYLTRANSFERASE 3A; SINEFUNGIN;

ARTICLE; CARBOXY TERMINAL SEQUENCE; CATALYSIS; DNA DETERMINATION; DNA METHYLATION; DNA METHYLTRANSFERASE INHIBITION TEST; FEASIBILITY STUDY; HIGH THROUGHPUT SCREENING; IC 50; MICHAELIS MENTEN KINETICS; POLYMERASE CHAIN REACTION; PRIORITY JOURNAL; PROCESS OPTIMIZATION; PROTEIN BINDING; PROTEIN DOMAIN;

CELL EXTRACTS; CELL LINE; DIMETHYL SULFOXIDE; DNA (CYTOSINE-5-)-METHYLTRANSFERASE; DNA METHYLATION; ENZYME INHIBITORS; HIGH-THROUGHPUT SCREENING ASSAYS; HUMANS; SOLVENTS; TRITIUM;

EID: 84885974734     PISSN: 03051048     EISSN: 13624962     Source Type: Journal    
DOI: 10.1093/nar/gkt753     Document Type: Article

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