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Volumn 12, Issue 9, 2011, Pages 1337-1345

C5-DNA Methyltransferase Inhibitors: From Screening to Effects on Zebrafish Embryo Development

(17) Ceccaldi, Alexandre a Rajavelu, Arumugam b Champion, Christine a Rampon, Christine c Jurkowska, Renata b Jankevicius, Gytis b Sénamaud Beaufort, Catherine a Ponger, Loïc a Gagey, Nathalie a Dali Ali, Hana a Tost, Jörg d Vriz, Sophie c Ros, Sindu e Dauzonne, Daniel e Jeltsch, Albert b Guianvarc'h, Dominique c Arimondo, Paola B a

a MUSÉUM NATIONAL D'HISTOIRE NATURELLE (France)

b JACOBS UNIVERSITY BREMEN (Germany)

c CNRS (France)

d CENTRE NATIONAL DE GÉNOTYPAGE (France)

e INSTITUT CURIE (France)

Author keywords

DNA methylation; DNMT; Flavones; High throughput screening; Inhibitors

Indexed keywords

AZACITIDINE; DNA METHYLTRANSFERASE; DNA METHYLTRANSFERASE 3A; DNA METHYLTRANSFERASE 3L; DNA METHYLTRANSFERASE INHIBITOR; FLAVANONE DERIVATIVE; FLAVONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DEMETHYLATION; DRUG MECHANISM; DRUG STRUCTURE; EMBRYO; EMBRYO DEVELOPMENT; ENZYME ACTIVITY; ENZYME INHIBITION; HIGH THROUGHPUT SCREENING; IC 50; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; ZEBRA FISH;

ANIMALS; BASE SEQUENCE; CRYSTALLOGRAPHY, X-RAY; DNA (CYTOSINE-5-)-METHYLTRANSFERASE; EMBRYONIC DEVELOPMENT; ENZYME INHIBITORS; MICE; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; SMALL MOLECULE LIBRARIES; ZEBRAFISH;

DANIO RERIO; MURINAE;

EID: 79958746640 PISSN: 14394227 EISSN: 14397633 Source Type: Journal
DOI: 10.1002/cbic.201100130 Document Type: Article

Times cited : (70)

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